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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

Mostrare 18 più sottocategorie

Trovati 5352 prodotti di "Proteina G/GPCR"

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  • Dasotraline
    Targetmol
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    Dasotraline

    CAS:
    <p>Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.</p>
    Formula:C16H15Cl2N
    Colore e forma:Solid
    Peso molecolare:292.2

    Ref: TM-T60607

  • Rolapitant hydrochloride hydrate
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    Rolapitant hydrochloride hydrate

    CAS:
    <p>Rolapitant (SCH-619734) is a selective NK1-receptor antagonist that may prevent nausea and vomiting induced by chemotherapy.</p>
    Formula:C25H29ClF6N2O3
    Colore e forma:Solid
    Peso molecolare:554.95

    Ref: TM-T68371

  • Irdabisant hydrochloride
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    Irdabisant hydrochloride

    CAS:
    <p>Irdabisant (CEP-26401) is a selective H3R inverse agonist, BBB-penetrable, with cognition-enhancing effects.</p>
    Formula:C18H24ClN3O2
    Colore e forma:Solid
    Peso molecolare:349.86

    Ref: TM-T61197

  • Spiperone hydrochloride
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    Spiperone hydrochloride

    CAS:
    <p>5-HT2A serotonin and selective D2-like dopamine receptor antagonist</p>
    Formula:C23H27ClFN3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:431.93

    Ref: TM-T23381

  • Tiapride
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    Tiapride

    CAS:
    <p>Tiapride, an atypical neuroleptic, is a selective dopamine D2-receptor antagonist with varying IC50 values for D1-D4.</p>
    Formula:C15H24N2O4S
    Colore e forma:Solid
    Peso molecolare:328.43

    Ref: TM-T60943

  • Melitracen hydrochloride
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    Melitracen hydrochloride

    CAS:
    <p>Melitracen hydrochloride (Thymeol hydrochloride) , an antidepressant, is used as potential dopamine D1/2 receptor antagonist to treat depression.</p>
    Formula:C21H26ClN
    Purezza:99.99%
    Colore e forma:Crystalline Solid
    Peso molecolare:327.90

    Ref: TM-T4274

  • THIQ
    Targetmol
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    THIQ

    CAS:
    <p>THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).</p>
    Formula:C33H41ClN6O2
    Purezza:98.93%
    Colore e forma:Solid
    Peso molecolare:589.17

    Ref: TM-T8485

  • Betazole
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    Betazole

    CAS:
    <p>Betazole, an oral H2 receptor agonist, stimulates gastric acid and raises bile duct pressure, used for gastric secretory testing.</p>
    Formula:C5H9N3
    Colore e forma:Solid
    Peso molecolare:111.15

    Ref: TM-T72005

  • Siponimod
    Targetmol
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    Siponimod

    CAS:
    <p>Siponimod (BAF312) modulates S1P1/S1P5 with EC50s of 0.39/0.98 nM; &gt;1000x selectivity over S1P2-4.</p>
    Formula:C29H35F3N2O3
    Purezza:97.08% - 99.40%
    Colore e forma:Solid
    Peso molecolare:516.59

    Ref: TM-T6403

  • Nuciferine
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    Nuciferine

    CAS:
    <p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>
    Formula:C19H21NO2
    Purezza:98.76% - 99.79%
    Colore e forma:Solid
    Peso molecolare:295.38

    Ref: TM-T3369

  • Lys-Bradykinin acetate(342-10-9 free base)
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    Lys-Bradykinin acetate(342-10-9 free base)

    CAS:
    <p>Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.</p>
    Formula:C58H89N17O14
    Purezza:99.86%
    Colore e forma:Solid
    Peso molecolare:1248.43

    Ref: TM-TP2268L

  • Flibanserin hydrochloride
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    Flibanserin hydrochloride

    CAS:
    <p>Flibanserin HCl: oral 5-HT1A agonist &amp; 5-HT2A antagonist, Ki values 1 nM &amp; 49 nM, for HSDD, has antidepressant/anxiolytic properties.</p>
    Formula:C20H22ClF3N4O
    Colore e forma:Solid
    Peso molecolare:426.87

    Ref: TM-T62324

  • Talnetant
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    Talnetant

    CAS:
    <p>Talnetant (SB 223412) is a selective NK3 receptor antagonist that can penetrate the brain and modulate dopamine.</p>
    Formula:C25H22N2O2
    Purezza:97.88%
    Colore e forma:Solid
    Peso molecolare:382.45

    Ref: TM-T7549

  • Tesmilifene fumarate
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    Tesmilifene fumarate

    CAS:
    <p>Tesmilifene fumarate (DPPE fumarate) (DPPE fumarate) is an H1C receptor antagonist。</p>
    Formula:C23H29NO5
    Purezza:99.86%
    Colore e forma:Solid
    Peso molecolare:399.48

    Ref: TM-T22746

  • Dolasetron
    Targetmol
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    Dolasetron

    CAS:
    <p>Dolasetron (MDL-73147)(MDL-73147) is a serotonin 5-HT3 receptor antagonist. Dolasetron is used to treat nausea and vomiting following chemotherapy.</p>
    Formula:C19H20N2O3
    Purezza:99.84% - 99.86%
    Colore e forma:White Powder
    Peso molecolare:324.37

    Ref: TM-T4568

  • ESI-09
    Targetmol
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    ESI-09

    CAS:
    <p>ESI-09 is a new-typel noncyclic nucleotide EPAC antagonist.The IC50 values of ESI-09 for EPAC1 and EPAC2 is 3.2 and 1.4 μM, respectively.</p>
    Formula:C16H15ClN4O2
    Purezza:97.24% - 99.57%
    Colore e forma:Solid
    Peso molecolare:330.77

    Ref: TM-T2244

  • CCG-50014
    Targetmol
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    CCG-50014

    CAS:
    <p>CCG-50014 is a potent and selective inhibitor of RGS4 with IC50 of 30 nM.</p>
    Formula:C16H13FN2O2S
    Purezza:98.53%
    Colore e forma:Solid
    Peso molecolare:316.35

    Ref: TM-T6434

  • Dazoxiben
    Targetmol
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    Dazoxiben

    CAS:
    <p>Dazoxiben (UK-37248) is a potent inhibitor of thromboxane (TX) synthase</p>
    Formula:C12H13ClN2O3
    Purezza:99.99%
    Colore e forma:Solid
    Peso molecolare:268.7

    Ref: TM-T7968

  • AnaMorelin hydrochloride
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    AnaMorelin hydrochloride

    CAS:
    <p>AnaMorelin hydrochloride (RC-1291 hydrochloride) is a novel ghrelin receptor agonist(EC50 : 0.74 nM, in the FLIPR assay).</p>
    Formula:C31H43ClN6O3
    Purezza:99.18% - ≥98%
    Colore e forma:Solid
    Peso molecolare:583.16

    Ref: TM-T7225

  • CS 2100
    Targetmol
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    CS 2100

    CAS:
    <p>CS 2100 (1-[[4-Ethyl-5-[5-(4-phenoxyphenyl)-1,2,4-oxadiazol-3-yl]-2-thienyl]methyl]-3-azetidinecarboxylic acid) is an S1P1 agonist.</p>
    Formula:C25H23N3O4S
    Purezza:99.19%
    Colore e forma:Solid
    Peso molecolare:461.53

    Ref: TM-T22697