Proteasi/Proteasoma
Gli inibitori delle proteasi e del proteasoma sono composti che bloccano l'attività delle proteasi e del proteasoma, che sono coinvolti nella degradazione e nel turnover delle proteine. Questi inibitori sono fondamentali per studiare la regolazione dell'omeostasi proteica, il controllo del ciclo cellulare e l'apoptosi. Gli inibitori delle proteasi e del proteasoma vengono anche utilizzati nel trattamento di malattie come il cancro, dove la degradazione anomala delle proteine svolge un ruolo nella progressione della malattia. Inibendo le proteasi o il proteasoma, questi composti possono indurre la morte cellulare nelle cellule tumorali e sono strumenti critici sia per la ricerca di base che per lo sviluppo terapeutico. Presso CymitQuimica, offriamo una vasta gamma di inibitori delle proteasi e del proteasoma di alta qualità per supportare la tua ricerca in biochimica, biologia cellulare e sviluppo di farmaci.
Sottocategorie di "Proteasi/Proteasoma"
- Acetil-CoA carbossilasi(38 prodotti)
- Cisteina proteasi(111 prodotti)
- DPP-4(27 prodotti)
- Glutaminasi(46 prodotti)
- Proteasi HIV(506 prodotti)
- PAI-1(26 prodotti)
- Inibitori della proteasi(50 prodotti)
- Ricettore attivato dalla proteasi(55 prodotti)
- Proteasoma(86 prodotti)
- Proteasi serina(54 prodotti)
- p97(15 prodotti)
Mostrare 3 più sottocategorie
Trovati 984 prodotti di "Proteasi/Proteasoma"
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Velpatasvir
CAS:Velpatasvir (GS-5816), also known as GS-5816, is a potent and selective Hepatitis C virus NS5A inhibitor.Formula:C49H54N8O8Purezza:99.17% - 99.83%Colore e forma:SolidPeso molecolare:883Ref: TM-T3334
5mg34,00€10mg49,00€25mg79,00€50mg98,00€100mg152,00€200mg219,00€500mg358,00€1mL*10mM (DMSO)54,00€Efegatran HCl
CAS:Efegatran (GYKI-14166, RGH-2958, LY294468) is a thrombin inhibitor in development by IVAX for thromboembolic disorders.Formula:C21H34Cl2N6O3Colore e forma:SolidPeso molecolare:489.442Brensocatib
CAS:Brensocatib (AZD7986) is a Dipeptidyl peptidase 1 (DPP1) inhibitor (pIC50s: 6.85, 7.7, 7.6, 7.8, and 7.8 in human, rat, mouse, rabbit, and dog, respectively).Formula:C23H24N4O4Purezza:97.55%Colore e forma:SolidPeso molecolare:420.46STK16-IN-1
CAS:STK16-IN-1 is an inhibitor of STK16 kinase (IC50: 295 nM).Formula:C17H12FN3OPurezza:99.52%Colore e forma:SolidPeso molecolare:293.32-Benzylsuccinic acid
CAS:2-Benzylsuccinic acid (DL-Benzylsuccinic acid) is a bacterial xenobiotic metabolite.Formula:C11H12O4Purezza:99.01% - ≥95%Colore e forma:SolidPeso molecolare:208.21Coblopasvir dihydrochloride
CAS:Coblopasvir dihydrochloride can be used to study chronic HCV infection and is a pan-genotypic nonstructural protein 5A (NS5A) inhibitor.Formula:C41H52Cl2N8O8Purezza:99.33%Colore e forma:SolidPeso molecolare:855.81Ref: TM-T25268L
1mg87,00€5mg187,00€10mg305,00€25mg518,00€50mg742,00€100mg1.017,00€1mL*10mM (DMSO)298,00€Grazoprevir
CAS:Grazoprevir (MK-5172) is a protease inhibitor targeting hepatitis C virus NS3/4A used for treating chronic HCV genotypes 1 or 4 infections. Cost-effective and quality-assured.Formula:C38H50N6O9SPurezza:99.36% - >99.99%Colore e forma:SolidPeso molecolare:766.9FT011
CAS:FT011, a direct anti-fibrotic agent,attenuates cardiac remodelling and dysfunction in experimental diabetic cardiomyopathy.Formula:C20H17NO5Purezza:98.98%Colore e forma:SolidPeso molecolare:351.35Tris(4-aminophenyl)methane
CAS:Tris(4-aminophenyl)methane (Leucopararosaniline), a triphenylmethane dye, is a weak HCV helicase inhibitor.Formula:C19H19N3Purezza:95.73%Colore e forma:Beige Solid CrystallinePeso molecolare:289.37Ilomastat
CAS:Ilomastat (GM6001) (GM6001, Galardin) is a broad spectrum matrix metalloprotease (MMP) inhibitor.Formula:C20H28N4O4Purezza:97.04% - 99.51%Colore e forma:SolidPeso molecolare:388.46Ref: TM-T2743
1mg46,00€2mg62,00€5mg89,00€10mg145,00€25mg255,00€50mg429,00€100mg620,00€200mg880,00€1mL*10mM (DMSO)94,00€TMC647055 Choline Hydroxide Salt
TMC647055 is a potent HCV NS5B inhibitor with low toxicity and good pharmacokinetics, under clinical evaluation.Formula:C37H53N5O8SPurezza:99.44%Colore e forma:SolidPeso molecolare:727.91Ref: TM-T21537L
1mg95,00€5mg200,00€10mg289,00€25mg520,00€50mg742,00€100mg1.018,00€1mL*10mM (DMSO)286,00€JNJ0966
CAS:JNJ0966 is a highly selective MMP-9 zymogen inhibitor (IC50: 440 nM).Formula:C16H16N4O2S2Purezza:99.46% - 99.62%Colore e forma:SolidPeso molecolare:360.45Ref: TM-T4783
2mg34,00€5mg46,00€10mg64,00€25mg126,00€50mg219,00€100mg315,00€200mg434,00€1mL*10mM (DMSO)35,00€UAMC00039 dihydrochloride
CAS:UAMC00039 dihydrochloride is a potent, reversible and competitive dipeptidyl peptidase II inhibitor with an IC50 of 0.48 nM.Formula:C16H26Cl3N3OPurezza:>99.99%Colore e forma:SolidPeso molecolare:382.76PythiDC
CAS:PythiDC is a selective collagen prolyl 4-hydroxylase inhibitor, neither causing general toxicity nor disrupting iron homeostasis.Formula:C10H6N2O4SPurezza:98.13%Colore e forma:SolidPeso molecolare:250.23Simeprevir
CAS:Simeprevir (TMC435) is a potent HCV NS3/4A protease inhibitor, and inhibits HCV replication with EC50 of 8 nM.Formula:C38H47N5O7S2Purezza:99.45% - 99.92%Colore e forma:SolidPeso molecolare:749.94Bz-RS-ISer(3-Ph)-Ome
CAS:Bz-RS-ISer(3-Ph)-Ome (Methyl (2R,3S)-3-(benzoylamino)-2-hydroxy-3-phenylpropanoate) is a paclitaxel derivative that inhibits the HSV replication cycle.
Formula:C17H17NO4Purezza:99.36% - 99.89%Colore e forma:White CrystalPeso molecolare:299.32Glecaprevir
CAS:Glecaprevir (ABT-493) is an HCV NS3/4A protease inhibitor, (IC50s: 3.5-11.3 nM).Formula:C38H46F4N6O9SPurezza:99.16% - 99.69%Colore e forma:SolidPeso molecolare:838.87Chlorcyclizine
CAS:CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Formula:C18H21ClN2Purezza:98.75%Colore e forma:SolidPeso molecolare:300.83VCH-916 free acid(1200133-34-1 free base)
CAS:VCH-916 is a novel nonnucleoside HCV NS5B polymerase inhibitor.Formula:C26H37NO4SPurezza:98.45%Colore e forma:SolidPeso molecolare:459.647-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
CAS:7-benzyl-5,6-dimethyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine is a inhibitor of Hepatitis C Virus(HCV).Formula:C15H16N4Purezza:99.22%Colore e forma:SolidPeso molecolare:252.31Samatasvir
CAS:Samatasvir (ATOLIHZIXHZSBA-BTSKBWHGSA-N) is a pan-genotypic inhibitor of the HCV non-structural protein 5A.Formula:C47H48N8O6S2Purezza:98.03%Colore e forma:SolidPeso molecolare:885.06Ref: TM-T9567
1mg55,00€5mg116,00€10mg187,00€25mg376,00€50mg632,00€100mg1.008,00€1mL*10mM (DMSO)197,00€Odanacatib
CAS:Odanacatib is an inhibitor of cathepsin K with potential anti-osteoporotic activity.Formula:C25H27F4N3O3SPurezza:98.53% - 99.53%Colore e forma:SolidPeso molecolare:525.56KP-457
CAS:KP-457 is a ADAM17 and a TNFα converting enzyme TACE inhibitor that blocks the production of soluble TNF (sTNF).Formula:C21H24N2O7S2Purezza:98.33%Colore e forma:SolidPeso molecolare:480.56Ref: TM-T77778
1mg96,00€5mg205,00€10mg334,00€25mg620,00€50mg982,00€100mg1.333,00€1mL*10mM (DMSO)219,00€(1S,2R)-Alicapistat
CAS:(1S,2R)-Alicapistat inhibits calpains 1 and 2, shows promise for Alzheimer's, and has an IC50 of 395 nM.Formula:C25H27N3O4Purezza:99.60%Colore e forma:SoildPeso molecolare:433.5Ref: TM-T60150
1mg64,00€5mg142,00€10mg197,00€25mg299,00€50mg400,00€100mg537,00€1mL*10mM (DMSO)167,00€(R)-Trolox
CAS:(R)-Trolox is a selective tyrosinase inhibitor used in food, cosmetics, and pharmaceutical products.Formula:C14H18O4Purezza:99.88%Colore e forma:SolidPeso molecolare:250.29Teneligliptin
CAS:Teneligliptin (MP-513), potent DPP-4 inhibitor, IC50 ~1 nM, blocks DPP-4 in human/rat plasma and recombinant forms.Formula:C22H30N6OSPurezza:99.73%Colore e forma:SolidPeso molecolare:426.58Ledipasvir
CAS:Ledipasvir (GS-5885) is a Hepatitis C Virus NS5A Inhibitor.Formula:C49H54F2N8O6Purezza:99.96%Colore e forma:SolidPeso molecolare:889Ref: TM-T6200
1mg35,00€2mg50,00€5mg74,00€10mg94,00€25mg150,00€50mg244,00€100mg421,00€500mg964,00€1mL*10mM (DMSO)94,00€Danoprevir
CAS:Danoprevir (RG7227) is a peptidomimetic inhibitor of the NS3/4A protease(IC50=0.2-3.5 nM) of hepatitis C virus (HCV).Formula:C35H46FN5O9SPurezza:98% - 99.80%Colore e forma:SolidPeso molecolare:731.83PSI
CAS:PSI is a proteasome inhibitor.Formula:C32H50N4O8Purezza:97% - 98.33%Colore e forma:SolidPeso molecolare:618.76Zampilimab
CAS:Zampilimab (UCB-7858) is a humanised monoclonal antibody targeting TGM2, inhibits the cross-linking transamidase activity of TG2, renal fibrosis.Purezza:95%Colore e forma:LiquidPeso molecolare:~150 kDaTriton X-45(n=4)
CAS:Triton X-45: nonionic, low HLB surfactant, dispersible in water, high Krafft point, relevant for HCV research.Formula:C22H38O5Colore e forma:SolidPeso molecolare:382.53KZR-504
CAS:KZR-504 is a selective inhibitor of immunoproteasome low molecular mass polypeptide 2 (LMP2) (IC50s: 51 nM, 4.274 μM for LMP2 and LMP7, respectively).Formula:C21H23N3O6Colore e forma:SolidPeso molecolare:413.42Isecarosmab
CAS:Isecarosmab (M6495) is a monoclonal antibody targeting ADAMTS-5, protect cartilage and inhibit ADAMTS-5-mediated degradation of aggrecan,osteoarthritis (OA).Purezza:95% - 98.0% (SDS-PAGE); 96.7% (SEC-HPLC)Colore e forma:LiquidPeso molecolare:28.05 kDaAnti-Human/Mouse denatured collagen type-I Antibody (XL313)
Anti-Human/Mouse denatured collagen type-I Antibody (XL313) is an IgG1, κ inhibitor derived from mice, targeting denatured collagen type-I in both human and mouse.Colore e forma:Odour LiquidLanadelumab
CAS:Lanadelumab (SHP643), a humanized IgG1 antibody, inhibits plasma kallikrein and its interaction with HMWK, supporting hereditary angioedema research.Purezza:95% - 97.4% (SDS-PAGE); 99.2% (SEC-HPLC)Colore e forma:LiquidPeso molecolare:145.70 kDaAnti-Matriptase Antibody
Anti-Matriptase Antibody is a human-derived antibody expressed in CHO cells, targeting Matriptase. It features a huIgG1 heavy chain and huκ light chain, with a predicted molecular weight (MW) of 150 kDa. The isotype control for Anti-Matriptase Antibody can be found in HumanIgG1kappa, Isotype Control.Colore e forma:Odour LiquidMG-132
CAS:Formula:C26H41N3O5Purezza:>95.0%(qNMR)Colore e forma:White to Light yellow powder to crystalPeso molecolare:475.63HCV-IN-30
CAS:HCV-IN-30 is an HCV NS5A replication complex inhibitor (IC50s: 901 and 102 nM for genotypes 1a and 1b replicons).Formula:C36H44N6O4Purezza:99.6%Colore e forma:SolidPeso molecolare:624.77S 2160
CAS:S 2160 is a synthetic chromogenic substrate for thrombin.Formula:C33H40N8O6Colore e forma:SolidPeso molecolare:644.72Carboxypeptidase G2 (CPG2) Inhibitor
CAS:Carboxypeptidase G2 (CPG2) Inhibitor (CPG2 Inhibitor) is a new CPG2 Inhibitor with antitumor activity.Formula:C13H15NO6SPurezza:99.96%Colore e forma:SolidPeso molecolare:313.33Cathepsin Inhibitor 1
CAS:Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively.Formula:C20H24ClN5O2Purezza:99.78%Colore e forma:SolidPeso molecolare:401.89Ref: TM-T6015
1mg46,00€5mg90,00€10mg144,00€25mg236,00€50mg371,00€100mg522,00€200mg743,00€1mL*10mM (DMSO)100,00€α-Glucosidase-IN-5
CAS:α-Glucosidase-IN-5 (compound 8) is isolated from a twig extract of Polyalthia cinnamomea which is a potent α-glucosidase inhibitor with an IC50 of 57.9 µM.Formula:C15H13NO3Colore e forma:SolidPeso molecolare:255.27BMS-363131
CAS:BMS-363131 (BMS363131) is a potent and selective trypsin inhibitor with an IC50 value of <1.7 nM.Formula:C28H40N6O5Purezza:97.99%Colore e forma:SolidPeso molecolare:540.65AZD5248
CAS:AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).Formula:C22H22N4O2Colore e forma:SolidPeso molecolare:374.44VA4 TG2 inhibitor
CAS:VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.Formula:C33H41N5O6SColore e forma:SolidPeso molecolare:635.77Kallikrein 5-IN-2
CAS:Kallikrein 5-IN-2 inhibits KLK5 (pIC50=7.1); may normalize skin shedding, lessen inflammation & itching.Formula:C23H22N6OColore e forma:SolidPeso molecolare:398.46Tyrosinase-IN-11
CAS:Tyrosinase-IN-11: potent inhibitor, IC50 - 50nM/64nM (L-tyrosinase/L-dopa), antioxidant, low toxicity, for hyperpigmentation study.Formula:C15H14O5Colore e forma:SolidPeso molecolare:274.27PMPA sodium
CAS:PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor.Formula:C6H11Na4O7PPurezza:98%Colore e forma:SolidPeso molecolare:318.08AL-9
CAS:AL-9 is a GT-1b and GT-2a replication inhibitor.Formula:C23H22N4O3Purezza:98%Colore e forma:SolidPeso molecolare:402.45RID-F
CAS:RID-F is an inhibitor of the nonpeptidic proteasome.Formula:C38H50N2O2Purezza:98%Colore e forma:SolidPeso molecolare:566.82BC-05
CAS:BC-05, an orally active inhibitor targeting CD13 and the proteasome, displays potent inhibition with IC50 values of 0.13 μM against human CD13 and 1.39 μM forFormula:C21H29BN2O9Purezza:98%Colore e forma:SolidPeso molecolare:464.27Tyrosinase-IN-7
CAS:Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.Formula:C15H10O5Purezza:99%Colore e forma:SolidPeso molecolare:270.24HCV-IN-34
CAS:HCV-IN-35, an oral HCV blocker, has an EC50 of 0.010 μM and a CC50 of 7.5 μM, indicating strong antiviral effects.Formula:C31H36ClN5Colore e forma:SolidPeso molecolare:514.1Azo-Resveratrol
CAS:Azo-Resveratrol is an analog of Resveratrol used as a potent tyrosinase inhibitor.Formula:C12H10N2O3Colore e forma:SolidPeso molecolare:230.22(3S,4S)-A2-32-01
(3S,4S)-A2-32-01, a less active (S,S)-enantiomer of A2-32-01. A2-32-01 is a potent caseinolytic protein proteases (ClpP) inhibitor .Formula:C19H27NO2Colore e forma:SolidPeso molecolare:301.42MMP-1-IN-1
MMP-1-IN-1 is a highly potent MMP-1 inhibitor with an IC 50 of 0.034 μM .Formula:C14H17ClN2O3Colore e forma:SolidPeso molecolare:296.75NAAA-IN-2
CAS:NAAA-IN-2, a selective inhibitor with 50 nM IC50, targets NAAA, an enzyme hydrolyzing PEA/OEA, and may aid inflammation and pain studies.Formula:C11H13N3O2SColore e forma:SolidPeso molecolare:251.3BI-L 45XX
CAS:BI-L 45XX, an anti-inflammatory benzimidazole derivative, has inhibitory effects on neutrophil function.Formula:C10H9F3N2O2SColore e forma:SolidPeso molecolare:278.25Tyrphostin 47
CAS:Tyrphostin 47 inhibits the protein-tyrosine kinase activity of EGF-R.Formula:C10H8N2O2SColore e forma:SolidPeso molecolare:220.25Levovirin valinate HCl
CAS:Levovirin valinate HCl is a valine ester prodrug of levovirin as a new investigational drug for the therapy of the hepatitis C virus.Formula:C13H22ClN5O6Purezza:98%Colore e forma:SolidPeso molecolare:379.8Ici 186756
CAS:Ici 186756 is a novel, effective, and selective inhibitor of human neutrophil elastase.Formula:C33H49N5O9Purezza:98%Colore e forma:SolidPeso molecolare:659.77TAPI-0
CAS:TAPI-0 is a matrix metalloprotease (MMP) and TACE inhibitor.Formula:C24H32N4O5Colore e forma:SolidPeso molecolare:456.53Tyrosinase-IN-10
CAS:Tyrosinase-IN-10 serves as a partially competitive inhibitor of tyrosinase, demonstrating an inhibition concentration (IC50) value of 1.6 μM against the enzyme'Formula:C16H12O4Colore e forma:SolidPeso molecolare:268.26Chymase-IN-2
CAS:Chymase-IN-2 is a modulator of chymase.Formula:C19H15ClF2NO3PSPurezza:98%Colore e forma:SolidPeso molecolare:441.82Calpain-2-IN-1
CAS:Calpain-2-IN-1 is a selective calpain-2 inhibitor with Ki values of 181 nM for calpain-1 and 7.8 nM for calpain-2, applicable for neurodegenerative diseases a.Formula:C28H37N3O7Purezza:98.05%Colore e forma:SolidPeso molecolare:527.61A-953227
CAS:A-953227: Selective calpain inhibitor with improved cathepsin selectivity, strong microsomal stability, and cellular efficacy.Formula:C25H20FN5O3Purezza:98%Colore e forma:SolidPeso molecolare:457.46HCV-IN-35
CAS:HCV-IN-35 is a potent inhibitor of HCV and shows potential for infectious disease research.Formula:C30H36ClN5Colore e forma:SolidPeso molecolare:502.09Duazomycin
CAS:Duazomycin, an antitumor substance and glutamine antagonist, is used as a chemotherapeutic agent.Formula:C8H11N3O4Colore e forma:SolidPeso molecolare:213.19Calpain Inhibitor XI
CAS:Calpain Inhibitor XI, a reversible covalent inhibitor of calpain-1, is utilized in the research of neurodegenerative disorders.Formula:C26H40N4O6Colore e forma:SolidPeso molecolare:504.62Moxicoumone
CAS:Moxicoumone is an anticoagulant agent.Formula:C22H30N2O6Purezza:98%Colore e forma:SolidPeso molecolare:418.48AM 4299 B
CAS:AM 4299 B is a novel inhibitor of a thiol protease.Formula:C16H27N3O7Purezza:98%Colore e forma:SolidPeso molecolare:373.4MDL 27399
CAS:MDL 27399 suppresses human neutrophil cathepsin G.Formula:C26H36N4O8Colore e forma:SolidPeso molecolare:532.59Tyrphostin A46
CAS:Tyrphostin A46 is an antagonist of the epidermal growth factor-urogastrone receptor.Formula:C10H8N2O3Purezza:98%Colore e forma:Off-White SolidPeso molecolare:204.18CAA0225
CAS:CAA0225 is a selective inhibitor of cathepsin L. CAA0225 is a probe for autophagic proteolysis.Formula:C28H29N3O5Colore e forma:SolidPeso molecolare:487.55MDK0734
CAS:MDK0734 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.Formula:C15H17N3O2Purezza:98%Colore e forma:SolidPeso molecolare:271.31Immunoproteasome inhibitor 1
CAS:Potent, reversible immunoproteasome inhibitor; Ki: β5c 1.18 μM, β1i 0.27 μM, β5i 1.91 μM; potential in treating cancer.Formula:C20H26N2O4Colore e forma:SolidPeso molecolare:358.43JO146
CAS:JO146为针对沙眼衣原体高温需要蛋白A(CtHtrA)的蛋白酶抑制剂，其对CtHtrA和人中性粒细胞弹性蛋白酶(HNE)的IC50值分别为21.86 μM和1.15 μM，可应用于细菌感染的抑制。Formula:C31H44N3O7PColore e forma:SolidPeso molecolare:601.67L-873724
CAS:L-873724: Selective, reversible cathepsin K inhibitor; IC50s—cat K: 0.2 nM, cat S: 178 nM, cat L: 264 nM, cat B: 5239 nM; inhibits bone resorption.Formula:C23H26F3N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:481.53(R)-ND-336
CAS:(R)-ND-336: potent, selective MMP-9 inhibitor (K i = 19 nM); inhibits MMP-2 (127 nM), MMP-14 (119 nM); studied for diabetic foot ulcers.Formula:C16H18ClNO3S2Colore e forma:SolidPeso molecolare:371.89PF-00356231 hydrochloride
CAS:PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.Formula:C25H21ClN2O3SPurezza:98.39%Colore e forma:SolidPeso molecolare:464.96Ref: TM-T12414
1mg67,00€5mg177,00€10mg284,00€25mg464,00€50mg642,00€100mg853,00€500mgPrezzo su richiestaMMP-2/9-IN-1
CAS:MMP-2/9-IN-1 (Compound 4a) is a potent dual inhibitor of MMP-2 (IC50: 56 nM) and MMP-9 (IC50: 38 nM). leading to DNA fragmentation.Formula:C14H16IN7SColore e forma:SolidPeso molecolare:441.29FQ
CAS:FQ is a novel reversible inhibitor of mixed-type tyrosinase.Formula:C14H9FN2OColore e forma:SolidPeso molecolare:240.23TAPI-1
CAS:TAPI1 (TAPI) , an ADAM17/TACE inhibitor, inhibits shedding of cytokine receptors.Formula:C26H37N5O5Purezza:≥95%Colore e forma:SolidPeso molecolare:499.6GLS1 Inhibitor-3
CAS:GLS1 Inhibitor-3 (compound C147) is a potent inhibitor of GLS1 (IC50: 27.98 nM) and exhibits anti-proliferative effects.Formula:C30H32N10O2SColore e forma:SolidPeso molecolare:596.71ADAMTS-5 Inhibitor
CAS:ADAMTS-5 Inhibitor is an inhibitor of ADAMTS-5 with an IC50 of 1.1 µM and can be used in studies about cartilage destruction in arthritis.Formula:C16H11ClF3N3OS3Purezza:99.66%Colore e forma:SolidPeso molecolare:449.92Ref: TM-T14124
1mg46,00€5mg93,00€10mg122,00€25mg193,00€50mg289,00€100mg414,00€200mg580,00€1mL*10mM (DMSO)96,00€HCV-IN-36
CAS:HCV-IN-36: oral HCV inhibitor, EC50 0.016 μM, CC50 8.78 μM, potent antiviral.Formula:C30H36ClN5Colore e forma:SolidPeso molecolare:502.09TNIK-IN-1
CAS:TNIK-IN-1 is an inhibitor of Traf2- and Nck-interacting kinase (TNIK).Formula:C19H17N5O3SPurezza:98%Colore e forma:SolidPeso molecolare:395.43Diethyl pyimDC
CAS:Diethyl pyimDC is an inhibitor of human collagen prolyl 4-hydroxylase 1 (CP4H1).Formula:C14H15N3O4Colore e forma:SolidPeso molecolare:289.29Aldumastat
CAS:Aldumastat (GLPG1972) is a highly potent, specific and orally active inhibitor of ADAMTS-5.Aldumastat is used for the study of osteoarthritis of the knee.Formula:C20H24F2N4O3Purezza:99.87%Colore e forma:SolidPeso molecolare:406.43BRD-8899
CAS:BRD-8899 is a STK33 inhibitor, with an IC 50 of 11 nM [1].Formula:C17H22N4O3SColore e forma:SolidPeso molecolare:362.45Tyrosinase-IN-5
CAS:Tyrosinase-IN-5 (16c) inhibits tyrosinase with 0.02 μM IC50, reduces melanogenesis, and is low-toxicity.Formula:C18H13N3O6Colore e forma:SolidPeso molecolare:367.31MK-4882
CAS:MK-4882 is an effective inhibitor of HCV NS5A.Formula:C42H50N8O7Purezza:98%Colore e forma:SolidPeso molecolare:778.9Elasnin
CAS:Elasnin is a reversible inhibitor of elastase for human granulocyte and pancreatic enzymes with IC50 values of 1.3 and 30 µg/ml, respectively.Formula:C24H40O4Colore e forma:SolidPeso molecolare:392.57ASPER-29
CAS:ASPER-29, an Asperphenamate analog, inhibits cathepsins L/S with IC50s of 6.03/5.02 μM, useful in cancer migration/invasion research.Formula:C31H29BrN2O5SColore e forma:SolidPeso molecolare:621.54CAY10704
CAS:CAY10704: Potent HCV inhibitor, EC50=17 nM, low cytotoxicity, good in mice, liver-targeted, not hepatotoxic, weak against dengue.Formula:C18H20Cl2N2Colore e forma:SolidPeso molecolare:335.27DPP-4-IN-1
CAS:DPP-4-IN-1 inhibits DPP-4 with 49 nM IC50, ideal for diabetes study, akin to Alogliptin.Formula:C19H19ClN6Colore e forma:SolidPeso molecolare:366.85Sortin1
CAS:Sortin1, a chemical genetic-hit compound, specifically induces mislocalization of both soluble and membrane-associated vacuolar markers in plants and yeast.Formula:C26H19NO6Purezza:98%Colore e forma:SolidPeso molecolare:441.43MDK7677
CAS:MDK7677 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.Formula:C12H10N4O3Colore e forma:SolidPeso molecolare:258.23Furaprofen
CAS:Furaprofen is an HCV inhibitor with anti-inflammatory activity that inhibits carrageenan-induced paw edema in rats.Formula:C17H14O3Purezza:98.49% - 99.52%Colore e forma:SolidPeso molecolare:266.29AA10 TG2 inhibitor
CAS:AA10 is an irreversible inhibitor of transglutaminase 2 (TG2).Formula:C32H36N4O5Colore e forma:SolidPeso molecolare:556.65
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