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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

Mostrare 19 più sottocategorie

Trovati 5838 prodotti di "Proteina G/GPCR"

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  • Betahistine mesylate
    Targetmol
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    Betahistine mesylate

    CAS:
    <p>Betahistine mesylate (Extovyl), an H1 agonist and vasodilator, treats Meniere's disease and vascular headaches; risks with asthma/ulcers.</p>
    Formula:C8H12N2·2(CH4O3S)
    Purezza:98% - 99.85%
    Colore e forma:Coa
    Peso molecolare:328.4

    Ref: TM-T0246L

  • BMY-14802
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    BMY-14802

    CAS:
    BMY-14802 (alpha-(4-fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazine butanol) is a selective and orally active sigma-1 antagonist with an IC50 of 112 nM.
    Formula:C18H22F2N4O
    Purezza:99.84%
    Colore e forma:Soild
    Peso molecolare:348.39

    Ref: TM-T67739

  • Logo CymitQuimica
    Targetmol
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    Calcitonin-13C6,15N4 TFA

    <p>Calcitonin-13CIC6,15NIC4(salmon) (Salmon calcitonin-13CIC6,15NIC4) TFA is a version of calcitonin(salmon) labeled with carbon-13 and nitrogen-15. This hormone regulates calcium and acts dualistically as an agonist to both amylin and calcitonin receptors, promoting bone formation while inhibiting bone resorption.</p>
    Formula:C1401C5H240N4315NO48S2·5C2HF3O2
    Colore e forma:Solid
    Peso molecolare:4007.93

    Ref: TM-T201476

  • Eledoisin
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    Eledoisin

    CAS:
    Eledoisin (Eledone peptide) is a specific agonist of NK2 and NK3 receptors.Eledoisin is an undecapeptide of mollusk origin, belonging to the tachykinin family
    Formula:C54H85N13O15S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1188.4

    Ref: TM-TP1177

  • Neurokinin A(4-10)
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    Neurokinin A(4-10)

    CAS:
    Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .
    Formula:C34H54N8O10S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:766.91

    Ref: TM-T7559

  • Logo CymitQuimica
    Targetmol
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    S1R agonist 2 hydrochloride

    Compound 8b hydrochloride, a selective S1R agonist, exhibits affinity with K i s of 1.1 nM for S1R and 88 nM for S2R.
    Formula:C21H28ClNO
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:345.91

    Ref: TM-T78087

  • Logo CymitQuimica
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    SLB1122168 formic

    SLB1122168 is a potent inhibitor of Spns2-mediated sphingosine-1-phosphate (S1P) release, exhibiting an IC50 value of 94 nM [1].
    Formula:C23H37N3O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:403.56

    Ref: TM-T78160

  • WAY-620645
    Targetmol
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    WAY-620645

    CAS:
    WAY-620645 is a CCK antagonist with antitumor and analgesic activities.
    Formula:C22H22N4O2
    Purezza:99.89%
    Colore e forma:Solid
    Peso molecolare:374.44

    Ref: TM-T9991

  • Edg-2 receptor inhibitor 1
    Targetmol
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    Edg-2 receptor inhibitor 1

    CAS:
    Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).
    Formula:C27H27NO5
    Purezza:99.47%
    Colore e forma:Solid
    Peso molecolare:445.51

    Ref: TM-T4521

  • L-796,778
    Targetmol
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    L-796,778

    CAS:
    <p>L-796,778 is an SST3 agonist and a selective ligand of SST3, which can increase the level of cAMP in the body.</p>
    Formula:C29H40N6O7
    Purezza:96.20%
    Colore e forma:Solid
    Peso molecolare:584.66

    Ref: TM-T32511

  • Logo CymitQuimica
    Targetmol
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    Survodutide TFA

    <p>Survodutide TFA (BI 456906 TFA) is a GCGR/GLP-1R dual agonist, a peptide compound used in obesity research.</p>
    Formula:C192H289N47O61·xC2HF3OC2
    Purezza:99.29% - 99.96%
    Colore e forma:Solid
    Peso molecolare:4231.62 (free base)

    Ref: TM-T78098

  • Dalcotidine
    Targetmol
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    Dalcotidine

    CAS:
    <p>Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, may lower relapse.</p>
    Formula:C18H29N3O2
    Purezza:99.11%
    Colore e forma:Solid
    Peso molecolare:319.44

    Ref: TM-T31195

  • N-Nitroso Atenolol
    Targetmol
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    N-Nitroso Atenolol

    CAS:
    N-Nitroso Atenolol is a derivative of Atenolol. At concentrations ranging from 0.1 to 1 mM, it induces DNA fragmentation in rat hepatocytes.
    Formula:C14H21N3O4
    Colore e forma:Solid
    Peso molecolare:295.33

    Ref: TM-T203130

  • (±)-9-Nor-9α-hydroxy Hexahydrocannabinol
    Targetmol
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    (±)-9-Nor-9α-hydroxy Hexahydrocannabinol

    CAS:
    (±)-9-Nor-9α-hydroxy Hexahydrocannabinol is a cannabinoid-structured compound that exhibits potent cannabinoid-like activity in both dogs and mice.
    Formula:C20H30O3
    Colore e forma:Solid
    Peso molecolare:318.45

    Ref: TM-T203604

  • Torososide B
    Targetmol
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    Torososide B

    CAS:
    Torososide B is an anti-allergic compound that inhibits leukotriene release from calcium ionophore A-stimulated rat peritoneal mast cells.
    Formula:C40H52O25
    Colore e forma:Solid
    Peso molecolare:932.83

    Ref: TM-T203084

  • CB2 receptor agonist 9
    Targetmol
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    CB2 receptor agonist 9

    CAS:
    CB2 receptor agonist 9 (Compound 33) is an orally active agonist of cannabinoid receptor 2 (CB2 receptor) with an EC50 of 16.2 nM. It inhibits the expression of TNF-α, IL-1β, and IL-6, demonstrating anti-inflammatory activity in a DSS-induced acute colitis model in mice.
    Formula:C16H23N3O2S
    Colore e forma:Solid
    Peso molecolare:321.44

    Ref: TM-T203517

  • SBI-810
    Targetmol
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    SBI-810

    CAS:
    SBI-810 is a functional selective β-arrestin-biased allosteric modulator of the neurotensin receptor 1 (NTSR1). In the presence of the endogenous ligand neurotensin (NT), SBI-810 regulates NTSR1 signaling through a G protein-specific mechanism. It fully antagonizes NT-induced Gq activation and partially antagonizes NT-induced Gi1 activation, allowing NTSR1 to activate GoA and G12.
    Formula:C27H34N4O2
    Colore e forma:Solid
    Peso molecolare:446.59

    Ref: TM-T203513

  • δ8-THC acetate
    Targetmol
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    δ8-THC acetate

    CAS:
    Delta8-THC acetate (Delta8-tetrahydrocannabinol) is a psychoactive cannabinoid that binds to the cannabinoid receptor 1 (CB1 receptor) and exhibits anti-nausea, appetite-stimulating, and anti-inflammatory effects. It may also offer neuroprotective benefits and has potential applications in research on anxiety and depression.
    Formula:C23H32O3
    Colore e forma:Solid
    Peso molecolare:356.5

    Ref: TM-T203037

  • Methamnetamine hydrochloride
    Targetmol
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    Methamnetamine hydrochloride

    CAS:
    Methamnetamine (PAL-1046) hydrochloride is a psychoactive substance derived from phenethylamine, known to cause excessive serotonin release.
    Formula:C14H18ClN
    Colore e forma:Solid
    Peso molecolare:235.75

    Ref: TM-T203312

  • Logo CymitQuimica
    Targetmol
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    AD353

    AD353 is a selective sigma-1 receptor ligand. It demonstrates high efficacy in models of capsaicin-induced allodynia and PGE2-induced mechanical hyperalgesia. Additionally, AD353 exhibits favorable pharmacokinetic properties.
    Formula:C23H30N2O2
    Colore e forma:Solid
    Peso molecolare:366.5

    Ref: TM-T203662