Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(1.003 prodotti)
- Recettore dell'adenosina(247 prodotti)
- Recettore adrenergico(3.010 prodotti)
- Recettore della bombesina(33 prodotti)
- Recettore della bradichinina(60 prodotti)
- CXCR(153 prodotti)
- CaSR(33 prodotti)
- Recettore dei cannabinoidi(215 prodotti)
- Colecistochinina(1 prodotti)
- Recettore della dopamina(435 prodotti)
- Recettore dell'endotelina(83 prodotti)
- Recettore GNRH(82 prodotti)
- GPCR19(33 prodotti)
- GRK(32 prodotti)
- GTPase(22 prodotti)
- Recettore del glucagone(190 prodotti)
- Proteina Hedgehog/Smoothened(48 prodotti)
- Recettore dell'istamina(381 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(26 prodotti)
- Recettore OX(41 prodotti)
- Recettore degli oppioidi(321 prodotti)
- PAFR(13 prodotti)
- PKA(51 prodotti)
- Recettore S1P(18 prodotti)
- SGLT(31 prodotti)
- Recettore Sigma(46 prodotti)
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Trovati 5838 prodotti di "Proteina G/GPCR"
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Azepexole hydrochloride
CAS:Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaestheticFormula:C9H16ClN3OPurezza:99.88% - 99.89%Colore e forma:SoildPeso molecolare:217.7KSK94 FA
KSK94 FA is a potent histamine H3 receptor antagonist that inhibits H3 receptors and is used in the study of neuropathic pain and obesity.Formula:C26H28N4O3Purezza:97.51%Colore e forma:SoildPeso molecolare:444.53GLP-1R Agonist DMB
CAS:GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).Formula:C13H15Cl2N3O2SPurezza:99.52%Colore e forma:SolidPeso molecolare:348.25AMK (hydrochloride)
CAS:AMK, a melatonin metabolite, scavenges oxygen, inhibits prostaglandin production, reduces lipid peroxidation, and affects Parkinson's in mouse studies.Formula:C12H17ClN2O3Colore e forma:SolidPeso molecolare:272.739-deoxy-9-methylene-16,16-dimethyl Prostaglandin E2
CAS:Meteneprost is a strong, long-lasting Prostaglandin E2 analog effective in ending early monkey pregnancies without causing fever or GI issues.Formula:C23H38O4Colore e forma:SolidPeso molecolare:378.5538-iso Prostaglandin E2 isopropyl ester
CAS:8-iso PGE2 isopropyl ester: lipophilic, hydrolyzes to acid in vivo, used as prodrug, less active than parent acid.Formula:C23H38O5Colore e forma:SolidPeso molecolare:394.54Vixticibart
Vixticibart is a humanized IgG4κ antibody targeting NPR1, with HumanIgG4(S228P) kappa serving as its corresponding isotype control.Neurokinin A(4-10)
CAS:Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .Formula:C34H54N8O10SPurezza:98%Colore e forma:SolidPeso molecolare:766.9116,16-dimethyl Prostaglandin E1
CAS:16,16-dimethyl Prostaglandin E1 is a PGE1 (T1626) analog that induces bronchoconstriction and vascular smooth muscle contraction and inhibits indomethacin-Formula:C22H38O5Colore e forma:SolidPeso molecolare:382.541[D-Pro2] Spantide I TFA
<p>[D-Pro2] Spantide I TFA is an analog of Spantide I, a selective antagonist of the NK1 receptor [1].</p>Formula:C75H108N20O13·xC2HF3O2Purezza:98%Colore e forma:SolidBMY-14802
CAS:BMY-14802 (alpha-(4-fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazine butanol) is a selective and orally active sigma-1 antagonist with an IC50 of 112 nM.Formula:C18H22F2N4OPurezza:99.84%Colore e forma:SoildPeso molecolare:348.39Lamprey LH-RH I
CAS:Lamprey LH-RH I triggers ovulation and raises steroid levels in lamprey, inactive in other species.Formula:C58H79N15O15Peso molecolare:1226.34G-Protein antagonist peptide acetate
G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G protein binding.Formula:C59H68N12O11SPurezza:98.06%Colore e forma:SolidPeso molecolare:1153.33DD202-114
CAS:DD202-114 is an effective and selective agonist of GLP1R. It promotes the accumulation of cAMP, reduces blood glucose levels, and decreases food intake. Additionally, DD202-114 holds potential for research in type 2 diabetes mellitus (T2DM) and obesity studies.Formula:C33H35FN4O5Peso molecolare:586.65Biotinyl-neuropeptide W-23 (human)
CAS:Biotinyl-neuropeptide W-23 (human) is a biotinylated form of neuropeptide W-23 (human), which functions as an agonist for the NPBW1 (GPR7) and NPBW2 (GPR8)Formula:C129H197N37O30S2Peso molecolare:2810.3CB2R/FAAH modulator-1
CAS:CB2R/FAAH modulator-1: agonizes CB2R, inhibits FAAH (IC50=4 μM), alters cytokine production; used in inflammation research. Ki: CB2R=14.8 nM, CB1R=241.3 nM.Formula:C24H27NO2Purezza:99.77%Colore e forma:SoildPeso molecolare:361.48PHI-27 (porcine)
CAS:PHI-27 (porcine) is a porcine-derived peptide consisting of 27 amino acids, utilized in the identification of peptide hormones and other bioactive peptides [1].Formula:C136H216N36O40Peso molecolare:2995.39(±)-Clopidogrel (hydrochloride)
CAS:Clopidogrel is an antithrombic compound whose active metabolite is a selective, irreversible antagonist of the platelet purinergic P2Y12 receptor (IC50 = 100 nMFormula:C16H17Cl2NO2SColore e forma:SolidPeso molecolare:358.28Y4R agonist-1
CAS:Y4R Agonist-1 is a potent agonist of the Y4 receptor, exhibiting a K_i (inhibition constant) value of 0.048 nM.Formula:C51H80N18O11Peso molecolare:1121.29Canagliflozin (Standard)
CAS:Canagliflozin (Standard) is the standard substance of Canagliflozin, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor that inhibits CHO cells expressing mSGLT2, rSGLT2, and hSGLT2 (IC50=2/3.7/4.4 nM). Canagliflozin can be used for the treatment of type II diabetes mellitus (T2DM).Formula:C24H25FO5SPeso molecolare:444.52SYL-4
CAS:SYL-4 is a potential P2Y12 receptor antagonist with a Ki value of 7.35 ± 1.72 for use in synthetic dyes.Formula:C20H15N3O5SPurezza:95.76%Colore e forma:SoildPeso molecolare:409.42Spiroxatrine
CAS:<p>Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.</p>Formula:C22H25N3O3Purezza:99.94%Colore e forma:SolidPeso molecolare:379.45Fedovapagon
CAS:<p>Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.</p>Formula:C27H34N4O3Purezza:99.33%Colore e forma:SolidPeso molecolare:462.58Cimetidine (Standard)
CAS:Cimetidine (Standard) is the standard substance of Cimetidine, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Cimetidine (SKF-92334) is a histamine congener, it competitively inhibits HISTAMINE binding to HISTAMINE H2 RECEPTORS. Cimetidine has a range of pharmacological actions. It inhibits GASTRIC ACID secretion, as well as PEPSIN and GASTRIN output.Formula:C10H16N6SPeso molecolare:252.344-(4-Chlorobenzyl)phthalazin-1(2H)-one
CAS:4-(4-Chlorobenzyl)phthalazin-1(2H)-one is a useful organic compound for research related to life sciences. The catalog number is T67610 and the CAS number is 53242-88-9.Formula:C15H11ClN2OColore e forma:SolidPeso molecolare:270.72Argipressin
CAS:Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.Formula:C46H65N15O12S2Purezza:98%Colore e forma:White PowderPeso molecolare:1084.231-Methyl-4-imidazoleacetic Acid (hydrochloride)
CAS:MIMA, a stable histamine byproduct from N-methylhistamine oxidation, indicates systemic mastocytosis via urinary levels.Formula:C6H9ClN2O2Colore e forma:SolidPeso molecolare:176.601PD176252
CAS:PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the growth and proliferation of a wide range of cancer cells.Formula:C32H36N6O5Purezza:99.00%Colore e forma:SolidPeso molecolare:584.67Sumanirole maleate
CAS:Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.Formula:C15H17N3O5Purezza:98%Colore e forma:SolidPeso molecolare:319.31(S)-(+)-Dimethindene maleate
CAS:<p>(S)-(+)-Dimethindene maleate is an orally available, selective muscarinic M2 receptor and histamine H1 receptor antagonist that inhibits muscarinic M1 receptors</p>Formula:C24H28N2O4Purezza:99.94%Colore e forma:SolidPeso molecolare:408.49MrgprX2 antagonist-1
CAS:MrgprX2 antagonist-1 (compound E23) is a MrgprX2 antagonist applicable to cutaneous inflammation.Formula:C15H15F5N4O2SPurezza:99.80%Peso molecolare:410.36GLP-1R modulator C5
CAS:GLP-1R modulator C5 is a GLP-1R modulator that enhances GLP-1 binding to GLP-1R via transmembrane sites and can be used in the study of type II diabetes.Formula:C24H21NO3Purezza:99.59%Colore e forma:SolidPeso molecolare:371.43(Rac)-Rotigotine hydrochloride
CAS:(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.Formula:C19H26ClNOSColore e forma:SolidPeso molecolare:351.93Quetiapine-d8 Fumarate
CAS:Quetiapine-d8 Fumarate is a deuterated compound of Quetiapine Fumarate. Quetiapine Fumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Formula:C25H21D8N3O6SColore e forma:SolidPeso molecolare:507.63Scopine hydrochloride
CAS:<p>Scopine hydrochloride (6,7-Epoxytropine hydrochloride) is the metabolite of anisodine, which is a α1-adrenergic receptor agonist.</p>Formula:C8H13NO2·HClPurezza:98%Colore e forma:White PowderPeso molecolare:191.66L-798106
CAS:L-798106 (CM9) is an EP3 receptor antagonist that inhibits EP4, EP1, and EP2 receptors and attenuates PGE2-induced cough.Formula:C27H22BrNO4SPurezza:98.97%Colore e forma:SolidPeso molecolare:536.44Furprofen
CAS:Furprofen, an NSAID, inhibits PGE synthesis, offers analgesic effects, and is orally taken for pain relief.Formula:C14H12O4Purezza:98.62% - 99.25%Colore e forma:SolidPeso molecolare:244.24SANT 2
CAS:SANT 2 is a Hedgehog (Hh) signaling pathway antagonist with potential anti-inflammatory and anti-cancer activities.Formula:C26H26ClN3O4Purezza:99.23%Colore e forma:SolidPeso molecolare:479.96TP-16
CAS:<p>TP-16 is a novel potent and selective EP4 antagonist that blocks the function of IMCs and enhances cytotoxic T cell-mediated tumor elimination in vivo.</p>Formula:C24H22FNO4SPurezza:98.53% - 99.15%Colore e forma:SolidPeso molecolare:439.5Tegaserod
CAS:Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).Formula:C16H23N5OPurezza:99.20% - 99.89%Colore e forma:SolidPeso molecolare:301.39Calcitonin (salmon)
CAS:<p>Calcitonin (salmon), a calcium regulating hormone, is used to treat osteoporosis in women who are at least 5 years past menopause.</p>Formula:C145H240N44O48S2Purezza:99.41% - 99.80%Colore e forma:PowderPeso molecolare:3431.85Quetiapine-d8 Hemifumarate
CAS:Quetiapine-d8 Hemifumarate is a deuterated compound of Quetiapine Hemifumarate. Quetiapine Hemifumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Formula:C25H21D8N3O6SColore e forma:SolidPeso molecolare:507.63V-0219
CAS:V-0219 is a positive allosteric modulator of GLP-1 and can be used in studies about obesity-associated diabetes.Formula:C20H25F3N4O2Purezza:99.91%Colore e forma:SoildPeso molecolare:410.43Eticlopride hydrochloride
CAS:Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).Formula:C17H25ClN2O3·HClPurezza:98%Colore e forma:SolidPeso molecolare:377.31Allura Red AC (Standard)
CAS:Allura Red AC (Standard) is the standard substance of Allura Red AC, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Allura Red AC (CI 16035) is a very important food azo dye used in the food, pharmaceutical, paper, cosmetic and textile industries.Allura Red AC promotes susceptibility to experimental colitis via mouse intestinal serotonin.Formula:C18H14N2Na2O8S2Colore e forma:Dark Maroon Solid PowderPeso molecolare:496.42Granisetron
CAS:<p>Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.</p>Formula:C18H24N4OColore e forma:SolidPeso molecolare:312.41GLP-1R modulator C16
CAS:GLP-1R modulator C16 is a variable modulator that significantly increases the binding affinity of GLP-4.Formula:C21H26ClFN2O3Purezza:99.6% - >99.99%Colore e forma:SolidPeso molecolare:408.89GLP-1R modulator L7-028
CAS:GLP-1R modulator L7-028 is a variant modulator that enhances affinity for GLP-1 and cAMP signaling.Formula:C24H28N2O3Purezza:98.76% - >99.99%Colore e forma:SolidPeso molecolare:392.49Pramipexole dihydrochloride
CAS:Pramipexole dihydrochloride could be used to treat Parkinson disease.Formula:C10H18ClN3SPurezza:98%Colore e forma:White Crystalline PowderPeso molecolare:247.79Neurotensin(8-13)
CAS:Neurotensin(8-13) is Neurotensin (NT) fragment, Neurotensin(8-13) results in a decrease in cell-surface NT1 receptors (NTR1) density.Formula:C38H64N12O8Purezza:99.95%Colore e forma:SolidPeso molecolare:816.99Fexofenadine-d6
CAS:Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.Formula:C32H39NO4Purezza:98%Colore e forma:SolidPeso molecolare:507.69Setiptiline maleate
CAS:Setiptiline maleate is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist, 5-HT serotonin receptor antagonist.Formula:C23H23NO4Purezza:99.94%Colore e forma:SolidPeso molecolare:377.43Piribedil D8
CAS:Piribedil D8 is the deuterium labeled Piribedil, which is an agent of antiparkinsonian.Formula:C16H18N4O2Purezza:98%Colore e forma:SolidPeso molecolare:306.39Gizzerosine
CAS:Gizzerosine, a biogenic amine formed during feed processing, is a toxicant that induces mortality in livestock.Formula:C11H20N4O2Colore e forma:SolidPeso molecolare:240.3Trimethobenzamide
CAS:<p>Trimethobenzamide (Ro 2-9578) is a D2 antagonist used to prevent nausea and vomiting.</p>Formula:C21H28N2O5Colore e forma:SolidPeso molecolare:388.46RU-SKI 43 Hydrochloride
CAS:RU-SKI 43 Hydrochloride is a selective Hedgehog acyltransferase inhibitor (IC50 850 nM) with reported anticancer activity in tumor biology studies.Formula:C22H31ClN2O2SPurezza:98%Colore e forma:SolidPeso molecolare:423.01SB-408124 Hydrochloride
CAS:SB-408124 Hydrochloride is a non-peptide OX1 receptor antagonist(Ki of 57 nM and 27 nM in both whole cell and membrane, respectively).Formula:C19H19ClF2N4OPurezza:98%Colore e forma:SolidPeso molecolare:392.831-Phenylbiguanide HCl
CAS:<p>Compound PDK0269, as 5-HT3 receptor agonists(3–100 μM, pEC50 5.05±0.06), acutely increased XII (hypoglossal) burst frequency and regularity, and decreased bursts/episode . Phenylbiguanide produced a dose-related (10-500 microM) increase in the release of dopamine (280-2000%). When nomifensine (5 microM) was included in the Ringer solution, the effect of Compound PDK0269 on the release of dopamine was ameliorated or inhibited.</p>Formula:C8H12ClN5Purezza:99.31%Colore e forma:SolidPeso molecolare:213.67Tiotidine
CAS:Tiotidine is a selective histamine H2-receptor antagonist (pA2=7.3-7.8 for guinea-pig right atrium).Formula:C10H16N8S2Purezza:98%Colore e forma:SolidPeso molecolare:312.42L 888607
CAS:L 888607 is an effective and selective CRTH2 agonist (Ki: 0.8 nM).Formula:C19H15ClFNO2SColore e forma:SolidPeso molecolare:375.84ML 00253764
CAS:melanocortin MC4 receptor antagonistFormula:C18H18BrFN2OColore e forma:SolidPeso molecolare:377.255-HT2B antagonist-1
CAS:Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.Formula:C11H14BrN5Purezza:99.965%Colore e forma:SolidPeso molecolare:296.17Ziprasidone D8
CAS:Ziprasidone D8, deuterium-labeled, is a potent antipsychotic, antagonizing 5-HT and dopamine receptors.Formula:C21H21ClN4OSPurezza:98%Colore e forma:SolidPeso molecolare:420.99Olanzapine D3
CAS:<p>Olanzapine D3 is the deuterium labeled Olanzapine.</p>Formula:C17H20N4SPurezza:98%Colore e forma:SolidPeso molecolare:315.45Lysosphingomyelin (d18:1)
CAS:<p>Sphingomyelins are phosphorylcholine, sphingosine, and fatty acid. Lysosphingomyelin, missing the fatty acid, activates diverse cellular pathways.</p>Formula:C23H49N2O5PColore e forma:SolidPeso molecolare:464.6284-Hydroxyatomoxetine D3
CAS:<p>4-Hydroxyatomoxetine D3, a deuterium variant, is Atomoxetine's active metabolite, metabolized by CYP2D6, an adrenergic reuptake blocker.</p>Formula:C17H21NO2Purezza:98%Colore e forma:SolidPeso molecolare:274.37Lanreotide
CAS:Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.Formula:C54H69N11O10S2Colore e forma:SolidPeso molecolare:1096.32Cariprazine D6
CAS:<p>Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).</p>Formula:C21H26D6Cl2N4OPurezza:98%Colore e forma:SolidPeso molecolare:433.45Calcium-Sensing Receptor Antagonists I
CAS:Calcium-Sensing Receptor Antagonists I functions as an antagonist to the parathyroid hormone receptors that sense calcium.Formula:C23H24N2O2Colore e forma:SolidPeso molecolare:360.45Ivabradine-d6 hydrochloride
CAS:Ivabradine HCl: novel If inhibitor, IC50 2.9 μM; lowers heart rate. Ivabradine D6 HCl is its deuterium variant.Formula:C27H37ClN2O5Purezza:98%Colore e forma:SolidPeso molecolare:511.08(+)-Penbutolol
CAS:(+)-Penbutolol is an antagonist of β-adrenoceptor(IC50 of 0.74 μM). (+)-Penbutolol is an optical isomer of l-penbutolol with Na+ channel-blocking action.Formula:C18H29NO2Colore e forma:SolidPeso molecolare:291.43Lecirelin
CAS:Lecirelin is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cysts.Formula:C59H84N16O12Colore e forma:SolidPeso molecolare:1209.4Thioridazine
CAS:Thioridazine: an antipsychotic, anti-anxiety drug, blocks dopamine D2, PI3K-Akt-mTOR; halts angiogenesis, kills cancer cells, targets CSCs.Formula:C21H26N2S2Colore e forma:SolidPeso molecolare:370.57Vilazodone-d8
CAS:Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.Formula:C26H27N5O2Purezza:98%Colore e forma:SolidPeso molecolare:449.573-O-Methyldopa-d3
CAS:3-O-Methyldopa-d3 is a deuterated compound of 3-O-Methyldopa. 3-O-Methyldopa has a CAS number of 300-48-1.Formula:C10H10D3NO4Peso molecolare:214.23Brombuterol hydrochloride
CAS:Brombuterol is an agonist of the β2-adrenergic receptor (β2-AR).1It has been used as an illicit feed additive to increase the muscle-to-fat ratio of livestock.Formula:C12H19Br2ClN2OColore e forma:SolidPeso molecolare:402.56Cetirizine D8
CAS:Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.Formula:C21H25ClN2O3Purezza:98%Colore e forma:SolidPeso molecolare:396.94Clomipramine D3 hydrochloride
CAS:Clomipramine D3 hydrochloride is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter blocker (Ki: 0.14, 54 and 3 nM).Formula:C19H24Cl2N2Colore e forma:SolidPeso molecolare:354.333-Hydroxy agomelatine D3
CAS:3-Hydroxy agomelatine D3 is a deuterated metabolite of Agomelatine and a 5-HT2C antagonist (IC50: 3.2 μM, Ki: 1.8 μM).Formula:C15H17NO3Purezza:98%Colore e forma:SolidPeso molecolare:262.32Dehydroaripiprazole
CAS:Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.Formula:C23H25Cl2N3O2Purezza:98.7%Colore e forma:SolidPeso molecolare:446.37Etofylline clofibrate
CAS:Etofylline clofibrate has a hypolipidemic and antithrombotic effect and it also has an agonistic interaction with intimal PGI2.Formula:C19H21ClN4O5Colore e forma:SolidPeso molecolare:420.85Mozavaptan hydrochloride
CAS:Mozavaptan is a vasopressin receptor antagonist.Formula:C27H30ClN3O2Colore e forma:SolidPeso molecolare:464Alosetron D3 Hydrochloride
CAS:<p>Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>Formula:C17H19ClN4OPurezza:98%Colore e forma:SolidPeso molecolare:333.83Zaloglanstat
CAS:Zaloglanstat (ISC-27864) is a selective, orally active mPGES-1 inhibitor with an IC50 of 5 nM, analgesic in osteoarthritis and inflammatory arthritis.Formula:C21H20ClF3N4O2Purezza:99.97%Colore e forma:SolidPeso molecolare:452.86Fluvoxamine
CAS:Fluvoxamine (DU-23000) is a selective, orally available 5-HT and serotonin reuptake inhibitor (SSRI) exhibiting antidepressant effects.Formula:C15H21F3N2O2Purezza:99.91%Colore e forma:SolidPeso molecolare:318.33TFLLR-NH2(TFA)
CAS:TFLLR-NH2 (TFA) is a selective PAR1 agonist with an EC50 of 1.9 μM. EC50: 1.9 μM (PAR1)Formula:C33H54F3N9O8Purezza:98%Colore e forma:SolidPeso molecolare:761.83BMS-986020 sodium
CAS:BMS-986020 sodium (AM152 sodium) is a high-affinity LPA1 antagonist for investigating idiopathic pulmonary fibrosis.Formula:C29H25N2NaO5Purezza:99.83%Colore e forma:SolidPeso molecolare:504.51Tetrahexyldecyl ascorbate
CAS:Tetrahexyldecyl ascorbate is a precursor of ascorbic acid, a more stable and permeable form of vitamin C. anti-hyperpigmentation antioxidant that inhibits MMP.Formula:C70H128O10Purezza:98%Colore e forma:SolidPeso molecolare:1129.76GB-88
CAS:GB-88 is an selective , oral non-peptide antagonist of PAR2, inhibits PAR2 activated Ca2+ release with an IC50 of 2 μM.Formula:C32H42N4O4Colore e forma:SolidPeso molecolare:546.7Doxazosin D8
CAS:Doxazosin D8, a deuterium-labeled version, is a selective AP1 adrenergic antagonist and a quinazoline derivative.Formula:C23H25N5O5Purezza:98%Colore e forma:SolidPeso molecolare:459.52Propranolol-d7 hydrochloride
CAS:Propranolol D7 HCl: deuterium-labeled, nonselective βAR antagonist.Formula:C16H22ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:302.85Levosalbutamol Hydrochloride
CAS:Levosalbutamol Hydrochloride is a β2-adrenergic receptor agonist. It is used to treat asthma and chronic obstructive pulmonary disease.Formula:C13H22ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:275.77Metipranolol hydrochloride
CAS:Metipranolol hydrochloride is a non-selective β-adrenergic receptor blocking agent.Formula:C17H28ClNO4Purezza:98%Colore e forma:SolidPeso molecolare:345.86(Rac)-Mirabegron-d5
CAS:(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.Formula:C21H24N4O2SPurezza:98%Colore e forma:SolidPeso molecolare:401.54Cudarolimab
CAS:<p>Cudarolimab (IBI-101) is a fully human anti-OX40 antibody with potential immune checkpoint inhibitory and anti-tumor activity for the study of cancer.</p>Purezza:97.5% (SDS-PAGE); 98.2% (SEC-HPLC) - 97.5% (SDS-PAGE); 98.2% (SEC-HPLC)Colore e forma:LiquidBombesin
CAS:Bombesin: 14-amino acid peptide from toad skin with two mammalian homologs, neuromedin B and gastrin-releasing peptide.Formula:C71H110N24O18SColore e forma:While Lyophilized PowderPeso molecolare:1619.85Hydroxyzine D8
CAS:Hydroxyzine D8, a deuterium-labeled version of Hydroxyzine, acts as a histamine H1-receptor antagonist.Formula:C21H27ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:382.95Asenapine hydrochloride
CAS:<p>Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.</p>Formula:C17H17Cl2NOColore e forma:SolidPeso molecolare:322.23β2AR/M-receptor agonist-2
CAS:<p>β2AR/M-receptor agonist-2 is a dual-function compound acting as a muscarinic antagonist and β2 adrenoceptor agonist (MABA).</p>Formula:C36H49ClN4O7SColore e forma:SolidPeso molecolare:717.31MRS-3777 hemioxalate
CAS:<p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>Formula:C17H19N5OC2H2O4Purezza:97.10%Colore e forma:SolidPeso molecolare:354.39
