Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

Mostrare 19 più sottocategorie

Trovati 5838 prodotti di "Proteina G/GPCR"

Purezza (%)

100

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CB2 PET Radioligand 1
CB2 PET Radioligand 1 (compound [18F]9) is a positron emission tomography (PET) radioligand with high affinity for the human cannabinoid receptor 2 (hCB2, Ki=7.
Formula:C₂₀H₁₉F₃N₄O
Purezza:98%
Colore e forma:Solid
Peso molecolare:388.39
Ref: TM-T79577
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Dp[Tyr(methyl)2,Arg8]-Vasopressin
CAS:
- 67269-08-3
Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].
Formula:C₄₉H₇₀N₁₄O₁₂S₂
Purezza:98%
Colore e forma:Solid
Peso molecolare:1111.3
Ref: TM-T80073
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ACTH (7-38) (human)
CAS:
- 68563-24-6
ACTH (7-38) (human) is a fragment (7-38) of the full human adrenocorticotropic hormone (ACTH (1-39)), also referred to as corticotropin inhibitory peptide (CIP
Formula:C₁₆₇H₂₅₇N₄₇O₄₆
Purezza:98%
Colore e forma:Solid
Peso molecolare:3659.11
Ref: TM-T80125
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PSB-1114 triethylamine
PSB-1114 triethylamine is a potent, enzymatically stable, P2Y2 receptor agonist with a 134 nM EC50, exhibiting greater than 50-fold selectivity over P2Y4 (EC50
Formula:C₁₀H₁₅F₂N₃O₁₃P₃S·xC₆H₁₅N
Purezza:98%
Colore e forma:Solid
Ref: TM-T78080
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FFN246
CAS:
- 2210244-83-8
FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation and
Formula:C₁₅H₁₃FN₂O
Purezza:98%
Colore e forma:Solid
Peso molecolare:256.27
Ref: TM-T78684
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(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS:
- 176714-12-8
(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].
Formula:C₅₂H₇₆N₁₄O₁₁S₂
Purezza:98%
Colore e forma:Solid
Peso molecolare:1137.38
Ref: TM-T80137
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PD 144418 oxalate
CAS:
- 1794760-28-3
PD 144418 oxalate: σ1 receptor ligand, Ki=0.08 nM; 1377 nM for σ2, minimal affinity elsewhere; potential antipsychotic.
Formula:C₂₀H₂₄N₂O₅
Purezza:98.76%
Colore e forma:Solid
Peso molecolare:372.42
Ref: TM-T39211
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Picumeterol FA
picumeterol FA is a potent and selective β2-adrenergic receptor agonist.
Formula:C₂₂H₃₁Cl₂N₃O₄
Purezza:99.8%
Colore e forma:Soild
Peso molecolare:472.4
Ref: TM-T68129L1
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SSTR4 agonist-1
CAS:
- 1638588-92-7
SSTR4agonist-1 (Compound 47) is a selective agonist of the somatostatin receptor 4 (SSTR4), with an EC50 of 4.7 nM. It has a half-life of over 130 minutes in human liver microsomes.
Formula:C₁₆H₂₃N₃O₂
Colore e forma:Solid
Peso molecolare:289.37
Ref: TM-T203033
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Atrial natriuretic peptide (3-28) (human)
CAS:
- 102686-43-1
Atrial natriuretic peptide (3-28) (human) (ANP (3-28) (human)), a peptide hormone produced by the atrial myocardium, plays a critical role in the regulation of
Formula:C₁₁₈H₁₈₇N₄₃O₃₆S₃
Purezza:98%
Colore e forma:Solid
Peso molecolare:2880.21
Ref: TM-T80438
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RS 56812
CAS:
- 143137-37-5
RS 56812 is a 5-HT3 receptor antagonist and agonist used in the study of cognitive disorders.
Formula:C₁₈H₂₁N₃O₂
Purezza:99.38%
Colore e forma:Soild
Peso molecolare:311.38
Ref: TM-T23264L
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Lanerkitug
Lanerkitug is a humanized IgG1λ2 antibody that targets CCR8, with HumanIgG1lambda2, Isotype Control serving as its corresponding isotype control.
Colore e forma:Odour Liquid
Ref: TM-T9901A-352
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L-threo Lysosphingomyelin (d18:1)
CAS:
- 105615-55-2
L-threo Lysosphingomyelin, a natural S1P receptor agonist, has EC50s: 19.3 nM (hS1P1), 131.8 nM (hS1P3), 313.3 nM (hS1P2).
Formula:C₂₃H₄₉N₂O₅P
Colore e forma:Solid
Peso molecolare:464.62
Ref: TM-T38452
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Preclamol hydrochloride
CAS:
- 88768-67-6
Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.
Formula:C₁₄H₂₂ClNO
Colore e forma:Solid
Peso molecolare:255.78
Ref: TM-T73684
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CACPD2011a-0001278239
CAS:
- 1030781-08-8
CACPD2011a-0001278239 is a β2AR hybrid agonist with high affinity binding to both the wild-type and T164I β2AR variants. It exhibits neither cytotoxicity nor mutagenicity, making it suitable for asthma research.
Formula:C₂₁H₂₂N₄O₄
Colore e forma:Solid
Peso molecolare:394.42
Ref: TM-T203578
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Tienoxolol FA
Tienoxolol FA, a beta-blocker for treating heart disease, hypertension, and ischemia.
Formula:C₂₂H₃₀N₂O₇S
Purezza:97.05% - 98.53%
Colore e forma:Soild
Peso molecolare:466.55
Ref: TM-T68161L
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ACTH (3-24) (human, bovine, mouse, ovine, porcine, rabbit, rat)
CAS:
- 1036763-00-4
ACTH (3-24) is the fragment 3-24 of ACTH, used in disease research including cancer and immune disorders.
Formula:C₁₂₄H₁₉₆N₃₈O₂₇S
Colore e forma:Solid
Peso molecolare:2683.19
Ref: TM-T76500
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a-Helical Corticotropin Releasing Factor (9-41)
CAS:
- 99658-03-4
α-Helical CRF (9-41) is a CRF antagonist that lowers in vivo plasma GH levels.
Formula:C₁₆₆H₂₇₃N₄₅O₅₄S₂
Colore e forma:Solid
Peso molecolare:3827.34
Ref: TM-T76204
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Esmolol acid hydrochloride
CAS:
- 83356-60-9
Esmolol acid (ASL-8123) hydrochloride is a mild antagonist of β-adrenergic receptors. It inhibits the heart rate and diastolic pressure responses induced by Isoproterenol in a dose-dependent manner and is applicable for renal failure research.
Formula:C₁₅H₂₄ClNO₄
Colore e forma:Solid
Peso molecolare:317.81
Ref: TM-T203119
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Cannabidivarinic acid
CAS:
- 31932-13-5
Cannabidivarinic acid (CBDVA), the carboxylic acid precursor to cannabidivarin (CBDV), is a non-psychoactive cannabinoid found in Cannabis and known for its anti-inflammatory properties.
Formula:C₂₀H₂₆O₄
Colore e forma:Solid
Peso molecolare:330.42
Ref: TM-T203665