Proteasi/Proteasoma
Gli inibitori delle proteasi e del proteasoma sono composti che bloccano l'attività delle proteasi e del proteasoma, che sono coinvolti nella degradazione e nel turnover delle proteine. Questi inibitori sono fondamentali per studiare la regolazione dell'omeostasi proteica, il controllo del ciclo cellulare e l'apoptosi. Gli inibitori delle proteasi e del proteasoma vengono anche utilizzati nel trattamento di malattie come il cancro, dove la degradazione anomala delle proteine svolge un ruolo nella progressione della malattia. Inibendo le proteasi o il proteasoma, questi composti possono indurre la morte cellulare nelle cellule tumorali e sono strumenti critici sia per la ricerca di base che per lo sviluppo terapeutico. Presso CymitQuimica, offriamo una vasta gamma di inibitori delle proteasi e del proteasoma di alta qualità per supportare la tua ricerca in biochimica, biologia cellulare e sviluppo di farmaci.
Sottocategorie di "Proteasi/Proteasoma"
- Acetil-CoA carbossilasi(36 prodotti)
- Cisteina proteasi(110 prodotti)
- DPP-4(23 prodotti)
- Glutaminasi(45 prodotti)
- Proteasi HIV(505 prodotti)
- PAI-1(26 prodotti)
- Inibitori della proteasi(50 prodotti)
- Ricettore attivato dalla proteasi(54 prodotti)
- Proteasoma(93 prodotti)
- Proteasi serina(55 prodotti)
- p97(15 prodotti)
Mostrare 3 più sottocategorie
Trovati 1045 prodotti di "Proteasi/Proteasoma"
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PKSI-527
CAS:PKSI-527 inhibits plasma kallikrein (Ki=0.81μM), selective vs. glandular kallikrein/thrombin/urokinase/Xa, reduces bradykinin, affects clotting times.Formula:C25H32ClN3O4Colore e forma:SolidPeso molecolare:473.99(Arg)9
CAS:(Arg)9 (Nona-L-arginine;Peptide R9) is a cell-penetrating peptide,and exhibits neuroprotective activity(IC50 of 0.78 μM, in the glutamic acid model).Formula:C54H110N36O10Colore e forma:SolidPeso molecolare:1423.69Tilpisertib
CAS:Tilpisertib is a serine/threonine kinase inhibitor (WO2017007689).Formula:C33H33ClN8OColore e forma:SolidPeso molecolare:593.13Pepstatin A
CAS:Formula:C34H63N5O9Purezza:>90.0%(HPLC)Colore e forma:White to Light yellow powder to crystalPeso molecolare:685.90Tanaproget
CAS:Tanaproget is an orally available, high-affinity, non-steroidal progesterone receptor (PR) agonist with an IC50 of 1.7 nM for hPR.Formula:C16H15N3OSPurezza:98%Colore e forma:SolidPeso molecolare:297.38S-Methylglutathione
CAS:S-Methylglutathione (S-Methyl glutathione) is a 1-chloro-2,4-dinitrobenzene coupling inhibitor, an XOCl scavenger, and inhibitor of glyoxalase 1.Formula:C11H19N3O6SPurezza:98%Colore e forma:SolidPeso molecolare:321.355-Amino-8-hydroxyquinoline
CAS:5-Amino-8-hydroxyquinoline(5A8HQ),Proteasome inhibitor. Potential anticancer agent.Formula:C9H8N2OPurezza:99.69%Colore e forma:SolidPeso molecolare:160.17DMP 777
CAS:DMP 777 is an orally active inhibitor of human leukocyte elastase.Formula:C31H40N4O6Colore e forma:SolidPeso molecolare:564.67Teneligliptin D8
CAS:Teneligliptin D8 a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting inhibitor of DPP-4.Formula:C22H30N6OSPurezza:98%Colore e forma:SolidPeso molecolare:434.63E-64d [for Biochemical Research]
CAS:Formula:C17H30N2O5Purezza:>95.0%(HPLC)Colore e forma:White to Almost white powder to crystalPeso molecolare:342.44Urokinase
CAS:Urokinase (uPA) is a serine protease that activates plasminogen to plasmin, crucial for thrombolysis and ECM degradation.
Colore e forma:SolidUbenimex
CAS:Formula:C16H24N2O4Purezza:>98.0%(HPLC)Colore e forma:White to Almost white powder to crystalPeso molecolare:308.38Glutaminase-IN-3
CAS:Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.Formula:C19H19F3N6O2SPurezza:98.51%Colore e forma:SolidPeso molecolare:452.45Ilomastat
CAS:Formula:C20H28N4O4Purezza:>95.0%(HPLC)(qNMR)Colore e forma:White to Light yellow powder to crystalPeso molecolare:388.47Saxagliptin
CAS:Saxagliptin (BMS-477118) is a selective and reversible DPP4 inhibitor with IC50 of 26 nM.Formula:C18H25N3O2Purezza:99.17% - 99.95%Colore e forma:SolidPeso molecolare:315.41Dolutegravir sodium
CAS:Dolutegravir sodium (GSK-1349572A) salt(DTG; GSK1349572) is an HIV integrase inhibitor(IC50: 2.7 nM), modest activity against raltegravir-resistant signature
Formula:C20H18F2N3NaO5Purezza:98% - 99.46%Colore e forma:SolidPeso molecolare:441.36Bortezomib-pinanediol
CAS:Bortezomib-pinanediol is a proteasome inhibitor. is a prodrug of Bortezomib.Formula:C29H39BN4O4Purezza:97.5%Colore e forma:Yellow SolidPeso molecolare:518.46NBD-557
CAS:NBD-557 is a potentially HIV-1 inhibitor.Formula:C17H24BrN3O2Purezza:99.52%Colore e forma:SolidPeso molecolare:382.3Ref: TM-T7382
1mg35,00€5mg74,00€10mg109,00€25mg210,00€50mg306,00€100mg434,00€200mg590,00€1mL*10mM (DMSO)82,00€Hepln-13
CAS:Hepln-13 is a hepsin inhibitor that acts by hindering prostate cancer bone metastasis.Formula:C17H13BrN2Purezza:97.67%Colore e forma:SolidPeso molecolare:325.2Ref: TM-T25492
1mg38,00€2mg50,00€5mg85,00€10mg126,00€25mg245,00€50mg364,00€100mg507,00€200mg700,00€1mL*10mM (DMSO)96,00€Sofosbuvir
CAS:Sofosbuvir (GS 7977) is a uridine monophosphate analog inhibitor of hepatitis C virus (HCV) polymerase NS5B that is used as an antiviral agent in the treatmentFormula:C22H29FN3O9PPurezza:99.77% - 99.82%Colore e forma:SolidPeso molecolare:529.45Alvelestat
CAS:Alvelestat (AZD9668) is an orally bioavailable, selective and reversible inhibitor of human neutrophil elastase (NE), with potential anti-inflammatory activity.Formula:C25H22F3N5O4SPurezza:98% - >99.99%Colore e forma:SolidPeso molecolare:545.53Ref: TM-T3107
1mg35,00€2mg46,00€5mg59,00€10mg88,00€25mg157,00€50mg230,00€100mg368,00€500mg877,00€1mL*10mM (DMSO)79,00€Lersivirine
CAS:Lersivirine (UK-453061)(UK 453061) is a second-generation non-nucleoside reverse transcriptase inhibitor (NNRTI) under development for HIV infection therapy.Formula:C17H18N4O2Purezza:98.01%Colore e forma:SolidPeso molecolare:310.35HIV-1 Nef-IN-1
CAS:HIV-1 Nef-IN-1 is an inhibitor of HIV-1 Nef protein. It efficiently competes for Nef-SH3Hck interactions(Kd : 6.7 μM).Formula:C18H16O2Purezza:99.90%Colore e forma:SolidPeso molecolare:264.324-Isopropylcatechol
CAS:4-Isopropylcatechol is a potent depigmenting agent and is of use in the topical therapy of selected patients with hypermelanosis.Formula:C9H12O2Purezza:97.93%Colore e forma:SolidPeso molecolare:152.19Ref: TM-T9065
1mg49,00€5mg101,00€10mg154,00€25mg248,00€50mg346,00€100mg472,00€200mg633,00€1mL*10mM (DMSO)88,00€Simeprevir
CAS:Simeprevir (TMC435) is a potent HCV NS3/4A protease inhibitor, and inhibits HCV replication with EC50 of 8 nM.Formula:C38H47N5O7S2Purezza:99.45% - 99.92%Colore e forma:SolidPeso molecolare:749.94SU 4942
CAS:SU-4942 is a modulator of tyrosine kinase signaling.Formula:C15H10BrNOPurezza:99% - 99.32%Colore e forma:SolidPeso molecolare:300.152-Benzylsuccinic acid
CAS:2-Benzylsuccinic acid (DL-Benzylsuccinic acid) is a bacterial xenobiotic metabolite.Formula:C11H12O4Purezza:99.01% - ≥95%Colore e forma:SolidPeso molecolare:208.21Anagliptin hydrochloride
CAS:Anagliptin (SK-0403) hydrochloride: potent, selective oral DPP-4 inhibitor; IC50: DPP-4 3.8 nM, DPP-8 68 nM, DPP-9 60 nM.Formula:C19H26ClN7O2Colore e forma:SolidPeso molecolare:419.91Ilomastat
CAS:Ilomastat (GM6001) (GM6001, Galardin) is a broad spectrum matrix metalloprotease (MMP) inhibitor.Formula:C20H28N4O4Purezza:97.04% - 99.51%Colore e forma:SolidPeso molecolare:388.46Ref: TM-T2743
1mg46,00€2mg62,00€5mg89,00€10mg145,00€25mg255,00€50mg429,00€100mg620,00€200mg880,00€1mL*10mM (DMSO)94,00€Tenofovir alafenamide hemifumarate
CAS:Tenofovir alafenamide hemifumarate (GS-7340 hemifumarate) is an oral phosphonoamidate prodrug of the HIV reverse transcriptase nucleotide inhibitor tenofovir.
Formula:C21H29N6O5PC4H4O4Purezza:99.33% - 99.96%Colore e forma:SolidPeso molecolare:534.51SB-3CT
CAS:SB-3CT is a potent and specific gelatinase inhibitor for MMP-2(Ki=13.9 nM) and MMP-9(Ki=600 nM).Formula:C15H14O3S2Purezza:98% - 99.38%Colore e forma:SolidPeso molecolare:306.4Ref: TM-T2009
1mg46,00€2mg62,00€5mg94,00€10mg150,00€25mg234,00€50mg349,00€100mg518,00€500mg1.134,00€1mL*10mM (DMSO)94,00€S-methyl-KE-298
CAS:S-methyl-KE-298 is the second main metabolite in plasma,is a methyl conjugate of deacetyl-KE-298.KE-298 inhibits matrix metalloproteinase (MMP-1) productionFormula:C13H16O3SPurezza:97.33%Colore e forma:SolidPeso molecolare:252.33Ref: TM-T4282
1mg88,00€5mg210,00€10mg338,00€25mg625,00€50mg938,00€100mg1.264,00€1mL*10mM (DMSO)188,00€Trelagliptin succinate
CAS:Trelagliptin succinate (SYR-472 succinate) is a long-acting inhibitor of dipeptidyl peptidase-4 (DPP-4), being developed for the treatment of type 2 diabetes (Formula:C22H26FN5O6Purezza:99.27% - 99.92%Colore e forma:SolidPeso molecolare:475.47Telaprevir
CAS:Telaprevir (Incivek) (VX-950) is an effective inhibitor of HCV NS3-4A serine protease (IC50: 0.35 μM).Formula:C36H53N7O6Purezza:96.9% - 98.89%Colore e forma:SolidPeso molecolare:679.85PF-00835231
CAS:PF-00835231 is a CoV-2 cysteine 3C-like protease (3CLpro) inhibitor, with IC50s of 0.27 nM and 4 nM for SARS CoV-2 and SARS CoV-1 3CLpro, respectively.PF-Formula:C24H32N4O6Purezza:97.83%Colore e forma:SolidPeso molecolare:472.53Ref: TM-T9458
1mg57,00€2mg81,00€5mg120,00€10mg187,00€25mg339,00€50mg510,00€100mg748,00€200mg1.035,00€1mL*10mM (DMSO)133,00€CGS 27023A
CAS:CGS 27023A is a non-peptidic, potent, and orally active stromelysin inhibitor.Formula:C18H24ClN3O5SPurezza:99.08%Colore e forma:SolidPeso molecolare:429.92Fostemsavir
CAS:Fostemsavir (BMS-663068) is an HIV-1 attachment inhibitor in development for the treatment of HIV-1 infection.Formula:C25H26N7O8PPurezza:98.95%Colore e forma:SolidPeso molecolare:583.49Ref: TM-T3523
1mg59,00€5mg120,00€10mg170,00€25mg283,00€50mg432,00€100mg622,00€200mg873,00€1mL*10mM (DMSO)156,00€2-Cyanopyrimidine
CAS:2-Cyanopyrimidine (m-Hydroxyphenylpropionic acid) is inhibitor of cathepsin K(IC50 : 170 nM)Formula:C5H3N3Purezza:99.27%Colore e forma:Crystalline SolidPeso molecolare:105.1Elvitegravir
CAS:Elvitegravir (JTK-303) is an HIV integrase inhibitor and CYP2C9 inducer.Formula:C23H23ClFNO5Purezza:98.43% - 99.57%Colore e forma:SolidPeso molecolare:447.88Picolamine
CAS:Picolamine acts as a potential inhibitor of DPP-4.Formula:C6H8N2Purezza:98.3%Colore e forma:Light Yellow LiquidPeso molecolare:108.14(R)-MG-132
CAS:(R)-MG-132 (Z-Leu-D-leu-leu-al) is the enantiomer of MG-132. (R)-MG-132 stereoisomer is a more potent proteasome inhibitor than MG-132.Formula:C26H41N3O5Purezza:99.90%Colore e forma:SolidPeso molecolare:475.62Ref: TM-T12628
2mg40,00€5mg60,00€10mg84,00€25mg127,00€50mg187,00€100mg283,00€200mg419,00€1mL*10mM (DMSO)74,00€Batimastat
CAS:Batimastat (BB94) (BB-94) is an effective, broad-spectrum matrix metalloprotease (MMP) inhibitor.Formula:C23H31N3O4S2Purezza:98.15% - 99.5%Colore e forma:SolidPeso molecolare:477.64Glutaminase C-IN-1
CAS:Glutaminase C-IN-1 (Compound 968) is a Glutaminase C allosteric inhibitor.Formula:C27H27BrN2OPurezza:99.68% - >99.99%Colore e forma:SolidPeso molecolare:475.42Ref: TM-T3964
2mg42,00€5mg60,00€10mg87,00€25mg162,00€50mg273,00€100mg378,00€200mg557,00€1mL*10mM (DMSO)67,00€MUN57694
CAS:MUN57694 is an inhibitor of 26S proteasome.Formula:C23H25N3O4Purezza:99%Colore e forma:SolidPeso molecolare:407.46Ref: TM-T9090
2mg38,00€5mg56,00€10mg90,00€25mg154,00€50mg221,00€100mg313,00€200mg437,00€1mL*10mM (DMSO)67,00€2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)-
CAS:2,4-Dioxaspiro(5.5)undec-8-ene, 3-(2-furanyl)- (Ulinastatin) ,as an urinary trypsin inhibitor (UTI), is a glycoprotein that is isolated from healthy human urineFormula:C13H16O3Purezza:99.53% - 99.81%Colore e forma:SolidPeso molecolare:220.26Ref: TM-T8802
1mg87,00€5mg172,00€10mg258,00€25mg425,00€50mg598,00€100mg810,00€500mg1.605,00€1mL*10mM (DMSO)155,00€Samatasvir
CAS:Samatasvir (ATOLIHZIXHZSBA-BTSKBWHGSA-N) is a pan-genotypic inhibitor of the HCV non-structural protein 5A.Formula:C47H48N8O6S2Purezza:98.03%Colore e forma:SolidPeso molecolare:885.06Ref: TM-T9567
1mg55,00€5mg116,00€10mg187,00€25mg376,00€50mg632,00€100mg1.008,00€1mL*10mM (DMSO)197,00€Dabigatran
CAS:Dabigatran (BIBR 953ZW), a thrombin inhibitor, prevents thrombus formation, reducing stroke and embolism risk in nonvalvular atrial fibrillation patients.Formula:C25H25N7O3Purezza:97.44% - 98.7%Colore e forma:Tan SolidPeso molecolare:471.51Ombitasvir
CAS:Ombitasvir (ABT-267) inhibits HCV protein NS5A, effective orally, EC50: 0.82-19.3 pM (genotypes 1-5), 366 pM (genotype 6a).Formula:C50H67N7O8Purezza:97.27% - 99.56%Colore e forma:SolidPeso molecolare:894.11Ref: TM-T7158
2mg43,00€5mg80,00€10mg111,00€25mg227,00€50mg329,00€100mg487,00€500mg1.026,00€1mL*10mM (DMSO)111,00€MDL-28170
CAS:MDL-28170 (Calpain Inhibitor III) is a Cysteine protease.Formula:C22H26N2O4Purezza:95.06%Colore e forma:SolidPeso molecolare:382.45Ref: TM-T2470
1mg34,00€2mg49,00€5mg71,00€10mg90,00€25mg128,00€50mg167,00€100mg284,00€1mL*10mM (DMSO)75,00€CTTHWGFTLC, CYCLIC acetate(244082-19-7 free base)
CTTHWGFTLC, CYCLIC acetate is an inhibitor for matrix metalloproteinases (MMP)-2 and MMP-9.Formula:C54H75N13O16S2Purezza:99.71%Colore e forma:SolidPeso molecolare:1226.39L-Albizziin
CAS:L-Albizziin (L-beta-Ureidoalanine) is a glutamase inhibitor and is a glutaminyl-tRNA synthetase inhibitor.Formula:C4H9N3O3Purezza:99.98%Colore e forma:White PowderPeso molecolare:147.13SB-734117
CAS:SB-734117 inhibits productive replication of several HCMV strains.Formula:C14H16N6OPurezza:99.72%Colore e forma:SolidPeso molecolare:284.32Ref: TM-T9580
1mg115,00€5mg249,00€10mg369,00€25mg562,00€50mg787,00€100mg1.054,00€200mg1.406,00€1mL*10mM (DMSO)235,00€Efegatran
CAS:Efegatran is a hematologic agent and platelet aggregation inhibitor.
Formula:C21H32N6O3Colore e forma:SolidPeso molecolare:416.52Y-29794 Tosylate
CAS:Y-29794 Tosylate (Y-29794) is an orally active, effective, and specific non-peptide-prolyl endopeptidase (PPCE) inhibitor.
Formula:C30H42N2O4S3Purezza:99.86%Colore e forma:SolidPeso molecolare:590.86Ref: TM-T35233
1mg52,00€2mg74,00€5mg96,00€10mg137,00€25mg217,00€50mg391,00€100mg582,00€500mg1.254,00€Raltegravir potassium
CAS:Raltegravir potassium (MK 0518 potassium salt) salt(MK0518 potassium salt) is a potent integrase (IN) inhibitor, used to treat HIV infection.Formula:C20H20FN6O5·KPurezza:98% - 99.55%Colore e forma:Off-White SolidPeso molecolare:482.51Carbobenzoxyproline
CAS:Carbobenzoxyproline (Carbobenzoxy-S-proline) is a prolidase inhibitor.Formula:C13H15NO4Purezza:99.79%Colore e forma:White To Light Yellow Crystal PowderPeso molecolare:249.26GK921
CAS:GK921 is a transglutaminase 2 (TGase) inhibitor.Formula:C21H20N4OPurezza:97.44% - 99.49%Colore e forma:SolidPeso molecolare:344.41Anagliptin
CAS:Anagliptin (SK-0403) is a potent Inhibitor of DPP-4(IC50 of 3.8 nM), for the treatment of type 2 diabetes mellitus.Formula:C19H25N7O2Purezza:97.59% - 99.98%Colore e forma:SolidPeso molecolare:383.45Ref: TM-T7133
1mg47,00€5mg92,00€10mg137,00€25mg224,00€50mg331,00€100mg502,00€200mg715,00€1mL*10mM (DMSO)97,00€Omarigliptin
CAS:Omarigliptin is a potent and selective oral dipeptidyl peptidase 4 (DPP4) inhibitor with IC50 value of 1.6 nM. Cost-effective and quality-assured.Formula:C17H20F2N4O3SPurezza:99.68% - 99.77%Colore e forma:SolidPeso molecolare:398.43Ref: TM-T2316
1mg38,00€2mg50,00€5mg80,00€10mg117,00€25mg200,00€50mg333,00€100mg477,00€500mg1.063,00€1mL*10mM (DMSO)131,00€Belnacasan
CAS:Belnacasan (VX-765) is an orally active IL-converting enzyme/caspase-1 inhibitor.Formula:C24H33ClN4O6Purezza:96.53% - 99.5%Colore e forma:SolidPeso molecolare:508.99Ref: TM-T6090
2mg37,00€5mg50,00€10mg86,00€25mg170,00€50mg235,00€100mg419,00€200mg617,00€1mL*10mM (DMSO)56,00€Thiamine disulfide
CAS:Thiamine disulfide (Algoneurina) , also known as thiamin or vitamin B1, is a vitamin found in food and manufactured as a dietary supplement and medication.Formula:C24H34N8O4S2Purezza:99.81% - 99.81%Colore e forma:CoaPeso molecolare:562.71GSK-A1
CAS:GSK-A1 is a specific inhibitor of PI4KA, also inhibited calcium-driven PRL secretion without affecting calcium signaling and Prl expression.Formula:C29H27FN6O4SPurezza:97.97% - 98.97%Colore e forma:SolidPeso molecolare:574.63NQ301
CAS:NQ301, an antithrombotic agent, inhibits collagen-challenged rabbit platelet aggregation (IC50: 10 mg/mL).Formula:C18H12ClNO3Purezza:99.74% - 99.76%Colore e forma:SolidPeso molecolare:325.75NSC 405020
CAS:NSC 405020 is a noncatalytic inhibitor of MT1-MMP.Formula:C12H15Cl2NOPurezza:96.93% - 99.07%Colore e forma:SolidPeso molecolare:260.162-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one
CAS:2-(2-bromophenyl)-5-chloro-4H-3,1-benzoxazin-4-one is an human neutrophil elastase inhibitor.Formula:C14H7BrClNO2Purezza:97.36%Colore e forma:SolidPeso molecolare:336.57JNJ0966
CAS:JNJ0966 is a highly selective MMP-9 zymogen inhibitor (IC50: 440 nM).Formula:C16H16N4O2S2Purezza:99.46% - 99.62%Colore e forma:SolidPeso molecolare:360.45Ref: TM-T4783
2mg34,00€5mg46,00€10mg64,00€25mg126,00€50mg219,00€100mg315,00€200mg434,00€1mL*10mM (DMSO)35,00€Voxilaprevir
CAS:Voxilaprevir is an inhibitor of hepatitis C virus (HCV) nonstructural (NS) protein 3/4A protease.Formula:C40H52F4N6O9SPurezza:99.83% - 99.98%Colore e forma:SolidPeso molecolare:868.93Ref: TM-T19862
1mg75,00€5mg295,00€10mg423,00€25mg708,00€50mg954,00€100mg1.288,00€200mg1.738,00€1mL*10mM (DMSO)394,00€Coblopasvir
CAS:Coblopasvir is a pan-genotypic non-structural protein 5A (NS5A) inhibitor. It can be used to study chronic hepatitis C virus infection.Formula:C41H50N8O8Purezza:99.33%Colore e forma:SolidPeso molecolare:782.88ML281
CAS:ML281 is a potent and selective STK33 inhibitor with IC50 of 14 nM.Formula:C22H19N3O2SPurezza:99.12% - 99.87%Colore e forma:SolidPeso molecolare:389.47Ref: TM-T3423
1mg35,00€5mg80,00€10mg97,00€25mg188,00€50mg311,00€100mg500,00€500mg1.093,00€1mL*10mM (DMSO)88,00€S 3304
CAS:S 3304 is a novel matrix metalloproteinases inhibitor which is specific for MMP-2 and MMP-9.Formula:C24H20N2O4S2Purezza:98.09%Colore e forma:SolidPeso molecolare:464.56Ref: TM-T16966
1mg44,00€2mg64,00€5mg111,00€10mg173,00€25mg298,00€50mg418,00€100mg567,00€200mg765,00€1mL*10mM (DMSO)114,00€Velpatasvir
CAS:Velpatasvir (GS-5816), also known as GS-5816, is a potent and selective Hepatitis C virus NS5A inhibitor.Formula:C49H54N8O8Purezza:99.17% - 99.83%Colore e forma:SolidPeso molecolare:883Ref: TM-T3334
5mg34,00€10mg49,00€25mg79,00€50mg98,00€100mg152,00€200mg219,00€500mg358,00€1mL*10mM (DMSO)54,00€Boc-Asp(OMe)-fluoromethyl ketone
CAS:Boc-Asp(OMe)-FMK is a broad-spectrum caspase inhibitor that blocks Fas-mediated processes without affecting IL-8 chemotaxis.
Formula:C11H18FNO5Purezza:≥98%Colore e forma:SolidPeso molecolare:263.26Paritaprevir
CAS:Paritaprevir (ABT450) 是一种非结构蛋白 3/4A 蛋白酶抑制剂，对 HCV 1a 和 HCV 1b 的 EC50 值分别为 1 和 0.21 nM。它也是SARS-CoV 3CLpro 的抑制剂，IC50为 1.31 μM。
Formula:C40H43N7O7SPurezza:99.72%Colore e forma:SolidPeso molecolare:765.88Ixazomib citrate
CAS:Ixazomib citrate (MLN9708), a prodrug of Ixazomib (MMLN-2238), is an oral 2nd-gen proteasome inhibitor with anti-cancer potential (IC50: 3.4 nM).Formula:C20H23BCl2N2O9Purezza:98.37% - >99.99%Colore e forma:SolidPeso molecolare:517.124-Phenoxybenzylamine
CAS:4-Phenoxybenzylamine inhibits the function of the NS3 protein by stabilizing an inactive conformation with an IC50 of about 500 μM against HCV NS3/4a .Formula:C13H13NOPurezza:97.26%Colore e forma:SolidPeso molecolare:199.25Dabigatran Etexilate Mesylate
CAS:Dabigatran Etexilate Mesylate (BIBR 1048MS) is the orally active prodrug of dabigatran. Dabigatran is a reversible and selective, direct thrombin inhibitor.Formula:C34H41N7O5·CH4O3SPurezza:99.91%Colore e forma:SolidPeso molecolare:723.84Ref: TM-T5133
5mg42,00€10mg57,00€25mg74,00€50mg95,00€100mg111,00€200mg169,00€500mg240,00€1mL*10mM (DMSO)64,00€Daclatasvir dihydrochloride
CAS:Daclatasvir dihydrochloride is an oral antiviral that treats chronic hepatitis C by inhibiting HCV's NS5A; rare liver enzyme elevation, seldom causes jaundice.Formula:C40H52Cl2N8O6Purezza:99.67%Colore e forma:SolidPeso molecolare:811.8Ref: TM-T1786
1g244,00€5mg42,00€10mg50,00€25mg60,00€50mg71,00€100mg81,00€500mg170,00€1mL*10mM (DMSO)52,00€Avatrombopag
CAS:Avatrombopag (YM477) is a new oral thrombopoietin (TPO) receptor agonist, activating TPO receptor and increasing megakaryocytic proliferation/differentiationFormula:C29H34Cl2N6O3S2Purezza:99.01% - 99.63%Colore e forma:SolidPeso molecolare:649.65Ref: TM-T7417
1mg57,00€5mg120,00€10mg187,00€25mg339,00€50mg540,00€100mg747,00€200mg1.035,00€1mL*10mM (DMSO)167,00€KKI-5 acetate(97145-43-2 free base)
KKI-5 acetate: Serine protease inhibitor, targets kallikrein/plasmin, potential anticancer and angioedema therapy.Formula:C37H59N11O11Purezza:99.44%Colore e forma:SolidPeso molecolare:833.95Mericitabine
CAS:Mericitabine (R-7128) is an HCV inhibitor that terminates RNA chains, halting replication.Formula:C18H26FN3O6Purezza:97.77% - 98.54%Colore e forma:SolidPeso molecolare:399.41Ref: TM-T16710
1mg49,00€5mg108,00€10mg150,00€25mg251,00€50mg369,00€100mg528,00€200mg720,00€1mL*10mM (DMSO)116,00€2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1λ*6*-BENZO[D]ISOTHIAZOL-3-ONE
CAS:2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA*6*-BENZO[D]ISOTHIAZOL-3-ONE targets the Neutrophil elastase (human).Formula:C8H6ClNO3SPurezza:97.28%Colore e forma:SolidPeso molecolare:231.66Ref: TM-T8602
2mg35,00€5mg50,00€10mg66,00€25mg108,00€50mg162,00€100mg235,00€200mg349,00€1mL*10mM (DMSO)50,00€Ivachtin
CAS:Ivachtin (Caspase-3 Inhibitor VII) is a nonpeptide, noncompetitive and reversibl caspase-3 inhibitor(IC50 = 23 nM) and is a modest inhibitor of the remaining
Formula:C20H21N3O7SPurezza:99.74%Colore e forma:SolidPeso molecolare:447.46Chlorcyclizine
CAS:CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Formula:C18H21ClN2Purezza:98.75%Colore e forma:SolidPeso molecolare:300.834-Butylresorcinol
CAS:4-Butylresorcinol (Butylresorcinol) is a potent inhibitor of tyrosinase(IC50 : 11.27 μM), and is used in cosmetics as a depigmenting agent.Formula:C10H14O2Purezza:99.48% - ≥95%Colore e forma:Light Beige Solid PowderPeso molecolare:166.22Rusalatide acetate (497221-38-2 free base)
CAS:Rusalatide acetate (TP508 amide acetate), a regenerated peptide, alleviates radiation-induced gastrointestinal injury by activating stem cells.Formula:C99H151N29O37SPurezza:>99.99%Colore e forma:SolidPeso molecolare:2371.5Ref: TM-TP1024
2mg40,00€5mg66,00€10mg95,00€25mg156,00€50mg225,00€100mg320,00€200mg434,00€1mL*10mM (DMSO)164,00€Ximelagatran
CAS:Ximelagatran, oral direct thrombin inhibitor, transforms to active melagatran in body.Formula:C24H35N5O5Purezza:95.48% - 99.60%Colore e forma:SolidPeso molecolare:473.57Dolutegravir
CAS:Dolutegravir (GSK1349572), HIV integrase inhibitor with IC50 of 2.7 nM, partly effective against some raltegravir-resistant HIV strains.
Formula:C20H19F2N3O5Purezza:98.97% - 99.75%Colore e forma:White To Pale Yellow SolidPeso molecolare:419.38STK16-IN-1
CAS:STK16-IN-1 is an inhibitor of STK16 kinase (IC50: 295 nM).Formula:C17H12FN3OPurezza:99.52%Colore e forma:SolidPeso molecolare:293.3KGP94
CAS:KGP94 is a potent, selective, and competitive inhibitor of the lysosomal endopeptidase enzyme.Formula:C14H12BrN3OSPurezza:99.6%Colore e forma:SolidPeso molecolare:350.23Ref: TM-T27730
1mg65,00€5mg138,00€10mg215,00€25mg359,00€50mg510,00€100mg692,00€200mg928,00€1mL*10mM (DMSO)152,00€Tris(4-aminophenyl)methane
CAS:Tris(4-aminophenyl)methane (Leucopararosaniline), a triphenylmethane dye, is a weak HCV helicase inhibitor.Formula:C19H19N3Purezza:95.73%Colore e forma:Beige Solid CrystallinePeso molecolare:289.37Boceprevir
CAS:Boceprevir (SCH 503034), an oral HCV NS3 protease inhibitor, has a Ki of 14 nM and EC90 of 350 nM.Formula:C27H45N5O5Purezza:95% - 99.16%Colore e forma:SolidPeso molecolare:519.68Ref: TM-T4988
1mg34,00€5mg66,00€10mg90,00€25mg137,00€50mg177,00€100mg260,00€200mg358,00€1mL*10mM (DMSO)75,00€Bemnifosbuvir
CAS:Bemnifosbuvir (AT-511) is a novel phosphoramidate prodrug of 2'-fluoro-2'-C-methylguanosine-5'-monophosphate that has potent in vitro activity against HCV.Formula:C24H33FN7O7PPurezza:99.35% - 99.54%Colore e forma:SolidPeso molecolare:581.53TAPI-1 trifluoroacetate (163847-77-6(free base))
TAPI-1 is an ADAM17/TACE inhibitor, which blocks shedding of cytokine receptors.Formula:C28H38F3N5O7Purezza:98.06%Colore e forma:SolidPeso molecolare:613.62(Arg)9 TFA (143413-47-2 free base)
CAS:(Arg)9 TFA (Peptide R9 TFA) is a cell-penetrating peptide. (Arg)9 TFA exhibits neuroprotective activity with an IC50 of 0.78 μM in the glutamic acid model.Formula:C56H111F3N36O12Purezza:>99.99%Colore e forma:SolidPeso molecolare:1537.71Letermovir
CAS:Letermovir (AIC246) (AIC246) is a novel anti-CMV compound (EC50: about 5 nM in fibroblast cells). It targets the pUL56 subunit of the viral terminase complex.Formula:C29H28F4N4O4Purezza:99.85% - 99.87%Colore e forma:SolidPeso molecolare:572.55Ref: TM-T5396
1mg84,00€5mg167,00€10mg268,00€25mg470,00€50mg670,00€100mg954,00€200mg1.288,00€1mL*10mM (DMSO)205,00€7-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
CAS:7-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine is a inhibitor of Hepatitis C Virus(HCV).Formula:C15H16N4Purezza:99.22%Colore e forma:SolidPeso molecolare:252.31LY 3000328
CAS:LY 3000328 (Cathepsin S inhibitor) is a selective inhibitor of cathepsin S.Cost-effective and quality-assured.Formula:C25H29FN4O5Purezza:97.83% - 99.54%Colore e forma:SolidPeso molecolare:484.52Ref: TM-TQ0116
1mg90,00€2mg130,00€5mg198,00€10mg263,00€25mg462,00€50mg672,00€100mg945,00€1mL*10mM (DMSO)207,00€2-PMPA
CAS:2-PMPA (2-(Phosphonomethyl)pentanedioic acid) is a potent and selective inhibitor of glutamate carboxypeptidase II (GCPII) (IC50=300 pM).Formula:C6H11O7PPurezza:97.4% - 99.5%Colore e forma:SolidPeso molecolare:226.12CA-074 methyl ester
CAS:CA-074 methyl ester (Cathepsin B Inhibitor IV) is a selective inhibitor of Cathepsin B (IC50=36.3 nM). neuroprotective effect. High-Quality, Low-Cost!Formula:C19H31N3O6Purezza:97.26% - 99.58%Colore e forma:SolidPeso molecolare:397.47(S,S)-TAPI-1
CAS:"(S,S)-TAPI-1, an isomer of TAPI-1, inhibits MMPs and TACE (ADAM17), reducing cell surface protein shedding."Formula:C26H37N5O5Colore e forma:SolidPeso molecolare:499.6
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