Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(939 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.945 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(148 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(407 prodotti)
- Recettore dell'endotelina(76 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(31 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(165 prodotti)
- Proteina Hedgehog/Smoothened(44 prodotti)
- Recettore dell'istamina(358 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(297 prodotti)
- PAFR(11 prodotti)
- PKA(48 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5352 prodotti di "Proteina G/GPCR"
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α-MSH, amide Acetate
<p>a-MSH, amide Acetate as an endogenous neuropeptide.</p>Formula:C79H113N21O21SPurezza:98.67%Colore e forma:SolidPeso molecolare:1724.94Phentolamine
CAS:<p>Phentolamine mesylate is an alpha-1 and alpha-2 selective adrenergic receptor antagonist</p>Formula:C17H19N3OPurezza:99.86% - 99.94%Colore e forma:Crystals SolidPeso molecolare:281.35Cenicriviroc
CAS:<p>Cenicriviroc (TAK-652), oral CCR2/CCR5 blocker, inhibits HIV-1/HIV-2, with strong anti-infective/anti-inflammatory effects.</p>Formula:C41H52N4O4SPurezza:97.87%Colore e forma:SolidPeso molecolare:696.94Xamoterol
CAS:<p>Xamoterol is a cardiac stimulant.</p>Formula:C16H25N3O5Colore e forma:SolidPeso molecolare:339.39γ-Mangostin
CAS:<p>Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.</p>Formula:C23H24O6Purezza:98.55% - 99.08%Colore e forma:SolidPeso molecolare:396.43Maraviroc
CAS:<p>Maraviroc: a CCR5 antagonist blocking HIV-1 entry; IC50s—MIP-1α: 3.3nM, MIP-1β: 7.2nM, RANTES: 5.2nM.</p>Formula:C29H41F2N5OPurezza:97.13% - 99.59%Colore e forma:Brown SolidPeso molecolare:513.67TS-011
CAS:<p>N-(3-Chloro-4-morpholinophenyl)-N'-hydroxyformimidamide (TS-011) is a selective 20-Hydroxyeicosatetraenoic acid synthesis inhibitor.</p>Formula:C11H14ClN3O2Purezza:99.48%Colore e forma:SolidPeso molecolare:255.7Dexmedetomidine hydrochloride
CAS:<p>Dexmedetomidine hydrochloride (Precedex) is a potent, selective, orally active α2-adrenoceptor agonist.Cost-effective and quality-assured.</p>Formula:C13H16N2·HClPurezza:99.94% - 99.94%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:236.74CAY10444
CAS:<p>CAY10444 is an S1P3 specific antagonist.</p>Formula:C15H29NO2SPurezza:99.15% - 99.61%Colore e forma:SolidPeso molecolare:287.46[Lys5,MeLeu9,Nle10]-NKA(4-10)
CAS:<p>Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).</p>Formula:C39H65N9O9Purezza:>99.99%Colore e forma:SolidPeso molecolare:803.99VUF 10166
CAS:<p>VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.</p>Formula:C13H15ClN4Purezza:99.66%Colore e forma:SolidPeso molecolare:262.74Buclizine
CAS:<p>Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects.</p>Formula:C28H33ClN2Colore e forma:SolidPeso molecolare:433.03Idalopirdine Hydrochloride
CAS:<p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>Formula:C20H20ClF5N2OPurezza:99.77%Colore e forma:SolidPeso molecolare:434.83Glasdegib
CAS:<p>Glasdegib (PF-04449913) (PF-04449913) is a potent, and orally bioavailable Smoothened (Smo) inhibitor with IC50 of 5 nM. Phase 2.</p>Formula:C21H22N6OPurezza:98.72%Colore e forma:SolidPeso molecolare:374.44BX471
CAS:<p>BX471 (BX 471) is a potent, selective non-peptide CCR1 antagonist.</p>Formula:C21H24ClFN4O3Purezza:98% - 99.94%Colore e forma:SolidPeso molecolare:434.89CYM-5520
CAS:<p>CYM-5520 is a noncompetitive allosteric agonist of S1P2</p>Formula:C21H19N3O2Purezza:99.47%Colore e forma:SolidPeso molecolare:345.39Lurasidone
CAS:<p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>Formula:C28H36N4O2SPurezza:99.78% - 99.91%Colore e forma:SolidPeso molecolare:492.68SAX-187 hydrochloride
CAS:<p>WAY-181187 is a potent, selective 5-HT6 agonist with high affinity (2.2-4.8 nM), and increases GABA in rat cortex at 3-30 mg/kg s.c.</p>Formula:C15H14Cl2N4O2S2Colore e forma:SolidPeso molecolare:417.33Exenatide
CAS:<p>Exenatide (Extendin-4) is a glucagon-like protein-1 (GLP-1) receptor agonist.</p>Formula:C186H286N50O62SPurezza:99.42%Colore e forma:SolidPeso molecolare:4247Harmine
CAS:<p>Harmine (Telepathine) is an alkaloid isolated from seeds of Peganum harmala.</p>Formula:C13H12N2OPurezza:98.29% - 99.92%Colore e forma:Off-White SolidPeso molecolare:212.25Fuscoside
CAS:<p>Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.</p>Formula:C26H31N3O4Purezza:98.13% - 99.66%Colore e forma:SolidPeso molecolare:449.54ML-18
CAS:<p>ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.</p>Formula:C32H35N5O5Purezza:98.62% - >99.99%Colore e forma:SolidPeso molecolare:569.65TG4-155
CAS:<p>TG4-155: brain-penetrant EP2 inhibitor, KB 2.4 nM; >1000x weaker at EP4, KB 11.4 μM; selective over other receptors/channels.</p>Formula:C23H26N2O4Purezza:97.2%Colore e forma:SolidPeso molecolare:394.46Fluphenazine decanoate
CAS:<p>Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.</p>Formula:C32H44F3N3O2SPurezza:98.14%Colore e forma:SolidPeso molecolare:591.77Ramosetron hydrochloride
CAS:<p>Ramosetron hydrochloride (YM-060) is a serotonin 5-HT3 receptor antagonist. It is used to treat diarrhea-predominant irritable bowel syndrome and nausea.</p>Formula:C17H18ClN3OPurezza:99.95%Colore e forma:SolidPeso molecolare:315.8Tianeptine
CAS:<p>Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。</p>Formula:C21H25ClN2O4SPurezza:99.04%Colore e forma:SolidPeso molecolare:436.95Seltorexant hydrochloride
CAS:<p>Seltorexant hydrochloride is a selective, orally active and high-affinity antagonist of OX2R with pKi values of 8.0 and 8.1 for human and rat OX2R.</p>Formula:C21H23ClFN7OPurezza:98%Colore e forma:SolidPeso molecolare:443.91AC 187 Acetate
<p>AC 187 Acetate is a potent antagonist of amylin receptor .AC 187 shows more selective for amylin receptor than calcitonin and CGRP receptors.</p>Formula:C129H209N37O42Purezza:99.71%Colore e forma:SolidPeso molecolare:2950.26Amezinium methylsulfate
CAS:<p>Amezinium methylsulfate (Lu-1631) has multiple mechanisms, including stimulation of α and β-1 receptors and inhibition of noradrenaline and tyramine uptake.</p>Formula:C12H15N3O5SPurezza:99.64%Colore e forma:SolidPeso molecolare:313.33Elagolix sodium
CAS:<p>Elagolix sodium (NBI-56418 sodium) is a GnRH receptor (GnRHR) antagonist ( IC50 and Ki of 0.25 and 3.7 nM, respectively).</p>Formula:C32H29F5N3NaO5Purezza:99.71%Colore e forma:SolidPeso molecolare:653.57Bimatoprost
CAS:<p>Bimatoprost (AGN 192024) is a cloprostenol-derived amide that is used as an antihypertensive agent in the treatment of open-angle glaucoma and ocular</p>Formula:C25H37NO4Purezza:98% - >99.99%Colore e forma:Crystalline SolidPeso molecolare:415.57Arformoterol Tartrate
CAS:<p>Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.</p>Formula:C23H30N2O10Purezza:99.98%Colore e forma:SolidPeso molecolare:494.49Neuromedin N acetate(92169-45-4 free base)
<p>Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct</p>Formula:C40H67N7O10Purezza:99.95%Colore e forma:SolidPeso molecolare:805.9Scyliorhinin II acetate
<p>Scyliorhinin II acetate is a selective agonist of the neurokinin-3 (NK3) receptor (Ki = 2.5 nM) in rat cerebral cortex.</p>Formula:C79H123N21O28S3Purezza:99.06%Colore e forma:SolidPeso molecolare:1911.14AdipoRon hydrochloride
CAS:<p>AdipoRon hydrochloride is a specific, orally active AdipoR agonist, capable of binding AdipoR1 (Kd: 1.8 μM) and AdipoR2 (Kd: 3.1 μM).</p>Formula:C27H29ClN2O3Colore e forma:SolidPeso molecolare:464.99PNU-282987
CAS:<p>PNU-282987 is a selective α7 nicotinic acetylcholine receptor(α7 nAChR) agonist with Ki of 26 nM; no affinity for α1β1γδ and α3β4 nAChRs (IC50 ≥ 60 μM).</p>Formula:C14H18Cl2N2OPurezza:99% - >99.99%Colore e forma:SolidPeso molecolare:301.21BMY 7378 dihydrochloride
CAS:<p>BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.</p>Formula:C22H33Cl2N3O3Purezza:97.32% - 99.08%Colore e forma:SolidPeso molecolare:458.42TC-G 1005
CAS:<p>TC-G 1005 is a potent and selective GPBA agonist (EC50 :0.72 nM; hTGR5).</p>Formula:C25H25N3O2Purezza:98.60% - 99.78%Colore e forma:SolidPeso molecolare:399.48Zatebradine
CAS:<p>Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).</p>Formula:C26H36N2O5Purezza:98%Colore e forma:SolidPeso molecolare:456.57SB-200646
CAS:<p>SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor</p>Formula:C15H14N4OPurezza:99.61%Colore e forma:SolidPeso molecolare:266.3Montelukast
CAS:<p>Montelukast (Singular), oral asthma med, linked to rare liver injury.</p>Formula:C35H36ClNO3SPurezza:98.56% - >99.99%Colore e forma:SolidPeso molecolare:586.18SKF-83566
CAS:<p>SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.</p>Formula:C17H18BrNOPurezza:95.00% - 99.82%Colore e forma:SolidPeso molecolare:332.23Chlorphenoxamine
CAS:<p>Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.</p>Formula:C18H22ClNOPurezza:99.44% - 99.85%Colore e forma:SolidPeso molecolare:303.83Norepinephrine bitartrate salt
CAS:<p>Norepinephrine bitartrate salt is an adrenergic neurotransmitter.</p>Formula:C12H17NO9Purezza:97.32% - 99.97%Colore e forma:SolidPeso molecolare:319.27Tasimelteon
CAS:<p>Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.</p>Formula:C15H19NO2Purezza:98.93% - 99.93%Colore e forma:SolidPeso molecolare:245.32Pramlintide acetate(151126-32-8 free base)
CAS:<p>Pramlintide acetate is a polypeptide analogue of human amylin. It serves as an antidiabetic agent and exhibits antineoplastic activity in colorectal cancer.</p>Formula:C173H271N51O55S2Purezza:>99.99%Colore e forma:SolidPeso molecolare:4009H4 Receptor antagonist 1
CAS:<p>H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.</p>Formula:C16H17ClN4OPurezza:98.81%Colore e forma:SolidPeso molecolare:316.79Urapidil
CAS:<p>Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.</p>Formula:C20H29N5O3Purezza:99.85% - >99.99%Colore e forma:SolidPeso molecolare:387.48Brexpiprazole
CAS:<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Formula:C25H27N3O2SPurezza:99.06% - 99.96%Colore e forma:SolidPeso molecolare:433.57GBR 12935
CAS:<p>GBR-12935: selective dopamine inhibitor, used in Parkinson's research.</p>Formula:C28H34N2OColore e forma:SolidPeso molecolare:414.58PF-04418948
CAS:<p>PF-04418948 is a potent EP2 receptor antagonist. Displays over 2000-fold selectivity for EP2 receptors over EP1, EP3, EP4, DP1 amd CRTH2 receptors.</p>Formula:C23H20FNO5Purezza:98.67% - 99.45%Colore e forma:SolidPeso molecolare:409.41UFP 803 acetate
UFP 803 acetate is a potent ligand of urotensin-II (UT) receptor. UFP-803 displays the activity of a lower residual agonist.Formula:C52H68N10O14S2Purezza:99.78%Colore e forma:SolidPeso molecolare:1121.29Vorapaxar
CAS:<p>Vorapaxar (MK-5348) (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).</p>Formula:C29H33FN2O4Purezza:98.77% - 99.93%Colore e forma:SolidPeso molecolare:492.58Octreotide Acetate
CAS:<p>Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.</p>Formula:C51H70N10O12S2Purezza:99.03% - 99.87%Colore e forma:Less To Off-White Lyophilised Solid Colourless To Off-White Lyophilised SolidPeso molecolare:1079.3M 1145 acetate
<p>M1145 acetate: chimeric peptide, selective GAL2 agonist, Ki=6.55 nM; >90x affinity vs GAL1, 76x vs GalR3. Enhances galanin signal.</p>Formula:C130H209N37O34Purezza:99.1%Colore e forma:SolidPeso molecolare:2834.28Decloxizine dihydrochloride
CAS:<p>Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.</p>Formula:C21H28N2O2·2ClHPurezza:99.73%Colore e forma:SolidPeso molecolare:413.39EST64454 hydrochloride
CAS:<p>EST64454 hydrochloride (EST64454) is a highly soluble σ1 receptor antagonist (Ki : 22 nM),has the potential for Pain Management.</p>Formula:C18H23ClF2N4O2Purezza:99.15%Colore e forma:SolidPeso molecolare:400.85Ritanserin
CAS:<p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>Formula:C27H25F2N3OSPurezza:99.77% - 99.89%Colore e forma:SolidPeso molecolare:477.57Betahistine
CAS:<p>Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.</p>Formula:C8H12N2Purezza:99.87% - 99.87%Colore e forma:Yellowish Liquid Liquid LiquidPeso molecolare:136.19Loxapine hydrochloride
CAS:<p>Loxapine hydrochloride, an oral anti-psychotic, inhibits dopamine and blocks 5-HT receptors.</p>Formula:C18H19Cl2N3OColore e forma:SolidPeso molecolare:364.27N-Acetylhistamine acetate
<p>N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.</p>Formula:C9H15N3O3Purezza:98%Colore e forma:SolidPeso molecolare:213.23Adrenocorticotropic Hormone (ACTH) (4-10) TFA
<p>Adrenocorticotropic Hormone (ACTH) (4-10) TFA (Acth (4-10)) is an agonist of potent melanocortin(MC4R) receptor .</p>Formula:C46H60F3N13O12SPurezza:98.49%Colore e forma:SolidPeso molecolare:1076.12SCH-37370
CAS:<p>SCH-37370 is an effective and orally active dual antagonist of platelet-activating factor and histamine.</p>Formula:C21H21ClN2OPurezza:99.07%Colore e forma:SolidPeso molecolare:352.86Ibrolipim
CAS:<p>Ibrolipim (NO-1886) attenuates high glucose-induced endothelial dysfunction in cultured human umbilical vein endothelial cells via PI3K/Akt pathway.</p>Formula:C19H20BrN2O4PPurezza:98.04%Colore e forma:SolidPeso molecolare:451.25FSLLRY-NH2 TFA(245329-02-6 free base)
<p>FSLLRY-NH2 TFA inhibits PAR2, reverses taxol-induced pain, and reduces itch in mice; blocks ERK and collagen in fibroblasts.</p>Formula:C41H61F3N10O10Purezza:99.32%Colore e forma:SolidPeso molecolare:910.99Ziprasidone mesylate
CAS:<p>Ziprasidone mesylate (CP-88059), an oral 5-HT & dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>Formula:C22H25ClN4O4S2Colore e forma:SolidPeso molecolare:509.04Sotagliflozin
CAS:<p>Sotagliflozin (LP-802034) is an orally bioavailable inhibitor of the sodium-glucose co-transporter subtype 1 (SGLT1) and 2 (SGLT2), with potential</p>Formula:C21H25ClO5SPurezza:99% - 99.86%Colore e forma:SolidPeso molecolare:424.94Mesdopetam
CAS:<p>Mesdopetam (IRL790), a D3 antagonist, has Ki=90 nM, IC50=9.8 μM, stabilizes psychomotors, used in Parkinson's research.</p>Formula:C12H18FNO3SColore e forma:SolidPeso molecolare:275.34Brompheniramine
CAS:<p>Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.</p>Formula:C16H19BrN2Colore e forma:SolidPeso molecolare:319.24M617 acetate
<p>M617 acetate is a selective agonist of galanin receptor 1 (GAL1).</p>Formula:C112H161N29O28Purezza:96.02%Colore e forma:SolidPeso molecolare:2361.65HS024
CAS:<p>HS024 is a highly potent melanocortin MC4 receptor antagonist, increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats.</p>Formula:C58H79N19O10S2Purezza:>99.99%Colore e forma:SolidPeso molecolare:1266.5SB-222200
CAS:<p>SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).</p>Formula:C26H24N2OPurezza:97.13%Colore e forma:SolidPeso molecolare:380.48GSK 789472 hydrochloride
CAS:<p>GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.</p>Formula:C15H22ClN3OPurezza:99.89%Colore e forma:SolidPeso molecolare:295.81Guanabenz Acetate
CAS:<p>Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor.</p>Formula:C8H8Cl2N4·C2H4O2Purezza:99% - 99.66%Colore e forma:White Solid From Acetonitrile White SolidPeso molecolare:291.13Decloxizine
CAS:<p>Decloxizine is a H1 receptor antagonist</p>Formula:C21H28N2O2Purezza:99.53%Colore e forma:White Or Similar To White PowderPeso molecolare:340.46Haloperidol decanoate
CAS:<p>Haloperidol decanoate (KD 16), an antipsychotic, treats schizophrenia and mood disorders as an intramuscular ester.</p>Formula:C31H41ClFNO3Purezza:99.57% - 99.72%Colore e forma:SolidPeso molecolare:530.11Pergolide
CAS:<p>Pergolide is a long-acting and orally active dopamine receptor D1/D2 agonist and ergoline derivative, used in the study of Parkinson's disease</p>Formula:C19H26N2SPurezza:99.95%Colore e forma:SolidPeso molecolare:314.49ACTH (1-17) acetate
<p>ACTH (1-17) acetate is a potent agonist at the human melanocortin 1 (MC1) receptor with high affinity(Ki = 0.21 nM).</p>Formula:C97H149N29O25SPurezza:98.53%Colore e forma:SolidPeso molecolare:2153.47Cimetidine hydrochloride
CAS:<p>Cimetidine (SKF-92334) is an oral H2 blocker with Ki 0.6 μM, anti-cancer and anti-inflammatory properties, used for ulcer research.</p>Formula:C10H17ClN6SColore e forma:SolidPeso molecolare:288.8S26131
CAS:<p>S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of</p>Formula:C31H34N2O4Purezza:99.77%Colore e forma:SolidPeso molecolare:498.614F 4PP oxalate
CAS:<p>4F 4PP oxalate is a 5-HT2A antagonist.</p>Formula:C22H26FNO·C2H2O4Purezza:97.34%Colore e forma:SolidPeso molecolare:429.49Domperidone monomaleate
CAS:<p>Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.</p>Formula:C26H28ClN5O6Colore e forma:SolidPeso molecolare:541.98ML221
CAS:<p>ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM in</p>Formula:C17H11N3O6SPurezza:97.74%Colore e forma:SolidPeso molecolare:385.35Loxapine
CAS:<p>Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.</p>Formula:C18H18ClN3OPurezza:99.88%Colore e forma:Pale Yellowish Crystals From Petroleum Ether SolidPeso molecolare:327.81LIXIVAPTAN
CAS:<p>Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)</p>Formula:C27H21ClFN3O2Purezza:98.36%Colore e forma:SolidPeso molecolare:473.93Isoetharine mesylate salt
CAS:<p>Isoetharine mesylate salt (Isoetarine mesilate) is a β-adrenergic receptor agonist.</p>Formula:C14H25NO6SPurezza:99.35% - 99.75%Colore e forma:SolidPeso molecolare:335.42Levobetaxolol hydrochloride
CAS:<p>Levobetaxolol hydrochloride ((S)-Betaxolol hydrochloride) is a beta blocker, used to lower the pressure in the eye in treating conditions such as glaucoma.</p>Formula:C18H29NO3·HClPurezza:98.80% - 99.69%Colore e forma:SolidPeso molecolare:343.89Neuropeptide EI, rat acetate
<p>Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.</p>Formula:C65H102N16O25Purezza:95.55%Colore e forma:SolidPeso molecolare:1507.6Motilin (26-47), human, porcine
CAS:<p>Motilin (26-47) binds Motilin receptors in hamster cells; Ki=2.3 nM, EC50=0.3 nM; same for humans, pigs.</p>Formula:C120H188N34O35SPurezza:98%Colore e forma:SolidPeso molecolare:2699.07Piperacetazine
CAS:<p>Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.</p>Formula:C24H30N2O2SPurezza:99.9% - 99.92%Colore e forma:SolidPeso molecolare:410.57MK 571
CAS:<p>MK 571 (L660711) is an orally active antagonist of CysLT1 receptor.</p>Formula:C26H27ClN2O3S2Purezza:98.69% - 99.65%Colore e forma:SolidPeso molecolare:515.09Bromodiphenhydramine
CAS:<p>Ambodryl, an antihistamine effective against many bacteria, aids in skin allergy studies.</p>Formula:C17H20BrNOColore e forma:SolidPeso molecolare:334.252-Pyridylethylamine dihydrochloride
CAS:<p>2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.</p>Formula:C7H12Cl2N2Purezza:99.42%Colore e forma:SolidPeso molecolare:195.09Eledoisin Related Peptide 2TFA
<p>Eledoisin Related Peptide 2TFA (Eledoisin Related Peptide 2TFA (2990-43-4(free base))) is a tachykinin receptor ligand.</p>Formula:C38H60F6N8O10SPurezza:99%Colore e forma:SolidPeso molecolare:934.99Almotriptan
CAS:<p>Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.</p>Formula:C17H25N3O2SPurezza:99.85%Colore e forma:Light Yellow Or White PowerPeso molecolare:335.46Escitalopram Oxalate
CAS:<p>Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.</p>Formula:C22H23FN2O5Purezza:97.39% - 99.73%Colore e forma:White SolidPeso molecolare:414.43Irdabisant hydrochloride
CAS:<p>Irdabisant (CEP-26401) is a selective H3R inverse agonist, BBB-penetrable, with cognition-enhancing effects.</p>Formula:C18H24ClN3O2Colore e forma:SolidPeso molecolare:349.86Romifidine hydrochloride
CAS:<p>Romifidine hydrochloride, an α2 adrenergic receptor agonist, induces sedation effects in vivo.</p>Formula:C9H10BrClFN3Colore e forma:SolidPeso molecolare:294.55SKF38393 hydrobromide
CAS:<p>SKF38393 hydrobromide is the salt form of SKF38393.a dopamine D1 receptor agonist that increases the expression of Shati/Nat8L mRNA in the NAc of mice;</p>Formula:C16H18BrNO2Purezza:98.99%Colore e forma:SolidPeso molecolare:336.22AM966
CAS:<p>AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.</p>Formula:C27H23ClN2O5Purezza:98.06% - 99.79%Colore e forma:SolidPeso molecolare:490.93
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