Apoptosi
Gli inibitori dell'apoptosi sono composti che prevengono o ritardano il processo di morte cellulare programmata, noto come apoptosi. Questi inibitori sono fondamentali per lo studio dei meccanismi di sopravvivenza cellulare e vengono utilizzati per indagare sulle malattie in cui l'apoptosi è disregolata, come il cancro, i disturbi neurodegenerativi e le malattie autoimmuni. Modulando l'apoptosi, questi inibitori possono aiutare nello sviluppo di terapie mirate a controllare la morte cellulare. Presso CymitQuimica, offriamo una vasta selezione di inibitori dell'apoptosi di alta qualità per supportare le tue ricerche in biologia cellulare, oncologia e campi correlati.
Sottocategorie di "Apoptosi"
- ASK(9 prodotti)
- BCL(3 prodotti)
- Caspasi(153 prodotti)
- FOXO1(2 prodotti)
- IAP(67 prodotti)
- Mdm2(12 prodotti)
- PD-1/PD-L1(93 prodotti)
- PDK(9 prodotti)
- PERK(26 prodotti)
- Chinasi di serina/treonina(18 prodotti)
- Survivin(14 prodotti)
- TNF(49 prodotti)
- c-RET(60 prodotti)
- p53(63 prodotti)
Mostrare 6 più sottocategorie
Trovati 6032 prodotti di "Apoptosi"
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IM-54
CAS:IM-54 is a cell-permeable, effective, and selective necrosis inhibitor.Formula:C19H23N3O2Purezza:99.24%Colore e forma:SolidPeso molecolare:325.4Ref: TM-T24160
1mg49,00€5mg104,00€10mg164,00€25mg281,00€50mg404,00€100mg567,00€1mL*10mM (DMSO)115,00€Topoisomerase II inhibitor 9
CAS:Topoisomerase II inhibitor 9: Topo II blocker (IC50: 0.97 μM), DNA intercalator (IC50: 43.51 μM), arrests G2/M in Hep G-2 cells and triggers apoptosis.
Formula:C22H17N7O3S2Colore e forma:SolidPeso molecolare:491.55S130
CAS:S130 is a high affinity, selectiveATG4B (a major cysteine protease) inhibitor (IC50 of 3.24 μM).It suppresses autophagy flux.Formula:C24H25N3O2Purezza:98%Colore e forma:SolidPeso molecolare:387.47KRAS G12D inhibitor 14
CAS:KRAS G12D inhibitor 14 is a potent inhibitor of KRAS G12D that binds KRAS G12D protein (Kd: 33 nM).
Formula:C20H19F3N4OSPurezza:>99.99%Colore e forma:SolidPeso molecolare:420.45RET-IN-22
CAS:RET-IN-22 (compound 17b) is a potent, selective, and orally active inhibitor of RET, exhibiting IC50 values of 20.9 nM for wild-type RET and 18.3 nM for RET-Formula:C29H31F3N6O4Colore e forma:SolidPeso molecolare:584.59CMLD012073
CAS:CMLD012073: Potent eIF4A inhibitor, halts eukaryotic translation; IC50 10 nM in NIH/3T3 cells.Formula:C30H30N2O7Purezza:98%Colore e forma:SolidPeso molecolare:530.57Topoisomerase I inhibitor 5
CAS:Topoisomerase I inhibitor 5 halts DNA replication, induces MCF-7 cell apoptosis, and overcomes drug resistance. IC50 value is noted.Formula:C24H24N2O2Colore e forma:SolidPeso molecolare:372.46CMLD010509
CAS:CMLD010509 (SDS-1-021) inhibits oncogenic proteins MDM2, CCND1, MYC, MAF, MCL-1 in multiple myeloma.Formula:C27H26BrNO7Purezza:98%Colore e forma:SolidPeso molecolare:556.4Methylisothiazolinone
CAS:Methylisothiazolinone (MI) is a powerful synthetic biocide and preservative within the group of isothiazolinones.Formula:C4H5NOSPurezza:99.78%Colore e forma:Colorless Prisms LiquidPeso molecolare:115.15Nampt-IN-3
CAS:Nampt-IN-3 simultaneously inhibit nicotinamide phosphoribosyltransferase (NAMPT) and HDAC (IC50s of 31 nM and 55 nM, respectively).Formula:C29H25N7O2Purezza:98%Colore e forma:SolidPeso molecolare:503.55CCT373567
CAS:CCT373567 is a potent degrader of the transcriptional repressor BCL6 (IC50: 2.9 nM) and exhibits anti-proliferative effects.Formula:C26H29ClF2N6O3Colore e forma:SolidPeso molecolare:547CEP-40125
CAS:CEP-40125 (RXDX-107) is a DNA alkylating agent for the study of advanced solid tumors.Formula:C28H45Cl2N3O2Purezza:98.28%Colore e forma:SolidPeso molecolare:526.58Topoisomerase II inhibitor 3
CAS:Acridone-based Topoisomerase II inhibitor 3 targets topo IIα/β (IC50: 0.17μM α, 0.23μM β), causes DNA damage, and induces apoptosis.Formula:C18H20N4O4Colore e forma:SolidPeso molecolare:356.38MMP-9-IN-4
CAS:MMP-9-IN-4 inhibits MMP-9 (IC50=7.46nM) and AKT (IC50=8.82nM), induces apoptosis and is used in cancer research.Formula:C28H19F3N4O6Colore e forma:SolidPeso molecolare:564.47Apoptotic agent-2
CAS:Apoptotic agent-2 reduces Bcl-2, boosts Bax & caspase-3, inducing apoptosis for cancer research.Formula:C25H16ClN7SColore e forma:SolidPeso molecolare:481.96Tezacitabine
CAS:Tezacitabine, a nucleoside analogue, inhibits ribonucleotide reductase, disrupts DNA replication, and induces apoptosis in tumor cells.Formula:C10H12FN3O4Colore e forma:SolidPeso molecolare:257.22Cinnabarinic acid
CAS:mGlu4 receptor agonistFormula:C14H8N2O6Purezza:98%Colore e forma:SolidPeso molecolare:300.22PDE5/HDAC-IN-1
CAS:PDE5/HDAC-IN-1 is a potent inhibitor of phosphodiesterase 5 (PDE5) and HDAC, with IC50 values of 46.3 nM and 14.5 nM, respectively.Formula:C27H29BrN4O4Colore e forma:SolidPeso molecolare:553.45RET-IN-12
CAS:RET-IN-12 is a RET inhibitor capable of acting on RET(WT) (IC50: 0.3 nM) and RET(V804M) (IC50: 1 nM).Formula:C30H30F3N5O4Colore e forma:SolidPeso molecolare:581.59Antitumor agent-44
CAS:Antitumor agent-44 (Compound 5n) elicits potent antitumor effects by inducing disruption of mitochondrial homeostasis, cell cycle arrest, and apoptosis in humanFormula:C24H15N3O3Colore e forma:SolidPeso molecolare:393.39BR102375
CAS:BR102375 is a non-TZD PPAR γ full agonist (EC50: 0.28 μM) for the treatment of type 2 diabetes.Formula:C31H34N6O4Purezza:98%Colore e forma:SolidPeso molecolare:554.64Flonoltinib
CAS:Flonoltinib (JAK2/FLT3-IN-1) is an orally active and efficient JAK2/FLT3 inhibitor with anti-cancer properties.Formula:C25H34FN7OPurezza:99.52%Colore e forma:SolidPeso molecolare:467.58NKP-1339
CAS:NKP-1339 (IT-139) induces G2/M cell cycle arrest, blockage of DNA synthesis, and induction of apoptosis via the mitochondrial pathway.Formula:C14H12Cl4N4NaRuPurezza:98%Colore e forma:SolidPeso molecolare:502.14GRI977143
CAS:GRI977143: selective LPA2 agonist (EC50=3.3μM), blocks caspases 3/7/8/9, limits DNA fragmentation.Formula:C22H17NO4SPurezza:99.08%Colore e forma:SolidPeso molecolare:391.44N1,N11-Diethylnorspermine
CAS:DENSPM: potent anticancer, spurs polyamine breakdown, triggers cytochrome c release and caspase 3, kills GBM via SSAT & H2O2.Formula:C13H32N4Colore e forma:SolidPeso molecolare:244.42W1131
CAS:W1131 is a potent STAT3 inhibitor and ferroptosis trigger, reducing cancer progression and 5-FU resistance.Formula:C23H19N5O4Colore e forma:SolidPeso molecolare:429.43LLL3
CAS:LLL3 is a small molecule STAT3 inhibitor.Formula:C16H10O4Colore e forma:SolidPeso molecolare:266.25PDK4-IN-1
CAS:PDK4-IN-1 is an anthraquinone derivative and a potent and orally active inhibitor of pyruvate dehydrogenase kinase 4 (PDK4)(IC50 value of 84 nM).Formula:C22H19N3O2Purezza:98%Colore e forma:SolidPeso molecolare:357.41VMY-1-103
CAS:VMY-1-103: a strong CDK inhibitor better than purvalanol B; halts prostate/breast cancer cell growth, induces apoptosis, may treat medulloblastoma.Formula:C34H42ClN9O4SColore e forma:SolidPeso molecolare:708.27PI3K/AKT-IN-2
CAS:PI3K/AKT-IN-2 inhibits PI3K/AKT, EMT, induces apoptosis, and blocks tubulin polymerization.Formula:C32H27BrO10Colore e forma:SolidPeso molecolare:651.45DC-CPin711
CAS:DC-CPin711: Potent, selective CBP bromodomain inhibitor, IC50=0.0626 μM; arrests G1 cell cycle, induces apoptosis.Formula:C23H22N4O2Colore e forma:SolidPeso molecolare:386.45Semapimod
CAS:Semapimod is an inhibitor of proinflammatory cytokine production, capable of suppressing TNF-α, IL-1β, and IL-6.Formula:C34H52N18O2Colore e forma:SolidPeso molecolare:744.9Didesmethylrocaglamide
CAS:Didesmethylrocaglamide, a Rocaglamide derivative, is a potent eukaryotic initiation factor 4A (eIF4A) inhibitor that exhibits strong growth-inhibitory effects,Formula:C27H27NO7Colore e forma:SolidPeso molecolare:477.51Mcl1-IN-4
CAS:Mcl1-IN-4 is an inhibitor of Mcl1 ( IC50:0.2 μM).Formula:C28H26N2O5SPurezza:98%Colore e forma:SolidPeso molecolare:502.58CRA-026440
CAS:CRA-026440(PCI-34051) is a highly potent HDAC inhibitor with inhibitory effects on HDAC1, HDAC2, HDAC3, HDAC6, HDAC8 and HDAC10 with Ki values of 4,14,11,15,7Formula:C23H24N4O4Purezza:96.42%Colore e forma:SolidPeso molecolare:420.46PDGFR-IN-1
CAS:PDGFR-IN-1 is a platelet-derived growth factor receptor (PDGFR) inhibitor, strongly inhibiting PDGFRα and PDGFRβ, useful for studying solid tumors.Formula:C25H30N8OPurezza:99.13% - 99.49%Colore e forma:SolidPeso molecolare:458.56Ref: TM-T62872
1mg170,00€5mg432,00€10mg655,00€25mg1.153,00€50mg1.665,00€100mg2.250,00€1mL*10mM (DMSO)434,00€BRD4 Inhibitor-15
CAS:BRD4 Inhibitor-15 targets BRD4 with 18 nM IC50, induces apoptosis in 22RV1 cells, and lowers c-Myc, aiding prostate cancer research.Formula:C22H21N3O2Colore e forma:SolidPeso molecolare:359.42IHMT-TRK-284
CAS:IHMT-TRK-284: Oral type II TRK inhibitor; targets TRKA, TRKB, TRKC (IC50s: 10.5, 0.7, 2.6 nM); selective and anti-tumor effective.Formula:C25H27N7OSColore e forma:SolidPeso molecolare:473.59LY5
CAS:LY5 is an inhibitor of STAT3 that acts by inhibiting cell viability, cell migration, and angiogenesis in medulloblastoma cells.Formula:C15H11N3O4SPurezza:98%Colore e forma:SolidPeso molecolare:329.33MSN-50
CAS:MSN-50, an inhibitor of Bax and Bak oligomerization, inhibits liposome permeabilization, prevents genotoxic cell death and promotes neuroprotection.Formula:C36H38BrN3O6Colore e forma:SolidPeso molecolare:688.61PD180970
CAS:PD180970 is an inhibitor of Bcr-Abl with IC50s of 5 nM, 0.8 nM and 50 nM for the autophosphorylation of p210Bcr-Abl, Src and Kit.Formula:C21H15Cl2FN4OPurezza:98.67%Colore e forma:SolidPeso molecolare:429.27Ref: TM-T23128
5mg55,00€10mg92,00€25mg137,00€50mg198,00€100mgPrezzo su richiesta1mL*10mM (DMSO)60,00€PARP-1-IN-2
CAS:PARP-1-IN-2 is a potent PARP1 inhibitor that crosses the blood-brain barrier (IC50: 149 nM).PARP-1-IN-2 showed significant antiproliferative activity against
Formula:C22H15Cl2N3O2Purezza:98.82%Colore e forma:SolidPeso molecolare:424.28PAK4-IN-2
CAS:PAK4-IN-2 inhibits PAK4 with IC50 2.7 nM, arrests MV4-11 cells at G0/G1, and induces apoptosis, promising for cancer research.Formula:C18H21ClN6Colore e forma:SolidPeso molecolare:356.85Verrucarin J
CAS:Verrucarin J, a Myrothecium fungus metabolite, triggers apoptosis in some cancer cells and fights Candida, Mucor, and JUNV (IC50: 1.2 ng/mL).Formula:C27H32O8Colore e forma:SolidPeso molecolare:484.54Prexasertib mesylate
CAS:Prexasertib (LY2606368), a Chk1/2 inhibitor, enhances therapy in acute lymphoblastic leukemia, causing DNA damage and antitumor effects.Formula:C19H23N7O5SPurezza:98%Colore e forma:SolidPeso molecolare:461.49ABT-100
CAS:ABT-100 is a potent, highly selective, and orally active farnesyl transferase inhibitor with broad-spectrum antitumor activity.Formula:C27H19F3N4O3Purezza:98%Colore e forma:SolidPeso molecolare:504.46RIPK1-IN-15
CAS:RIPK1-IN-15 (Compound 2.5) is a potent RIPK1 inhibitor that has the potential in neurodegenerative, autoimmune, and inflammatory diseases research [1].Formula:C19H19N3O2Colore e forma:SolidPeso molecolare:321.37HDAC-IN-31
CAS:HDAC-IN-31: Oral HDAC inhibitor; targets HDAC1, 2, 3; weak on HDAC8; potential in fighting lymphoma.Formula:C25H24N4O2Colore e forma:SolidPeso molecolare:412.48AG6033
CAS:AG6033, a novel CRBN modulator, degrades GSPT1/IKZF1 and inhibits various tumors.Formula:C30H23N5O4Colore e forma:SolidPeso molecolare:517.53CMLD012072
CAS:CMLD012072 is a potent eukaryotic initiation factor 4A (eIF4A) inhibitor with potent anti-neoplastic activity. It can induce RNA clamping of eIF4A1 and eIF4A2.Formula:C32H32N2O7Purezza:98%Colore e forma:SolidPeso molecolare:556.61VRT-043198
CAS:VRT-043198, a VX-765 metabolite, is a potent ICE/caspase-1 inhibitor, crossing the blood-brain barrier with K i of 0.8/0.6 nM.Formula:C22H29ClN4O6Colore e forma:SolidPeso molecolare:480.94HJC0416
CAS:HJC0416 is a potent orally bioavailable signal transducer and activator of transcription 3 inhibitor.Formula:C18H17ClN2O4SPurezza:98%Colore e forma:SolidPeso molecolare:392.86CDK1/Cyc B-IN-1
CAS:CDK1/Cyc B-IN-1: Potent CDK1/Cyc B inhibitor, IC50 97 nM, induces apoptosis, arrests G2/M cycle, halts cancer growth.Formula:C14H12ClN3O2S2Colore e forma:SolidPeso molecolare:353.85SDZ 224-015
CAS:SDZ 224-015 is an inhibitor of interleukin-1β (IL-1β) converting enzyme and caspase-1 with anti-COVID-19 and anti-inflammatory activity.Formula:C30H35Cl2N3O9Purezza:95.49% - 95.49%Colore e forma:SolidPeso molecolare:652.52Epofolate
CAS:Epofolate: folate receptor-targeted antimitotic, delivers epothilone to cancer cells, inhibits mitosis, may halt tumor growth. Check clinical trials.Formula:C67H92N16O22S3Colore e forma:SolidPeso molecolare:1569.74Vin-C01
CAS:Vin-C01, a potent protector of pancreatic β-cells (EC50=0.22μM), aids in type 2 diabetes research by preventing STZ-induced β-cell apoptosis.Formula:C20H24N2OColore e forma:SolidPeso molecolare:308.42Esuberaprost Sodium
CAS:Famitinib (SHR1020), an oral drug, inhibits c-kit, VEGFR-2, and PDGFRβ (IC50: 2.3/4.7/6.6 nM) and triggers apoptosis in gastric cancer.Formula:C23H27FN4O2Colore e forma:SolidPeso molecolare:410.48Oxythiamine chloride HCl
CAS:Oxythiamine chloride is a thiamine antagonist and anticancer agent that inhibits transketolase, affecting RNA/DNA synthesis and inducing apoptosis.Formula:C12H17Cl2N3O2SColore e forma:SolidPeso molecolare:338.25PI3Kα-IN-6
CAS:PI3Kα-IN-6 (Compound 5b) is a PI3Kα inhibitor that exhibits anticancer effects without toxicity to normal cells.Formula:C16H15IN2OSColore e forma:SolidPeso molecolare:410.27Prinomastat hydrochloride
CAS:Prinomastat HCl, an oral MMP (1, 3, 9) inhibitor, IC50s: 79, 6.3, 5.0 nM, shows antitumor activity.
Formula:C18H22ClN3O5S2Purezza:98%Colore e forma:SolidPeso molecolare:459.97Topoisomerase I inhibitor 2
CAS:ZML-8 selectively inhibits Top1, blocks G2/M phase, causes DNA damage, and induces apoptosis with anti-tumor properties.Formula:C18H15NO3Colore e forma:SolidPeso molecolare:293.32PDE5-IN-3
CAS:PDE5-IN-3: Inhibits PDE5 (1.57 nM), EGFR (5.827 μM), Wnt pathway (1286.96 ng/mL), induces apoptosis, and has antitumor effects.Formula:C21H14BrN5O2Colore e forma:SolidPeso molecolare:448.27Dipin
CAS:Dipin is an Antineoplastic.Formula:C12H24N6O2P2Purezza:98%Colore e forma:SolidPeso molecolare:346.31PHA-690509
CAS:PHA-690509 is a cyclin-dependent kinase 2 inhibitor. It potentially for the treatment of cancer.Formula:C17H21N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:331.43Antitumor agent-83
Antitumor agent-83 activates BAX protein, impedes tumor growth, triggers apoptosis, and is stable in vitro.Formula:C29H30N6O2Colore e forma:SolidPeso molecolare:494.59Atopaxar
CAS:Atopaxar (E5555), a reversible PAR-1 thrombin receptor antagonist, interferes with platelet signaling.Formula:C29H38FN3O5Purezza:97.07% - 98.07%Colore e forma:SolidPeso molecolare:527.63CAY10506
CAS:CAY10506, a hybrid lipoic acid-TZD, activates PPARγ to control glucose and lipid levels with an EC50 of 10 μM.Formula:C20H26N2O4S3Colore e forma:SolidPeso molecolare:454.63PhiKan 083 hydrochloride
CAS:PhiKan 083 HCl: carbazole, binds Y220C (Kd 167 μM), affinity in Ln229 (Kd 150 μM).Formula:C16H19ClN2Purezza:98%Colore e forma:SolidPeso molecolare:274.79Mutant p53 modulator-1
CAS:Mutant p53 modulator-1 inhibits cancer with p53 mutations; see patent WO2021231474A1, compound 231B.Formula:C27H32F4N8O2Colore e forma:SolidPeso molecolare:576.59FKGK 18
CAS:FKGK 18: GVIA iPLA2 inhibitor, 99.9% at 0.091 fraction, selective, IC50 ~50 nM–3 μM, reduces blood glucose and diabetes in NOD mice.Formula:C16H15F3OColore e forma:SolidPeso molecolare:280.28QM31
CAS:QM31 is a selective Apaf-1 inhibitor(inbitita formation of the apoptosome with IC50 of 7.9μM).Formula:C39H38Cl4N4O4Purezza:98%Colore e forma:SolidPeso molecolare:768.56RIP1 kinase inhibitor 6
CAS:RIP1 Kinase Inhibitor 6 is a potent and selective inhibitor of RIP1 kinase, demonstrating inhibitory activity with an IC50 of less than 100 nM in a human R1P1Formula:C19H18F2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:360.35EGFR-IN-59
CAS:EGFR-IN-59: EGFR inhibitor, IC50 = 190 nM, induces apoptosis, cytotoxic to A549 cells (IC50 = 8.62 μM) and WI38 cells (IC50 = 52.6 μM). Use: Various cancers.Formula:C27H23N5O4SColore e forma:SolidPeso molecolare:513.57RET-IN-8
CAS:RET-IN-8 is an inhibitor of rearrangement kinase (RET) during transfection and can be used in cancer research.Formula:C27H30N6O3Colore e forma:SolidPeso molecolare:486.57Sanazole
CAS:Sanazole is a 3-nitrotriazole cpd. It can affect the human cervical cancer cell line.Formula:C7H11N5O4Colore e forma:SolidPeso molecolare:229.19DX2-201
CAS:DX2-201 is a potent and selective inhibitor of oxidative phosphorylation (OXPHOS) complex I (IC50: 312 nM) and exhibits anticancer activity.Formula:C18H28N2O6S2Colore e forma:SolidPeso molecolare:432.55SB-218078
CAS:SB-218078 is less potently inhibits Cdc2 (IC50: 250 nM) and PKC (IC50: 1000 nM).Formula:C24H15N3O3Purezza:98%Colore e forma:SolidPeso molecolare:393.39EGFR-IN-46
CAS:EGFR-IN-46: Potent EGFR/FAK inhibitor (IC50: 20.17 & 14.25 nM), curbs cancer cell growth, triggers apoptosis.Formula:C27H32F3N3O3Colore e forma:SolidPeso molecolare:503.56Tubulin/HDAC-IN-1
CAS:Tubulin/HDAC-IN-1 is a dual inhibitor for tubulin & HDAC8, blocking polymerization & targeting HDAC8 (IC50: 150 nM), and induces cancer cell apoptosis.Formula:C21H18N4O3Colore e forma:SolidPeso molecolare:374.39PD-1/PD-L1-IN-14
CAS:PD-1/PD-L1-IN-14 (compound 17) is an inhibitor of PD-1/PD-L1 interaction (IC50=27.8 nM).Formula:C24H24N4O2Colore e forma:SolidPeso molecolare:400.47T-3256336
CAS:T-3256336 is an oral IAP blocker targeting cIAP-1, cIAP-2, and XIAP.Formula:C31H45F2N5O5Purezza:98%Colore e forma:SolidPeso molecolare:605.72BTK-IN-9
CAS:BTK-IN-9 reversibly inhibits BTK, disrupts mitochondria, boosts ROS, and triggers apoptosis in Z138 cells, impeding condyloma cell growth.Formula:C25H19N7O4Colore e forma:SolidPeso molecolare:481.46Pentabromophenol
CAS:Pentabromophenol (NSC-5717) suppressed TGF-β response by accelerating the turnover rate of TGF-β receptors.Formula:C6HBr5OPurezza:99.83%Colore e forma:Monoclinic Prisms From Acetic Acid; Needles From Alcohol Physical Description Light Brown Powder Insoluble In Water (Ntp 1992)Peso molecolare:488.59RIPK1-IN-3
CAS:RIPK1-IN-3 is a RIPK1 inhibitor, with anti-inflammatory proprieties.Formula:C22H19F3N6O3Purezza:98%Colore e forma:SolidPeso molecolare:472.42Anti-inflammatory agent 11
CAS:Potent anti-inflammatory compound 16 combats tuberculosis, inhibiting Mtb H37Rv and M299 (MICs: 1.3, 6.9 μM) and reduces NO, TNF-α, IL-1β production.Formula:C14H14N4OSColore e forma:SolidPeso molecolare:286.35DCP-LA
CAS:DCP-LA (FR236924), linoleic acid derivatives, selective and direct activation of PKCε.Formula:C20H36O2Purezza:98%Colore e forma:SolidPeso molecolare:308.5MCL-1/BCL-2-IN-4
CAS:MCL-1/BCL-2-IN-4 is a selective and potent Mcl-1 and Bcl-2 dual inhibitor.Formula:C26H23BrN2O5SPurezza:98%Colore e forma:SolidPeso molecolare:555.44EL-102
CAS:EL-102 is a HIF1α inhibitor with anticancer activity that inhibits microtubule protein polymerization and can be used to study prostate cancer.Formula:C19H16N2O3S2Purezza:99.34%Colore e forma:SolidPeso molecolare:384.47Ref: TM-T15205
1mg93,00€5mg205,00€10mg331,00€25mg515,00€50mg700,00€100mg1.044,00€1mL*10mM (DMSO)173,00€Irbesartan HCl
CAS:Irbesartan: angiotensin II blocker; treats hypertension by inhibiting receptor binding.Formula:C25H29ClN6OPurezza:98%Colore e forma:SolidPeso molecolare:465(E)-[6]-Dehydroparadol
CAS:(E)-[6]-Dehydroparadol ((6)-Dehydroparadol), an oxidative metabolite of [6]-Shogaol, is a potent Nrf2 activator.Formula:C17H24O3Purezza:99.85%Colore e forma:SolidPeso molecolare:276.37Ref: TM-T13436
1mg42,00€2mg34,00€5mg52,00€10mg73,00€25mg122,00€50mg166,00€100mg231,00€500mg872,00€1mL*10mM (DMSO)58,00€K-7174 dihydrochloride
CAS:K-7174 dihydrochloride is a novel cell adhesion inhibitor; inhibits the expression of vascular cell adhesion molecule-1 (VCAM-1) induced by either IL-1β or TNF-Formula:C33H50Cl2N2O6Purezza:99.15%Colore e forma:SolidPeso molecolare:641.67PARP14 inhibitor H10
CAS:PARP14 inhibitor H10 is a selective inhibitor against PARP14 with IC50 of 490 nMFormula:C24H27N7O7SPurezza:98%Colore e forma:SolidPeso molecolare:557.58DJ001
CAS:DJ001: specific PTPσ inhibitor, non-competitive, IC50=1.43 μM, aids hematopoietic stem cell regeneration.Formula:C15H12N2O3Purezza:99.54%Colore e forma:SolidPeso molecolare:268.27Ref: TM-T11053
1mg39,00€5mg89,00€10mg124,00€25mg198,00€50mg280,00€100mg376,00€200mg520,00€1mL*10mM (DMSO)87,00€CDK8/19-IN-1
CAS:CDK8/19-IN-1 is a selective and oral bioavailable CDK8/19 dual inhibitor (IC50s: 0.46 nM, 0.99 nM, and 270 nM for CDK8, CDK19, and CDK9).Formula:C19H18N4O4S2Purezza:98%Colore e forma:SolidPeso molecolare:430.5Psammaplysene A
CAS:Psammaplysene A is a FOXO1a nuclear export inhibitor.Formula:C27H35Br4N3O3Purezza:98%Colore e forma:SolidPeso molecolare:769.2W146 TFA
CAS:W146 TFA is a selective sphingosine-1-phosphate receptor 1 ( S1PR1 ) antagonist with an EC 50 value of 398 nM.Formula:C18H28F3N2O6PColore e forma:SolidPeso molecolare:456.399MYRA-A
CAS:MYRA-A is an inducer of apoptosis in a Myc-dependent manner that acts by inhibiting Myc-driven transformation and disrupting MYC-Max interaction.Formula:C19H20N2O4Purezza:98%Colore e forma:SolidPeso molecolare:340.37Epirubicin
CAS:Epirubicin, a doxorubicin derivative, is an antineoplastic, inhibits topoisomerase, DNA/RNA synthesis, and Foxp3, reducing T cell activity.Formula:C27H29NO11Colore e forma:SolidPeso molecolare:543.52SLMP53-2
CAS:SLMP53-2 is a mutant p53 reactivator that restores the wild-type-like conformation and DNA-binding ability of mutp53-Y220C through enhanced interaction withFormula:C26H22N2O2Colore e forma:SolidPeso molecolare:394.47pan-HER-IN-1
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