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Apoptosi

Apoptosi

Gli inibitori dell'apoptosi sono composti che prevengono o ritardano il processo di morte cellulare programmata, noto come apoptosi. Questi inibitori sono fondamentali per lo studio dei meccanismi di sopravvivenza cellulare e vengono utilizzati per indagare sulle malattie in cui l'apoptosi è disregolata, come il cancro, i disturbi neurodegenerativi e le malattie autoimmuni. Modulando l'apoptosi, questi inibitori possono aiutare nello sviluppo di terapie mirate a controllare la morte cellulare. Presso CymitQuimica, offriamo una vasta selezione di inibitori dell'apoptosi di alta qualità per supportare le tue ricerche in biologia cellulare, oncologia e campi correlati.

Sottocategorie di "Apoptosi"

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Trovati 5618 prodotti di "Apoptosi"

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  • HDAC1/6-IN-1

    CAS:
    <p>HDAC1/6-IN-1, a dual HDAC1 (89 nM) and HDAC6 (13 nM) inhibitor, blocks cancer cell cycle, triggers apoptosis, and halts metastasis.</p>
    Formula:C32H45N7O4
    Colore e forma:Solid
    Peso molecolare:591.74
  • Metallo-β-lactamase-IN-5

    CAS:
    <p>Metallo-β-lactamase-IN-5 (compound 5c) is a powerful inhibitor of metallo-β-lactamases (MBLs).</p>
    Formula:C19H16N4O3
    Colore e forma:Solid
    Peso molecolare:348.36
  • Topoisomerase II inhibitor 11

    CAS:
    <p>Topoisomerase II inhibitor 11 (compound 3d) is a potent inhibitor of Topoisomerase II (IC50: 2.89 μM).</p>
    Formula:C27H21BrCl2N2O2S
    Colore e forma:Solid
    Peso molecolare:588.34
  • Anisperimus

    CAS:
    <p>Anisperimus (LF 15-0195) is an immunosuppressant that prevents CNS autoimmunity by promoting the development of regulatory CD4 T cells expressing Foxp3.</p>
    Formula:C18H39N7O3
    Purezza:98.10%
    Colore e forma:Solid
    Peso molecolare:401.55
  • CX-5011

    CAS:
    <p>CX-5011, a CK2 inhibitor, induces Rac1 activation and promotes apoptosis, effectively causing cancer cell death [1] [2].</p>
    Formula:C20H12N4O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:340.33
  • NBI-42902

    CAS:
    <p>NBI-42902 is a potent GnRH receptor antagonist (Ki=0.56 nm, Kd=0.19 nm), suppressing serum LH in macaques without causing histamine release.</p>
    Formula:C27H24F3N3O3
    Colore e forma:Solid
    Peso molecolare:495.49
  • ADU-S100

    CAS:
    <p>ADU-S100 (MIW815) is a STING agonist that significantly induces the production of IFN-β,TNF-α,IL-6,and MCP-1,induces TBK1 and IRF3 phosphorylation,antitumour.</p>
    Formula:C20H24N10O10P2S2
    Purezza:99.83%
    Colore e forma:Solid
    Peso molecolare:690.54
  • hnRNPK-IN-1

    CAS:
    <p>hnRNPK-IN-1 binds hnRNPK tightly (Kd 4.6-2.6 μM), disrupting c-myc transcription and inducing apoptosis in Hela cells.</p>
    Formula:C23H21N3O5
    Colore e forma:Solid
    Peso molecolare:419.43
  • CDK6/PIM1-IN-1

    CAS:
    <p>CDK6/PIM1-IN-1: A dual inhibitor for CDK6 (39 nM IC50) &amp; PIM1 (88 nM), also targets CDK4 (3.6 nM IC50), halts AML cell growth, and induces apoptosis.</p>
    Formula:C25H28FN9
    Colore e forma:Solid
    Peso molecolare:473.55
  • BRD0476

    CAS:
    <p>BRD0476 prevents pancreatic β-cell death by blocking IFN-γ-induced JAK2 &amp; STAT1 without inhibiting JAK kinase activity.</p>
    Formula:C35H38N4O8S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:674.76
  • Jolkinolide B

    CAS:
    <p>Jolkinolide B is a bioactive diterpene isolated from the roots of Euphorbia fischeriana Steud.</p>
    Formula:C20H26O4
    Purezza:99.39% - 99.7%
    Colore e forma:Solid
    Peso molecolare:330.42
  • VEGFR-2-IN-28

    CAS:
    <p>VEGFR-2-IN-28 is a potent inhibitor of VEGFR-2 (IC50: 0.83 μM). VEGFR-2-IN-28 induces apoptosis and exhibits antitumor effects.</p>
    Formula:C26H17N7O7
    Colore e forma:Solid
    Peso molecolare:539.46
  • VS 8

    CAS:
    <p>VS 8: potent oral VEGFR-2 inhibitor, anti-angiogenic, induces cancer cell apoptosis &amp; migration, acts on CSCs.</p>
    Formula:C26H20F3N3O3
    Colore e forma:Solid
    Peso molecolare:479.45
  • SPRC

    CAS:
    <p>"SPRC, a synthetic antioxidant, boosts H2S production, activates STAT3, and guards against doxorubicin heart damage."</p>
    Formula:C6H9NO2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:159.21
  • EGFR-IN-52

    CAS:
    <p>EGFR-IN-52, a potent EGFR inhibitor, has IC50s: 0.358 μM (wild-type), 86.02 μM (L858R-TK), 432.67 μM (T790M-TK); induces cancer cell apoptosis.</p>
    Formula:C19H18N4O3S
    Colore e forma:Solid
    Peso molecolare:382.44
  • Anticancer agent 67

    CAS:
    <p>Anticancer agent 67 is a ciprofloxacin analogue, an anticancer agent that induces apoptosis and increases sub-G1 cell populations in MCF-7 cells.</p>
    Formula:C26H24F2N6O2S2
    Colore e forma:Solid
    Peso molecolare:554.63
  • Quinidine Monosulfate

    CAS:
    <p>Quinidine Monosulfate: an oral antiarrhythmic, CYP450db inhibitor, K+ blocker (IC50 19.9 μM), used in malaria research.</p>
    Formula:C40H50N4O8S
    Colore e forma:Solid
    Peso molecolare:746.92
  • DAT-230

    CAS:
    <p>DAT-230 is a microtubule inhibitor effective against cancer cells, causing cell cycle arrest and apoptosis via caspase activation.</p>
    Formula:C20H21NO2S
    Colore e forma:Solid
    Peso molecolare:339.45
  • HX 630

    CAS:
    <p>RXR agonist</p>
    Formula:C28H27NO2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:441.58
  • Telomerase-IN-4

    CAS:
    <p>Telomerase-IN-4 is a potent inhibitor of telomerase with antiproliferative properties and induces apoptosis [1].</p>
    Formula:C21H18N4OS2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:406.52