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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5378 prodotti di "Proteina G/GPCR"

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  • JNJ-26070109

    CAS:
    <p>JNJ-26070109, an antagonist of cholecystokinin CCK2 receptor, inhibits gastric acid secretion and prevents omeprazole-induced acid rebound in the rat.</p>
    Formula:C23H17BrF2N4O3S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:547.37
  • Ro 19-1400

    CAS:
    <p>Ro 19-1400, a platelet-activating factor antagonist, directly inhibits immunoglobulin E-dependent mediator release.</p>
    Formula:C31H56N2O8S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:616.85
  • (Rac)-E1R

    CAS:
    <p>(Rac)-E1R is the racemate of E1R. (Rac)-E1R is a sigma-1 receptor positive allosteric (Sig1R PAM) modulator of for the treatment of cognition/memory disorders.</p>
    Formula:C13H16N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:232.28
  • GSK 189254 HCl

    CAS:
    <p>GSK 189254A: histamine H3 antagonist, treats narcolepsy, may improve cognition and help with dementia, neuropathic pain.</p>
    Formula:C21H26ClN3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:387.9
  • Resomelagon

    CAS:
    <p>Resomelagon (AP1189), an oral melanocortin receptor agonist, triggers Ca2+ and ERK1/2 activation; useful in obesity and inflammation studies.</p>
    Formula:C14H14N6O2
    Colore e forma:Solid
    Peso molecolare:298.3
  • ONO-2952

    CAS:
    <p>ONO-2952, a selective TSPO antagonist with Ki: 0.33-9.30 nM, may treat irritable bowel syndrome, reducing stress without causing amnesia.</p>
    Formula:C22H20ClFN2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:398.86
  • S-3608

    CAS:
    <p>S-3608 is an atypical dopamine agonist.</p>
    Formula:C16H20ClN3OS
    Colore e forma:Solid
    Peso molecolare:337.87
  • Panamesine

    CAS:
    <p>Panamesine (EMD 57445) is a high affinity receptor ligand for sigma (IC50: 6 nM) with potential for atypical antipsychotic studies.</p>
    Formula:C23H26N2O6
    Colore e forma:Solid
    Peso molecolare:426.46
  • (-)-S-Timolol

    CAS:
    <p>(-)-S-Timolol is an antagonist of the beta-Adrenergic .</p>
    Formula:C13H26N4O4S
    Colore e forma:Solid
    Peso molecolare:334.44
  • Inupadenant

    CAS:
    <p>Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].</p>
    Formula:C25H26F2N8O4S2
    Colore e forma:Solid
    Peso molecolare:604.65
  • A3AR antagonist 1

    CAS:
    <p>A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.</p>
    Formula:C32H24N4O4S
    Colore e forma:Solid
    Peso molecolare:560.62
  • FR260010

    CAS:
    <p>FR260010 is a novel potent serotonin 5-HT2C receptor antagonist.</p>
    Formula:C22H19N5
    Colore e forma:Solid
    Peso molecolare:353.42
  • Trimazosin

    CAS:
    <p>Trimazosin, a quinazoline derivative and prazosin relative, lowers blood pressure by blocking alpha1-adrenoceptors.</p>
    Formula:C20H29N5O6
    Colore e forma:Solid
    Peso molecolare:435.47
  • SMO-IN-3

    CAS:
    <p>SMO-IN-3: Strong SMO blocker, disrupts Hh pathway (IC50=34.09 nM), hinders Daoy cell growth, has anticancer properties.</p>
    Formula:C27H25F4N3O2
    Colore e forma:Solid
    Peso molecolare:499.5
  • CM572

    CAS:
    <p>CM572 is a selective putative sigma-2 antagonist.</p>
    Formula:C22H23FN4O2S
    Colore e forma:Solid
    Peso molecolare:426.51
  • CAY10680

    CAS:
    <p>CAY10680 inhibits MAO-B (IC50=34.9 nM) &amp; A2A receptors (Ki=39.5 nM), sparing other adenosine types &amp; MAO-A, may treat Parkinson's.</p>
    Formula:C18H16N2O2S
    Colore e forma:Solid
    Peso molecolare:324.4
  • FR-194921

    CAS:
    <p>FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.</p>
    Formula:C23H23N5O
    Colore e forma:Solid
    Peso molecolare:385.46
  • RP101442

    CAS:
    <p>RP101442: Ozanimod metabolite, selective S1PR1 agonist, EC50: 2.6 nM (S1PR1), 171 nM (S1PR5).</p>
    Formula:C23H22N4O3
    Colore e forma:Solid
    Peso molecolare:402.45
  • ZM 169369

    CAS:
    <p>ICI 169369, a 5-HT2/5-HT1C antagonist, can evoke endothelium-dependent relaxation in rabbit aorta.</p>
    Formula:C19H20N2S
    Colore e forma:Solid
    Peso molecolare:308.44
  • Immepip

    CAS:
    <p>Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.</p>
    Formula:C9H15N3
    Colore e forma:Solid
    Peso molecolare:165.24
  • Phenyltoloxamine

    CAS:
    <p>Phenyltoloxamine (Bistrimin): antihistamine with sedative, analgesic properties, and Sigma-1 receptor affinity (Ki=160 nM).</p>
    Formula:C17H21NO
    Colore e forma:Solid
    Peso molecolare:255.35
  • CP 93129 dihydrochloride

    CAS:
    <p>5-HT1B agonist, potent and highly selective</p>
    Formula:C12H14ClN3O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:251.71
  • CCG-2046

    CAS:
    <p>CCG-2046 is a chemical inhibitor targeting RGS4, demonstrating an inhibition concentration (IC50) of 4.3 μM for the interaction between RGS4 and Gαo signal.</p>
    Formula:C11H10N4
    Colore e forma:Solid
    Peso molecolare:198.22
  • COR167

    CAS:
    <p>COR167 is a CB2 agonist with immunomodulatory effects, protective brain properties, and antinociception.</p>
    Formula:C28H38N2O2
    Colore e forma:Solid
    Peso molecolare:434.61
  • CGS 12066B dimaleate

    CAS:
    <p>5-HT1B full agonist</p>
    Formula:C25H25F3N4O8
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:566.48
  • Mizolastine dihydrochloride

    CAS:
    <p>Mizolastine dihydrochloride is a histamine H1-receptor antagonist (IC50: 47 nM).</p>
    Formula:C24H27Cl2FN6O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:505.42
  • CH 141

    CAS:
    <p>CH 141 is a new type of peripheral vasodilator.</p>
    Formula:C19H21N3O
    Colore e forma:Solid
    Peso molecolare:307.39
  • CID1172084

    CAS:
    CID1172084, a novel high-potent GPR55 agonist, interacts with cannabinoid receptors.
    Formula:C23H18FN5O2S2
    Colore e forma:Solid
    Peso molecolare:479.55
  • Oxyfedrine

    CAS:
    <p>Oxyfedrine: oral β-adrenoreceptor agonist, vasodilator for cardiovascular research.</p>
    Formula:C19H23NO3
    Colore e forma:Solid
    Peso molecolare:313.39
  • CP 135807

    CAS:
    <p>CP 135807 is a 5-HT1D receptor agonist.</p>
    Formula:C19H21N5O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:351.4
  • SSTR4 agonist 2

    CAS:
    <p>SSTR4 agonist 2, a potent SSTR4 subtype activator, may aid in researching nociceptive and inflammatory disorders.</p>
    Formula:C18H24N4O
    Colore e forma:Solid
    Peso molecolare:312.41
  • GB-110

    CAS:
    <p>GB-110, a potent PAR2 agonist, triggers Ca2+ release in HT29 cells with a 0.28 μM EC50, is orally active and nonpeptidic.</p>
    Formula:C33H48N6O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:608.77
  • GSK334429

    CAS:
    <p>GSK334429 is an antagonist of histamine H3 receptor.</p>
    Formula:C20H29F3N4O
    Colore e forma:Solid
    Peso molecolare:398.47
  • Piroheptine HCl

    CAS:
    <p>Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.</p>
    Formula:C22H26ClN
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:339.9
  • Bromerguride

    CAS:
    <p>Bromerguride is a dopamine antagonist with the activity of antipsychotic.</p>
    Formula:C20H25BrN4O
    Colore e forma:Solid
    Peso molecolare:417.34
  • S-5751

    CAS:
    <p>S-5751, a prostanoid DP (DP1) antagonist, is used potentially for the treatment of bronchial asthma.</p>
    Formula:C25H31NO4S
    Colore e forma:Solid
    Peso molecolare:441.58
  • Methylcarbamyl PAF C-16

    CAS:
    <p>Methylcarbamyl PAF C-16 (Carbamyl-PAF) is a PAF analog with PAF agonistic properties, activating inflammation in pregnancy tissues and promoting preterm birth.</p>
    Formula:C26H55N2O7P
    Colore e forma:Solid
    Peso molecolare:538.7
  • PF-04781340

    CAS:
    PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.
    Formula:C17H21N3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:267.37
  • AK-IN-1

    CAS:
    <p>AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.</p>
    Formula:C22H21N3O4
    Colore e forma:Solid
    Peso molecolare:391.42
  • SC 51089 free base

    CAS:
    <p>SC 51089 free base is a selective antagonist of the prostaglandin E2 EP1 receptor, demonstrating neuroprotective activity.</p>
    Formula:C22H19ClN4O3
    Colore e forma:Solid
    Peso molecolare:422.86
  • Metrenperone

    CAS:
    <p>Metrenperone is used as a S(2)-receptor blocker.</p>
    Formula:C24H26FN3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:407.48
  • CCG-271423

    CAS:
    <p>CCG-271423: potent GRK5 inhibitor (IC50: 0.0021 μM), less on GRK2 (IC50: 44 μM); lowers Ca2+ events and heart cell contractility.</p>
    Formula:C28H26N4O3
    Colore e forma:Solid
    Peso molecolare:466.53
  • LY 302148

    CAS:
    <p>LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.</p>
    Formula:C19H23FN4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:326.41
  • BMS-193884

    CAS:
    <p>BMS-193884 is an oral endothelin antagonist for the treatment of congestive heart failure (CHF) and pulmonary arterial hypertension.</p>
    Formula:C20H17N3O4S
    Colore e forma:Solid
    Peso molecolare:395.43
  • O-2093

    CAS:
    <p>anandamide uptake inhibitor</p>
    Formula:C34H43Cl2NO3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:584.62
  • ATC0065

    CAS:
    <p>ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.</p>
    Formula:C25H29BrF3N5O
    Colore e forma:Solid
    Peso molecolare:552.43
  • Acetylaszonalenin

    CAS:
    <p>Acetylaszonalenin, from A. flavipes, is an NK1 receptor antagonist with a Ki of 170 μM, blocking substance P.</p>
    Formula:C25H25N3O3
    Colore e forma:Solid
    Peso molecolare:415.48
  • Usmarapride

    CAS:
    <p>Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.</p>
    Formula:C23H31N5O6
    Colore e forma:Solid
    Peso molecolare:473.53
  • SKF 77434 hydrobromide

    CAS:
    <p>SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.</p>
    Formula:C19H22BrNO2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:376.29
  • (R)-(+)-8-Hydroxy-DPAT hydrobromide

    CAS:
    <p>5-HT1A serotonin receptor agonist</p>
    Formula:C16H26BrNO
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:328.29
  • VUF8507

    CAS:
    <p>Vuf8507 is an allosteric regulator of adenosine receptor.</p>
    Formula:C21H15N3O
    Colore e forma:Solid
    Peso molecolare:325.36
  • PD 81723

    CAS:
    <p>Allosteric potentiator at the adenosine A1 receptor</p>
    Formula:C14H12F3NOS
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:299.31
  • GAT228

    CAS:
    <p>GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].</p>
    Formula:C22H18N2O2
    Colore e forma:Solid
    Peso molecolare:342.39
  • 3-epi-Vitamin D3

    CAS:
    <p>3-epi-Vitamin D3 (Epicholecalciferol), an analogue of Vitamin D3, serves as a Hedgehog pathway inhibitor, exhibiting potency with an IC50 value of 39.2 μM in</p>
    Formula:C27H44O
    Colore e forma:Solid
    Peso molecolare:384.64
  • Fenmetozole Tosylate

    CAS:
    <p>Fenmetozole Tosylate , acts as an antidepressant drug. is an antagonist of the actions of ethanol, also antagonizes α2-adrenergic receptor,</p>
    Formula:C17H18Cl2N2O4S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:417.31
  • Agroclavine

    CAS:
    <p>Agroclavine is a clavine type of ergot alkaloid with D1 dopamine and a-adrenoceptor agonistic properties.</p>
    Formula:C16H18N2
    Colore e forma:Solid
    Peso molecolare:238.33
  • ADRA1D receptor antagonist 1 free base

    CAS:
    <p>ADRA1D antagonist blocks bladder contractions; Ki=1.6 nM, IC30=15 nM, useful in overactive bladder research.</p>
    Formula:C15H13ClN4O
    Colore e forma:Solid
    Peso molecolare:300.74
  • Fonazine

    CAS:
    <p>Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.</p>
    Formula:C19H25N3O2S2
    Colore e forma:Solid
    Peso molecolare:391.55
  • Lidanserin

    CAS:
    <p>Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.</p>
    Formula:C26H31FN2O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:454.53
  • Atigliflozin

    CAS:
    <p>Atigliflozin is an antihyperglycaemic drug candidate.</p>
    Formula:C18H22O7S
    Colore e forma:Solid
    Peso molecolare:382.43
  • Ro 363 hydrochloride

    CAS:
    <p>Ro 363 hydrochloride: selective β1-adrenoceptor agonist, boosts heart contraction, lowers diastolic pressure.</p>
    Formula:C19H26ClNO6
    Colore e forma:Solid
    Peso molecolare:399.87
  • FG-5893

    CAS:
    <p>FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.</p>
    Formula:C27H29F2N3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:465.53
  • ASP7657

    CAS:
    <p>ASP7657 is a novel, potent, and selective prostaglandin EP4 receptor antagonist.</p>
    Formula:C28H26F3N3O3
    Colore e forma:Solid
    Peso molecolare:509.52
  • Octoclothepin maleate salt

    CAS:
    <p>Octoclothepin maleate salt is a D2 dopamine receptor antagonist and 5-HT2 serotonin receptor antagonist.</p>
    Formula:C23H25ClN2O4S
    Colore e forma:Solid
    Peso molecolare:460.97
  • ICI 192605

    CAS:
    <p>ICI 192605 is a potent thromboxane A2 receptor (TP receptor) antagonist.</p>
    Formula:C22H23ClO5
    Colore e forma:Solid
    Peso molecolare:402.87
  • AL-3138

    CAS:
    <p>AL-3138 is a prostaglandin F2alpha (PGF2alpha) analogue which antagonizes FP prostanoid receptor-mediated inositol phosphates generation.</p>
    Formula:C20H33FO4
    Colore e forma:Solid
    Peso molecolare:356.47
  • CCR8 antagonist 2

    CAS:
    <p>CCR8 antagonist 2 blocks CCR8 activity, mainly on Treg and Th2 cells, for treating related diseases. See WO2022000443A1, compound 220.</p>
    Formula:C23H30ClN3O3S
    Colore e forma:Solid
    Peso molecolare:464.02
  • PQ-69

    CAS:
    <p>PQ-69 is a selective adenosine A1 receptor antagonist with inverse agonist activity.</p>
    Formula:C20H19FN4O
    Colore e forma:Solid
    Peso molecolare:350.39
  • Autotaxin-IN-6

    CAS:
    <p>Autotaxin-IN-6 is a strong ATX inhibitor with a 30 nM IC50, potentially aiding anticancer research by hindering cell migration.</p>
    Formula:C35H54BNO6
    Colore e forma:Solid
    Peso molecolare:595.62
  • Izuforant

    CAS:
    <p>Izuforant (JW1601) has anti-inflammatory effects, binds h5-HT3R (IC50: 9.1 μM), and blocks H4R orally (IC50: 36 nM).</p>
    Formula:C12H12BrN7
    Colore e forma:Solid
    Peso molecolare:334.17
  • Methyldopate hydrochloride

    CAS:
    <p>Methyldopate HCl is an agent of antihypertensive.</p>
    Formula:C12H18ClNO4
    Colore e forma:Solid
    Peso molecolare:275.73
  • Fluprostenol methyl ester

    CAS:
    <p>Fluprostenol, a vet-approved luteolytic, has an isopropyl ester, travoprost, used as an eye pressure reducer. CAY10532 is its methyl ester form.</p>
    Formula:C24H31F3O6
    Colore e forma:Solid
    Peso molecolare:472.49
  • SB 207710

    CAS:
    SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.
    Formula:C19H27IN2O4
    Colore e forma:Solid
    Peso molecolare:474.33
  • QCC-374

    CAS:
    <p>QCC-374 is a prostanoid agonist. It potentially for the treatment of pulmonary arterial hypertension.</p>
    Formula:C28H33N3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:443.58
  • UK 1745

    CAS:
    <p>UK 1745 is a novel drug of cardiotonic.</p>
    Formula:C16H23ClN2O2
    Colore e forma:Solid
    Peso molecolare:310.82
  • CP-195543

    CAS:
    <p>CP-195543 is an effective leukotriene B4 antagonist for the treatment of inflammatory diseases.</p>
    Formula:C24H19F3O4
    Colore e forma:Solid
    Peso molecolare:428.4
  • LY288513

    CAS:
    <p>Selective CCK2 receptor antagonist</p>
    Formula:C22H18BrN3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:436.3
  • GSK-269984B

    CAS:
    <p>GSK-269984B is a novel antagonist of EP1 receptor.</p>
    Formula:C20H14Cl2FNO3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:406.23
  • Guanethidine

    CAS:
    <p>Guanethidine sulphate, made in 1959, lowers blood pressure by disrupting neurotransmitters in sympathetic nerves.</p>
    Formula:C10H22N4
    Colore e forma:Solid
    Peso molecolare:198.31
  • EP4 receptor antagonist 4

    CAS:
    <p>EP4 receptor antagonist 4 is an agonist of EP4 receptor (human pEC 50 = 6.3) [1].</p>
    Formula:C19H14N2OS
    Colore e forma:Solid
    Peso molecolare:318.39
  • SKF-75670 Hydrobromide

    CAS:
    <p>SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.</p>
    Formula:C17H20BrNO2
    Colore e forma:Solid
    Peso molecolare:350.25
  • Zicronapine

    CAS:
    <p>Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.</p>
    Formula:C22H27ClN2
    Colore e forma:Solid
    Peso molecolare:354.92
  • A 55453

    CAS:
    <p>A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.</p>
    Formula:C25H32N6O3
    Colore e forma:Solid
    Peso molecolare:464.56
  • FRG8701

    CAS:
    <p>FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.</p>
    Formula:C22H30N2O4S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:418.55
  • WB403

    CAS:
    <p>WB403 activates TGR5, lowers fasting/postprandial glucose and HbA1c, enhances glucose tolerance, and normalizes pancreatic α/β-cells in diabetic mice.</p>
    Formula:C19H19BrN2OS
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:403.34
  • PD-135666

    CAS:
    <p>PD-135666 is an antagonist of CCK receptor.</p>
    Formula:C33H39N3O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:557.68
  • S-777469

    CAS:
    <p>S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.</p>
    Formula:C23H27FN2O4
    Colore e forma:Solid
    Peso molecolare:414.47
  • CB2 receptor agonist 3

    CAS:
    <p>GP 2A is a selective agonist of CB2 receptor.</p>
    Formula:C24H23Cl2N3O
    Colore e forma:Solid
    Peso molecolare:440.36
  • ATL-801

    CAS:
    <p>ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.</p>
    Formula:C24H25N7O3
    Colore e forma:Solid
    Peso molecolare:459.5
  • Latanoprost ethyl amide

    CAS:
    <p>Lat-NEt, a latanoprost analog, is an ocular hypotensive prodrug with slower hydrolysis, converting to free acids in corneal tissue.</p>
    Formula:C25H39NO4
    Colore e forma:Solid
    Peso molecolare:417.58
  • Edivoxetine

    CAS:
    <p>Edivoxetine (LY2216684) is a selective norepinephrine reuptake inhibitor for ADHD and depression.</p>
    Formula:C18H26FNO4
    Colore e forma:Solid
    Peso molecolare:339.4
  • ChemR23-IN-1

    CAS:
    <p>ChemR23-IN-1 inhibits human and mouse ChemR23 (IC50: 38 nM, 100 nM) and stops CAL-1 chemotaxis induced by Chemerin in vitro.</p>
    Formula:C28H29N7O2
    Colore e forma:Solid
    Peso molecolare:495.58
  • Bopindolol (malonate)

    CAS:
    <p>Bopindolol is a non-selective β-adrenergic receptor antagonist.</p>
    Formula:C26H32N2O7
    Colore e forma:Solid
    Peso molecolare:484.549
  • MG 1

    CAS:
    <p>MG 1 is a potent alpha-1 adrenergic receptor antagonist.</p>
    Formula:C17H25N3O2
    Purezza:98.98% - >99.99%
    Colore e forma:Solid
    Peso molecolare:303.4
  • hA2AAR antagonist 1

    CAS:
    <p>Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.</p>
    Formula:C15H15N5O
    Colore e forma:Solid
    Peso molecolare:281.31
  • Eplivanserin

    CAS:
    Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.
    Formula:C19H21FN2O2
    Purezza:97.04%
    Colore e forma:Solid
    Peso molecolare:328.38
  • EMDT

    CAS:
    <p>EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.</p>
    Formula:C15H22N2O
    Purezza:97.66% - 99.78%
    Colore e forma:Solid
    Peso molecolare:246.35
  • Nedocromil

    CAS:
    <p>Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).</p>
    Formula:C19H17NO7
    Purezza:95% - 97.34%
    Colore e forma:Solid
    Peso molecolare:371.34
  • Quinpirole Hydrochloride

    CAS:
    <p>Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and mice</p>
    Formula:C13H22ClN3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:255.79
  • Iprindole

    CAS:
    <p>Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].</p>
    Formula:C19H28N2
    Purezza:99.54%
    Colore e forma:Solid
    Peso molecolare:284.44