Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(939 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.945 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(148 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(407 prodotti)
- Recettore dell'endotelina(76 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(31 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(165 prodotti)
- Proteina Hedgehog/Smoothened(44 prodotti)
- Recettore dell'istamina(358 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(297 prodotti)
- PAFR(11 prodotti)
- PKA(48 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5352 prodotti di "Proteina G/GPCR"
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Ralmitaront
CAS:<p>Ralmitaront (RO6889450) is a potent, orally active partial agonist of the trace amine-associated receptor 1 (TAAR1).</p>Formula:C17H22N4O2Purezza:99.71% - 99.79%Colore e forma:SolidPeso molecolare:314.38Chlorpheniramine
CAS:<p>Chlorpheniramine is an H1 anti-histamine agent for IgE-mediated inflammation that is commonly used for allergic diseases.</p>Formula:C16H19ClN2Colore e forma:SolidPeso molecolare:274.79MRT-10
CAS:<p>MRT-10 is a Smoothened (Smo) receptor antagonist.</p>Formula:C24H23N3O5SPurezza:99.73%Colore e forma:SolidPeso molecolare:465.52Icatibant Acetate
CAS:<p>Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.</p>Formula:C61H93N19O15SPurezza:99.68%Colore e forma:SolidPeso molecolare:1364.57MK-2894 sodium salt
CAS:<p>MK-2894 sodium salt is a highly potent and selective antagonist of second generation EP4.</p>Formula:C25H22F3NNaO3SPurezza:98%Colore e forma:SolidPeso molecolare:496.5Terazosin
CAS:<p>Terazosin: oral α1-blocker, relaxes blood vessels, treats BPH and hypertension.</p>Formula:C19H25N5O4Colore e forma:SolidPeso molecolare:387.43Melanotan I
CAS:<p>Melanotan I is a non-specific melanocortin receptor (MCR) agonist, an α-melanocyte-stimulating hormone (α-MSH) analog, which is injected subcutaneously to</p>Formula:C78H111N21O19Purezza:>99.99%Colore e forma:SolidPeso molecolare:1646.85Nomifensine maleate
CAS:<p>Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.</p>Formula:C20H22N2O4Purezza:98.46%Colore e forma:SolidPeso molecolare:354.4Siponimod hemifumarate
CAS:<p>Siponimod (BAF-312) is a potent S1P receptor modulator for multiple sclerosis research.</p>Formula:C62H74F6N4O10Colore e forma:SolidPeso molecolare:1149.282Hemokinin 1 (mouse) acetate(208041-90-1 free base)
<p>Mouse Hemokinin-1 acetate: NK1 receptor agonist, Ki=0.175 nM; NK2 Ki=560 nM.</p>Formula:C63H104N22O17SPurezza:98.33%Colore e forma:SolidPeso molecolare:1473.72Bupranolol
CAS:<p>Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.</p>Formula:C14H22ClNO2Purezza:97.63%Colore e forma:SolidPeso molecolare:271.78Felypressin
CAS:<p>Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.</p>Formula:C46H65N13O11S2Purezza:99.65%Colore e forma:SolidPeso molecolare:1040.22NIBR-0213
CAS:<p>NIBR-0213 is a potent and selective competitive S1P1 antagonist.Cost-effective and quality-assured.</p>Formula:C27H29ClN2O3Purezza:98.36% - 99.34%Colore e forma:SolidPeso molecolare:464.98d[Cha4]-AVP acetate(500170-27-4 free base)
<p>'d[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'</p>Formula:C52H75N13O13S2Purezza:99.86%Colore e forma:SolidPeso molecolare:1154.37Dobutamine tartrate
CAS:<p>Dobutamine tartrate is a cardiotonic.</p>Formula:C22H29NO9Colore e forma:SolidPeso molecolare:451.472Emedastine
CAS:<p>Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.</p>Formula:C17H26N4OPurezza:97.1% - 97.76%Colore e forma:OilPeso molecolare:302.41Ozanimod
CAS:<p>Ozanimod (RPC-1063) (RPC1063) is a specific oral S1P Receptor 1 modulator.</p>Formula:C23H24N4O3Purezza:98.68% - 99.58%Colore e forma:SolidPeso molecolare:404.46Lys-[Des-Arg9]Bradykinin,TFA
<p>Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2</p>Formula:C54H75F6N13O15Purezza:97.35%Colore e forma:SolidPeso molecolare:1260.24MDL 100009
CAS:<p>MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.</p>Formula:C22H28FNO3Purezza:98.96%Colore e forma:SolidPeso molecolare:373.46GRK5-IN-2
CAS:<p>GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor.</p>Formula:C20H20N4O4Purezza:99.92%Colore e forma:SolidPeso molecolare:380.4IPSU
CAS:<p>IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus OX1 receptors.</p>Formula:C23H27N5O2Purezza:97.05%Colore e forma:SolidPeso molecolare:405.49Spiperone hydrochloride
CAS:<p>5-HT2A serotonin and selective D2-like dopamine receptor antagonist</p>Formula:C23H27ClFN3O2Purezza:98%Colore e forma:SolidPeso molecolare:431.93Midaglizole
CAS:<p>Midaglizole, an α2-adrenoceptor blocker, raises blood pressure and lowers glucose.</p>Formula:C16H17N3Colore e forma:SolidPeso molecolare:251.33Liraglutide
CAS:<p>Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.</p>Formula:C172H265N43O51Purezza:97.65% - 99.04%Colore e forma:SolidPeso molecolare:3751.25MK-3697
CAS:<p>MK-3697, an isonicotinamide small molecule, acts as a potent and selective Orexin 2 receptor antagonist (Ki: 0.95 nM).</p>Formula:C23H21N5O3SPurezza:97.69% - 98.15%Colore e forma:SolidPeso molecolare:447.51Otenabant hydrochloride
CAS:<p>Otenabant hydrochloride (Otenabant) (CP-945598) is a competitive, high affinity, selective antagonist of the CB1 receptor (Ki: 0.7 nM).</p>Formula:C25H26Cl3N7OPurezza:99.79% - ≥95%Colore e forma:SolidPeso molecolare:546.88Conivaptan hydrochloride
CAS:<p>Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and</p>Formula:C32H26N4O2·HClPurezza:98.33% - 99.86%Colore e forma:SolidPeso molecolare:535.04Opaganib
CAS:<p>Opaganib (ABC294640) is an orally active and specific sphingosine kinase-2 (SphK2) inhibitor (IC50: 60 μM).</p>Formula:C23H25ClN2OPurezza:98.86% - 99.85%Colore e forma:SolidPeso molecolare:380.91Pipamperone HCl
CAS:<p>Pipamperone blocks 5-HT2A/B/C, D2/D3/D4, α1/α2 receptors; favors 5-HT2A/D4 over D2; negligible affinity for H1, mACh. Highly selective at low doses.</p>Formula:C21H31ClFN3O2Colore e forma:SolidPeso molecolare:411.95K 41498 aceate
<p>K41498 acetate, a potent CRF2 antagonist (Ki: 0.66/0.62 nM for CRF2α/β) with 425 nM for CRF1; blocks aSvg-30 effect on cAMP in cells.</p>Purezza:96.4%Colore e forma:LiquidPeso molecolare:N/ASarpogrelate hydrochloride
CAS:<p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>Formula:C24H32ClNO6Purezza:99.73%Colore e forma:Colorless LiquidPeso molecolare:465.97Betaxolol
CAS:<p>Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.</p>Formula:C18H29NO3Purezza:99.01%Colore e forma:White Crystalline SolidPeso molecolare:307.43Human growth hormone-releasing factor acetate
<p>Human growth hormone-releasing factor acetate is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) on</p>Purezza:99.26%Colore e forma:LiquidPeso molecolare:N/AGuanabenz hydrochloride
CAS:<p>Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.</p>Formula:C8H9Cl3N4Purezza:99.45%Colore e forma:SolidPeso molecolare:267.54ACH-000143
CAS:<p>ACH-000143 是一种可口服的褪黑素受体激动剂，对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。</p>Formula:C13H16ClN3O3Purezza:98.15%Colore e forma:SolidPeso molecolare:297.74Senktide
CAS:<p>Senktide is an agonist of tachykinin NK3 receptor.</p>Formula:C40H55N7O11SPurezza:99.84% - >99.99%Colore e forma:White PowderPeso molecolare:841.97Linzagolix
CAS:<p>Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by Kissei</p>Formula:C22H15F3N2O7SPurezza:99.33%Colore e forma:SolidPeso molecolare:508.42HAEGTFT acetate(926018-95-3 free base)
<p>HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.</p>Formula:C35H51N9O14Purezza:>99.99%Colore e forma:SolidPeso molecolare:821.84Nelotanserin
CAS:<p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>Formula:C18H15BrF2N4O2Purezza:98.42% - 99.88%Colore e forma:SolidPeso molecolare:437.24T-1095
CAS:<p>T-1095 is an inhibitor of renal glucose reabsorption and the expression of Na+-glucose cotransporters (SGLTs) and facilitative glucose transporter 2 (GLUT2).</p>Formula:C26H28O11Purezza:99.78%Colore e forma:SolidPeso molecolare:516.49CS 2100
CAS:<p>CS 2100 (1-[[4-Ethyl-5-[5-(4-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]-2-thienyl]methyl]-3-azetidinecarboxylic acid) is an S1P1 agonist.</p>Formula:C25H23N3O4SPurezza:99.19%Colore e forma:SolidPeso molecolare:461.53BA 1 acetate(183241-31-8 free base)
<p>BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.</p>Formula:C59H80N14O13Purezza:95.3%Colore e forma:SolidPeso molecolare:1193.35PRX-07034 hydrochloride
CAS:<p>PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.</p>Formula:C21H29Cl2N3O4SPurezza:98.5%Colore e forma:SolidPeso molecolare:490.44Dasotraline hydrochloride
CAS:<p>Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.</p>Formula:C16H16Cl3NPurezza:98.92% - 99.6%Colore e forma:SolidPeso molecolare:328.66ACTH 1-14 acetate(25696-21-3 free base)
<p>ACTH 1-14 acetate regulates cortisol and androgen, is part of the hypothalamic-pituitary-adrenal stress response.</p>Formula:C79H113N21O22SPurezza:>99.99%Colore e forma:SolidPeso molecolare:1740.96Nuciferine
CAS:<p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>Formula:C19H21NO2Purezza:98.76% - 99.79%Colore e forma:SolidPeso molecolare:295.38Conopressin S acetate(111317-90-9 free base)
<p>Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b</p>Formula:C43H77N17O12S2Purezza:99.79%Colore e forma:SolidPeso molecolare:1088.32Lys-Bradykinin acetate(342-10-9 free base)
CAS:<p>Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.</p>Formula:C58H89N17O14Purezza:99.86%Colore e forma:SolidPeso molecolare:1248.43Ambrisentan sodium
CAS:<p>Ambrosentan (BSF 208075) sodium is a selective and oral effective antagonist of ET type A receptor ( ETAR ).</p>Formula:C22H21N2NaO4Colore e forma:SolidPeso molecolare:400.41Secretin (33-59), rat
CAS:<p>Secretin (33-59), rat (Secretin (rat)) is a classical hormone in the gastrointestinal system and a neuropeptide.</p>Formula:C129H216N42O42Purezza:98.12%Colore e forma:SolidPeso molecolare:3027.35Methyldopa hydrate
CAS:<p>Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.</p>Formula:C10H13NO4H2OPurezza:99.67%Colore e forma:White SolidPeso molecolare:238.24BMS-986278
CAS:<p>BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb values of 6.9 nM and 4.0 nM for human and mouse LPA1,</p>Formula:C22H31N5O5Purezza:99.86%Colore e forma:SolidPeso molecolare:445.51Ketanserin tartrate
CAS:<p>Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.</p>Formula:C26H28FN3O9Purezza:99.68%Colore e forma:SolidPeso molecolare:545.51Pentoxyverine
CAS:<p>Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.</p>Formula:C20H31NO3Purezza:97.11%Colore e forma:SolidPeso molecolare:333.47WAY-100635 maleate
CAS:<p>WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).</p>Formula:C25H34N4O2·xC4H4O4Purezza:>99.99%Colore e forma:White SolidPeso molecolare:538.645KB-5492 free base
CAS:<p>KB-5492 free base is an antiulcer agent that inhibits sigma receptors and can be used to study gastric lesions and gastric secretion.</p>Formula:C23H30N2O6Purezza:97.10% - 97.94%Colore e forma:SolidPeso molecolare:430.49L-368,899 hydrochloride
CAS:<p>L-368,899 hydrochloride is an OXTR antagonist that prevents oxytocin-induced antiabnormal pain and anti-nausea, and may be used in the study of depression.</p>Formula:C26H43ClN4O5S2Purezza:99.59%Colore e forma:SolidPeso molecolare:591.23Bucindolol
CAS:<p>Bucindolol (BMY 13105) is a novel and potent β1-adrenergic receptor blocker that mediates vasodilation and can be used to study chronic heart failure.</p>Formula:C22H25N3O2Purezza:99.9%Colore e forma:SolidPeso molecolare:363.45Levocetirizine Dihydrochloride
CAS:<p>Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.</p>Formula:C21H27Cl3N2O3Purezza:99.89%Colore e forma:White Or Off-White Crystalline PowderPeso molecolare:461.81Tandospirone
CAS:<p>Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.</p>Formula:C21H29N5O2Purezza:99.94%Colore e forma:SolidPeso molecolare:383.49Alfuzosin
CAS:<p>Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and urethral dysfunction.</p>Formula:C19H27N5O4Purezza:99.64%Colore e forma:White Crystaline PowderPeso molecolare:389.45Jatrorrhizine chloride
CAS:<p>Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.</p>Formula:C20H20ClNO4Purezza:99.79%Colore e forma:SolidPeso molecolare:373.8ACT-462206
CAS:<p>ACT-462206 is a Orexin 1/Orexin 2 receptor antagonist.ACT-462206 is highly potent and can be used to study sleep and anxiety.</p>Formula:C20H24N2O4SPurezza:99.45%Colore e forma:SolidPeso molecolare:388.48Opipramol
CAS:<p>Opipramol (Ensidon) is a compound with antidepressant activity, a sigma (σ) receptor agonist, and anxiolytic activity.</p>Formula:C23H29N3OPurezza:99.84% - 99.98%Colore e forma:SolidPeso molecolare:363.5Fenoterol hydrobromide
CAS:<p>Fenoterol hydrobromide is a beta2-adrenergic receptor agonist and bronchodilator used in the study of cardiovascular diseases such as asthma and bronchitis.</p>Formula:C17H22BrNO4Purezza:99.88%Colore e forma:SolidPeso molecolare:384.27Latrepirdine dihydrochloride
CAS:<p>Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.</p>Formula:C21H25N3·2HClPurezza:98.45%Colore e forma:SolidPeso molecolare:392.37UCM 608
CAS:<p>UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces an increase in GDP-GTP exchange.</p>Formula:C19H20N2O2Purezza:98.88%Colore e forma:SolidPeso molecolare:308.37Fenoprofen
CAS:<p>Fenoprofen (LILLY-5385) is a non-steroidal anti-inflammatory compound and a modifier enhancer of the melanocortin receptor, increasing ERK1/2 activation.</p>Formula:C15H14O3Purezza:98.4%Colore e forma:SolidPeso molecolare:242.27Rizatriptan
CAS:<p>Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.</p>Formula:C15H19N5Purezza:99.74%Colore e forma:SolidPeso molecolare:269.35GRK6-IN-2
CAS:<p>GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 has been studied in multiple myeloma.</p>Formula:C21H21FN6Purezza:98.94%Colore e forma:SolidPeso molecolare:376.43(S)-Mirtazapine
CAS:<p>(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.</p>Formula:C17H19N3Purezza:99.37%Colore e forma:SolidPeso molecolare:265.35AF-710B
CAS:<p>AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.</p>Formula:C20H27N3OSPurezza:98.62% - 99.89%Colore e forma:SolidPeso molecolare:357.51S1RA
CAS:<p>S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2</p>Formula:C20H23N3O2Purezza:99.45%Colore e forma:SolidPeso molecolare:337.42Renzapride
CAS:<p>Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.</p>Formula:C16H22ClN3O2Purezza:98.97% - 99.09%Colore e forma:SolidPeso molecolare:323.82A2ti-1
CAS:<p>A2ti-1 is an annexin A2/S100A10 heterotetramer (A2t) inhibitor that inhibits Src activation and can be used to study human papillomavirus type 16 infection.</p>Formula:C20H22N4O2SPurezza:99.86%Colore e forma:SolidPeso molecolare:382.48INCB 3284
CAS:INCB 3284, a potent human CCR2 antagonist with an IC50 of 3.7 nM, is researchable for acute liver failure and inhibits MCP-1/hCCR2 binding.Formula:C26H31F3N4O4Purezza:97.81% - 99.42%Colore e forma:SolidPeso molecolare:520.54Nebentan potassium
CAS:<p>Nebentan potassium (YM598) is an ETA receptor antagonist that inhibits pulmonary arterial hypertension and is used in the study of neurologic diseases.</p>Formula:C24H20KN5O5SPurezza:99.05%Colore e forma:SolidPeso molecolare:529.61GAT211
CAS:<p>GAT211 (AZ-4) is a cannabinoid 1 receptor (CB1R) positive allosteric modulator (PAM) for the study of epilepsy.</p>Formula:C22H18N2O2Purezza:99.7%Colore e forma:SolidPeso molecolare:342.39Atipamezole
CAS:<p>Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.</p>Formula:C14H16N2Purezza:99.88%Colore e forma:Off-White To Light Yellow Crystal PowderPeso molecolare:212.29Canagliflozin hemihydrate
CAS:<p>Canagliflozin hemihydrate (TA 7284) treats type 2 diabetes by blocking SGLT2, leading to glucose excretion in urine.</p>Formula:C48H52F2O11S2Purezza:99.42% - 99.96%Colore e forma:SolidPeso molecolare:907.05Medetomidine
CAS:<p>Medetomidine (MPV785 free base) is a selective α2-adrenoceptor agonist, with sedative and analgesic and vasoconstrictive hypoxic , in small animal anesthesia.</p>Formula:C13H16N2Purezza:99.88%Colore e forma:SolidPeso molecolare:200.28Protein deglycase DJ-1 against-1
CAS:<p>Protein deglycase DJ-1 against-1 penetrate the BBB and bind to DJ-1 protein,restoring neuronal cellular death in a neurotoxin MPTP-induced model of PD.</p>Formula:C24H23N3O4Purezza:97.23%Colore e forma:SolidPeso molecolare:417.46(R)-Mirtazapine
CAS:<p>(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.</p>Formula:C17H19N3Purezza:99.75%Colore e forma:SolidPeso molecolare:265.35SID 7969543
CAS:<p>SID 7969543 is a selective SF-1 inhibitor with potential anticancer activity, inhibits SF-1-triggered luciferase expression and can be used for cancer research.</p>Formula:C24H24N2O7Purezza:98.94%Colore e forma:SolidPeso molecolare:452.46Citalopram
CAS:<p>Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.</p>Formula:C20H21FN2OPurezza:99.78% - 99.89%Colore e forma:SolidPeso molecolare:324.39WIN 51,708
CAS:<p>WIN 51,708 is an antagonist of neurokinin-1 receptor.</p>Formula:C29H33N3OPurezza:99%Colore e forma:SolidPeso molecolare:439.59LP-533401 hydrochloride
CAS:<p>LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.</p>Formula:C27H23ClF4N4O3Purezza:98%Colore e forma:SolidPeso molecolare:562.94CGP 20712 A
CAS:<p>CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that reverses RKT-induced gastric relaxation.</p>Formula:C24H29F3N4O8SPurezza:99.37%Colore e forma:SolidPeso molecolare:590.57Poly-D-lysine hydrobromide (MW 30000-70000)
CAS:<p>Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant PrP from SN56 neuroblastoma cells.</p>Formula:(C6H14N2O2)x·xHBrColore e forma:SolidPeso molecolare:227.102SB 243213
CAS:<p>SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.</p>Formula:C22H19F3N4O2Purezza:98.78% - 99.86%Colore e forma:SolidPeso molecolare:428.41Dexpramipexole
CAS:<p>Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.</p>Formula:C10H17N3SPurezza:99.78%Colore e forma:SolidPeso molecolare:211.33Clopidogrel thiolactone
CAS:<p>Clopidogrel thiolactone (2-oxoclopidogrel), a P2Y12 receptor inhibitor, is an antiplatelet aggregation compound.</p>Formula:C16H16ClNO3SPurezza:98.79%Colore e forma:SolidPeso molecolare:337.82Atogepant
CAS:<p>Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist for the study of migraine.</p>Formula:C29H23F6N5O3Purezza:99.66%Colore e forma:SolidPeso molecolare:603.52Trabodenoson
CAS:<p>Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.</p>Formula:C15H20N6O6Purezza:99.94%Colore e forma:SolidPeso molecolare:380.36CP-105696
CAS:<p>CP-105696 is a potent and selective leukotriene B4 (LTB4) receptor antagonist for the study of allograft rejection.</p>Formula:C28H28O4Purezza:99.78%Colore e forma:SolidPeso molecolare:428.52Trazpiroben
CAS:<p>Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.</p>Formula:C31H39N3O4Purezza:99.41% - >99.99%Colore e forma:SolidPeso molecolare:517.66Rotigotine
CAS:<p>Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.</p>Formula:C19H25NOSPurezza:99.04% - 99.88%Colore e forma:SolidPeso molecolare:315.47CB1/2 agonist 3
CAS:<p>CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.</p>Formula:C25H41NO2Purezza:98.78%Colore e forma:SolidPeso molecolare:387.6Ozanimod hydrochloride
CAS:<p>Ozanimod (RPC-1063) HCl is a selective S1P1/S1P5 modulator with high affinity, used in relapsing MS research.</p>Formula:C23H25ClN4O3Purezza:99.81%Colore e forma:SolidPeso molecolare:440.92S-Methoprene
CAS:<p>S-Methoprene (ZR2458), a juvenile hormone analog, acts as an insecticide influencing redox activity and male sex differentiation.</p>Formula:C19H34O3Purezza:97.05% - 98.55%Colore e forma:SolidPeso molecolare:310.47
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