Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(993 prodotti)
- Recettore dell'adenosina(246 prodotti)
- Recettore adrenergico(3.004 prodotti)
- Recettore della bombesina(33 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(153 prodotti)
- CaSR(33 prodotti)
- Recettore dei cannabinoidi(212 prodotti)
- Recettore della dopamina(433 prodotti)
- Recettore dell'endotelina(79 prodotti)
- Recettore GNRH(77 prodotti)
- GPCR19(32 prodotti)
- GRK(32 prodotti)
- GTPase(22 prodotti)
- Recettore del glucagone(182 prodotti)
- Proteina Hedgehog/Smoothened(47 prodotti)
- Recettore dell'istamina(381 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(26 prodotti)
- Recettore OX(41 prodotti)
- Recettore degli oppioidi(310 prodotti)
- PAFR(12 prodotti)
- PKA(51 prodotti)
- Recettore S1P(18 prodotti)
- SGLT(31 prodotti)
- Recettore Sigma(46 prodotti)
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Trovati 5745 prodotti di "Proteina G/GPCR"
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Methimepip dihydrobromide
CAS:Methimepip dihydrobromide is a selective H3R agonist.Formula:C10H19Br2N3Colore e forma:SolidPeso molecolare:341.091Prolactin Releasing Peptide (1-31), human acetate
Prolactin Releasing Peptide (1-31), human (acetate), is a potent GPR10 ligand with high affinity, eliciting prolactin secretion.Formula:C162H26N56O44SPeso molecolare:3724.17Vapiprost hydrochloride
CAS:Vapiprost hydrochloride is a biochemicla.Formula:C30H40ClNO4Colore e forma:SolidPeso molecolare:514.1Spantide II
CAS:<p>Spantide II is an antagonist of tachykinin.</p>Formula:C86H104Cl2N18O13Purezza:98%Colore e forma:SolidPeso molecolare:1668.77Bertilimumab
CAS:<p>Bertilimumab (CAT 213; iCo-008), a human monoclonal antibody that targets eotaxin-1 (CCL11), shows promise in the research of allergic disorders [1].</p>Colore e forma:LiquidAcmopatide
CAS:Acmopatide (Compound E-153) is a dual agonist of GIP and GLP-1 receptors and can be utilized in diabetes research.Colore e forma:SolidBiotin-Gastrin Releasing Peptide, human TFA
Biotin-Gastrin Releasing Peptide, human TFA, is a biotinylated form of the gastrin-releasing peptide (GRP). GRP is a neuropeptide known for its growth-stimulating and tumorigenic properties.Colore e forma:Odour SolidNeuropeptide Y (human)
CAS:<p>Neuropeptide Y (29-64), amide, human is a biologically active 36-amino acid peptide.</p>Formula:C189H285N55O57SPurezza:98%Colore e forma:SolidPeso molecolare:4271.68Galanin (1-16), mouse, porcine, rat TFA
Galanin (1-16) agonizes hippocampal receptors; Kd 3 nM. Active on locus coeruleus neurons in mice, pigs, rats.Formula:C80H117F3N20O23Purezza:98%Colore e forma:SolidPeso molecolare:1783.915-keto Latanoprost
CAS:Latanoprost, a PG analog for ocular pressure, metabolizes into 15-keto latanoprost, a less potent variant reducing intraocular pressure and pupil size.Formula:C26H38O5Colore e forma:SolidPeso molecolare:430.58Neuropeptide Y5 receptor ligand-1
CAS:Neuropeptide Y5 receptor ligand-1 (Compound 54), a carbazole derivative, acts as a powerful antagonist to the neuropeptide Y5 (NPY-5) receptor [1].Formula:C19H17N3O2Colore e forma:SolidPeso molecolare:319.36GB-110 hydrochloride
GB-110 HCl: potent, nonpeptidic oral PAR2 agonist; triggers Ca2+ release in HT29 cells; EC50 0.28 μM.Formula:C33H49ClN6O5Colore e forma:SolidPeso molecolare:645.23U92016A
CAS:U92016A is a highly potent and selective agonist of 5-HT1A receptor.Formula:C19H25N3Purezza:98%Colore e forma:SolidPeso molecolare:295.42HTL22562
CAS:HTL22562 is a calcitonin gene-related peptide (CGRP) receptor antagonist for acute treatment of migraine.Formula:C40H49N11O5Colore e forma:SolidPeso molecolare:763.904Moxilubant HCl
CAS:Moxilubant HCl: small molecule LTB4R antagonist for immune, skin, musculoskeletal disorders, and research in psoriasis, arthritis.Formula:C26H38ClN3O4Purezza:99.94%Colore e forma:SoildPeso molecolare:492.05Zovaglutide
CAS:Zovaglutide is a GLP-1 receptor agonist that is utilized in diabetes research.Colore e forma:SolidSU 4029 dihydrochloride
CAS:SU 4029 dihydrochloride is a bioactive chemical.Formula:C9H21Cl2N3OColore e forma:SolidPeso molecolare:258.19[Gly8]-GLP-1(7-37) acetate
[Gly8]-GLP-1(7-37) acetate is a derivative of GLP-1, where glycine at position 8 is replaced with alanine. [Gly8]-GLP-1(7-37) acetate is also a peptide fragment of the GLP-1 receptor (GLP-1R) agonist, Dulaglutide.Colore e forma:Odour SolidNK3R-IN-2
NK3R-IN-2 is an orally active NK3R inhibitor with an IC50 of 330.50 nM against human NK3R. It can penetrate the blood-brain barrier and exhibits excellent NK3R binding affinity in CHO-K1 cells (IC50= 87.31 nM). NK3R-IN-2 effectively suppresses luteinizing hormone (LH) levels and is applicable for research on hormone-related diseases.Colore e forma:Odour SolidPACAP (6-38), human, ovine, rat
CAS:<p>PACAP (6-38) in humans, sheep, rats: a strong inhibitor of PACAP 38, outperforms PACAP (6-27) in blocking PACAP-27-induced adenylate cyclase.</p>Formula:C182H300N56O45SPurezza:98%Colore e forma:SolidPeso molecolare:4024.74SLP7111228
CAS:SLP7111228 is an effective and selective SphK1 inhibitor (Ki = 48 nM).Formula:C22H33N5OColore e forma:SolidPeso molecolare:383.53Substance P (1-9)
CAS:Substance P (1-9), a nonapeptide, slows its own inactivation and stimulates neurons.Formula:C52H77N15O12Purezza:98%Colore e forma:SolidPeso molecolare:1104.266β-Prostaglandin I1
CAS:6β-PGI1 is a stable PGI2 analog resistant to hydrolysis in aqueous solutions.Formula:C20H34O5Colore e forma:SolidPeso molecolare:354.487GIP/GLP-1 dual receptor agonist-1 sodium
GIP/GLP-1 dual receptor agonist-1 (Compound 4) (sodium) functions as a GIP/GLP-1 receptor agonist. This compound is applicable for research into metabolic disorders and liver diseases, including non-alcoholic steatohepatitis (NASH) and non-alcoholic fatty liver disease (NAFLD).Colore e forma:Odour SolidGRP (porcine)
CAS:GRP: agonist for GRPR, stimulates amygdala GABA release reducing fear in mice, aids mitogenesis, GI function, and appetite control.Formula:C126H198N38O31S2Purezza:98%Colore e forma:SolidPeso molecolare:2805.31BE-24566B
CAS:BE-24566B, a polyketide from S. violaceusniger, inhibits various bacteria and blocks ET receptors (ETA IC50=11 μM, ETB=3.9 μM).Formula:C27H24O7Colore e forma:SolidPeso molecolare:460.482PACAP (6-27) (human, chicken, mouse, ovine, porcine, rat) (trifluoroacetate salt)
PACAP (6-27) is an antagonist for PACAP receptors with varying IC50s; blocks cAMP in neuroblastoma and breast cancer cells.Colore e forma:LiquidOrexin B, rat, mouse
CAS:Orexin B, rat, mouse is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.Formula:C126H215N45O34SPurezza:98%Colore e forma:SolidPeso molecolare:2936.45Beraprost
CAS:Beraprost is a stable prostacyclin analog.Formula:C24H30O5Colore e forma:SolidPeso molecolare:398.49Prepro VIP (81-122), human
CAS:Prepro VIP (81-122), human is a prepro-vasoactive intestinal polypeptide (VIP) derived peptide, corresponding to residues 81-122.Formula:C202H325N53O64SPurezza:98%Colore e forma:SolidPeso molecolare:4552.13SDV-Exendin-3/4
SDV-Exendin-3/4 is a 32-amino acid peptide.Formula:NAPurezza:98%Colore e forma:SolidPeso molecolare:3443.87Esprolol
CAS:<p>Esprolol (ACC-9369 free base) is a novel beta-adrenergic antagonist used to study exertional angina.</p>Formula:C17H27NO4Purezza:71.58% - 99.16%Colore e forma:SoildPeso molecolare:309.4Petrelintide acetate
<p>Petrelintide (ZP8396) acetate is an amylin analog with potential for weight reduction, suitable for diabetes research.</p>Formula:C185H305N49O61·xC2H4O2Colore e forma:SolidPeso molecolare:4191.69 (free base)PAMP-12(human, porcine)
CAS:Potent endogenous peptide agonist of Mas related GPR X2 (MRGPRX2, EC50 = 57.2 nM). Corresponds to amino acids 9 to 20 of proadrenomedullin.Formula:C77H119N25O14Purezza:98%Colore e forma:SolidPeso molecolare:1618.95CTP-amiodarone
CTP-amiodarone, a cellular-penetrating conjugate of myocardial cell-targeting peptide and Amiodarone, exhibits anti-arrhythmic activity by blocking Na+, K+, and Ca2+ channels as well as β-adrenergic receptors.Formula:C97H131F3I2N20O25S2Colore e forma:SolidPeso molecolare:2352.13Mapenterol hydrochloride
CAS:<p>Mapenterol hydrochloride is an agonist of β2-adrenergic receptor.</p>Formula:C14H21Cl2F3N2OPurezza:98.11% - 99.98%Colore e forma:SolidPeso molecolare:361.23KISS1-305
CAS:KISS1-305: Metastin analog, prototype peptide, resists protease degradation, suboptimal KISS1R agonist.Formula:C56H76N16O12Purezza:98%Colore e forma:SolidPeso molecolare:1165.3Acetyl neurotensin (8-13)
CAS:Acetyl neurotensin (8-13), the most concise analog of neurotensin, retains complete binding and pharmacological properties [1].Formula:C40H66N12O9Peso molecolare:859.03Sufotidine
CAS:Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.Formula:C20H31N5O3SPurezza:99.03% - 99.92%Colore e forma:SolidPeso molecolare:421.56[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide
[D-Leu6, Val7]-LH-RH (1-9) Ethyl Amide is a LHRH peptide analogue.Formula:C58H82N16O12Peso molecolare:1195.37Tamuzimod
CAS:Tamuzimod, an effective immunomodulator, exhibits modulatory activity on S1P Receptors with EC50 values below 1 μM [1] [2].Formula:C21H13Cl3F3N5O3Colore e forma:SolidPeso molecolare:546.71Ro60-0175
CAS:<p>Ro60-0175 is a selective 5-HT2B and 5-HT2C serotonin receptor agonist, often used as fumarate.</p>Formula:C11H12ClFN2Purezza:97.09%Colore e forma:SolidPeso molecolare:226.68(Des-Bromo)-Neuropeptide B (1-23) (human)
CAS:'(Des-Bromo)-Neuropeptide B (1-23) (human)' is an agonist for orphan G-protein-coupled receptors, exhibiting a K i of 1.2 nM for GPR7 (NPBW1) and 341 nM forFormula:C107H162N30O30Peso molecolare:2348.61DOTA-EB-TATE
DOTA-EB-TATE is formed by combining the SST peptide derivative DOTA-octreotate with an Evans blue analog (EB). This peptide drug conjugate (PDC) enhances the pharmacokinetics of SSTR2 analogs and reduces PRRT toxicity. Additionally, DOTA-EB-TATE serves in the synthesis/research of radiopharmaceutical conjugates (RDC).Formula:C105H133N21O30S5Peso molecolare:2329.63Anti-GLP-1R Antibody
<p>Anti-GLP-1R Antibody is an anti-GLP-1R antibody that can be used for immunohistochemistry of paraffin sections.</p>Purezza:98.3% (SDS-PAGE); 97.2% (SEC-HPLC) - 98.3% (SDS-PAGE); 97.2% (SEC-HPLC)Colore e forma:Odour LiquidHPP-9
HPP-9, a Proteolysis-Targeting Chimera (PROTAC) derived from Hedgehog Pathway Inhibitor-1 (HPI-1) with a pIC50 value of 6.71, is designed to degrade BETFormula:C49H52N6O11Colore e forma:SolidPeso molecolare:900.97Firazorexton
CAS:Firazorexton is a potent orexin type 2 receptor (OX2R) agonist.Formula:C22H25F3N2O4SColore e forma:SolidPeso molecolare:470.51PROTAC(H-PGDS)-8
CAS:PROTAC(H-PGDS)-8 is a PROTAC degrader targeting Hematopoietic prostaglandin D synthase (H-PGDS), exhibiting an IC50 of 0.14 μM [1].Formula:C41H40N8O7Colore e forma:SolidPeso molecolare:756.819-deoxy-9-methylene Prostaglandin E2
CAS:9-deoxy-9-methylene PGE2: stable PGE2 analog with similar effects, less side effects, equal potency in rats, gerbils, primates.Formula:C21H34O4Colore e forma:SolidPeso molecolare:350.499(-)-Eseroline fumarate
CAS:(-)-Eseroline fumarate, a Physostigmine metabolite and AChE inhibitor, triggers cancer cell LDH release and neuronal cell death.Formula:C17H22N2O5Colore e forma:SolidPeso molecolare:334.37ACT-1016-0707
CAS:<p>ACT-1016-0707 is a selective, insurmountable LPA1 antagonist with antifibrotic and anti-inflammatory activity in lung fibrosis models</p>Formula:C19H23ClN4O4SPurezza:99.905%Colore e forma:SolidPeso molecolare:438.93Hemokinin 1, human TFA
<p>Hemokinin-1 is a human TFA and selective NK1 agonist; also activates NK2 & NK3 and induces opioid-independent analgesia.</p>Formula:C56H85F3N14O16SColore e forma:SolidPeso molecolare:1299.42Sorbinicate
CAS:<p>Sorbinicate is an antihypercholesterolaemic and vasodilating nicotinic acid ester.</p>Formula:C42H32N6O12Purezza:98%Colore e forma:SolidPeso molecolare:812.74Human growth hormone-releasing factor TFA
<p>Human growth hormone-releasing factor TFA is a hypothalamic peptide that promotes GH secretion by targeting pituitary GHRHR.</p>Formula:C217H359F3N72O68SColore e forma:SolidPeso molecolare:5153.67Ecnoglutide
CAS:Ecnoglutide (XW003) is a glucagon-like peptide 1 (GLP-1) receptor agonist [1] .Formula:C194H304N48O61Colore e forma:SolidPeso molecolare:4284.76Levitide
CAS:Levitide is a neurohormone-like peptide which is from the skin of Xenopus laevis.Formula:C66H119N21O19SPurezza:98%Colore e forma:SolidPeso molecolare:1542.85K-(D-1-Nal)-FwLL-NH2 TFA
<p>K-(D-1-Nal)-FwLL-NH2 TFA: potent ghrelin inverse agonist; Ki=4.9 nM (COS7), 31 nM (HEK293T); blocks Gq/G13 signaling.</p>Formula:C53H68F3N9O8Colore e forma:SolidPeso molecolare:1016.16ANQ-11125 TFA
<p>ANQ-11125 TFA is a motilin antagonist with a pKd of 8.24, inhibiting motilide contractions in rabbits.</p>Formula:C88H126F3N19O23Colore e forma:SolidPeso molecolare:1875.05Neuropeptide Y (18-36) (porcine)
CAS:<p>"Neuropeptide Y (18-36) (porcine) is a NPY heart receptor blocker, halts I-NPY binding, aids in heart failure research."</p>Formula:C112H174N36O27Colore e forma:SolidPeso molecolare:2456.8ORG 2766
CAS:<p>ORG 2766 is an ACTH 4-9 (H-Met(O)-Glu-His-Phe-D-Lys-Phe-OH) analog and neurotrophic peptide.</p>Formula:C40H55N9O11SColore e forma:SolidPeso molecolare:869.99Secretoneurin, rat
CAS:Secretoneurin, rat, a 33-amino acid polypeptide, is generated by proteolytic processing of secretogranin II (SgII).Formula:C159H252N40O58Purezza:98%Colore e forma:SolidPeso molecolare:3651.95Selepressin acetate
<p>Selepressin acetate is a useful organic compound for research related to life sciences and the catalog number is T73654.</p>Formula:C48H77N13O13S2Colore e forma:SolidPeso molecolare:1108.33[Ala2] Endothelin-3, human
CAS:<p>[Ala2] Endothelin-3, a linear ET-3 analog with Ala replacing Cys, stimulates endothelial cell migration.</p>Formula:C120H166N26O32S4Colore e forma:SolidPeso molecolare:2613.02Dotanoc
CAS:<p>Dotanoc is a ligand to make gallium Ga 68-DOTANOC, which is a gallium Ga 68-radiolabeled analog of somatostatin.</p>Formula:C69H94N14O17S2Colore e forma:SolidPeso molecolare:1455.71Gastrin I, rat
CAS:Gastrin I, rat is a peptide hormone that effectively stimulates gastric acid secretion.Formula:C94H128N22O31S2Colore e forma:SolidPeso molecolare:2126.3Neuropeptide Y (3-36) (porcine)
CAS:<p>Neuropeptide Y (3-36) (porcine) is a potent, selective agonist at NPY Y2 receptors, increasing feeding in rats.</p>Formula:C176H271N53O54Colore e forma:SolidPeso molecolare:3993.36Kisspeptin-54(human) TFA
<p>Endogenous kisspeptin-54(human) TFA targets KISS1/GPR54 receptors; Ki: 1.81 nM (rat), 1.45 nM (human); inhibits metastasis, boosts gonadotropin.</p>Formula:C258H401N79O78·C2HF3O2Colore e forma:SolidPeso molecolare:5971.45Cyclic SSTR agonist octreotide
Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .Formula:C53H71N11O14S2Colore e forma:SolidPeso molecolare:1150.33[Asu1,6-Arg8]Vasopressin
CAS:[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.Formula:C48H68N14O12Colore e forma:SolidPeso molecolare:1033.14(2R,2R)-PF-07258669
CAS:<p>(2R,2R)-PF-07258669' is an antagonist for the MC4R (melanocortin 4 receptor), primarily studied for its role in regulating appetite and energy expenditure.</p>Formula:C25H27FN6O2Colore e forma:SolidPeso molecolare:462.52Melanostatin, frog
CAS:<p>Melanostatin, frog, is an inhibitor of α-melanocyte-stimulating hormone (α-MSH) release, with an IC50 of 60 nM [1] [2].</p>Formula:C189H285N53O57SColore e forma:SolidPeso molecolare:4243.67α-CGRP(human) TFA
<p>α-CGRP(human) TFA is a 37-amino acid regulatory neuropeptide that is extensively located within the central and peripheral nervous system, functioning as a</p>Formula:C165H268F3N51O51S2Colore e forma:SolidPeso molecolare:3903.33Neuropeptide Y (3-36) (human, rat)
CAS:<p>Neuropeptide Y (3-36) is a Y2 receptor agonist that limits norepinephrine release, produced by DPP4 from NPY.</p>Formula:C175H269N53O54SColore e forma:SolidPeso molecolare:4011.5Prepro-ANF (56-92), human
CAS:<p>Human prepro-ANF (56-92) activates renal guanylate cyclase and boosts its activity.</p>Formula:C173H270N44O57Colore e forma:SolidPeso molecolare:3878.26Protease-Activated Receptor-1, PAR-1 Agonist TFA
<p>PAR-1 Agonist TFA: Selective peptide, mimics thrombin, activates PAR-1 receptor.</p>Colore e forma:Liquid(Trp7,β-Ala8)-Neurokinin A (4-10)
CAS:<p>(Trp7,β-Ala8)-Neurokinin A (4-10) is a potent neurokinin-3 (NK3) antagonist [1] .</p>Formula:C41H57N9O10SColore e forma:SolidPeso molecolare:868.01Cyclosomatostatin TFA
<p>Cyclosomatostatin TFA blocks SST receptor, reduces CRC cell growth, ALDH+ size, and sphere-formation.</p>Formula:C46H58F3N7O8Colore e forma:SolidPeso molecolare:893.99Sauvagine TFA
<p>Sauvagine TFA: frog-derived, 40-amino-acid CRF agonist; stimulates ACTH release, affects diuresis, cardiovascular system, endocrine glands.</p>Formula:C204H347F3N56O65S1Colore e forma:SolidPeso molecolare:4713.33Physalaemin
CAS:Physalaemin is a non-mammalian tachykinin.Formula:C58H84N14O16SPurezza:98%Colore e forma:SolidPeso molecolare:1265.45GR 82334
CAS:<p>Tachykinin NK1 receptor antagonist.</p>Formula:C69H91N15O16Purezza:98%Colore e forma:SolidPeso molecolare:1386.57Orforglipron hemicalcium hydrate
CAS:Orforglipron hemicalcium hydrate (LY3502970 hemicalcium hydrate; GLP-1 receptor agonist 1 hemicalcium hydrate) represents the hemicalcium hydrate form of the calcium salt of Orforglipron, an orally active agonist targeting the Glucagon-like peptide-1 receptor (GLP-1R). This compound has demonstrated efficacy in mitigating type 2 diabetes [1].Formula:C48H48F2N10O5Ca·H2OColore e forma:SolidPeso molecolare:921.02Quinelorane
CAS:Quinelorane is dextrorotary isomer.Formula:C14H22N4Colore e forma:SolidPeso molecolare:246.35[Lys4] Sarafotoxin S6c
CAS:<p>[Lys4] Sarafotoxin S6c: potent partial endothelin receptor agonist; causes pig coronary contraction, EC50=1.5 nM.</p>Formula:C105H153N27O36S5Colore e forma:SolidPeso molecolare:2529.82[Tyr22] Calcitonin Gene Related Peptide, (22-37), rat
CAS:[Tyr22] CGRP (22-37), rat is a fragment of rat CGRP, targeting its receptor and adenylate cyclase, produced by thyroid and stored in the nervous system.Formula:C82H120N20O25Colore e forma:SolidPeso molecolare:1785.95Angiopeptin
CAS:<p>Angiopeptin is a synthetic octapeptide analog of somatostatin; suppresses accelerated transplant atherosclerosis in rabbit heart arteries.</p>Formula:C54H71N11O10S2Colore e forma:SolidPeso molecolare:1098.34ZL-1101
<p>ZL-1101 is a human monoclonal antibody (mAb) targeting TNFRSF4/OX40/CD134.</p>Colore e forma:Odour Liquida-Helical Corticotropin Releasing Factor (9-41)
CAS:<p>α-Helical CRF (9-41) is a CRF antagonist that lowers in vivo plasma GH levels.</p>Formula:C166H273N45O54S2Colore e forma:SolidPeso molecolare:3827.34Dexbrompheniramine
CAS:Dexbrompheniramine: oral H1 antagonist, antihistamine for hay fever and urticaria research.Formula:C16H19BrN2Colore e forma:SolidPeso molecolare:319.2415(S)-15-methyl Prostaglandin D2
CAS:15(S)-15-methyl PGD2 is a stable PGD2 analog that induces vasoconstriction, raises blood pressure, and shows strong antifertility effects.Formula:C21H34O5Colore e forma:SolidPeso molecolare:366.49Adenosine receptor antagonist 1
CAS:A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.Formula:C22H15ClFN7OColore e forma:SolidPeso molecolare:447.86MEN 11270
CAS:<p>B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.</p>Formula:C60H90N20O11SPurezza:98%Colore e forma:SolidPeso molecolare:1299.56Dipentylone hydrochloride
CAS:Dipentylone hydrochloride (Bk-dmbdp HCl) is a psychoactive synthetic cathinone and sympathomimetic stimulant. Its inhibitory activity towards the dopamine transporter (IC50=0.233µM) is tenfold higher than that towards NET and SERT, inhibiting dopamine uptake and stimulating locomotor activity in mice.Formula:C14H20ClNO3Purezza:99.94%Colore e forma:SolidPeso molecolare:285.77Linzagolix choline
CAS:Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.Formula:C27H28F3N3O8SPurezza:99.64%Colore e forma:SolidPeso molecolare:611.59Methdilazine
CAS:Methdilazine: oral antibiotic, histamine antagonist, fights mycobacterium (MIC 5-15 μg/mL) for infectious disease research.Formula:C18H20N2SColore e forma:SolidPeso molecolare:296.43α-CGRP(human)
CAS:Endogenous calcitonin gene-related peptide receptor (CGRP) agonist.Formula:C163H267N51O49S2Purezza:98%Colore e forma:SolidPeso molecolare:3789.33Stressin I
Potent CRF1 agonist; Ki: 1.5 nM (CRF1), 224 nM (CRF2). Boosts ACTH, enhances stool frequency after i.p. administration.Formula:C203H337N57O56Purezza:98%Colore e forma:SolidPeso molecolare:4472.24GLP-1 receptor agonist 9 citrate
<p>GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.</p>Formula:C38H39ClFN3O12Purezza:98.76%Colore e forma:SolidPeso molecolare:784.18ELA-11(human)
CAS:<p>Apelin receptor agonist with high affinity (Ki = 14 nM). Blocks cAMP production and promotes β-arrestin activation; derived from ELA-32.</p>Formula:C58H90N16O13S2Purezza:98%Colore e forma:SolidPeso molecolare:1283.57GLP-1R agonist 14
CAS:GLP-1R agonist 14, also known as Compound 14, is a potent agonist of the GLP-1 receptor, demonstrating an EC50 range of 0-20 nM against human GLP-1 [1].Formula:C45H42F2N10O5Colore e forma:SolidPeso molecolare:840.88SR 142948 dihydrochloride
SR 142948 dihydrochloride is a selective oral non-peptide NT antagonist, IC50 <4 nM, with brain penetration and potential for psychiatric research.Formula:C39H53Cl2N5O6Colore e forma:SolidPeso molecolare:758.77
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