CymitQuimica logo
Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

Mostrare 18 più sottocategorie

Trovati 5378 prodotti di "Proteina G/GPCR"

Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
prodotti per pagina.
  • Neuropeptide FF
    Targetmol
    + Info

    Neuropeptide FF

    CAS:
    <p>Endogenous antiopioid peptide and agonist at NPFF1 and NPFF2 receptors (Ki values are 2.82 and 0.21 nM respectively).</p>
    Formula:C54H76N14O10
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1081.27

    Ref: TM-TP1074

  • Neuropeptide Y 13-36 (porcine)
    Targetmol
    + Info

    Neuropeptide Y 13-36 (porcine)

    CAS:
    <p>Neuropeptide Y 13-36 (porcine) is a selective neuropeptide Y2 receptor agonist.</p>
    Formula:C135H209N41O36
    Colore e forma:Solid
    Peso molecolare:2982.408

    Ref: TM-T36447

  • Vicasinabin
    Targetmol
    + Info

    Vicasinabin

    CAS:
    <p>Vicasinabin: potent CB2 agonist; researches chronic pain, atherosclerosis, bone mass, neuroinflammation.</p>
    Formula:C15H22N10O
    Colore e forma:Solid
    Peso molecolare:358.41

    Ref: TM-T38912

  • Logo CymitQuimica
    Targetmol
    + Info

    Colulintide

    CAS:
    <p>Colulintide is an analog of amylin, utilized in obesity research.</p>
    Colore e forma:Solid

    Ref: TM-TP3252

  • Adenosine receptor antagonist 1
    Targetmol
    + Info

    Adenosine receptor antagonist 1

    CAS:
    <p>A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.</p>
    Formula:C22H15ClFN7O
    Colore e forma:Solid
    Peso molecolare:447.86

    Ref: TM-T40307

  • Logo CymitQuimica
    Targetmol
    + Info

    Galanin-Like Peptide (porcine)

    CAS:
    <p>Galanin-Like Peptide (porcine) is a 60 amino acid neuropeptide originally isolated from the porcine hypothalamus.</p>
    Formula:C281H443N81O78
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:6204.02

    Ref: TM-T80145

  • Val9-Oxytocin
    Targetmol
    + Info

    Val9-Oxytocin

    CAS:
    <p>Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor.</p>
    Formula:C46H72N12O12S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1049.27

    Ref: TM-T80136

  • Dp[Tyr(methyl)2,Arg8]-Vasopressin
    Targetmol
    + Info

    Dp[Tyr(methyl)2,Arg8]-Vasopressin

    CAS:
    <p>Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].</p>
    Formula:C49H70N14O12S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1111.3

    Ref: TM-T80073

  • Osanetant
    Targetmol
    + Info

    Osanetant

    CAS:
    Osanetant produces anxiolytic- and antidepressant-like effects. Osanetant is a selective NK3 receptor antagonist. It is researched for schizophrenia.
    Formula:C35H41Cl2N3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:606.62

    Ref: TM-T16408

  • Logo CymitQuimica
    Targetmol
    + Info

    CB2 PET Radioligand 1

    <p>CB2 PET Radioligand 1 (compound [18F]9) is a positron emission tomography (PET) radioligand with high affinity for the human cannabinoid receptor 2 (hCB2, Ki=7.</p>
    Formula:C20H19F3N4O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:388.39

    Ref: TM-T79577

  • Logo CymitQuimica
    Targetmol
    + Info

    5-HT6R antagonist 1

    <p>Compound 8 (5-HT6R antagonist 1), a 5-HT6R antagonist (K i : 5 nM), not only demonstrates inhibition of platelet aggregation and excellent metabolic stability</p>
    Formula:C17H22F2N6O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:364.39

    Ref: TM-T79684

  • Logo CymitQuimica
    Targetmol
    + Info

    AD186

    <p>AD186, a potent and selective S1R agonist, exhibits dissociation constants (Kis) of 2.7 nM for S1R and 27 nM for S2R.</p>
    Formula:C22H28N2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:320.47

    Ref: TM-T78915

  • Logo CymitQuimica
    Targetmol
    + Info

    A3AR modulator 1

    <p>MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.</p>
    Formula:C23H25IN4
    Colore e forma:Solid
    Peso molecolare:484.38

    Ref: TM-T74993

  • (±)5(6)-EET
    Targetmol
    + Info

    (±)5(6)-EET

    CAS:
    <p>5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes.</p>
    Formula:C20H32O3
    Colore e forma:Solid
    Peso molecolare:320.473

    Ref: TM-T36070

  • (R)-(+)-Atenolol
    Targetmol
    + Info

    (R)-(+)-Atenolol

    CAS:
    <p>(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.</p>
    Formula:C14H22N2O3
    Purezza:98.72%
    Colore e forma:Solid
    Peso molecolare:266.34

    Ref: TM-T0007L

  • Logo CymitQuimica
    Targetmol
    + Info

    A3AR agonist 1

    <p>A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effective</p>
    Formula:C28H34N6O6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:550.61

    Ref: TM-T79372

  • Des-Arg9-[Leu8]-Bradykinin acetate
    Targetmol
    + Info

    Des-Arg9-[Leu8]-Bradykinin acetate

    CAS:
    <p>Des-Arg9-[Leu8]-Bradykinin acetate is a potent antagonist of the bradykinin receptor 1 (B1R), utilized in renal fibrosis research [1].</p>
    Formula:C43H67N11O12
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:930.06

    Ref: TM-T80072

  • Logo CymitQuimica
    Targetmol
    + Info

    Galanin-Like Peptide (rat)

    CAS:
    <p>Galanin-Like Peptide (rat), a neuropeptide comprising 60 amino acids, plays a crucial role in regulating feeding, body weight, and energy metabolism [1].</p>
    Formula:C288H461N87O83S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:6502.34

    Ref: TM-T80146

  • [Des-His1,Glu9]-Glucagon amide
    Targetmol
    + Info

    [Des-His1,Glu9]-Glucagon amide

    CAS:
    <p>Glucagon blocker with pA2 of 7.2; no agonist effect. Boosts insulin; prevents glucagon-driven hyperglycemia in rabbits and diabetic rats.</p>
    Formula:C148H221N41O47S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3358.68

    Ref: TM-TP2033

  • SB-408124
    Targetmol
    + Info

    SB-408124

    CAS:
    SB408124: Non-peptide, OX1 receptor antagonist, Ki 57 nM (whole cell) and 27 nM (membrane), 50x more selective than OX2.
    Formula:C19H18F2N4O
    Purezza:99.81%
    Colore e forma:Solid
    Peso molecolare:356.37

    Ref: TM-T6658