Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(939 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.945 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(148 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(407 prodotti)
- Recettore dell'endotelina(76 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(31 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(165 prodotti)
- Proteina Hedgehog/Smoothened(44 prodotti)
- Recettore dell'istamina(358 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(297 prodotti)
- PAFR(11 prodotti)
- PKA(48 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5352 prodotti di "Proteina G/GPCR"
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TSHR antagonist S37
CAS:<p>TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).</p>Formula:C25H20N2O3S2Purezza:98.35%Colore e forma:SolidPeso molecolare:460.57NF-56-EJ40 hydrochloride
CAS:<p>NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.</p>Formula:C27H31Cl2N3O3Purezza:99.33%Colore e forma:SoildPeso molecolare:516.46UCM-1306
CAS:<p>UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive function in PD.</p>Formula:C14H14FNO2SPurezza:99.98%Colore e forma:SoildPeso molecolare:279.33MP-A08
CAS:<p>MP-A08 selectively inhibits SPHK1; targets SphK1 & SphK2 with Ki of 6.9 μM & 27 μM, respectively.</p>Formula:C27H25N3O4S2Purezza:97.44%Colore e forma:SolidPeso molecolare:519.64YNT-185
CAS:<p>YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,</p>Formula:C33H37N5O5SPurezza:99.67%Colore e forma:SolidPeso molecolare:615.74Zolmitriptan
CAS:<p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>Formula:C16H21N3O2Purezza:99.69% - 99.91%Colore e forma:White Or Kind Of White PowderPeso molecolare:287.36Urocortin (rat) acetate
<p>Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.</p>Purezza:97.76%Colore e forma:SoildPalonosetron hydrochloride
CAS:<p>Palonosetron hydrochloride (RS 25259) is a 5-HT3 antagonist used in the prevention and treatment of chemotherapy-induced nausea and vomiting.</p>Formula:C19H24N2O·HClPurezza:99.84% - 99.92%Colore e forma:White SolidPeso molecolare:332.87Sonepcizumab
CAS:<p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>Purezza:SDS-PAGE:95% SEC-HPLC:98.90%Colore e forma:LiquidPeso molecolare:146.43 kDaFosopamine(HCl)
CAS:<p>Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.</p>Formula:C9H15ClNO5PPurezza:99.84%Colore e forma:SolidPeso molecolare:283.65Buflomedil hydrochloride
CAS:<p>Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.</p>Formula:C17H26ClNO4Purezza:99.7% - 99.91%Colore e forma:White Or Off-White Crystalline PowderPeso molecolare:343.85Granisetron hydrochloride
CAS:<p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>Formula:C18H25ClN4OPurezza:99.88% - 99.93%Colore e forma:White To Off-White Crystalline SolidPeso molecolare:348.87p-MPPI hydrochloride
CAS:<p>p-MPPI hydrochloride is a selective antagonist of 5-HT1A receptor, and has antidepressant and anxiolytic-like effects.</p>Formula:C25H28ClIN4O2Purezza:99.95%Colore e forma:SolidPeso molecolare:578.87Rimonabant hydrochloride
CAS:<p>Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂， Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。</p>Formula:C22H22Cl4N4OPurezza:98.24% - 99.5%Colore e forma:Off-White To White Crystalline PowderPeso molecolare:500.25Acetophenazine dimaleate
CAS:<p>Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.</p>Formula:C31H37N3O10SPurezza:99.39% - 99.48%Colore e forma:SolidPeso molecolare:643.71Ramelteon
CAS:<p>Ramelteon (TAK-375) is a Melatonin Receptor Agonist. The mechanism of action of ramelteon is as a Melatonin Receptor Agonist.</p>Formula:C16H21NO2Purezza:97.21% - 99.92%Colore e forma:Crystalline SolidPeso molecolare:259.342',5'-Dideoxyadenosine
CAS:<p>2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).</p>Formula:C10H13N5O2Purezza:99.55%Colore e forma:White SolidPeso molecolare:235.24Ketotifen fumarate
CAS:<p>Ketotifen fumarate (HC 20511 fumarate) is a cycloheptathiophene blocker of histamine H1 receptors and release of inflammatory mediators.</p>Formula:C23H23NO5SPurezza:99.25% - 99.73%Colore e forma:SolidPeso molecolare:425.50Terazosin hydrochloride
CAS:<p>Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.</p>Formula:C19H26ClN5O4Purezza:99.69% - 99.91%Colore e forma:SolidPeso molecolare:423.89PF429242 dihydrochloride
CAS:<p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>Formula:C25H37Cl2N3O2Purezza:99.68%Colore e forma:SolidPeso molecolare:482.49Indacaterol maleate
CAS:<p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>Formula:C28H32N2O7Purezza:99.03% - 99.67%Colore e forma:SolidPeso molecolare:508.56Terbutaline Sulfate
CAS:Terbutaline Sulfate (Terbutaline hemisulfate) is a selective beta-2 adrenergic agonist used as a bronchodilator and tocolytic.Formula:C12H19NO3H2SO4Purezza:99.47% - 99.94%Colore e forma:Crystalline PowderPeso molecolare:274.32Agomelatine
CAS:<p>Agomelatine (Valdoxan), like melatonin, boosts mood by targeting melatonin and 5-HT2C receptors.</p>Formula:C15H17NO2Purezza:99.92%Colore e forma:White SolidPeso molecolare:243.3LCKLSL hydrochloride
<p>LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.</p>Formula:C30H58ClN7O8SPurezza:98.02% - 99.31%Colore e forma:SolidPeso molecolare:712.34Nylidrin hydrochloride
CAS:<p>Nylidrin HCl inhibits IgG1-induced histamine release in guinea pigs and IgE-induced release in rat mast cells & human basophils.</p>Formula:C19H26ClNO2Purezza:99.35%Colore e forma:SolidPeso molecolare:335.87Isoxsuprine hydrochloride
CAS:<p>Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.</p>Formula:C18H24ClNO3Purezza:99.38%Colore e forma:Crystals From Water SolidPeso molecolare:337.84Dopexamine hydrochloride
CAS:<p>Dopexamine hydrochloride (FPL60278AR) is a β2-adrenoceptor agonist that modulates inflammation and protects organs without affecting hemodynamics.</p>Formula:C22H34Cl2N2O2Purezza:98.55%Colore e forma:SolidPeso molecolare:429.42PF-5190457
CAS:<p>PF-5190457 is an effective and selective ghrelin receptor inverse agonist (pKi: 8.36).</p>Formula:C29H32N6OSPurezza:99.34%Colore e forma:SolidPeso molecolare:512.67Ifenprodil
CAS:<p>Ifenprodil (RC61-91) inhibits NMDA receptor subunits GluN1 & GluN2B, GIRK channels, and affects alpha1, serotonin, sigma receptors.</p>Formula:C21H27NO2Purezza:99.58%Colore e forma:White Crystalline PowderPeso molecolare:325.44Promethazine hydrochloride
CAS:<p>Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.</p>Formula:C17H20N2S·HClPurezza:99.85%Colore e forma:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecolare:320.882-Bromo-6-methoxynaphthalene
CAS:<p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>Formula:C11H9BrOPurezza:98.51%Colore e forma:White To Off-White PowderPeso molecolare:237.09Ketanserin
CAS:<p>Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.</p>Formula:C22H22FN3O3Purezza:99.19% - 99.73%Colore e forma:SolidPeso molecolare:395.43Prucalopride
CAS:<p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these receptors.</p>Formula:C18H26ClN3O3Purezza:>99.99%Colore e forma:SolidPeso molecolare:367.87Terlipressin Acetate
CAS:<p>Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).</p>Formula:C56H82N16O19S2Purezza:98.50% - 99.69%Colore e forma:SolidPeso molecolare:1347.5Venlafaxine hydrochloride
CAS:<p>Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.</p>Formula:C17H28ClNO2Purezza:97.32% - 99.86%Colore e forma:White Crystalline PowderPeso molecolare:313.86Fluparoxan hydrochloride
CAS:<p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>Formula:C10H11ClFNO2Purezza:99.98%Colore e forma:SoildPeso molecolare:231.65Chlorprothixene hydrochloride
CAS:<p>Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.</p>Formula:C18H18ClNS·HClPurezza:99.76%Colore e forma:White PowderPeso molecolare:352.32JP1302 dihydrochloride
CAS:<p>JP1302 dihydrochloride: selective α2C-adrenoceptor antagonist; Ki=28 nM, Kb=16 nM.</p>Formula:C24H26Cl2N4Purezza:99.61%Colore e forma:SolidPeso molecolare:441.4Talastine
CAS:<p>Talastine is an antihistamine compound that can induce an allergic rash.</p>Formula:C19H21N3OPurezza:98.50% - 99.44%Colore e forma:SolidPeso molecolare:307.39CP-809101 hydrochloride
CAS:<p>CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).</p>Formula:C15H18Cl2N4OPurezza:99.5%Colore e forma:SolidPeso molecolare:341.24Methyldopa
CAS:<p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>Formula:C10H13NO4Purezza:98.95% - 99.86%Colore e forma:Less Or Almost Colorless Crystals Or White To Yellowish-White FinePeso molecolare:211.21Fenspiride hydrochloride
CAS:<p>Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.</p>Formula:C15H20N2O2·HClPurezza:99.64% - 99.92%Colore e forma:SolidPeso molecolare:296.79Timonacic
CAS:<p>Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.</p>Formula:C4H7NO2SPurezza:99.99%Colore e forma:SolidPeso molecolare:133.17Amiselimod hydrochloride
CAS:<p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>Formula:C19H31ClF3NO3Purezza:99.55%Colore e forma:SolidPeso molecolare:413.9Alverine citrate
CAS:<p>Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.</p>Formula:C26H35NO7Purezza:98.53% - 99.43%Colore e forma:CoaPeso molecolare:473.57Dexpramipexole dihydrochloride
CAS:<p>Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine</p>Formula:C10H19Cl2N3SPurezza:99.75% - 99.88%Colore e forma:SolidPeso molecolare:284.25Filorexant
CAS:<p>Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki <3 nM).</p>Formula:C24H25FN4O2Purezza:98.88%Colore e forma:SolidPeso molecolare:420.48Pemirolast potassium
CAS:<p>Pemirolast potassium, a pyrimidinone antiallergic, blocks antigen-induced Ca²⁺ influx in mast cells.</p>Formula:C10H7KN6OPurezza:98.91% - 99.63%Colore e forma:Crystals From Dimethylformamide Crystalline SolidPeso molecolare:266.31Clonidine hydrochloride
CAS:<p>Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.</p>Formula:C9H10Cl3N3Purezza:99.16% - 99.86%Colore e forma:SolidPeso molecolare:266.55Cyproheptadine hydrochloride sesquihydrate
CAS:<p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>Formula:C21H24ClNOPurezza:99.77% - >99.99%Colore e forma:White To Slightly Yellowish Crystalline SolidPeso molecolare:341.88Cericlamine
CAS:<p>Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.</p>Formula:C12H17Cl2NOPurezza:99.38%Colore e forma:SolidPeso molecolare:262.18Silodosin
CAS:<p>Silodosin (KAD 3213) is an alpha-Adrenergic Blocker. The mechanism of action of silodosin is as an Adrenergic alpha-Antagonist.</p>Formula:C25H32F3N3O4Purezza:99.282% - 99.76%Colore e forma:Colorless To Pink SolidPeso molecolare:495.53Ondansetron hydrochloride dihydrate
CAS:<p>Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.</p>Formula:C18H19N3O·HCl·2H2OPurezza:99.92%Colore e forma:White Crystal PowderPeso molecolare:365.86Rimonabant
CAS:<p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>Formula:C22H21Cl3N4OPurezza:98% - 99.91%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:463.79Adrenalone hydrochloride
CAS:<p>Adrenalone HCl: α1-adrenoceptor agonist, topical hemostatic, vasoconstrictor, prolongs local anesthesia.</p>Formula:C9H11NO3·HClPurezza:99.94%Colore e forma:SolidPeso molecolare:217.65Ro 10-5824 dihydrochloride
CAS:<p>Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).</p>Formula:C17H22Cl2N4Purezza:99.79%Colore e forma:SolidPeso molecolare:353.29Fluoxetine hydrochloride
CAS:<p>Fluoxetine HCl (Lilly110140), a selective serotonin reuptake inhibitor (SSRI), is an antidepressant with fewer side effects.</p>Formula:C17H19ClF3NOPurezza:99.6% - 99.98%Colore e forma:White To Off-White Crystalline Solid White To Off-White PowderPeso molecolare:345.787Carvedilol EP IMpurity E
CAS:<p>Carvedilol EP IMpurity E (Carvedilol USP E) is used as a pharmaceutical intermediate.</p>Formula:C9H14ClNO2Purezza:99.53%Colore e forma:White To Almost White Solid CrystallinePeso molecolare:203.666Azacyclonol
CAS:<p>Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.</p>Formula:C18H21NOPurezza:99.46%Colore e forma:Solid PowderPeso molecolare:267.37Ciliobrevin D
CAS:<p>Ciliobrevin D is a AAA+ ATPase motor cytoplasmic dynein inhibitor.</p>Formula:C17H8Cl3N3O2Purezza:98.09%Colore e forma:SolidPeso molecolare:392.62Pamabrom
CAS:<p>Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.</p>Formula:C11H18BrN5O3Purezza:99.84% - >99.99%Colore e forma:CoaPeso molecolare:348.2ALLO-2
CAS:<p>ALLO-2 is a Inhibitor of Drug-Resistant Smo Mutant.It inhibits Smo agonist Hh-Ag1.5-induced luciferase expression in TM3-Gli-Luc cells with IC50 of 6 nM.</p>Formula:C18H12F3N5OPurezza:99.19%Colore e forma:SolidPeso molecolare:371.32Fezolinetant
CAS:<p>Fezolinetant (ESN-364) is a neurokinin-3 receptor antagonist that is being investigated for menopausal hot flashes.Cost-effective and quality-assured.</p>Formula:C16H15FN6OSPurezza:98.62% - 99.7%Colore e forma:SolidPeso molecolare:358.39Orphenadrine hydrochloride
CAS:<p>Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.</p>Formula:C18H23NO·HClPurezza:99.88%Colore e forma:Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)Peso molecolare:305.85Talipexole dihydrochloride
CAS:<p>Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and</p>Formula:C10H17Cl2N3SPurezza:99.89%Colore e forma:Light Yellow SolidPeso molecolare:282.23GTS-21 dihydrochloride
CAS:<p>GTS-21 dihydrochloride (DMBX-anabaseine) is a nAChRs agonist. nAChRs are neuron receptor proteins that activated by the binding of the neurotransmitter ACh.</p>Formula:C19H20N2O2·2HClPurezza:98.54% - >99.99%Colore e forma:SolidPeso molecolare:381.3Roluperidone
CAS:<p>Roluperidone (CYR-101) is a novel cyclic amide derivative.</p>Formula:C22H23FN2O2Purezza:96.46% - 97.77%Colore e forma:SolidPeso molecolare:366.43INCB-9471
CAS:<p>INCB-9471 is a CCR5 antagonist with anti-HIV activity and inhibits the interaction between HIV-1 gp120.</p>Formula:C30H40F3N5O2Purezza:98.80%Colore e forma:SolidPeso molecolare:559.666Nepafenac
CAS:<p>Nepafenac (AHR 9434) is an NSAID that acts as a cyclooxygenase inhibitor.</p>Formula:C15H14N2O2Purezza:98.94% - 99.43%Colore e forma:SolidPeso molecolare:254.28Paroxetine hydrochloride
CAS:<p>Paroxetine hydrochloride (Paroxetine HCl) is a serotonin uptake inhibitor that is effective in the treatment of depression.</p>Formula:C19H21ClFNO3Purezza:98% - 99.99%Colore e forma:White Crystalline PowderPeso molecolare:365.826Efloxate
CAS:<p>Efloxate (Angorlisin), a vasodilator, is utilized in the treatment of chronic coronary insufficiency.</p>Formula:C19H16O5Purezza:99.66%Colore e forma:SolidPeso molecolare:324.33Enrasentan
CAS:<p>Enrasentan (sb-217242) is a mixed antagonist of ET(A) and ET(B) receptors that reduces blood pressure and protects myocardial function.</p>Formula:C29H30O8Purezza:97.9% - 98.39%Colore e forma:SolidPeso molecolare:506.54Risperidone
CAS:<p>Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.</p>Formula:C23H27FN4O2Purezza:99.73%Colore e forma:Crystalline SolidPeso molecolare:410.48SR59230A
CAS:<p>SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).</p>Formula:C23H29NO6Purezza:98.84%Colore e forma:SolidPeso molecolare:415.48Aniracetam
CAS:<p>Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.</p>Formula:C12H13NO3Purezza:99.88% - 99.89%Colore e forma:White Crystalline Or Crystalline PowdePeso molecolare:219.24HJC0197
CAS:<p>HJC0197 is a selective Epac antagonist; blocks cAMP-induced activation with IC50=5.9 μM for Epac2.</p>Formula:C19H21N3OSPurezza:98.05%Colore e forma:SolidPeso molecolare:339.45JNJ-39758979
CAS:<p>JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).</p>Formula:C11H19N5Purezza:98.33% - 99.62%Colore e forma:SolidPeso molecolare:221.3Terbutaline
CAS:<p>Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite of bambuterol</p>Formula:C12H19NO3Purezza:99.12%Colore e forma:SolidPeso molecolare:225.3RS102895 hydrochloride
CAS:<p>RS102895 hydrochloride is a potent antagonist of CCR2(IC50 of 360 nM).</p>Formula:C21H22ClF3N2O2Purezza:98.95%Colore e forma:SolidPeso molecolare:426.86Relamorelin
CAS:<p>Relamorelin(BIM28131, RM131) is a selective and potent ghrelin/growth hormone secretagogue receptor (GHSR) agonist.Cost-effective and quality-assured.</p>Formula:C43H50N8O5SPurezza:99.26% - >99.99%Colore e forma:SolidPeso molecolare:790.97AM-8123
CAS:<p>AM-8123: oral APJ agonist, potent, inhibits cAMP, activates Gα, key for cardiovascular research.</p>Formula:C27H33N7O5SPurezza:99.59% - 99.76%Colore e forma:SolidPeso molecolare:567.66Ranitidine Hydrochloride
CAS:<p>Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.</p>Formula:C13H23ClN4O3SPurezza:99.30% - 99.49%Colore e forma:SolidPeso molecolare:350.86Perphenazine
CAS:<p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>Formula:C21H26ClN3OSPurezza:99.3% - 99.99%Colore e forma:SolidPeso molecolare:403.97Sarizotan 2HCl
CAS:<p>Sarizotan 2HCl is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant effects for the study of Parkinsonian movement disorders.</p>Formula:C22H23Cl2FN2OPurezza:98.83%Colore e forma:SoildPeso molecolare:421.34Molindone hydrochloride
CAS:<p>Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.</p>Formula:C16H24N2O2·HClPurezza:99% - 99.99%Colore e forma:SolidPeso molecolare:312.84ONC206
CAS:<p>ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations and</p>Formula:C23H22F2N4OPurezza:99.38% - 99.81%Colore e forma:SolidPeso molecolare:408.44Maprotiline hydrochloride
CAS:<p>Maprotiline hydrochloride (Psymion) is a tetracyclic antidepressant akin to tricyclics with similar side effects.</p>Formula:C20H24ClNPurezza:99.68% - 99.84%Colore e forma:White PowderPeso molecolare:313.864Vapreotide acetate
CAS:<p>Vapreotide acetate (BMY-41606 acetate) is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM).</p>Formula:C59H74N12O11S2Purezza:99.89%Colore e forma:SolidPeso molecolare:1191.42Evocalcet
CAS:<p>Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).</p>Formula:C24H26N2O2Purezza:98.88% - 99.68%Colore e forma:SolidPeso molecolare:374.48Sertraline hydrochloride
CAS:<p>Sertraline hydrochloride (Sertraline HCl) is a selective serotonin uptake inhibitor that is used in the treatment of depression.</p>Formula:C17H18Cl3NPurezza:99.12% - 99.89%Colore e forma:Solid PowderPeso molecolare:342.691Clomipramine hydrochloride
CAS:<p>Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the liver.</p>Formula:C19H23ClN2·HClPurezza:99.04% - 99.47%Colore e forma:White To Slightly Yellow Crystalline PowderPeso molecolare:351.31(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid
CAS:<p>(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.</p>Formula:C20H29N3O8Purezza:99.72%Colore e forma:SoildPeso molecolare:439.46Naftifine hydrochloride
CAS:<p>Naftifine HCl: synthetic antifungal; inhibits squalene epoxidase, disrupting fungal cell sterol synthesis.</p>Formula:C21H22ClNPurezza:98.75% - 99.84%Colore e forma:SolidPeso molecolare:323.86Amp579 TFA
<p>Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.</p>Formula:C24H29ClF3N5O5SPurezza:96.56%Colore e forma:SoildPeso molecolare:592.03Dynarrestin
CAS:<p>Dynarrestin inhibits cytoplasmic dynein 1/2, preventing microtubule sliding without affecting ATP hydrolysis or ciliogenesis.</p>Formula:C22H23F2N3O2SPurezza:99.64%Colore e forma:SolidPeso molecolare:431.5Trimipramine maleate
CAS:<p>Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.</p>Formula:C24H30N2O4Purezza:99.47%Colore e forma:SolidPeso molecolare:410.51Tetrabenazine
CAS:<p>Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.</p>Formula:C19H27NO3Purezza:98% - 99.91%Colore e forma:White To Off-White White To Off-White SolidPeso molecolare:317.42Tolamolol
CAS:<p>Tolamolol is a selective β-adrenergic blocker that significantly reduces the degree of exercise-induced inhibition of the S-T segment and can be used in the</p>Formula:C19H24N2O4Purezza:98.59%Colore e forma:SolidPeso molecolare:344.4Ritodrine hydrochloride
CAS:<p>Ritodrine hydrochloride (NSC 291565), a phenethylamine derivative, reduces uterine contractions by increasing cAMP and decreasing calcium in myometrial cells.</p>Formula:C17H21NO3·HClPurezza:99% - 99.52%Colore e forma:SolidPeso molecolare:323.82Imidazolidinyl urea
CAS:<p>Imidazolidinyl urea (Imidurea) is an antimicrobial preservative used in cosmetics.</p>Formula:C11H16N8O8Purezza:98.6%Colore e forma:White Fluid Powder With Slight Characteristic OdorPeso molecolare:388.29Asenapine Maleate
CAS:<p>Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.</p>Formula:C21H20ClNO5Purezza:99.28%Colore e forma:SolidPeso molecolare:401.84Atomoxetine hydrochloride
CAS:<p>Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.</p>Formula:C17H22ClNOPurezza:99.86%Colore e forma:White SolidPeso molecolare:291.82Rebamipide
CAS:<p>Rebamipide (OPC12759) is a drug enhancing gastric defense by stimulating COX2, prostaglandins, and mucus, while reducing TNF alpha and free radicals.</p>Formula:C19H15ClN2O4Purezza:99.48% - 99.61%Colore e forma:White PowderPeso molecolare:370.79(S)-(-)-Atenolol
CAS:<p>(S)-(-)-Atenolol has beta-adrenergic blocking effects.</p>Formula:C14H22N2O3Purezza:99.31% - 99.81%Colore e forma:SolidPeso molecolare:266.34Amitriptyline hydrochloride
CAS:<p>Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive</p>Formula:C20H24ClNPurezza:97% - 99.94%Colore e forma:Crystals White To Off-White PowderPeso molecolare:313.86Metaraminol tartrate
CAS:<p>Metaraminol tartrate (Metaradrine tartrate) is a sympathomimetic agent that acts predominantly at alpha-1 adrenergic receptors.</p>Formula:C13H19NO8Purezza:99.68%Colore e forma:White PowderPeso molecolare:317.29PF-4348235 2HCl
<p>PF-4348235 2HCl is an adrenergic agonist and muscarinic receptor antagonist, and is a bronchodilator.</p>Formula:C36H51Cl3N4O7SPurezza:99.85%Colore e forma:SolidPeso molecolare:790.24Carteolol hydrochloride
CAS:<p>Carteolol hydrochloride is a nonselective beta-blocker used to treat hypertension, arrhythmias, angina, and glaucoma.</p>Formula:C16H24N2O3·HClPurezza:99.84% - 99.91%Colore e forma:SolidPeso molecolare:328.83Glycerol phenylbutyrate
CAS:<p>Glycerol phenylbutyrate (HPN-100) (GPB) is a new generation ammonia scavenger drug and it also is a sigma-2 (σ2) receptor ligand (pKi: 8.02).</p>Formula:C33H38O6Purezza:98.54% - 99.74%Colore e forma:SolidPeso molecolare:530.65Clozapine
CAS:<p>Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.</p>Formula:C18H19ClN4Purezza:99.91% - 99.93%Colore e forma:Yellow Crystals From Acetone-Petroleum Ether SolidPeso molecolare:326.82Strontium ranelate
CAS:<p>Strontium ranelate (S12911), a strontium (II) salt of the ranelic acid, is a medication for osteoporosis and can slow the course of osteoarthritis of the knee.</p>Formula:C12H6N2O8S·2SrPurezza:98.97%Colore e forma:Crystalline SolidPeso molecolare:513.49Triprolidine hydrochloride monohydrate
CAS:Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.Formula:C19H25ClN2OPurezza:99.68% - 99.81%Colore e forma:White Crystalline PowderPeso molecolare:332.87Promethazine
CAS:<p>Promethazine (Proazamine) is an analogue of anti-glaucoma prostaglandin (PG) .</p>Formula:C17H20N2SPurezza:99.76%Colore e forma:CrystalsPeso molecolare:284.42CCX140
CAS:<p>CCX140 (CCX140-B) (CCX140-B) is an antagonist of CCR2.</p>Formula:C20H13ClF3N5O3SPurezza:99.66% - 99.95%Colore e forma:SolidPeso molecolare:495.86CCR2-RA-[R]
CAS:<p>CCR2-RA-[R] is a C-C chemokine receptor type 2 (CCR2) allosteric antagonist (IC50: 103 nM).</p>Formula:C18H19ClFNO3Purezza:99.7%Colore e forma:SolidPeso molecolare:351.8Tirzepatide monosodium salt
<p>Tirzepatide sodium salt (LY3298176 sodium salt) is a GIP and GLP-1 receptor agonist with neuroprotective activity and can be used to treat obesity.</p>Formula:C225H347N48O68NaPurezza:99.69%Colore e forma:SoildPeso molecolare:4835.51GANT 58
CAS:<p>GANT 58 (NSC-75503) is a potent antagonist of Gli. Which inhibits GLI1-induced transcription (IC50: 5 μM).</p>Formula:C24H16N4SPurezza:99.53%Colore e forma:SolidPeso molecolare:392.48Isoprenaline hydrochloride
CAS:<p>Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac stimulating properties.</p>Formula:C11H18ClNO3Purezza:98% - 99.65%Colore e forma:Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)Peso molecolare:247.719Fenoterol
CAS:Fenoterol is an agonist of β2-adrenergic receptor It is classed as sympathomimetic beta agonist and asthma medication.Formula:C17H21NO4Purezza:98.29%Colore e forma:SolidPeso molecolare:303.35Aripiprazole Lauroxil
CAS:<p>Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.</p>Formula:C36H51Cl2N3O4Purezza:99.64%Colore e forma:SolidPeso molecolare:660.71CYM50308
CAS:<p>CYM50308 is a high affinity agonist of sphingosine-1-phosphate receptor 4 (S1P4-R) (EC50: 56 nM).</p>Formula:C20H21F2N3O2SPurezza:99.43% - 99.77%Colore e forma:SolidPeso molecolare:405.46Olopatadine hydrochloride
CAS:<p>Olopatadine hydrochloride (ALO4943A) is an antihistamine with mast-cell stabilizing properties used as eye drops in the treatment of ALLERGIC CONJUNCTIVITIS.</p>Formula:C21H23NO3·HClPurezza:99.62% - 99.64%Colore e forma:White SolidPeso molecolare:373.87PF-04995274
CAS:<p>PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.</p>Formula:C23H32N2O6Purezza:99.52%Colore e forma:SolidPeso molecolare:432.51Tolazoline hydrochloride
CAS:<p>Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonary</p>Formula:C10H13ClN2Purezza:99.67%Colore e forma:Pale Yellow Crystalline SolidPeso molecolare:196.68Pipamperone
CAS:<p>Pipamperone (McN-JR 3345) binds 5-HT2A closely as receptor.</p>Formula:C21H30FN3O2Purezza:99.85%Colore e forma:White PowderPeso molecolare:375.48Prasugrel
CAS:<p>Prasugrel (CS-747) is a piperazine derivative and PLATELET AGGREGATION INHIBITOR that is used to prevent THROMBOSIS in patients with ACUTE CORONARY SYNDROME;</p>Formula:C20H20FNO3SPurezza:99.62% - 99.82%Colore e forma:White SolidPeso molecolare:373.44Capeserod
CAS:<p>Capeserod is a potential 5-HT4 receptor (5-hydroxytryptamine receptor 4) agonist for the study of digestive disorders and neurological disorders.</p>Formula:C23H25ClN4O4Purezza:98.10% - 99.94%Colore e forma:SolidPeso molecolare:456.92Mianserin hydrochloride
CAS:<p>Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.</p>Formula:C18H21ClN2Purezza:99.63% - 99.82%Colore e forma:White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film CoatedPeso molecolare:300.83ML-109
CAS:<p>ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)</p>Formula:C31H29N3O5Purezza:98.63%Colore e forma:SolidPeso molecolare:523.58Mirtazapine
CAS:<p>Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.</p>Formula:C17H19N3Purezza:99.98%Colore e forma:SolidPeso molecolare:265.35Doxylamine succinate
CAS:<p>Doxylamine Succinate is a pyridine derivate histamine H1 antagonist with pronounced sedative properties.</p>Formula:C21H28N2O5Purezza:99.61%Colore e forma:5 1 (Ntp 1992)Peso molecolare:388.46Nicergoline
CAS:<p>Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with vascular origins.</p>Formula:C24H26BrN3O3Purezza:98% - 99.80%Colore e forma:SolidPeso molecolare:484.39Ogerin
CAS:<p>Ogerin: GPR68 modulator, blocks mice fear recall, A2A inverse agonist/antagonist (Ki 220 nM), weak 5-HT2B antagonist (Ki 736 nM).</p>Formula:C17H17N5OPurezza:99.5% - 99.75%Colore e forma:SolidPeso molecolare:307.35NS-2028
CAS:<p>NS-2028 is a selective sGC inhibitor, affecting both basal and NO-activated activities; used in nitric oxide research.</p>Formula:C9H5BrN2O3Purezza:99.44%Colore e forma:A Crystalline SolidPeso molecolare:269.05Domperidone
CAS:<p>Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.</p>Formula:C22H24ClN5O2Purezza:98% - 99.82%Colore e forma:SolidPeso molecolare:425.91EMPA
CAS:<p>EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nM</p>Formula:C23H26N4O4SPurezza:99.11%Colore e forma:SolidPeso molecolare:454.54Ziprasidone
CAS:<p>Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.</p>Formula:C21H21ClN4OSPurezza:99.55%Colore e forma:Tan SolidPeso molecolare:412.94Carboprost tromethamine
CAS:<p>Carboprost tromethamine, a synthetic 15-methyl analogue of prostaglandin F2α, effectively promotes uterine contractions and significantly reduces bleeding</p>Formula:C25H47NO8Purezza:>99.99%Colore e forma:SolidPeso molecolare:489.64Doxofylline
CAS:<p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>Formula:C11H14N4O4Purezza:99.958% - >99.99%Colore e forma:SolidPeso molecolare:266.25Iloperidone
CAS:<p>Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.</p>Formula:C24H27FN2O4Purezza:99.42%Colore e forma:SolidPeso molecolare:426.48Chlorpheniramine maleate
CAS:<p>Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.</p>Formula:C20H23ClN2O4Purezza:99.64% - 99.98%Colore e forma:Odorless White Crystalline Solid Or White Powder With A Bitter TastePeso molecolare:390.87[Leu15]-Gastrin I, human
CAS:<p>[Leu15]-Gastrin I, human is a variant of Gastrin I, modulating the binding of cholecystokinin to mucosal membranes.</p>Formula:C98H126N20O31Purezza:98.02% - 98.84%Colore e forma:SolidPeso molecolare:2080.16Carbazochrome sodium sulfonate
CAS:<p>Carbazochrome sodium sulfonate (AC-17) (AC-17) is an antihemorrhagic for the treatment of hemorrhoids.</p>Formula:C10H11N4NaO5SPurezza:99.63%Colore e forma:Orange Yellow Crystalline PowderPeso molecolare:322.03(R)-Terazosin
CAS:<p>R-Terazosin is the active R-enantiomer and potent α1-adrenoceptor antagonist (Ki: α1a 6.51 nM, α1b 1.01 nM, α1d 1.97 nM).</p>Formula:C19H25N5O4Purezza:98.87% - 98.96%Colore e forma:SolidPeso molecolare:387.43Luzindole
CAS:<p>Luzindole (N-0774) is a selective melatonin receptor antagonist.</p>Formula:C19H20N2OPurezza:98.53%Colore e forma:Off-White Amorphous SolidPeso molecolare:292.37Desvenlafaxine
CAS:<p>Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.</p>Formula:C16H25NO2Purezza:99.46% - 99.81%Colore e forma:White Crystalline PowderPeso molecolare:263.38Lintopride HCl
CAS:<p>Lintopride HCl is a 5HT-4 antagonist.</p>Formula:C14H20Cl2N4O2Purezza:98.42% - 98.81%Colore e forma:SoildPeso molecolare:347.24Mirabegron
CAS:<p>Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.</p>Formula:C21H24N4O2SPurezza:99.64%Colore e forma:Light Yellow To Yellow SolidPeso molecolare:396.51YT 146
CAS:<p>YT 146 is a biochemical.</p>Formula:C18H25N5O4Purezza:98.81% - 99.25%Colore e forma:SolidPeso molecolare:375.42Quipazine dimaleate
CAS:<p>Quipazine dimaleate is a selective 5-HT3 agonist.</p>Formula:C21H23N3O8Purezza:>99.99%Colore e forma:SolidPeso molecolare:445.42Leronlimab
CAS:<p>Leronlimab (PRO 140), a humanized IgG4 monoclonal antibody, targets CCR5 to combat HIV and cancer.</p>Purezza:SDS-PAGE:95.0%;SEC-HPLC:99.6%Colore e forma:LiquidPeso molecolare:146.66 kDaOzagrel
CAS:<p>Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of</p>Formula:C13H12N2O2Purezza:97.90% - 99.38%Colore e forma:White PowderPeso molecolare:228.25Alprenolol
CAS:<p>Alprenolol (Alpheprol) is a non-selective β-adrenergic receptor (β-AR) antagonist that is also an antagonist of the serotonin (5-HT) receptor subtypes 5-HT1A</p>Formula:C15H23NO2Purezza:99.72% - 99.78%Colore e forma:SolidPeso molecolare:249.35Olodaterol
CAS:Olodaterol is a novel, long-acting beta2-adrenergic agonist (LABA) that exerts its pharmacological effect by binding and activating beta2-adrenergic receptorsFormula:C21H26N2O5Purezza:98.9%Colore e forma:SolidPeso molecolare:386.45Evatanepag
CAS:<p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>Formula:C25H28N2O5SPurezza:97.09%Colore e forma:SolidPeso molecolare:468.57Tropisetron hydrochloride
CAS:<p>Tropisetron hydrochloride (Tropisetron HCl) is a selective, competitive serotonin 5-HT3 receptor antagonist, with antinauseant and antiemetic activities.</p>Formula:C17H21ClN2O2Purezza:99.72% - 99.83%Colore e forma:SolidPeso molecolare:320.82Loxapine succinate
CAS:<p>Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.</p>Formula:C22H24ClN3O5Purezza:99.69%Colore e forma:White To Of-White SolidPeso molecolare:445.9Clopidogrel
CAS:<p>Clopidogrel (SR-25990C), a P2Y12 receptor antagonist, decreases platelet aggregation.</p>Formula:C16H16ClNO2SPurezza:98.23% - 98.83%Colore e forma:White PowderPeso molecolare:321.82Pericyazine
CAS:<p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>Formula:C21H23N3OSPurezza:99.61%Colore e forma:SolidPeso molecolare:365.49Avexitide acetate
CAS:<p>Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.</p>Formula:C155H246N40O53SPurezza:96.64% - 98.65%Colore e forma:SolidPeso molecolare:3549.91Amisulpride
CAS:<p>Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the US.</p>Formula:C17H27N3O4SPurezza:99.97%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:369.48Mebhydrolin napadisylate
CAS:<p>Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic</p>Formula:C19H20N2C10H8O6S2Purezza:99.35% - 99.96%Colore e forma:White Or Almost White CrystallinePeso molecolare:420.52DSP-4 hydrochloride
CAS:<p>DSP-4 hydrochloride is a neurotoxin that degrades noradrenergic neurons in rats and crosses the blood-brain barrier.</p>Formula:C11H16BrCl2NPurezza:99.9%Colore e forma:SolidPeso molecolare:313.06Heptaminol hydrochloride
CAS:<p>Heptaminol hydrochloride (RP-2831 hydrochloride), a vasoconstrictor, is used in the therapy of hypotension, especially orthostatic hypotension.</p>Formula:C8H20ClNOPurezza:98.61%Colore e forma:White Crystalline PowderPeso molecolare:181.71CI 169369
CAS:<p>CI 169369 is a selective 5-HT2 receptor antagonist used in the study of anxiety and depression.</p>Formula:C19H21ClN2SPurezza:98.97%Colore e forma:SoildPeso molecolare:344.9Iobenguane sulfate
CAS:<p>Iobenguane sulfate is used in radioiodinated form to diagnose and treat adrenergic tumors.</p>Formula:C8H10IN3H2O4SPurezza:99.04%Colore e forma:SolidPeso molecolare:324.12Moxonidine
CAS:<p>Moxonidine (BDF5895) is a selective agonist at the imidazoline receptor subtype 1, acting as an antihypertensive drug.</p>Formula:C9H12ClN5OPurezza:99.81% - 99.94%Colore e forma:CrystalPeso molecolare:241.68N6-Ethyladenosine
CAS:<p>N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).</p>Formula:C12H17N5O4Purezza:99.96%Colore e forma:SolidPeso molecolare:295.29GR 103691
CAS:<p>GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).</p>Formula:C30H35N3O3Purezza:98.94% - 99.29%Colore e forma:SolidPeso molecolare:485.62CB1 antagonist 2
CAS:<p>CB1 antagonist 2 (AM4113) is caimabinoid 1 (CB1) antagonist which inhibits CB1 in vivo with an IC50 of 25.5 nM.</p>Formula:C17H12Cl3N3OPurezza:99.75%Colore e forma:SolidPeso molecolare:380.66Romergoline 2HCl
<p>Romergoline 2HCl is a D1 agonist and D2 antagonist used in the study of Parkinson's disease.</p>Formula:C20H24Cl2N4O2Purezza:99.01% - 99.40%Colore e forma:SoildPeso molecolare:423.34Flunarizine dihydrochloride
CAS:<p>Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.</p>Formula:C26H28Cl2F2N2Purezza:99.53% - 99.89%Colore e forma:White Crystalline Powder Odorless And TastelessPeso molecolare:477.42Seganserin
CAS:<p>Seganserin, a 5-HT2 antagonist, negates fluoxetine and quipazine's effects on hyperphagia, depression, and pain.</p>Formula:C29H27F2N3OPurezza:99.22%Colore e forma:SolidPeso molecolare:471.54DF-1012 FA
<p>DF-1012 FA is a structural analog of DF-1012, a neuropeptide inhibitor used in the study of asthma and cough.</p>Formula:C17H22N4O3Purezza:99.15% - 99.97%Colore e forma:SolidPeso molecolare:330.382SEP-363856 hydrochloride
CAS:<p>SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.</p>Formula:C9H14ClNOSPurezza:99.86% - 99.99%Colore e forma:SolidPeso molecolare:219.73Quetiapine hemifumarate
CAS:Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Formula:C46H54N6O8S2Purezza:99.32% - >99.99%Colore e forma:White Crystalline SolidPeso molecolare:883.09Frovatriptan succinate hydrate
CAS:<p>Frovatriptan treats all migraine types, nausea, vomiting, light/sound sensitivity, and prevents menstrual migraines; it targets 5-HT1B/D and 5-HT7 receptors.</p>Formula:C18H25N3O6Purezza:99.66%Colore e forma:SolidPeso molecolare:379.41Phenoxybenzamine hydrochloride
CAS:<p>Phenoxybenzamine hydrochloride: non-selective, irreversible alpha-blocker; antihypertensive, vasodilator, may cause tachycardia, potential carcinogen.</p>Formula:C18H23Cl2NOPurezza:98.04% - >99.99%Colore e forma:Antihypertensive DrugPeso molecolare:340.3Tipepidine hydrochloride
CAS:<p>Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.</p>Formula:C15H18ClNS2Purezza:99.97%Colore e forma:SolidPeso molecolare:311.89Bisoprolol hemifumarate
CAS:Bisoprolol, a selective beta-1 adrenergic receptor antagonist, selectively and competitively binds to and blocks beta-1 adrenergic receptors in the heart,Formula:C20H33NO6Purezza:98.69% - 99.84%Colore e forma:White To Offf-White PowderPeso molecolare:383.49Cloperastine hydrochloride
CAS:<p>Cloperastine hydrochloride (HT-11 hydrochloride) is a type of flavonoid.</p>Formula:C20H25Cl2NOPurezza:97.74% - 99.42%Colore e forma:SolidPeso molecolare:366.33Nardeterol HCl
<p>Nardeterol HCl is a β-adrenergic receptor partial agonist used in the study of the central nervous system.CAS 번호13460-73-83-4</p>Formula:C20H25ClFN3O2Purezza:97.72% - 98.65%Colore e forma:SoildPeso molecolare:393.88MK-0812 Succinate
CAS:<p>MK-0812 Succinate is an effective and selective CCR2 antagonist.</p>Formula:C28H40F3N3O7Purezza:98.62% - 99.93%Colore e forma:SolidPeso molecolare:587.63Retatrutide sodium salt
<p>Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study of type 2 diabetes mellitus.</p>Purezza:99.97%Colore e forma:SoildJ-113863
CAS:<p>J-113863 is also a potent antagonist of the human CCR3 (IC50 of 0.58 nM) , but a weak antagonist of the mouse CCR3 (IC50 of 460 nM).</p>Formula:C30H37Cl2IN2O2Purezza:95.11%Colore e forma:SolidPeso molecolare:655.44Degarelix acetate(214766-78-6 free base)
CAS:<p>Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .</p>Formula:C84H107ClN18O18Purezza:98.66%Colore e forma:SolidPeso molecolare:1692.34(±) Clopidogrel hydrogen sulfate
CAS:<p>(±) Clopidogrel hydrogen sulfate (Iscover) , an antiplatelet agent pharmacologically and structurally analogous to ticlopidine, is used to inhibit blood clots</p>Formula:C16H16ClNO2S·H2SO4Purezza:98.67% - 99.04%Colore e forma:Colorless To Light Yellow LiquidPeso molecolare:419.9SB 258585
CAS:<p>SB 258585: Selective 5-HT6 antagonist, binds human receptors, used in cognitive and antipsychotic assays.</p>Formula:C18H22IN3O3SPurezza:99.8%Colore e forma:SoildPeso molecolare:487.36H4R antagonist 3
CAS:<p>H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R antagonist 3 has potential inflammatory activity for the study of</p>Formula:C19H21ClN4SPurezza:98%Colore e forma:SolidPeso molecolare:372.92CB2R/FAAH modulator-2
CAS:<p>CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH.</p>Formula:C24H33NO2Purezza:99.15%Colore e forma:SoildPeso molecolare:367.52Galantide acetate
<p>Galantide acetate, a non-specific galanin receptor antagonist, is a peptide consisting of fragments of galanin and substance P.</p>Formula:C106H155N25O28SPurezza:97.8% - 97.91%Colore e forma:SolidPeso molecolare:2259.58[18F]-Labeled L-dopa precursor
CAS:<p>[18F]-Labeled L-dopa precursor is a precursor for synthesis of 18F-labeled L-dopa[1].</p>Formula:C35H36N2O7Colore e forma:SolidPeso molecolare:596.67Des His1, Glu8 Exendin-4
<p>Des His1, Glu8 Exendin-4 is a glucagon-like peptide-1 receptor (GLP1R) antagonist that regulates blood glucose and is used in the study of diabetes and obesity.</p>Formula:C179H277N47O59SPurezza:99.92%Colore e forma:SolidPeso molecolare:4063.46Setmelanotide
CAS:<p>Setmelanotide (BIM-22493) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).</p>Formula:C49H68N18O9S2Purezza:98%Colore e forma:SolidPeso molecolare:1117.31GIP/GLP-1 dual receptor agonist-1
CAS:<p>Compound 4: GIP/GLP-1 agonist for metabolic/fatty liver disease research.</p>Colore e forma:SolidCGRP 8-37 (rat)
CAS:<p>CGRP 8-37 (rat) is a CGRP receptor antagonist, a CGRP fragment with potential anti-injury effects that induces arterial relaxation.</p>Formula:C138H224N42O41Purezza:99.28%Colore e forma:SolidPeso molecolare:3127.51Oxmetidine
CAS:<p>Oxmetidine (SKF 92994) is an H2R antagonist that inhibits transmembrane calcium flux in the cardiovascular system and is used in the study of duodenal ulcers.</p>Formula:C19H21N5O3SPurezza:99.67%Colore e forma:SolidPeso molecolare:399.47SLB1122168 formic
<p>SLB1122168 is a potent inhibitor of Spns2-mediated sphingosine-1-phosphate (S1P) release, exhibiting an IC50 value of 94 nM [1].</p>Formula:C23H37N3O3Purezza:98%Colore e forma:SolidPeso molecolare:403.56S1R agonist 2 hydrochloride
<p>Compound 8b hydrochloride, a selective S1R agonist, exhibits affinity with K i s of 1.1 nM for S1R and 88 nM for S2R.</p>Formula:C21H28ClNOPurezza:98%Colore e forma:SolidPeso molecolare:345.91Calcitonin-13C6,15N4 TFA
<p>Calcitonin-13CIC6,15NIC4(salmon) (Salmon calcitonin-13CIC6,15NIC4) TFA is a version of calcitonin(salmon) labeled with carbon-13 and nitrogen-15. This hormone regulates calcium and acts dualistically as an agonist to both amylin and calcitonin receptors, promoting bone formation while inhibiting bone resorption.</p>Formula:C1401C5H240N4315NO48S2·5C2HF3O2Colore e forma:SolidPeso molecolare:4007.93
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