Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(939 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.945 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(148 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(407 prodotti)
- Recettore dell'endotelina(76 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(31 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(165 prodotti)
- Proteina Hedgehog/Smoothened(44 prodotti)
- Recettore dell'istamina(358 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(297 prodotti)
- PAFR(11 prodotti)
- PKA(48 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5352 prodotti di "Proteina G/GPCR"
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NPY 5RA972
CAS:<p>NPY 5RA972 is a neuropeptide Y Y5 receptor antagonist</p>Formula:C21H25N3O2Purezza:99.02% - 99.56%Colore e forma:SolidPeso molecolare:351.44RS 504393
CAS:RS 504393 is a highly selective CCR2 chemokine receptor antagonist (IC50s: 89 nM and > 100 μM for human recombinant CCR2 and CCR1).Formula:C25H27N3O3Purezza:98.64% - 99.62%Colore e forma:SolidPeso molecolare:417.5Idazoxan hydrochloride
CAS:<p>Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.</p>Formula:C11H12N2O2·HClPurezza:99.42% - 99.84%Colore e forma:SolidPeso molecolare:240.691-[(5-methylisoxazol-3-yl)methyl]piperazine
CAS:<p>1-[(5-methylisoxazol-3-yl)methyl]piperazine (Piperazine, 1-[(5-methyl-3-isoxazolyl)methyl]- (9CI)) is a P2Y12 inhibitor.</p>Formula:C9H15N3OPurezza:95%Colore e forma:SolidPeso molecolare:181.23Chlorphenesin
CAS:<p>Chlorphenesin (Chlorophenesin) is an antigen-associated immunosuppressant that inhibits IgE-mediated histamine release. It is also used as an antimycotic agent.</p>Formula:C9H11ClO3Purezza:99.59%Colore e forma:SolidPeso molecolare:202.63SBI-115
CAS:<p>SBI-115 is an antagonist of TGR5. SBI-115 decreases hepatic cystogenesis with polycystic liver diseases via inhibiting TGR5</p>Formula:C14H13ClN2O4SPurezza:99.53% - 99.78%Colore e forma:SolidPeso molecolare:340.78ZK 756326
CAS:<p>ZK 756326: Selective CCR8 agonist, IC50 1.8 μM (human), 2.6 μM (mouse), no CCR4/5, CXCR3/4 action, 28-fold selectivity vs 26 GPCRs, anti-HIV fusion.</p>Formula:C21H28N2O3Purezza:99.43%Colore e forma:SolidPeso molecolare:356.46AZD2098
CAS:AZD2098 is a potent CC-chemokine receptor 4 (CCR4) inhibitor used for asthma research.Formula:C11H9Cl2N3O3SPurezza:99.80% - >99.99%Colore e forma:SolidPeso molecolare:334.18AC-55541
CAS:<p>AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.</p>Formula:C25H20BrN5O3Purezza:98% - 99.33%Colore e forma:SolidPeso molecolare:518.36Dolasetron
CAS:<p>Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.</p>Formula:C19H20N2O3Purezza:99.84% - 99.86%Colore e forma:White PowderPeso molecolare:324.37Litorin acetate(55749-97-8 Free base)
<p>Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.</p>Formula:C53H72N14O13SPurezza:98.61%Colore e forma:SolidPeso molecolare:1145.29Nifenalol
CAS:<p>Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.</p>Formula:C11H16N2O3Purezza:98%Colore e forma:SolidPeso molecolare:224.26Tetradecyl Phosphonate
CAS:<p>Tetradecyl Phosphonate 是溶血磷脂酸 1 (LPA1)、LPA2 和 LPA3 受体的泛拮抗剂。</p>Formula:C14H31O3PPurezza:99.95%Colore e forma:White To Off-White PowderPeso molecolare:278.37Sevoflurane
CAS:<p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>Formula:C4H3F7OPurezza:98%Colore e forma:Less Oil Colorless OilPeso molecolare:200.05ML-SI3
CAS:<p>CCG-143140 is a GLP-1 receptor inverse agonists.</p>Formula:C23H31N3O3SPurezza:99.75%Colore e forma:SolidPeso molecolare:429.58ACH-000143
CAS:<p>ACH-000143 是一种可口服的褪黑素受体激动剂，对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。</p>Formula:C13H16ClN3O3Purezza:98.15%Colore e forma:SolidPeso molecolare:297.74CB1-IN-1
CAS:<p>CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.</p>Formula:C33H31Cl2F3N6O3S2Purezza:99.08% - 99.76%Colore e forma:SolidPeso molecolare:751.67Linzagolix
CAS:<p>Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei</p>Formula:C22H15F3N2O7SPurezza:99.33%Colore e forma:SolidPeso molecolare:508.42Org 27569
CAS:<p>Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity and</p>Formula:C24H28ClN3OPurezza:>99.99% - ≥95%Colore e forma:SolidPeso molecolare:409.95ARN272
CAS:<p>ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).</p>Formula:C27H20N4O2Purezza:98.23%Colore e forma:SolidPeso molecolare:432.47BMS-813160
CAS:<p>BMS-813160 is the first dual CCR2/CCR5 antagonist to enter Clinical development for cardiovascular.</p>Formula:C25H40N8O2Purezza:99.66% - 99.79%Colore e forma:SolidPeso molecolare:484.64HAEGTFT acetate(926018-95-3 free base)
<p>HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.</p>Formula:C35H51N9O14Purezza:>99.99%Colore e forma:SolidPeso molecolare:821.84MK-0557
CAS:<p>MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).</p>Formula:C22H19FN4O3Purezza:99.88%Colore e forma:SolidPeso molecolare:406.41RS102895
CAS:<p>RS102895 is a potent CCR2 antagonist (IC50: 360 nM) and shows no effect on CCR1.</p>Formula:C21H21F3N2O2Purezza:97.64% - 99.80%Colore e forma:SolidPeso molecolare:390.4BD-1047 dihydrobromide
CAS:<p>BD-1047 dihydrobromide (BD1047.2HBr) , a selective functional antagonist of sigma receptors, has antipsychotic activity in animal models predictive of efficacy</p>Formula:C13H22Br2Cl2N2Purezza:98.13% - 99.39%Colore e forma:SolidPeso molecolare:437.04Vercirnon
CAS:<p>Vercirnon (Traficet-EN) is a selective and potent antagonist of CCR9 (IC50: 10 nM). It is also used in the research of inflammatory bowel diseases.</p>Formula:C22H21ClN2O4SPurezza:99.23%Colore e forma:SolidPeso molecolare:444.93Namodenoson
CAS:<p>Namodenoson (2-Cl-IB-MECA) is an adenosine A3 receptor agonist.</p>Formula:C18H18ClIN6O4Purezza:98.97%Colore e forma:SolidPeso molecolare:544.73Bepotastine
CAS:<p>Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.</p>Formula:C21H25ClN2O3Purezza:99.75%Colore e forma:SolidPeso molecolare:388.89Felypressin
CAS:<p>Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.</p>Formula:C46H65N13O11S2Purezza:99.65%Colore e forma:SolidPeso molecolare:1040.22Flibanserin hydrochloride
CAS:<p>Flibanserin HCl: oral 5-HT1A agonist & 5-HT2A antagonist, Ki values 1 nM & 49 nM, for HSDD, has antidepressant/anxiolytic properties.</p>Formula:C20H22ClF3N4OColore e forma:SolidPeso molecolare:426.87Bromodiphenhydramine hydrochloride
CAS:<p>Bromodiphenhydramine hydrochloride is a new antihistaminic in the control of cutaneous.</p>Formula:C17H21BrClNOPurezza:97.29%Colore e forma:SolidPeso molecolare:370.71Cariprazine
CAS:<p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>Formula:C21H32Cl2N4OPurezza:99.68% - 99.87%Colore e forma:SolidPeso molecolare:427.41BA 1 acetate(183241-31-8 free base)
<p>BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.</p>Formula:C59H80N14O13Purezza:95.3%Colore e forma:SolidPeso molecolare:1193.35Blarcamesine hydrochloride
CAS:Blarcamesine hydrochloride (AVex-73 hydrochloride) is a Sigma-1 Receptor agonist (IC50: 860 nM).Formula:C19H24ClNOPurezza:99.57% - 99.9%Colore e forma:SolidPeso molecolare:317.85Nelociguat
CAS:<p>Nelociguat (BAY60-4552) is an sGC stimulator, crucial in NO signal pathways.</p>Formula:C19H17FN8O2Purezza:99.19%Colore e forma:SolidPeso molecolare:408.39Velneperit
CAS:<p>Velneperit (S2367) is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.</p>Formula:C17H24F3N3O3SPurezza:99.70%Colore e forma:SolidPeso molecolare:407.45THIQ
CAS:<p>THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).</p>Formula:C33H41ClN6O2Purezza:98.93%Colore e forma:SolidPeso molecolare:589.17M871 acetate
<p>M871 acetate is a selective galanin GAL2 receptor antagonist (Ki values are 13.1 and 420 nM at GAL2 and GAL1 receptors, respectively).It blocks pronociceptive</p>Formula:C110H167N27O30Purezza:99.84%Colore e forma:SolidPeso molecolare:2347.67SB-203186 hydrochloride
CAS:<p>SB 203186 hydrochloride is a potent 5-HT4 receptor antagonist</p>Formula:C16H20N2O2·HClPurezza:99.64%Colore e forma:SolidPeso molecolare:308.81Atipamezole hydrochloride
CAS:<p>Atipamezole is a synthetic α2 adrenergic receptor antagonist.</p>Formula:C14H16N2·HClPurezza:99.74%Colore e forma:SolidPeso molecolare:248.75ARC-239
CAS:<p>ARC-239 is an agonist of α2-adrenergic receptor.</p>Formula:C24H29N3O3Colore e forma:SolidPeso molecolare:407.51AM281
CAS:<p>AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.</p>Formula:C21H19Cl2IN4O2Purezza:98.6% - >99.99%Colore e forma:White To Off-White SolidPeso molecolare:557.21Bindarit
CAS:<p>Bindarit is a selective inhibitor of monocyte chemoattractant proteins MCP-1/CCL2, MCP-3/CCL7 and MCP-2/CCL8.Cost-effective and quality-assured.</p>Formula:C19H20N2O3Purezza:98.35% - 98.55%Colore e forma:SolidPeso molecolare:324.37Eltoprazine hydrochloride
CAS:<p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>Formula:C12H17ClN2O2Purezza:99.35%Colore e forma:SolidPeso molecolare:256.73Ebastine
CAS:<p>Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.</p>Formula:C32H39NO2Purezza:99.65% - 99.93%Colore e forma:White To Off-White PowderPeso molecolare:469.66Canagliflozin
CAS:<p>Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor. Canagliflozin is used to treat type II diabetes mellitus. Cost-effective and quality-assured.</p>Formula:C24H25FO5SPurezza:98.01% - >99.99%Colore e forma:SolidPeso molecolare:444.52BPTU
CAS:<p>BPTU (BMS-646786) is an allosteric antagonist of P2Y1 (EC50 = 0.06-0.3 μM).</p>Formula:C23H22F3N3O3Purezza:99.37% - 99.89%Colore e forma:SolidPeso molecolare:445.43ICI 89406
CAS:<p>ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.</p>Formula:C19H22N4O3Purezza:99.92%Colore e forma:SolidPeso molecolare:354.4MK-571 sodium
CAS:<p>MK-571 sodium, a CysLT1 antagonist and MRP2 inhibitor, obstructs drug efflux and hampers enterocyte phase-2 conjugation of flavonoids.</p>Formula:C26H27ClN2O3S2·NaPurezza:97.86% - 99.58%Colore e forma:SolidPeso molecolare:537.07LY 78335
CAS:<p>LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.</p>Formula:C8H10Cl3NPurezza:99.30% - 99.81%Colore e forma:SolidPeso molecolare:226.53Laropiprant sodium
<p>Laropiprant sodium is a potent and selective DP receptor antagonist with Ki values of 0.57 nM for TP receptors and 2.95 nM for DP receptors.</p>Colore e forma:SolidLys-[Des-Arg9]Bradykinin,TFA
<p>Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2</p>Formula:C54H75F6N13O15Purezza:97.35%Colore e forma:SolidPeso molecolare:1260.24GLP-1(7-37) acetate(106612-94-6 free base)
CAS:<p>Glp-1(7-37) acetate is an intestinal insulin hormone that enhances glucose-induced insulin secretion.</p>Formula:C151H228N40O47Purezza:98.89%Colore e forma:SolidPeso molecolare:3355.67Ralinepag
CAS:<p>Ralinepag (APD811) is a potent, orally bioavailable agonist of non-prostanoid prostacyclin (IP) receptor, with EC50s of 8.5 nM, 530 nM and 850 nM for human and</p>Formula:C23H26ClNO5Purezza:99.79% - 99.85%Colore e forma:SolidPeso molecolare:431.91Etelcalcetide hydrochloride
CAS:<p>Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary hyperparathyroidism.</p>Formula:C38H73N21O10S2HClPurezza:>99.99%Colore e forma:SolidPeso molecolare:1353.33Dasotraline hydrochloride
CAS:<p>Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.</p>Formula:C16H16Cl3NPurezza:98.92% - 99.6%Colore e forma:SolidPeso molecolare:328.66JNJ-31020028
CAS:<p>JNJ-31020028 is a selective brain penetrant antagonist of neuropeptide Y2 receptor with high affinity (pIC50=8.07, human; pIC50=8.22, rat).</p>Formula:C34H36FN5O2Purezza:95.92% - 99.65%Colore e forma:SolidPeso molecolare:565.68Nuciferine
CAS:<p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>Formula:C19H21NO2Purezza:98.76% - 99.79%Colore e forma:SolidPeso molecolare:295.38Senktide
CAS:<p>Senktide is an agonist of tachykinin NK3 receptor.</p>Formula:C40H55N7O11SPurezza:99.84% - >99.99%Colore e forma:White PowderPeso molecolare:841.97Levalbuterol tartrate
CAS:<p>Levalbuterol tartrate is a short-acting β2-adrenergic receptor agonist and the R enantiomer of salbutamol.Cost-effective and quality-assured.</p>Formula:C17H27NO9Purezza:98.97% - 99.79%Colore e forma:SolidPeso molecolare:389.39Sarpogrelate hydrochloride
CAS:<p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>Formula:C24H32ClNO6Purezza:99.73%Colore e forma:Colorless LiquidPeso molecolare:465.979-FLUORENOL
CAS:<p>9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.</p>Formula:C13H10OPurezza:99.98%Colore e forma:Off-White Crystalline PowderPeso molecolare:182.223-AQC
CAS:<p>3-AQC is a competitive antagonist of 5-HT3.</p>Formula:C20H21N5O4Purezza:99.45%Colore e forma:SolidPeso molecolare:395.41Dioxopromethazine
CAS:<p>Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.</p>Formula:C17H20N2O2SPurezza:98%Colore e forma:SolidPeso molecolare:316.42Montelukast dicyclohexylamine
CAS:<p>Montelukast (MK0476), a selective CysLT1 antagonist, treats asthma, liver injury, and is researched for COVID-19.</p>Formula:C47H59ClN2O3SColore e forma:SolidPeso molecolare:767.5ENMD-1068 HBr
CAS:<p>ENMD-1068 HBr is a novel Proteinase-Activated Receptor 2 antagonist.</p>Formula:C15H30BrN3O2Colore e forma:SolidPeso molecolare:364.32T-1095
CAS:<p>T-1095 is an inhibitor of renal glucose reabsorption and the expression of Na+-glucose cotransporters (SGLTs) and facilitative glucose transporter 2 (GLUT2).</p>Formula:C26H28O11Purezza:99.78%Colore e forma:SolidPeso molecolare:516.49BAR 501 impurity
CAS:<p>BAR 501 impurity 在 BAR501 制剂中发现的一种杂质，可作为 G 蛋白偶联胆汁酸激活受体 (GP-BAR1) 的激动剂。 BAR501 杂质 (10 µM) 在 GP-BAR1 报告基因检测中诱导荧光素酶活性增加 150%。</p>Formula:C26H46O3Purezza:98.78%Colore e forma:SolidPeso molecolare:406.64PF-06291874
CAS:<p>PF-06291874 (Glucagon receptor antagonists-4) (Glucagon receptor antagonists-4) is a highly effective and orally active antagonist of the glucagon receptor.</p>Formula:C26H28F3N3O4Purezza:99.12% - 99.27%Colore e forma:SolidPeso molecolare:503.51Haloperidol decanoate
CAS:<p>Haloperidol decanoate (KD 16), an antipsychotic, treats schizophrenia and mood disorders as an intramuscular ester.</p>Formula:C31H41ClFNO3Purezza:99.57% - 99.72%Colore e forma:SolidPeso molecolare:530.11D3-βArr
CAS:<p>D3-βArr (NCGC00379308) is a positive allosteric modulator for thyrotropin receptor (TSHR), which initiates translocation of β-Arr 1 (EC50: 11.6 μM) by direct</p>Formula:C20H23N5Purezza:98.82%Colore e forma:SolidPeso molecolare:333.43Talastine HCl
CAS:<p>Talastine is an antihistamine drug.</p>Formula:C19H22ClN3OPurezza:98%Colore e forma:SolidPeso molecolare:343.865'-N-Ethylcarboxamidoadenosine
CAS:<p>NECA, an adenosine receptor agonist, boosts brain extravasation of fluorescein and dextran without affecting the blood-brain barrier.</p>Formula:C12H16N6O4Purezza:98.95% - ≥95%Colore e forma:PowderPeso molecolare:308.29Serotonin hydrochloride
CAS:<p>Serotonin hydrochloride (Serotonin HCl) is an endogenous 5-HT receptor agonist, a monoamine neurotransmitter in the CNS, and a catechol O-methyltransferase (</p>Formula:C10H13ClN2OPurezza:98.05% - 99.93%Colore e forma:White To Cream PowderPeso molecolare:212.676Hemokinin 1 (human) acetate(491851-53-7 free base)
<p>Hemokinin 1 acetate: Human SP homolog, NK1 agonist (IC50: NK1 1.8 nM), proliferates B-cells, antihypertensive.</p>Formula:C56H88N14O16SPurezza:97.82%Colore e forma:SolidPeso molecolare:1245.45Veralipride
CAS:<p>Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.</p>Formula:C17H25N3O5SPurezza:99.65%Colore e forma:SolidPeso molecolare:383.46ML-097
CAS:ML-097 (CID-2160985) is a pan activator of Ras-related GTPasesFormula:C14H11BrO3Purezza:99.12%Colore e forma:SolidPeso molecolare:307.139Lys-[Des-Arg9]Bradykinin acetate
<p>Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and</p>Formula:C52H77N13O13Purezza:99.93%Colore e forma:SolidPeso molecolare:1092.27Droxidopa hydrochloride
CAS:<p>Droxidopa (L-DOPS) HCI is an oral norepinephrine precursor for nOH and ADHD research, raising standing BP and easing orthostatic hypotension.</p>Formula:C9H12ClNO5Colore e forma:SolidPeso molecolare:249.65Pranlukast hemihydrate
CAS:<p>Pranlukast hemihydrate (ONO-1078 hemihydrate) is an LT antagonist with anti-asthmatic activity.</p>Formula:C27H23N5O40·5H2OPurezza:99.28%Colore e forma:SolidPeso molecolare:490.52AR-M 1896 Acetate
<p>AR-M 1896 Acetate is the selective agonist of GalR2.</p>Formula:C56H85N13O16Purezza:99.76%Colore e forma:SolidPeso molecolare:1196.35Amperozide
CAS:<p>Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.</p>Formula:C23H29F2N3OPurezza:99.68%Colore e forma:SolidPeso molecolare:401.49AM966
CAS:<p>AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.</p>Formula:C27H23ClN2O5Purezza:98.06% - 99.79%Colore e forma:SolidPeso molecolare:490.93Phentolamine hydrochloride
CAS:<p>Phentolamine hydrochloride is a blocking agent of adrenergic α receptor that is orally active [1].</p>Formula:C17H20ClN3OColore e forma:SolidPeso molecolare:317.82Sitaxsentan sodium
CAS:<p>Sitaxsentan sodium (TBC11251 sodium salt) is a highly selective antagonist of endothelin A receptors.</p>Formula:C18H14ClN2O6S2·NaPurezza:98.39% - 99.01%Colore e forma:SolidPeso molecolare:476.89GLP-1(7-36), amide
CAS:<p>GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.</p>Formula:C149H226N40O45Purezza:99.85%Colore e forma:White PowderPeso molecolare:3297.63Pergolide
CAS:<p>Pergolide is a long-acting and orally active dopamine receptor D1/D2 agonist and ergoline derivative, used in the study of Parkinson's disease</p>Formula:C19H26N2SPurezza:99.95%Colore e forma:SolidPeso molecolare:314.49Fuscoside
CAS:<p>Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.</p>Formula:C26H31N3O4Purezza:98.13% - 99.66%Colore e forma:SolidPeso molecolare:449.54Irdabisant hydrochloride
CAS:<p>Irdabisant (CEP-26401) is a selective H3R inverse agonist, BBB-penetrable, with cognition-enhancing effects.</p>Formula:C18H24ClN3O2Colore e forma:SolidPeso molecolare:349.86Hemokinin 1 (mouse) acetate(208041-90-1 free base)
<p>Mouse Hemokinin-1 acetate: NK1 receptor agonist, Ki=0.175 nM; NK2 Ki=560 nM.</p>Formula:C63H104N22O17SPurezza:98.33%Colore e forma:SolidPeso molecolare:1473.72PD 168568
CAS:<p>PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.</p>Formula:C22H27N3OColore e forma:SolidPeso molecolare:349.47Phosphorylcholine chloride
CAS:<p>Phosphorylcholine chloride, an antigenic component found on the surface of numerous commensal and pathogenic bacteria inhabiting the upper airway, is integral</p>Formula:C5H15ClNO4PPurezza:99.481% - 99.85%Colore e forma:SolidPeso molecolare:219.6Ziprasidone mesylate
CAS:<p>Ziprasidone mesylate (CP-88059), an oral 5-HT & dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>Formula:C22H25ClN4O4S2Colore e forma:SolidPeso molecolare:509.04d[Cha4]-AVP acetate(500170-27-4 free base)
<p>'d[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'</p>Formula:C52H75N13O13S2Purezza:99.86%Colore e forma:SolidPeso molecolare:1154.37NIBR-0213
CAS:<p>NIBR-0213 is a potent and selective competitive S1P1 antagonist.Cost-effective and quality-assured.</p>Formula:C27H29ClN2O3Purezza:98.36% - 99.34%Colore e forma:SolidPeso molecolare:464.98Rolapitant hydrochloride hydrate
CAS:<p>Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.</p>Formula:C25H29ClF6N2O3Colore e forma:SolidPeso molecolare:554.95Cannabigerol
CAS:<p>Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also</p>Formula:C21H32O2Purezza:99.59% - 99.92%Colore e forma:SolidPeso molecolare:316.48Elinzanetant
CAS:<p>Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.</p>Formula:C33H35F7N4O3Purezza:98% - 99.13%Colore e forma:SolidPeso molecolare:668.64Pancreatic Polypeptide, rat acetate
<p>Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4.</p>Purezza:97.53%Colore e forma:SolidPeso molecolare:N/AOXA (17-33) acetate
<p>OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).</p>Formula:C79H125N23O22Purezza:98.52%Colore e forma:SolidPeso molecolare:1748.98
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