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Apoptosi

Apoptosi

Gli inibitori dell'apoptosi sono composti che prevengono o ritardano il processo di morte cellulare programmata, noto come apoptosi. Questi inibitori sono fondamentali per lo studio dei meccanismi di sopravvivenza cellulare e vengono utilizzati per indagare sulle malattie in cui l'apoptosi è disregolata, come il cancro, i disturbi neurodegenerativi e le malattie autoimmuni. Modulando l'apoptosi, questi inibitori possono aiutare nello sviluppo di terapie mirate a controllare la morte cellulare. Presso CymitQuimica, offriamo una vasta selezione di inibitori dell'apoptosi di alta qualità per supportare le tue ricerche in biologia cellulare, oncologia e campi correlati.

Sottocategorie di "Apoptosi"

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Trovati 5592 prodotti di "Apoptosi"

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  • ASK1-IN-3

    CAS:
    <p>ASK1-IN-3, selective ASK1 inhibitor with 33.8 nM IC50; inhibits cell cycle kinases; induces apoptosis in HepG2 cells.</p>
    Formula:C18H18N8O2
    Colore e forma:Solid
    Peso molecolare:378.39
  • MDM2-IN-1

    CAS:
    <p>MDM2-IN-1 is a synthetic MDM2-p53 interaction (MDM2) inhibitor and contains the trans (D-)configuration.</p>
    Formula:C23H21Cl2FN2O3
    Colore e forma:Solid
    Peso molecolare:463.33
  • PERK-IN-3

    CAS:
    <p>PERK-IN-3 is a potent inhibitor of PERK(IC50 of 7.4 nM).</p>
    Formula:C22H16F2N4O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:406.38
  • c-Met-IN-9

    CAS:
    <p>c-Met-IN-9 is a 4-phenoxypyridine derivative and a c-Met kinase inhibitor (IC50: 12 nM). c-Met-IN-9 induces apoptosis and shows antitumour effects.</p>
    Formula:C25H19F2N5O3
    Colore e forma:Solid
    Peso molecolare:475.45
  • TRAF-STOP inhibitor 6877002

    CAS:
    <p>TRAF-STOP 6877002 inhibits CD40-TRAF6, curbing leukocyte recruitment and macrophage activation/proliferation in plaques.</p>
    Formula:C17H17NO
    Purezza:99.76%
    Colore e forma:Solid
    Peso molecolare:251.32
  • BLM-IN-1

    CAS:
    <p>BLM-IN-1: BLM inhibitor, KD 1.81 μM, IC50 0.95 μM; causes DNA damage, apoptosis, stops cancer cell growth.</p>
    Formula:C28H35FN4O
    Colore e forma:Solid
    Peso molecolare:462.6
  • DAT-230

    CAS:
    <p>DAT-230 is a microtubule inhibitor effective against cancer cells, causing cell cycle arrest and apoptosis via caspase activation.</p>
    Formula:C20H21NO2S
    Colore e forma:Solid
    Peso molecolare:339.45
  • PI3Kδ-IN-10

    CAS:
    <p>PI3Kδ-IN-10 is a highly potent and orally active PI3Kδ inhibitor (IC50= 2 nM).</p>
    Formula:C19H16ClN9
    Colore e forma:Solid
    Peso molecolare:405.84
  • Caspase-9 Inhibitor III

    CAS:
    <p>Caspase-9 Inhibitor III (Ac-LEHD-cmk) blocks caspase-9, protects against ischemic heart damage.</p>
    Formula:C24H35ClN6O9
    Colore e forma:Solid
    Peso molecolare:587.02
  • HLI 373

    CAS:
    <p>HLI373: potent Hdm2 (ubiquitin ligase) inhibitor, induces apoptosis in tumor cells, has antimalarial properties.</p>
    Formula:C18H23N5O2
    Colore e forma:Solid
    Peso molecolare:341.41
  • OXPHOS-IN-1

    CAS:
    <p>OXPHOS-IN-1 inhibits oxidative phosphorylation; halts MIA PaCa-2 (IC50: 2.34 μM) and BxPC-3 cells growth (IC50: 13.82 μM).</p>
    Formula:C19H29N3O6S2
    Colore e forma:Solid
    Peso molecolare:459.58
  • Caspase-3/7 activator 3


    <p>Caspase-3/7 activator 3 triggers apoptosis with tumor selectivity and anti-proliferative effects.</p>
    Formula:C24H27NO5
    Colore e forma:Solid
    Peso molecolare:409.47
  • Anticancer agent 63

    CAS:
    <p>Compound 3h fights various cancers; most effective on MCF-7 (IC50 3.4 μM). Triggers apoptosis; alters Bcl-2, IL-2, Caspase-3 levels, has antioxidant effects.</p>
    Formula:C17H24F3NOSe
    Colore e forma:Solid
    Peso molecolare:394.33
  • PSB 0474

    CAS:
    <p>P2Y6 receptor agonist</p>
    Formula:C17H20N2O13P2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:522.29
  • MMP-9-IN-5

    CAS:
    <p>MMP-9-IN-5: MMP-9 and AKT inhibitor (IC50: 4.49 nM and 1.34 nM), induces apoptosis for cancer research.</p>
    Formula:C27H20IN3O4
    Colore e forma:Solid
    Peso molecolare:577.37
  • GW-3333

    CAS:
    <p>GW-3333 inhibits matrix metalloproteinases and TNF-Converting Enzyme, showing potential as an antiarthritic therapy.</p>
    Formula:C22H36N4O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:420.55
  • Anticancer agent 47

    CAS:
    <p>Compound 4j: potent anticancer agent; halts cell growth, induces apoptosis and G0/G1 arrest; significant in vivo tumor reduction.</p>
    Formula:C19H14N2O4S
    Colore e forma:Solid
    Peso molecolare:366.39
  • Antiproliferative agent-19


    Antiproliferative agent-19 induces apoptosis and G2/M cell cycle arrest in lung cancer cells.
    Formula:C26H23NO
    Colore e forma:Solid
    Peso molecolare:365.47
  • Bcl-2/Mcl-1-IN-1

    CAS:
    <p>Bcl-2/Mcl-1-IN-1 is an inhibitor of Bcl-2 (Ki: 4.53 μM) and Mcl-1 (Ki: 1.19 μM).Bcl-2/Mcl-1-IN-1 can be used in cancer research.</p>
    Formula:C28H23NO3
    Colore e forma:Solid
    Peso molecolare:421.49
  • EGFR/HER2/TS-IN-1

    CAS:
    <p>EGFR/HER2/TS-IN-1 inhibits EGFR (0.203 μM), HER2 (0.088 μM), TS (0.168 μM), and induces apoptosis in MCF7 cells.</p>
    Formula:C24H15N5O4S2
    Colore e forma:Solid
    Peso molecolare:501.54