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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5352 prodotti di "Proteina G/GPCR"

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  • B-Raf IN 14
    Targetmol
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    B-Raf IN 14

    CAS:
    <p>B-Raf IN 14 is a BRAF inhibitor.</p>
    Formula:C15H14BrN5O3S
    Purezza:98.32%
    Colore e forma:Solid
    Peso molecolare:424.27

    Ref: TM-T72070

  • [Ala17]-MCH acetate
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    [Ala17]-MCH acetate

    <p>[Ala17]-MCH acetate is a selective ligand for MCHR1 with a Ki of 0.16 nM and Kd of 0.37 nM(Eu3+ chelate-labeled).</p>
    Formula:C99H159N29O28S4
    Purezza:98.92%
    Colore e forma:Solid
    Peso molecolare:2331.76

    Ref: TM-TP1997L

  • Orexin B, human
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    Orexin B, human

    CAS:
    <p>Orexin B, human agonizes Orexin receptors (OX1 Ki=420 nM, OX2 Ki=36 nM), promotes feeding in rats, and is a neuropeptide.</p>
    Formula:C123H212N44O35S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:2899.34

    Ref: TM-TP1139

  • Adrenocorticotropic Hormone (ACTH) (1-39), rat
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    Adrenocorticotropic Hormone (ACTH) (1-39), rat

    CAS:
    <p>ACTH (1-39), rat: potent MC2 agonist, forms fragments in vitro, isolated by HPLC, characterized by amino acids and NH2-terminus.</p>
    Formula:C210H315N57O57S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:4582.23

    Ref: TM-TP1249

  • Bombinakinin M acetate
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    Bombinakinin M acetate

    <p>Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and is</p>
    Formula:C102H163N31O26
    Purezza:99.80%
    Colore e forma:Solid
    Peso molecolare:2239.58

    Ref: TM-TP2075L

  • 5-OMe-UDP trisodium salt
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    5-OMe-UDP trisodium salt

    CAS:
    <p>Potent P2Y6 agonist</p>
    Formula:C10H16N2O13P2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:434.19

    Ref: TM-T22525

  • CB1R agonist 1
    Targetmol
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    CB1R agonist 1

    <p>CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.</p>
    Formula:C20H18F3N3O3S
    Colore e forma:Solid
    Peso molecolare:437.435

    Ref: TM-T206337

  • Cortistatin 14, human, rat acetate
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    Cortistatin 14, human, rat acetate

    <p>Cortistatin 14, human, rat acetate is a neuropeptide having structural similarity to somatostatin-14 and shows anticonvulsive, neuroprotective effects and</p>
    Formula:C80H112N18O19S2
    Purezza:97.86%
    Colore e forma:Solid
    Peso molecolare:1693.98

    Ref: TM-TP1188L

  • 4-Chloromethamphetamine hydrochloride
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    4-Chloromethamphetamine hydrochloride

    CAS:
    <p>4-Chloromethamphetamine hydrochloride is a novel psychoactive substance belonging to the amphetamine class.</p>
    Formula:C10H15Cl2N
    Colore e forma:Solid
    Peso molecolare:220.14

    Ref: TM-T203542

  • CB2R probe 1
    Targetmol
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    CB2R probe 1

    CAS:
    <p>CB2R Probe 1, a cannabinoid 2 receptor (CB2R) fluorescent probe, exhibits both safety and environmental friendliness, boasting a dissociation constant (K i) of</p>
    Formula:C36H42N4O4
    Colore e forma:Solid
    Peso molecolare:594.74

    Ref: TM-T74604

  • Dipentylone hydrochloride
    Targetmol
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    Dipentylone hydrochloride

    CAS:
    <p>Dipentylone hydrochloride (Bk-dmbdp HCl) is a psychoactive synthetic cathinone and sympathomimetic stimulant. Its inhibitory activity towards the dopamine transporter (IC50=0.233µM) is tenfold higher than that towards NET and SERT, inhibiting dopamine uptake and stimulating locomotor activity in mice.</p>
    Formula:C14H20ClNO3
    Purezza:99.94%
    Colore e forma:Solid
    Peso molecolare:285.77

    Ref: TM-T205977

  • Jatrorrhizine hydroxide
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    Jatrorrhizine hydroxide

    CAS:
    <p>Jatrorrhizine hydroxide: alkaloid from Coptis chinensis; neuroprotective, antimicrobial, antiplasmodial, antioxidant; AChE inhibitor, affects 5-HT/NE uptake.</p>
    Formula:C20H21NO5
    Colore e forma:Solid
    Peso molecolare:355.38

    Ref: TM-T75436

  • Azaline B
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    Azaline B

    CAS:
    <p>Azaline B is an antagonist of the gonadotropin-releasing hormone (GnRH), with an IC50 of 1.37 nM. It is utilized in research related to pathologies associated with sex hormones, ovulation induction, and male contraception.</p>
    Formula:C80H102ClN23O12
    Colore e forma:Solid
    Peso molecolare:1613.27

    Ref: TM-TP2707

  • VIP36
    Targetmol
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    VIP36

    <p>VIP36 is an agonist of the cannabinoid type 1 receptor (CB1) with analgesic properties. It reduces the recruitment of inhibitory proteins, thereby exerting its pain-relieving effects, and is applicable in research related to chronic pain.</p>
    Formula:C27H35FN6O4
    Colore e forma:Solid
    Peso molecolare:526.603

    Ref: TM-T206705

  • Logo CymitQuimica
    Targetmol
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    Cyclic AC253

    <p>Cyclic AC253 is an amylin receptor antagonist with an IC50 of 0.3 μM. It offers neuroprotective effects against Aβ toxicity and mitigates Aβ-induced impairments in hippocampal long-term potentiation. Additionally, Cyclic AC253 is capable of penetrating the blood-brain barrier.</p>
    Formula:C126H202N42O40S2
    Peso molecolare:3007.45049

    Ref: TM-TP3648

  • Logo CymitQuimica
    Targetmol
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    GRL018-21

    <p>GRL018-21 is a potent, highly selective inhibitor of G protein-coupled receptor kinase 5 (GRK5), exhibiting an IC50 of 10 nM [1].</p>
    Colore e forma:Odour Solid

    Ref: TM-T82258

  • LTD4 antagonist 2
    Targetmol
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    LTD4 antagonist 2

    CAS:
    <p>LTD4 antagonist 2 (compound 6) functions as a leukotriene D4 (LTD4) antagonist with an IC50 of 2.8 μM for the cysteinyl leukotriene 1 receptor (CysLT1R). Additionally, it acts as an agonist for the G protein-coupled bile acid receptor 1 (GPBAR1), making it applicable for research into colitis, metabolic syndrome, and other GPBAR1- and CysLT1R-related diseases.</p>
    Formula:C17H13NO3
    Colore e forma:Solid
    Peso molecolare:279.29

    Ref: TM-T203302

  • INCB 3284 dimesylate
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    INCB 3284 dimesylate

    CAS:
    <p>INCB 3284 dimesylate: oral CCR2 antagonist, blocks MCP-1/hCCR2 binding (IC50: 3.7 nM), potential in acute liver failure research.</p>
    Formula:C28H39F3N4O10S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:712.76

    Ref: TM-T11647

  • Logo CymitQuimica
    Targetmol
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    Imelciment

    CAS:
    <p>Imelciment (REGN-9035) is a humanised monoclonal antibody targeting NPR1, which can be used for research into heart failure.</p>
    Purezza:95%
    Colore e forma:Soild

    Ref: TM-T9901A-366

  • BIIE-0246
    Targetmol
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    BIIE-0246

    CAS:
    <p>BIIE-0246 is a potent and highly selective non-peptide neuropeptide Y (NPY) Y2 receptor antagonist. With an IC50 of 15 nM.</p>
    Formula:C49H57N11O6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:896.05

    Ref: TM-T14572