
Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(942 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.949 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(149 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(410 prodotti)
- Recettore dell'endotelina(75 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(32 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(166 prodotti)
- Proteina Hedgehog/Smoothened(45 prodotti)
- Recettore dell'istamina(359 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(298 prodotti)
- PAFR(11 prodotti)
- PKA(49 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5378 prodotti di "Proteina G/GPCR"
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JNJ-26070109
CAS:<p>JNJ-26070109, an antagonist of cholecystokinin CCK2 receptor, inhibits gastric acid secretion and prevents omeprazole-induced acid rebound in the rat.</p>Formula:C23H17BrF2N4O3SPurezza:98%Colore e forma:SolidPeso molecolare:547.37Ro 19-1400
CAS:<p>Ro 19-1400, a platelet-activating factor antagonist, directly inhibits immunoglobulin E-dependent mediator release.</p>Formula:C31H56N2O8SPurezza:98%Colore e forma:SolidPeso molecolare:616.85(Rac)-E1R
CAS:<p>(Rac)-E1R is the racemate of E1R. (Rac)-E1R is a sigma-1 receptor positive allosteric (Sig1R PAM) modulator of for the treatment of cognition/memory disorders.</p>Formula:C13H16N2O2Purezza:98%Colore e forma:SolidPeso molecolare:232.28GSK 189254 HCl
CAS:<p>GSK 189254A: histamine H3 antagonist, treats narcolepsy, may improve cognition and help with dementia, neuropathic pain.</p>Formula:C21H26ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:387.9Resomelagon
CAS:<p>Resomelagon (AP1189), an oral melanocortin receptor agonist, triggers Ca2+ and ERK1/2 activation; useful in obesity and inflammation studies.</p>Formula:C14H14N6O2Colore e forma:SolidPeso molecolare:298.3ONO-2952
CAS:<p>ONO-2952, a selective TSPO antagonist with Ki: 0.33-9.30 nM, may treat irritable bowel syndrome, reducing stress without causing amnesia.</p>Formula:C22H20ClFN2O2Purezza:98%Colore e forma:SolidPeso molecolare:398.86S-3608
CAS:<p>S-3608 is an atypical dopamine agonist.</p>Formula:C16H20ClN3OSColore e forma:SolidPeso molecolare:337.87Panamesine
CAS:<p>Panamesine (EMD 57445) is a high affinity receptor ligand for sigma (IC50: 6 nM) with potential for atypical antipsychotic studies.</p>Formula:C23H26N2O6Colore e forma:SolidPeso molecolare:426.46(-)-S-Timolol
CAS:<p>(-)-S-Timolol is an antagonist of the beta-Adrenergic .</p>Formula:C13H26N4O4SColore e forma:SolidPeso molecolare:334.44Inupadenant
CAS:<p>Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].</p>Formula:C25H26F2N8O4S2Colore e forma:SolidPeso molecolare:604.65A3AR antagonist 1
CAS:<p>A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.</p>Formula:C32H24N4O4SColore e forma:SolidPeso molecolare:560.62FR260010
CAS:<p>FR260010 is a novel potent serotonin 5-HT2C receptor antagonist.</p>Formula:C22H19N5Colore e forma:SolidPeso molecolare:353.42Trimazosin
CAS:<p>Trimazosin, a quinazoline derivative and prazosin relative, lowers blood pressure by blocking alpha1-adrenoceptors.</p>Formula:C20H29N5O6Colore e forma:SolidPeso molecolare:435.47SMO-IN-3
CAS:<p>SMO-IN-3: Strong SMO blocker, disrupts Hh pathway (IC50=34.09 nM), hinders Daoy cell growth, has anticancer properties.</p>Formula:C27H25F4N3O2Colore e forma:SolidPeso molecolare:499.5CM572
CAS:<p>CM572 is a selective putative sigma-2 antagonist.</p>Formula:C22H23FN4O2SColore e forma:SolidPeso molecolare:426.51CAY10680
CAS:<p>CAY10680 inhibits MAO-B (IC50=34.9 nM) & A2A receptors (Ki=39.5 nM), sparing other adenosine types & MAO-A, may treat Parkinson's.</p>Formula:C18H16N2O2SColore e forma:SolidPeso molecolare:324.4FR-194921
CAS:<p>FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.</p>Formula:C23H23N5OColore e forma:SolidPeso molecolare:385.46RP101442
CAS:<p>RP101442: Ozanimod metabolite, selective S1PR1 agonist, EC50: 2.6 nM (S1PR1), 171 nM (S1PR5).</p>Formula:C23H22N4O3Colore e forma:SolidPeso molecolare:402.45ZM 169369
CAS:<p>ICI 169369, a 5-HT2/5-HT1C antagonist, can evoke endothelium-dependent relaxation in rabbit aorta.</p>Formula:C19H20N2SColore e forma:SolidPeso molecolare:308.44Immepip
CAS:<p>Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.</p>Formula:C9H15N3Colore e forma:SolidPeso molecolare:165.24Phenyltoloxamine
CAS:<p>Phenyltoloxamine (Bistrimin): antihistamine with sedative, analgesic properties, and Sigma-1 receptor affinity (Ki=160 nM).</p>Formula:C17H21NOColore e forma:SolidPeso molecolare:255.35CP 93129 dihydrochloride
CAS:<p>5-HT1B agonist, potent and highly selective</p>Formula:C12H14ClN3OPurezza:98%Colore e forma:SolidPeso molecolare:251.71CCG-2046
CAS:<p>CCG-2046 is a chemical inhibitor targeting RGS4, demonstrating an inhibition concentration (IC50) of 4.3 μM for the interaction between RGS4 and Gαo signal.</p>Formula:C11H10N4Colore e forma:SolidPeso molecolare:198.22COR167
CAS:<p>COR167 is a CB2 agonist with immunomodulatory effects, protective brain properties, and antinociception.</p>Formula:C28H38N2O2Colore e forma:SolidPeso molecolare:434.61CGS 12066B dimaleate
CAS:<p>5-HT1B full agonist</p>Formula:C25H25F3N4O8Purezza:98%Colore e forma:SolidPeso molecolare:566.48Mizolastine dihydrochloride
CAS:<p>Mizolastine dihydrochloride is a histamine H1-receptor antagonist (IC50: 47 nM).</p>Formula:C24H27Cl2FN6OPurezza:98%Colore e forma:SolidPeso molecolare:505.42CH 141
CAS:<p>CH 141 is a new type of peripheral vasodilator.</p>Formula:C19H21N3OColore e forma:SolidPeso molecolare:307.39CID1172084
CAS:CID1172084, a novel high-potent GPR55 agonist, interacts with cannabinoid receptors.Formula:C23H18FN5O2S2Colore e forma:SolidPeso molecolare:479.55Oxyfedrine
CAS:<p>Oxyfedrine: oral β-adrenoreceptor agonist, vasodilator for cardiovascular research.</p>Formula:C19H23NO3Colore e forma:SolidPeso molecolare:313.39CP 135807
CAS:<p>CP 135807 is a 5-HT1D receptor agonist.</p>Formula:C19H21N5O2Purezza:98%Colore e forma:SolidPeso molecolare:351.4SSTR4 agonist 2
CAS:<p>SSTR4 agonist 2, a potent SSTR4 subtype activator, may aid in researching nociceptive and inflammatory disorders.</p>Formula:C18H24N4OColore e forma:SolidPeso molecolare:312.41GB-110
CAS:<p>GB-110, a potent PAR2 agonist, triggers Ca2+ release in HT29 cells with a 0.28 μM EC50, is orally active and nonpeptidic.</p>Formula:C33H48N6O5Purezza:98%Colore e forma:SolidPeso molecolare:608.77GSK334429
CAS:<p>GSK334429 is an antagonist of histamine H3 receptor.</p>Formula:C20H29F3N4OColore e forma:SolidPeso molecolare:398.47Piroheptine HCl
CAS:<p>Piroheptine HCl is an agent of anticholinergic that acts by inhibiting dopamine uptake and completely preventing loss of striatal dopamine in MPTP-treated mice.</p>Formula:C22H26ClNPurezza:98%Colore e forma:SolidPeso molecolare:339.9Bromerguride
CAS:<p>Bromerguride is a dopamine antagonist with the activity of antipsychotic.</p>Formula:C20H25BrN4OColore e forma:SolidPeso molecolare:417.34S-5751
CAS:<p>S-5751, a prostanoid DP (DP1) antagonist, is used potentially for the treatment of bronchial asthma.</p>Formula:C25H31NO4SColore e forma:SolidPeso molecolare:441.58Methylcarbamyl PAF C-16
CAS:<p>Methylcarbamyl PAF C-16 (Carbamyl-PAF) is a PAF analog with PAF agonistic properties, activating inflammation in pregnancy tissues and promoting preterm birth.</p>Formula:C26H55N2O7PColore e forma:SolidPeso molecolare:538.7PF-04781340
CAS:PF-04781340 is an effective, selective, and CNS penetrant agonist of 5-HT2C receptor.Formula:C17H21N3Purezza:98%Colore e forma:SolidPeso molecolare:267.37AK-IN-1
CAS:<p>AK-IN-1: competitive adenosine inhibitor, not ATP; inhibits AK 86-89% at 2-10 µM; promising for ischaemia, inflammation, seizure research.</p>Formula:C22H21N3O4Colore e forma:SolidPeso molecolare:391.42SC 51089 free base
CAS:<p>SC 51089 free base is a selective antagonist of the prostaglandin E2 EP1 receptor, demonstrating neuroprotective activity.</p>Formula:C22H19ClN4O3Colore e forma:SolidPeso molecolare:422.86Metrenperone
CAS:<p>Metrenperone is used as a S(2)-receptor blocker.</p>Formula:C24H26FN3O2Purezza:98%Colore e forma:SolidPeso molecolare:407.48CCG-271423
CAS:<p>CCG-271423: potent GRK5 inhibitor (IC50: 0.0021 μM), less on GRK2 (IC50: 44 μM); lowers Ca2+ events and heart cell contractility.</p>Formula:C28H26N4O3Colore e forma:SolidPeso molecolare:466.53LY 302148
CAS:<p>LY 302148 , a 5-HT1F receptor agonist, inhibits neurogenic dural inflammation in guinea pigs. It has potential for migraine therapeutics.</p>Formula:C19H23FN4Purezza:98%Colore e forma:SolidPeso molecolare:326.41BMS-193884
CAS:<p>BMS-193884 is an oral endothelin antagonist for the treatment of congestive heart failure (CHF) and pulmonary arterial hypertension.</p>Formula:C20H17N3O4SColore e forma:SolidPeso molecolare:395.43O-2093
CAS:<p>anandamide uptake inhibitor</p>Formula:C34H43Cl2NO3Purezza:98%Colore e forma:SolidPeso molecolare:584.62ATC0065
CAS:<p>ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.</p>Formula:C25H29BrF3N5OColore e forma:SolidPeso molecolare:552.43Acetylaszonalenin
CAS:<p>Acetylaszonalenin, from A. flavipes, is an NK1 receptor antagonist with a Ki of 170 μM, blocking substance P.</p>Formula:C25H25N3O3Colore e forma:SolidPeso molecolare:415.48Usmarapride
CAS:<p>Usmarapride (SUVN-D4010) is an oral 5-HT4 receptor agonist, crosses BBB, with an EC50 of 44 nM, for Alzheimer's research.</p>Formula:C23H31N5O6Colore e forma:SolidPeso molecolare:473.53SKF 77434 hydrobromide
CAS:<p>SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.</p>Formula:C19H22BrNO2Purezza:98%Colore e forma:SolidPeso molecolare:376.29(R)-(+)-8-Hydroxy-DPAT hydrobromide
CAS:<p>5-HT1A serotonin receptor agonist</p>Formula:C16H26BrNOPurezza:98%Colore e forma:SolidPeso molecolare:328.29VUF8507
CAS:<p>Vuf8507 is an allosteric regulator of adenosine receptor.</p>Formula:C21H15N3OColore e forma:SolidPeso molecolare:325.36PD 81723
CAS:<p>Allosteric potentiator at the adenosine A1 receptor</p>Formula:C14H12F3NOSPurezza:98%Colore e forma:SolidPeso molecolare:299.31GAT228
CAS:<p>GAT228, an allosteric ligand for the cannabinoid receptor 1 (CB1), functions as the enantiomer of GAT211 [1].</p>Formula:C22H18N2O2Colore e forma:SolidPeso molecolare:342.393-epi-Vitamin D3
CAS:<p>3-epi-Vitamin D3 (Epicholecalciferol), an analogue of Vitamin D3, serves as a Hedgehog pathway inhibitor, exhibiting potency with an IC50 value of 39.2 μM in</p>Formula:C27H44OColore e forma:SolidPeso molecolare:384.64Fenmetozole Tosylate
CAS:<p>Fenmetozole Tosylate , acts as an antidepressant drug. is an antagonist of the actions of ethanol, also antagonizes α2-adrenergic receptor,</p>Formula:C17H18Cl2N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:417.31Agroclavine
CAS:<p>Agroclavine is a clavine type of ergot alkaloid with D1 dopamine and a-adrenoceptor agonistic properties.</p>Formula:C16H18N2Colore e forma:SolidPeso molecolare:238.33ADRA1D receptor antagonist 1 free base
CAS:<p>ADRA1D antagonist blocks bladder contractions; Ki=1.6 nM, IC30=15 nM, useful in overactive bladder research.</p>Formula:C15H13ClN4OColore e forma:SolidPeso molecolare:300.74Fonazine
CAS:<p>Forazine (dimethiazide) is a phenothiazine drug used in the treatment of migraine and is a serotonin antagonist and a histamine antagonist.</p>Formula:C19H25N3O2S2Colore e forma:SolidPeso molecolare:391.55Lidanserin
CAS:<p>Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.</p>Formula:C26H31FN2O4Purezza:98%Colore e forma:SolidPeso molecolare:454.53Atigliflozin
CAS:<p>Atigliflozin is an antihyperglycaemic drug candidate.</p>Formula:C18H22O7SColore e forma:SolidPeso molecolare:382.43Ro 363 hydrochloride
CAS:<p>Ro 363 hydrochloride: selective β1-adrenoceptor agonist, boosts heart contraction, lowers diastolic pressure.</p>Formula:C19H26ClNO6Colore e forma:SolidPeso molecolare:399.87FG-5893
CAS:<p>FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.</p>Formula:C27H29F2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:465.53ASP7657
CAS:<p>ASP7657 is a novel, potent, and selective prostaglandin EP4 receptor antagonist.</p>Formula:C28H26F3N3O3Colore e forma:SolidPeso molecolare:509.52Octoclothepin maleate salt
CAS:<p>Octoclothepin maleate salt is a D2 dopamine receptor antagonist and 5-HT2 serotonin receptor antagonist.</p>Formula:C23H25ClN2O4SColore e forma:SolidPeso molecolare:460.97ICI 192605
CAS:<p>ICI 192605 is a potent thromboxane A2 receptor (TP receptor) antagonist.</p>Formula:C22H23ClO5Colore e forma:SolidPeso molecolare:402.87AL-3138
CAS:<p>AL-3138 is a prostaglandin F2alpha (PGF2alpha) analogue which antagonizes FP prostanoid receptor-mediated inositol phosphates generation.</p>Formula:C20H33FO4Colore e forma:SolidPeso molecolare:356.47CCR8 antagonist 2
CAS:<p>CCR8 antagonist 2 blocks CCR8 activity, mainly on Treg and Th2 cells, for treating related diseases. See WO2022000443A1, compound 220.</p>Formula:C23H30ClN3O3SColore e forma:SolidPeso molecolare:464.02PQ-69
CAS:<p>PQ-69 is a selective adenosine A1 receptor antagonist with inverse agonist activity.</p>Formula:C20H19FN4OColore e forma:SolidPeso molecolare:350.39Autotaxin-IN-6
CAS:<p>Autotaxin-IN-6 is a strong ATX inhibitor with a 30 nM IC50, potentially aiding anticancer research by hindering cell migration.</p>Formula:C35H54BNO6Colore e forma:SolidPeso molecolare:595.62Izuforant
CAS:<p>Izuforant (JW1601) has anti-inflammatory effects, binds h5-HT3R (IC50: 9.1 μM), and blocks H4R orally (IC50: 36 nM).</p>Formula:C12H12BrN7Colore e forma:SolidPeso molecolare:334.17Methyldopate hydrochloride
CAS:<p>Methyldopate HCl is an agent of antihypertensive.</p>Formula:C12H18ClNO4Colore e forma:SolidPeso molecolare:275.73Fluprostenol methyl ester
CAS:<p>Fluprostenol, a vet-approved luteolytic, has an isopropyl ester, travoprost, used as an eye pressure reducer. CAY10532 is its methyl ester form.</p>Formula:C24H31F3O6Colore e forma:SolidPeso molecolare:472.49SB 207710
CAS:SB 207710 is a selective and high affinity antagonist of 5-HT4 receptor.Formula:C19H27IN2O4Colore e forma:SolidPeso molecolare:474.33QCC-374
CAS:<p>QCC-374 is a prostanoid agonist. It potentially for the treatment of pulmonary arterial hypertension.</p>Formula:C28H33N3O2Purezza:98%Colore e forma:SolidPeso molecolare:443.58UK 1745
CAS:<p>UK 1745 is a novel drug of cardiotonic.</p>Formula:C16H23ClN2O2Colore e forma:SolidPeso molecolare:310.82CP-195543
CAS:<p>CP-195543 is an effective leukotriene B4 antagonist for the treatment of inflammatory diseases.</p>Formula:C24H19F3O4Colore e forma:SolidPeso molecolare:428.4LY288513
CAS:<p>Selective CCK2 receptor antagonist</p>Formula:C22H18BrN3O2Purezza:98%Colore e forma:SolidPeso molecolare:436.3GSK-269984B
CAS:<p>GSK-269984B is a novel antagonist of EP1 receptor.</p>Formula:C20H14Cl2FNO3Purezza:98%Colore e forma:SolidPeso molecolare:406.23Guanethidine
CAS:<p>Guanethidine sulphate, made in 1959, lowers blood pressure by disrupting neurotransmitters in sympathetic nerves.</p>Formula:C10H22N4Colore e forma:SolidPeso molecolare:198.31EP4 receptor antagonist 4
CAS:<p>EP4 receptor antagonist 4 is an agonist of EP4 receptor (human pEC 50 = 6.3) [1].</p>Formula:C19H14N2OSColore e forma:SolidPeso molecolare:318.39SKF-75670 Hydrobromide
CAS:<p>SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.</p>Formula:C17H20BrNO2Colore e forma:SolidPeso molecolare:350.25Zicronapine
CAS:<p>Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.</p>Formula:C22H27ClN2Colore e forma:SolidPeso molecolare:354.92A 55453
CAS:<p>A 55453 is a radiated ionophore used as a reversibl, high-affinity alpha 1-adrenergic receptor probe.</p>Formula:C25H32N6O3Colore e forma:SolidPeso molecolare:464.56FRG8701
CAS:<p>FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.</p>Formula:C22H30N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:418.55WB403
CAS:<p>WB403 activates TGR5, lowers fasting/postprandial glucose and HbA1c, enhances glucose tolerance, and normalizes pancreatic α/β-cells in diabetic mice.</p>Formula:C19H19BrN2OSPurezza:98%Colore e forma:SolidPeso molecolare:403.34PD-135666
CAS:<p>PD-135666 is an antagonist of CCK receptor.</p>Formula:C33H39N3O5Purezza:98%Colore e forma:SolidPeso molecolare:557.68S-777469
CAS:<p>S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.</p>Formula:C23H27FN2O4Colore e forma:SolidPeso molecolare:414.47CB2 receptor agonist 3
CAS:<p>GP 2A is a selective agonist of CB2 receptor.</p>Formula:C24H23Cl2N3OColore e forma:SolidPeso molecolare:440.36ATL-801
CAS:<p>ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.</p>Formula:C24H25N7O3Colore e forma:SolidPeso molecolare:459.5Latanoprost ethyl amide
CAS:<p>Lat-NEt, a latanoprost analog, is an ocular hypotensive prodrug with slower hydrolysis, converting to free acids in corneal tissue.</p>Formula:C25H39NO4Colore e forma:SolidPeso molecolare:417.58Edivoxetine
CAS:<p>Edivoxetine (LY2216684) is a selective norepinephrine reuptake inhibitor for ADHD and depression.</p>Formula:C18H26FNO4Colore e forma:SolidPeso molecolare:339.4ChemR23-IN-1
CAS:<p>ChemR23-IN-1 inhibits human and mouse ChemR23 (IC50: 38 nM, 100 nM) and stops CAL-1 chemotaxis induced by Chemerin in vitro.</p>Formula:C28H29N7O2Colore e forma:SolidPeso molecolare:495.58Bopindolol (malonate)
CAS:<p>Bopindolol is a non-selective β-adrenergic receptor antagonist.</p>Formula:C26H32N2O7Colore e forma:SolidPeso molecolare:484.549MG 1
CAS:<p>MG 1 is a potent alpha-1 adrenergic receptor antagonist.</p>Formula:C17H25N3O2Purezza:98.98% - >99.99%Colore e forma:SolidPeso molecolare:303.4hA2AAR antagonist 1
CAS:<p>Compound 4a, also known as hA2AAR antagonist 1, is a highly selective hA2AAR antagonist with a Ki value of 5 nM. It is useful in the field of immuno-oncology research.</p>Formula:C15H15N5OColore e forma:SolidPeso molecolare:281.31Eplivanserin
CAS:Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.Formula:C19H21FN2O2Purezza:97.04%Colore e forma:SolidPeso molecolare:328.38EMDT
CAS:<p>EMDT oxalate is a selective 5-HT6 agonist, and has antidepressant effects.</p>Formula:C15H22N2OPurezza:97.66% - 99.78%Colore e forma:SolidPeso molecolare:246.35Nedocromil
CAS:<p>Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).</p>Formula:C19H17NO7Purezza:95% - 97.34%Colore e forma:SolidPeso molecolare:371.34Quinpirole Hydrochloride
CAS:<p>Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and mice</p>Formula:C13H22ClN3Purezza:98%Colore e forma:SolidPeso molecolare:255.79Iprindole
CAS:<p>Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].</p>Formula:C19H28N2Purezza:99.54%Colore e forma:SolidPeso molecolare:284.44
