Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(939 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.945 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(148 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(407 prodotti)
- Recettore dell'endotelina(76 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(31 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(165 prodotti)
- Proteina Hedgehog/Smoothened(44 prodotti)
- Recettore dell'istamina(358 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(297 prodotti)
- PAFR(11 prodotti)
- PKA(48 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
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Trovati 5352 prodotti di "Proteina G/GPCR"
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[Ala1,3,11,15]-Endothelin
CAS:<p>Selective ETB endothelin receptor agonist (IC50 values are 0.33 and 2200 nM for displacing [125I]-ET-1 from ETB and ETA receptors respectively).</p>Formula:C109H163N25O32SPurezza:98%Colore e forma:SolidPeso molecolare:2368Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
CAS:<p>Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), acts as a weak agonist at the antidiuretic receptor but is a potent</p>Formula:C45H63N15O11S2Colore e forma:SolidPeso molecolare:1054.21Pexopiprant
CAS:<p>Pexopiprant, a potent oral antagonist of the prostaglandin D2 receptor 2 (DP2) with a K i value less than 100nM, is a valuable compound for asthma research.</p>Formula:C21H17Cl2F2NO4Colore e forma:SolidPeso molecolare:456.27P2Y14R antagonist 3
<p>P2Y14R antagonist 3 (compound A) is an orally active P2Y14R antagonist with an IC50 of 23.60 nM and a Kd of 7.26 μM. It mitigates lung injury in mice induced by Lipopolysaccharides (LPS) and can be utilized in the study of inflammatory diseases.</p>Formula:C26H25N5O5Colore e forma:SolidPeso molecolare:487.51CB2R agonist 3
<p>CB2R agonist 3, a potent activator of cannabinoid receptor 2 (CB2R), exhibits an EC50 value of 0.37μM, indicative of its significant role in the immune system [</p>Purezza:98%Colore e forma:Odour SolidPROTAC(H-PGDS)-8
CAS:<p>PROTAC(H-PGDS)-8 is a PROTAC degrader targeting Hematopoietic prostaglandin D synthase (H-PGDS), exhibiting an IC50 of 0.14 μM [1].</p>Formula:C41H40N8O7Colore e forma:SolidPeso molecolare:756.81Angiopeptin TFA
CAS:Angiopeptin TFA: somatostatin analogue, sst2/sst5 partial agonist (IC50: 0.26/6.92 nM), suppresses GH & IGF-1, for atherosclerosis research.Formula:C58H73F6N11O14S2Colore e forma:SolidPeso molecolare:1326.39Piperulin A
CAS:<p>Piperulin A effectively inhibits platelet-activating factor receptor (PAFR) by specifically blocking its binding to isolated rabbit platelet plasma membranes,</p>Formula:C23H28O6Colore e forma:SolidPeso molecolare:400.46Somatostatin-28 (1-14)
CAS:<p>Somatostatin-28 (1-14) is a truncated neuropeptide from prosomatostatin cleavage.</p>Formula:C61H105N23O21SPurezza:98%Colore e forma:SolidPeso molecolare:1528.71LCKLSL acetate
<p>LCKLSL acetate is a potent AnxA2 inhibitor, blocking tPA binding and plasmin production, with anti-angiogenic effects.</p>Formula:C32H61N7O10SPurezza:99.9%Colore e forma:SolidPeso molecolare:735.93RC-3095 TFA
CAS:<p>RC-3095 TFA (RC-3095 (TFA)) is a bombesin/gastrin-releasing peptide (BN/GRP) antagonist with potential anticancer activity.</p>Formula:C58H80F3N15O11Purezza:98%Colore e forma:SolidPeso molecolare:1220.34Cagrilintide acetate
<p>.Cagrilintide is a long-acting amylin analog,treat diabetes and obesity by reducing appetite through activation of the AMY3R and calcitonin receptor.</p>Formula:C196H316N54O61S2Purezza:99.88%Colore e forma:SolidPeso molecolare:4469.06Edg-2 receptor inhibitor 1
CAS:<p>Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).</p>Formula:C27H27NO5Purezza:99.47%Colore e forma:SolidPeso molecolare:445.51[D-Trp34]-Neuropeptide Y
CAS:<p>Potent NPY Y5 receptor agonist (pEC50 = 7.82); highly selective; induces hyperphagia, body weight gain; orally active.</p>Formula:C196H289N55O56Purezza:98%Colore e forma:SolidPeso molecolare:4311.77[D-Phe12,Leu14]-Bombesin
CAS:<p>Bombesin receptor blocker; stops binding in rat brain (IC50=2 μM), hinders amylase release (IC50=4 μM), reduces appetite suppression in vivo.</p>Formula:C77H113F3N22O20Purezza:98%Colore e forma:SolidPeso molecolare:1724.9Phenylethanolamine A
CAS:<p>Phenylethanolamine A is a β-adrenergic agonist and a byproduct of the Ractopamine synthesis process.</p>Formula:C19H24N2O4Colore e forma:SolidPeso molecolare:344.40LUF6096
CAS:<p>LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically while</p>Formula:C22H21Cl2N3OPurezza:99.5%Colore e forma:SolidPeso molecolare:414.33CCK (26-30) (sulfated)
CAS:<p>CCK (26-30) is a digestive and satiety-related peptide fragment inhibiting [125I]CCK-33 binding by 10% at 0.1 mM.</p>Formula:C33H41N7O12S2Colore e forma:SolidPeso molecolare:791.85Satavaptan
CAS:<p>Satavaptan is a vasopressin V2 receptor antagonist. Satavaptan improves the control of ascites in cirrhosis.</p>Formula:C33H45N3O8SColore e forma:SolidPeso molecolare:643.79VVZ-149
<p>VVZ-149 is an antagonist of both serotonin receptor 2A (5HT2A) and glycine transporter type 2 (GlyT2), with potential anti-nociceptive activity.</p>Colore e forma:SolidFR167344 free base
CAS:<p>FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.</p>Formula:C30H28BrCl2N5O4Purezza:98%Colore e forma:SolidPeso molecolare:673.38Misoprostol
CAS:<p>Misoprostol, a prostaglandin E1 derivative, has a strong inhibitory effect on gastric acid secretion, while having a contractile effect on pregnancy.</p>Formula:C22H38O5Purezza:99.78%Colore e forma:Water-Soluble Viscous LiquidPeso molecolare:382.53Galantide acetate
<p>Galantide acetate, a non-specific galanin receptor antagonist, is a peptide consisting of fragments of galanin and substance P.</p>Formula:C106H155N25O28SPurezza:97.8% - 97.91%Colore e forma:SolidPeso molecolare:2259.58Atrial natriuretic peptide (3-28) (human)
CAS:<p>Atrial natriuretic peptide (3-28) (human) (ANP (3-28) (human)), a peptide hormone produced by the atrial myocardium, plays a critical role in the regulation of</p>Formula:C118H187N43O36S3Purezza:98%Colore e forma:SolidPeso molecolare:2880.21CB2R/FAAH modulator-2
CAS:<p>CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH.</p>Formula:C24H33NO2Purezza:99.15%Colore e forma:SoildPeso molecolare:367.52Cortistatin-8 acetate
<p>Cortistatin-8 acetate: synthetic corticosteroid analog, GHS-R antagonist; doesn't affect acyl GH release or hesperidin response.</p>Formula:C49H72N12O11S2Purezza:99.01%Colore e forma:SoildPeso molecolare:1069.3PEN (rat)
CAS:<p>PEN (rat) is an Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.</p>Formula:C102H169N27O33Purezza:98%Colore e forma:SolidPeso molecolare:2301.62γ-Glu-Abu TFA
<p>Gamma-Glu-AbuTFA is the TFA salt form of Gamma-Glu-Abu. This compound acts as an agonist for the calcium sensing receptor (CaSR), activating CaSR in HEK-293 cells with an EC50 of 0.21 μM.</p>Formula:C11H17F3N2O7Colore e forma:SolidPeso molecolare:346.26Conessine hydrobromide
CAS:<p>Conessine hydrobromide is a naturally occurring steroid alkaloid and has been used in traditional herbal medicine as a treatment for amoebic dysentery.</p>Formula:C24H41BrN2Colore e forma:SolidPeso molecolare:437.51Boc-Phe-Leu-Phe-Leu-Phe
CAS:<p>Boc-Phe-Leu-Phe-Leu-Phe is a chemotactic peptide antagonist that inhibits the release of peptide leukotrienes induced by FMLP.</p>Formula:C44H59N5O8Colore e forma:SolidPeso molecolare:785.97Muscarinic toxin 3
CAS:<p>Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57</p>Formula:C319H489N89O97S8Purezza:98%Colore e forma:SolidPeso molecolare:7379.35Luseogliflozin hydrate
CAS:<p>Luseogliflozin hydrate: SGLT2 inhibitor, IC50 2.26 nM, oral, for type 2 diabetes research.</p>Formula:C23H32O7SColore e forma:SolidPeso molecolare:452.56RXFP3/4 agonist 1
CAS:<p>RXFP3/4 agonist 1 is a relaxin family peptide 3/4 receptor (RXFP3/4) agonist(EC50s of 82/2 nM, respectivley).</p>Formula:C20H22ClN5OPurezza:98%Colore e forma:SolidPeso molecolare:383.88M40
CAS:<p>Potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in rat</p>Formula:C94H145N23O24Purezza:98%Colore e forma:SolidPeso molecolare:1981.338-iso Prostaglandin E2
CAS:<p>"8-iso PGE2: Isoprostane from arachidonic acid, potent rat renal vasoconstrictor, reduces GFR and renal flow by 80%, no BP effect."</p>Formula:C20H32O5Colore e forma:SolidPeso molecolare:352.47Vapitadine
CAS:<p>Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.</p>Formula:C17H20N4OPurezza:99.77% - 99.86%Colore e forma:SoildPeso molecolare:296.371a,1b-dihomo Prostaglandin E1
CAS:<p>1a,1b-dihomo Prostaglandin E1 is a class of prostaglandin compounds.</p>Formula:C22H38O5Colore e forma:SolidPeso molecolare:382.541Galcanezumab
CAS:<p>Galcanezumab: humanized IgG4 antibody that targets CGRP for migraine and cluster headache prevention/treatment.</p>Purezza:> 95%Colore e forma:LiquidPeso molecolare:144.08 kDa4-Hydroxy MET
CAS:4-Hydroxy MET (4-HO-MET) is a tryptamine-based new psychoactive substance (NPS), structurally similar to the endogenous neurotransmitter serotonin. It has hallucinogenic properties that affect mood, movement, and cognitive functions.Formula:C13H18N2OColore e forma:SolidPeso molecolare:218.3NPC 567 acetate
<p>NPC 567 acetate is a bradykinin B2 antagonist and can be used in studies about the treatment of allergic airway disease.</p>Formula:C62H91N19O15Purezza:97.72%Colore e forma:SolidPeso molecolare:1342.5Urocortin II, human TFA
<p>hUcn II, a CRF family member, targets CRF2 receptor, has time-linked stress regulation effects, showing mild motor suppression and delayed anxiolytic action.</p>Formula:C196H340F3N63O56SPurezza:98%Colore e forma:SolidPeso molecolare:4564.3UCM 549
CAS:<p>UCM 549 is a bioactive chemical.</p>Formula:C19H21NO2Colore e forma:SolidPeso molecolare:295.38FSCPX
CAS:<p>FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.</p>Formula:C23H27FN4O6SPurezza:98%Colore e forma:SolidPeso molecolare:506.55Seglitide acetate
CAS:<p>Seglitide acetate (MK-678) is a selective agonist of sst2 somatostatin receptor.</p>Formula:C46H60N8O9Purezza:98.87%Colore e forma:SolidPeso molecolare:869.02BAM(8-22) TFA
<p>BAM(8-22) TFA activates Mrgprs, induces mouse scratching, and is a proenkephalin A derivative.</p>Formula:C93H128F3N25O25SColore e forma:SolidPeso molecolare:2085.22GFB-024
<p>GFB-024 is a humanized antibody targeting CB1, which can be used to study obesity.</p>Colore e forma:LiquidPeso molecolare:145.5kDaECPLA
CAS:<p>ECPLA is an LSD analog and a potent 5-HT2A agonist (EC50 of 14.6 nM), capable of stimulating Gq-mediated calcium flux. It exhibits high affinity for most serotonin receptors, α2-adrenergic receptors, and D2-like dopamine receptors.</p>Formula:C21H25N3OColore e forma:SolidPeso molecolare:335.44α-MSH TFA
CAS:<p>α-Melanocyte-stimulating hormone (α-MSH) is a 13-amino acid peptide hormone produced by post-translational processing of proopiomelanocortin (POMC) in the</p>Formula:C79H110F3N21O21SColore e forma:SolidPeso molecolare:1778.93K1-70
<p>K1-70 is a humanized antibody targeting TSHR, used in the study of autoimmune diseases and endocrine disorders.</p>Colore e forma:LiquidPeso molecolare:145.5kDa(+)-OSU 6162
CAS:<p>(+)-OSU 6162 (Piperidine, 3-[3-(methylsulfonyl)phenyl]-1-propyl-, (3R)-) is an agonist of 5-HT Receptor with anti-Alzheimer and antidepressant activities.</p>Formula:C15H23NO2SPurezza:98.19%Colore e forma:SoildPeso molecolare:281.41SR-140603
CAS:<p>SR-140603, the less potent enantiomer of SR 140333, is used as the negative control.</p>Formula:C37H45Cl3N2O2Purezza:98%Colore e forma:SolidPeso molecolare:656.12ANQ-11125 TFA
<p>ANQ-11125 TFA is a motilin antagonist with a pKd of 8.24, inhibiting motilide contractions in rabbits.</p>Formula:C88H126F3N19O23Colore e forma:SolidPeso molecolare:1875.05α-Helical CRF(9-41)
CAS:<p>Corticotropin-releasing factor receptor antagonist (Ki values are 17, 5 and 0.97 at human CRF1, rat CRF2α and mouse CRF2β receptors respectively).</p>Formula:C166H274N46O53S2Purezza:98%Colore e forma:SolidPeso molecolare:3827K-(D-1-Nal)-FwLL-NH2 TFA
<p>K-(D-1-Nal)-FwLL-NH2 TFA: potent ghrelin inverse agonist; Ki=4.9 nM (COS7), 31 nM (HEK293T); blocks Gq/G13 signaling.</p>Formula:C53H68F3N9O8Colore e forma:SolidPeso molecolare:1016.16Antisauvagine-30 TFA
<p>aSvg-30 TFA: potent CRF2 receptor antagonist, Kd 1.4 nM (mCRFR2β), 150 nM (CRFR1).</p>Formula:C163H275N48F3O49SColore e forma:SolidPeso molecolare:3764.28Peptide 401
CAS:<p>Peptide 401: AMP from bee/wasp venom, triggers histamine release, reduces paw swelling.</p>Formula:C110H192N40O24S4Purezza:98%Colore e forma:SolidPeso molecolare:2587.22SGLT1/2-IN-2
CAS:<p>SGLT1/2-IN-2 is a chemical compound with robust dual inhibitory properties, exhibiting potent activities against SGLT1 (IC50 = 96 nM) and SGLT2 (IC50 = 1.3 nM).</p>Formula:C23H26F2O7Colore e forma:SolidPeso molecolare:452.451Cortagine
<p>Potent CRF1 agonist, EC50 = 0.18 nM in rats. Exhibits in vivo anxiolytic and antidepressant effects; reduces mouse defensive behavior.</p>Formula:C192H323N55O63SPurezza:98%Colore e forma:SolidPeso molecolare:4442.06Neuropeptide Y(29-64)
CAS:<p>Neuropeptide Y(29-64) is a 36 amino acid peptide, a fragment of Neuropeptide Y.</p>Formula:C189H284N54O58SPurezza:98%Colore e forma:SolidPeso molecolare:4272.7GLP-1(28-36)amide acetate
<p>GLP-1(28-36)amide acetate inhibits mitochondrial permeability transition with antioxidant, anti-diabetic and cardioprotection activities.</p>Formula:C56H89N15O11Purezza:99.9500%Colore e forma:SolidPeso molecolare:1148.4Exendin-3/4 (59-86)
<p>Exendin-3/4 (59-86) is a Exendin-4 peptide derivative.</p>Formula:NAPurezza:98%Colore e forma:SolidPeso molecolare:3055.495-MeO-pyr-T
CAS:<p>5-MeO-pyr-T (5-Methoxy pyrrolidinyltryptamine) acts as a 5-HT1AR agonist, exhibiting Ki values of 0.577 μM and 373 μM for 5-HT1AR and 5-HT2AR, respectively. It inhibits the reuptake of 5-HT and triggers its release. Additionally, 5-MeO-pyr-T can induce reduced motor activity.</p>Formula:C15H20N2OColore e forma:SolidPeso molecolare:244.33CCR8 agonist 1
<p>CCR8 agonist1 (Compound 2) is an activator of CCR8 and is applicable in studies related to autoimmune diseases.</p>Formula:C22H29NO3Colore e forma:SolidPeso molecolare:355.47TRV045
CAS:<p>TRV045 is a selective agonist of the sphingosine-1-phosphate (S1P) subtype 1 receptor and does not impact lymphocyte trafficking. It possesses antiepileptic properties.</p>Formula:C18H18N4O3Colore e forma:SolidPeso molecolare:338.36ONO-8711
CAS:<p>ONO-8711 is a potent and selective competitive antagonist of EP1 receptor with Kis of 0.6 nM and 1.7 nM for human and mouse EP1, respectively.</p>Formula:C22H30ClNO4SColore e forma:SolidPeso molecolare:440MMC(TMZ)-TOC TFA
<p>MMC(TMZ)-TOC TFA exhibits high binding affinity and selectivity for the somatostatin receptor subtype 2 (SSTR2). It targets the delivery of TMZ to SSTR2-positive tumor cells, making MMC(TMZ)-TOC TFA useful for cancer research.</p>Formula:C74H99F3N20O21S2Colore e forma:SolidPeso molecolare:1725.82Metipranolol
CAS:<p>Metipranolol (Betamann) is a type of β- Adrenergic receptors（ β- A potent antagonist of adrenergic receptor on guinea pig atria β 1- Adrenergic receptors and rat uterus β The 2-adrenergic receptor exhibited the beta blocking potentials (pA2) of 8.3 and 8.4, respectively. It is also a potent substituent in the 3H DHA binding assay, with a ligand concentration of 0.7 nM and a Ki of 39 ± 24 nM.</p>Formula:C17H27NO4Purezza:98.37%Colore e forma:SolidPeso molecolare:309.4ALEPH hydrochloride
CAS:<p>ALEPH (hydrochloride) acts as a partial agonist of h5-HT2A and h5-HT2B receptors, with EC50 values of 10.3 nM and 19.2 nM, respectively. It can induce head twitch responses in mice, with an ED50 of 0.80 mg/kg.</p>Formula:C12H20ClNO2SColore e forma:SolidPeso molecolare:277.81Human growth hormone-releasing factor TFA
<p>Human growth hormone-releasing factor TFA is a hypothalamic peptide that promotes GH secretion by targeting pituitary GHRHR.</p>Formula:C217H359F3N72O68SColore e forma:SolidPeso molecolare:5153.67Adrenomedullin (AM) (22-52), human acetate
<p>Adrenomedullin (AM) (22-52), human acetate is an antagonist of calcitonin generelated peptide receptor in the hindlimb vascular bed of the cat and an</p>Formula:C161H256N46O50Purezza:99.42%Colore e forma:SolidPeso molecolare:3636.09(R,R)-Palonosetron Hydrochloride
CAS:<p>(R,R)-Palonosetron Hydrochloride is the active enantiomer of Palonosetron</p>Formula:C19H25ClN2OPurezza:98%Colore e forma:SolidPeso molecolare:332.87Tabernanthalog
CAS:<p>TBG is a 5-HT2A agonist reducing alcohol/heroin cravings and promoting neuroplasticity with antidepressant effects in rodents.</p>Formula:C14H18N2OPurezza:99.82% - 99.89%Colore e forma:SoildPeso molecolare:230.31Ala-parafluoroPhe-Arg-Cha-Cit-Tyr-NH2
CAS:<p>Ala-parafluoroPhe-Arg-Cha-Cit-Tyr-NH2 is a biologically active peptide functioning as a selective agonist for Protease Activated Receptor 1 (PAR-1), a subtype</p>Formula:C42H63FN12O8Colore e forma:SolidPeso molecolare:883.02Antidepressant agent 4
<p>Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.</p>Formula:C19H38ClN5O2SColore e forma:SolidPeso molecolare:436.06Hemopressin(rat)
CAS:<p>Peptide inhibitor for ep24.15, neurolysin & ACE with Ki 27.76, 3.43, 1.87 μM. Lowers blood pressure, modulates CB1 receptor, reduces pain & food intake.</p>Formula:C53H77N13O12Purezza:98%Colore e forma:SolidPeso molecolare:1088.27Ethylpropyltryptamine
CAS:<p>Ethylpropyltryptamine (EPT) is an orally active novel psychoactive substance. It is predicted to act as a partial agonist of the 5-HT2A receptor.</p>Formula:C15H22N2Colore e forma:SolidPeso molecolare:230.35Litoxetine HCl
<p>Litoxetine HCl, an SSRI and 5-HT antagonist, treats urinary incontinence and relaxes rat oesophageal muscles without antimuscarinic effects.</p>Formula:C16H20ClNOPurezza:99.56% - 99.75%Colore e forma:SoildPeso molecolare:277.79JNJ-39933673
CAS:<p>JNJ-39933673 is a bio-active chemical.</p>Formula:C48H54F2N2O11Colore e forma:SolidPeso molecolare:872.96Sauvagine
CAS:<p>CRF receptor agonist; Ki: 9.4 nM (hCRF-R1), 9.9 nM (rCRF-R2a), 3.8 nM (mCRF-R2b) for 125I-[D-Tyr1]astressin binding inhibition.</p>Formula:C202H346N56O63SPurezza:98%Colore e forma:SolidPeso molecolare:4599.35Neuropeptide Y (22-36)
CAS:<p>Neuropeptide Y (22-36) is a 15-amino acid fragment of NPY, which is abundant in the mammalian brain and involved in multiple physiological functions.</p>Formula:C85H139N29O21Purezza:98%Colore e forma:SolidPeso molecolare:1903.19Clomipramine D3
CAS:<p>Clomipramine D3 is deuterium-labeled Clomipramine, blocking serotonin, norepinephrine, dopamine transporters (Ki: 0.14, 54, 3 nM).</p>Formula:C19H23ClN2Purezza:98%Colore e forma:SolidPeso molecolare:317.87tetranor-PGDM
CAS:<p>PGD2, made by H-PGDS in mast cells and lipocalin-PGD-synthase in the brain, aids sleep, cools the body, and inhibits platelet aggregation.</p>Formula:C16H24O7Colore e forma:SolidPeso molecolare:328.361PD 142893
CAS:<p>PD 142893 is a functional endothelin-stimulated vasoconstriction antagonist.</p>Formula:C50H65N7O10Purezza:98%Colore e forma:SolidPeso molecolare:924.09Eloralintide sodium
<p>Eloralintide sodium (LY-3841136 sodium) is an AMYR (amylin receptor) agonist applicable for studying type 2 diabetes and obesity.</p>Formula:C201H319N49O65S2·xNaPurezza:98.66%Colore e forma:SolidPeso molecolare:4526.1 (free base)Albiglutide Fragment
CAS:<p>Albiglutide fragment is a 30-amino-acid sequence of modified human GLP-1 (fragment 7-36).</p>Formula:C148H224N40O45Purezza:98%Colore e forma:SolidPeso molecolare:3283.6L-770644
CAS:<p>L-770644 is an agonist of B3 adrenergic receptor.</p>Formula:C30H37N7O4SColore e forma:SolidPeso molecolare:591.72PY-60
CAS:<p>PY-60 can effectively activate YAP transcriptional activity against annexin A2 (ANXA2).Cost-effective and quality-assured.</p>Formula:C16H15N3O2SPurezza:99.5% - 99.67%Colore e forma:SolidPeso molecolare:313.37SSTR4 agonist-1
CAS:<p>SSTR4agonist-1 (Compound 47) is a selective agonist of the somatostatin receptor 4 (SSTR4), with an EC50 of 4.7 nM. It has a half-life of over 130 minutes in human liver microsomes.</p>Formula:C16H23N3O2Colore e forma:SolidPeso molecolare:289.37GIP/GLP-1 dual receptor agonist-1
CAS:<p>Compound 4: GIP/GLP-1 agonist for metabolic/fatty liver disease research.</p>Colore e forma:SolidTocrifluor T1117
CAS:<p>Fluorescent form of AM 251, CB1 receptor antagonist</p>Formula:C56H53Cl2N7O5Purezza:98%Colore e forma:SolidPeso molecolare:974.97Motilin, canine
CAS:<p>Motilin canine, a 22-amino acid peptide, functions as a robust gastrointestinal smooth muscle contraction agonist.</p>Formula:C120H194N36O34Purezza:98%Colore e forma:SolidPeso molecolare:2685.05Bamosiran
CAS:<p>Bamosiran, a small interfering RNA (siRNA), specifically targets the β-adrenergic receptor 2 to reduce intraocular pressure.</p>Colore e forma:Solid5-HT1AR agonist 2
<p>5-HT1AR Agonist 2 (Compound 4f) is a potent agonist of the 5-HT1A receptor with a Ki value of 10.0 nM. It also binds to SERT, D2, and 5-HT6 receptors with Ki values of 2.8 nM, 23 nM, and 192 nM, respectively. Furthermore, this compound demonstrates stability in microsomes and induces hypothermia in mice.</p>Formula:C31H31N5O3Colore e forma:SolidPeso molecolare:521.61Octodrine
CAS:<p>Octodrine (2-Amino-6-methylheptane) is primarily used as a pharmaceutical intermediate for Octamylamine; it also functions as a local anesthetic and vasoconstrictor.</p>Formula:C8H19NPurezza:99.98%Colore e forma:Clear Colorless To Light Yellow LiquidPeso molecolare:129.24Alosetron
CAS:<p>Alosetron, a 5-HT3 antagonist, is used for the management of severe diarrhea-predominant irritable bowel syndrome (IBS) in women only.</p>Formula:C17H18N4OPurezza:98%Colore e forma:Crystalline PowderPeso molecolare:294.36Zebrafish Kisspeptin-1
CAS:<p>Zebrafish Kisspeptin-1 is the core sequence of the neuropeptide kisspeptin-1, which plays a crucial role in regulating the release of gonadotropin-releasing hormone (GnRH) and modulating the reproductive system.</p>Formula:C58H84N16O15Colore e forma:SolidPeso molecolare:1245.39Bremelanotide
CAS:<p>Bremelanotide is a synthetic peptide analog of alpha-MSH and is an agonist at melanocortin receptors including the MC3R and MC4R.</p>Formula:C50H68N14O10Purezza:98%Colore e forma:White PowderPeso molecolare:1025.16Spantide acetate
<p>Spantide acetate is a selective antagonist of NK1 receptor with Kis of 230 nM and 8150 nM for NK1 and NK2.</p>Formula:C77H112N20O15Purezza:98.9200%Colore e forma:SolidPeso molecolare:1557.84Phoenixin-14 TFA
<p>Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.</p>Formula:C75H110N18O20·xC2HF3O2Purezza:99.11%Colore e forma:SolidPeso molecolare:1583.78 (free base)Kisspeptin-10, rat TFA
<p>Kisspeptin-10, a rat TFA, constricts blood vessels, inhibits vessel growth, and counters Methotrexate reproductive toxicity.</p>Formula:C65H84F3N17O17Colore e forma:SolidPeso molecolare:1432.46LMN-NKA acetate
<p>LMN-NKA acetate is a modified Neurokinin A (4-10) and selective NK2R (Neurokinin 2 receptor) agonist induces bladder contraction smooth muscle contraction.</p>Formula:C41H68N8O12Colore e forma:SolidPeso molecolare:865.03CB2 receptor agonist 2
CAS:<p>CB2 receptor agonist 2 (ZINC72105556): potent, Ki=8.5 nM, high selectivity for CB2.</p>Formula:C30H36N2O4Purezza:99.75%Colore e forma:SolidPeso molecolare:488.62Setmelanotide
CAS:<p>Setmelanotide (BIM-22493) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM and 0.28 nM, respectively).</p>Formula:C49H68N18O9S2Purezza:98%Colore e forma:SolidPeso molecolare:1117.31Maridebart
CAS:<p>Maridebart is a humanized IgG1-kappa monoclonal antibody that targets the GIPR (gastric inhibitory polypeptide receptor) [1].</p>Colore e forma:LiquidHemokinin 1, human
CAS:<p>Endogenous P-like compound, NK1 receptor agonist; IC50: NK1-1.8 nM, NK3-370 nM, NK2-480 nM; boosts B-cell growth, antiapoptotic, lowers blood pressure in vivo.</p>Formula:C54H84N14O14SPurezza:98%Colore e forma:SolidPeso molecolare:1185.4sGnRH-A
CAS:<p>sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.</p>Formula:C64H83N17O12Colore e forma:SolidPeso molecolare:1282.45Calcitonin Gene Related Peptide (CGRP) II, rat TFA
<p>Rat CGRP II TFA: potent vasodilator and CGRP receptor activator for cardiovascular research.</p>Formula:C165H268F3N51O52S2Colore e forma:SolidPeso molecolare:3919.33KSK67
CAS:<p>KSK67 is a selective dual antagonist of sigma-2 and histamine H3 receptors with inhibitory effects on H3 receptors, sigma-1, and sigma-2 receptors, with Ki</p>Formula:C22H27N3O2Purezza:99.11%Colore e forma:SoildPeso molecolare:365.47SB 258585
CAS:<p>SB 258585: Selective 5-HT6 antagonist, binds human receptors, used in cognitive and antipsychotic assays.</p>Formula:C18H22IN3O3SPurezza:99.8%Colore e forma:SoildPeso molecolare:487.36Obestatin(rat)
CAS:<p>Endogenous peptide that suppresses food intake and body weight-gain</p>Formula:C114H174N34O31Purezza:98%Colore e forma:SolidPeso molecolare:2516.81Cetirizine Impurity C
CAS:<p>Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.</p>Formula:C21H25ClN2O3Colore e forma:SolidPeso molecolare:388.89GB-6
CAS:<p>GB-6, a short linear peptide that selectively binds to the gastrin releasing peptide receptor (GRPR), shows potential as a high-contrast imaging probe due to</p>Formula:C32H45N11O8Purezza:98%Colore e forma:SolidPeso molecolare:711.77SAE-14
CAS:<p>GPR183, a chemotactic receptor aiding B cell maturation, binds 7α,25-OHC; studied in IBD research.</p>Formula:C19H19F3N2O2Purezza:99.85%Colore e forma:SolidPeso molecolare:364.36SC 31391
CAS:<p>SC 31391 is a PGE1 analog.</p>Formula:C24H32O6Colore e forma:SolidPeso molecolare:416.51(R)-(+)-Atenolol
CAS:<p>(R)-(+)-Atenolol ((R)-Atenolol) is a cardioselective beta-1 adrenergic blocker, which properties are similar to propranolol, but without a negative inotropic effect.</p>Formula:C14H22N2O3Purezza:98.72%Colore e forma:SolidPeso molecolare:266.34Bradykinin (1-7)
CAS:<p>Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.</p>Formula:C35H52N10O9Purezza:98%Colore e forma:White Lyophilized PowderPeso molecolare:756.85[Des-His1,Glu9]-Glucagon amide
CAS:<p>Glucagon blocker with pA2 of 7.2; no agonist effect. Boosts insulin; prevents glucagon-driven hyperglycemia in rabbits and diabetic rats.</p>Formula:C148H221N41O47SPurezza:98%Colore e forma:SolidPeso molecolare:3358.68Pancreatic Polypeptide, human
CAS:<p>Endogenous high affinity agonist for human NPY Y4 receptor (Ki = 0.056 nM). Believed to play an important role in the function of the gastrointestinal tract.</p>Formula:C185H287N53O54S2Purezza:98%Colore e forma:SolidPeso molecolare:4181.71LGnRH-III, lamprey
CAS:<p>GnRH III triggers luteinizing and follicle-stimulating hormone release, part of the conserved GnRH family.</p>Formula:C59H74N18O14Purezza:98%Colore e forma:SolidPeso molecolare:1259.335-OMe-UDP trisodium salt
CAS:<p>Potent P2Y6 agonist</p>Formula:C10H16N2O13P2Purezza:98%Colore e forma:SolidPeso molecolare:434.19Imnopitant dihydrochloride
CAS:<p>Imnopitant dihydrochloride is a neurokinin NK1 receptor antagonist [1] .</p>Formula:C28H30Cl2F6N4OColore e forma:SolidPeso molecolare:623.46γ1-MSH
CAS:<p>Endogenous melanocortin MC3 receptor agonist (pKi = 7.46) that displays ~ 40-fold selectivity over MC4.</p>Formula:C72H97N21O14SPurezza:98%Colore e forma:SolidPeso molecolare:1512.76GLP-1R agonist 27
<p>GLP-1R agonist 27 (compound 21) is a potent and orally active GLP-1R agonist. It enhances the accumulation of cyclic adenosine monophosphate (cAMP), reduces blood glucose levels, and decreases food intake. GLP-1R agonist 27 shows potential for research in obesity and type 2 diabetes mellitus (T2DM).</p>Formula:C32H33N5O4SeColore e forma:SolidPeso molecolare:630.6Amitraz
CAS:<p>Amitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine demodectic mange.</p>Formula:C19H23N3Purezza:99.88%Colore e forma:White/Pale Yellow Crystalline SolidPeso molecolare:293.41Benzomalvin A
CAS:<p>Benzomalvin A is a filamentous fungal secondary metabolite.</p>Formula:C24H19N3O2Colore e forma:SolidPeso molecolare:381.43ACTH (1-14)
CAS:<p>ACTH (1-14) is a pituitary hormone fragment that controls cortisol and androgen levels.</p>Formula:C77H109N21O20SPurezza:98%Colore e forma:SolidPeso molecolare:1680.88Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate
CAS:<p>Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate is an NPR-A agonist and ANP hormone. Carperitide increases cGMP levels and reduces the heart's workload.</p>Formula:C129H207N45O41S3Purezza:99.78%Colore e forma:SoildPeso molecolare:3140.5Vicasinabin
CAS:<p>Vicasinabin: potent CB2 agonist; researches chronic pain, atherosclerosis, bone mass, neuroinflammation.</p>Formula:C15H22N10OColore e forma:SolidPeso molecolare:358.41Galanin (1-16), mouse, porcine, rat TFA
<p>Galanin (1-16) agonizes hippocampal receptors; Kd 3 nM. Active on locus coeruleus neurons in mice, pigs, rats.</p>Formula:C80H117F3N20O23Purezza:98%Colore e forma:SolidPeso molecolare:1783.9sGC activator 2
<p>sGC activator 2 (Compound 16a) acts as an activator of soluble guanylate cyclase (sGC), enhancing the production of cGMP and exhibiting vasoprotective and anti-inflammatory properties.</p>Formula:C21H21FN8O3Colore e forma:SolidPeso molecolare:452.44UKH-1114
CAS:<p>UKH-1114 is a potent σ2 receptor/Tmem97 agonist with a Ki value of 46 nM, demonstrating antinociceptive effects against mechanical hypersensitivity. This compound alleviates mechanical hypersensitivity in mice caused by nerve injury without inducing motor impairment and is a promising candidate for neuropathic pain research.</p>Formula:C22H24F3NOColore e forma:SolidPeso molecolare:375.43Gulgafafusp alfa
CAS:<p>Gulgafafusp alfa is a human IgG2κ monoclonal antibody that selectively binds to the glucagon-like peptide 1 receptor (GLP1R) [1].</p>Colore e forma:LiquidCasopitant
CAS:<p>Casopitant (GW679769) is an orally active neurokinin-1 (NK1) receptor antagonist, researched for its potential use in managing chemotherapy-induced nausea and vomiting (CINV) and postoperative nausea and vomiting (PONV).</p>Formula:C30H35F7N4O2Colore e forma:SolidPeso molecolare:616.61BAY-6672
CAS:<p>BAY-6672 is, a selective,oral, highly potent human prostaglandin F (FP) receptor antagonist, exerts antifibrotic effects by inhibiting PGF₂α activity.</p>Formula:C26H27BrClN3O3Purezza:99.51%Colore e forma:SolidPeso molecolare:544.87PAF C-18
CAS:<p>PAF C-18 is a natural phospholipid molecule belonging to the platelet-activating factor (PAF) family,, involved in hemostasis and thrombosis by binding to PAFR.</p>Formula:C28H58NO7PPurezza:>99.99%Colore e forma:SolidPeso molecolare:551.74Amylin (8-37), rat
CAS:<p>Amylin (8-37), rat, an analog of IAPP, blocks insulin's effects on muscle glucose uptake and glycogen storage.</p>Formula:C140H227N43O43Purezza:98%Colore e forma:SolidPeso molecolare:3200.61(R)-V-0219 hydrochloride
<p>(R)-V-0219 hydrochloride: Oral GLP-1R PAM, enantiomer of V-0219, triggers Ca2+ flux in hGLP-1R HEK cells.</p>Formula:C20H26ClF3N4O2Colore e forma:SolidPeso molecolare:446.89Lys-γ3-MSH(human)
CAS:<p>Pro-opiomelanocortin (POMC) derived peptide that stimulates lipolysis</p>Formula:C128H193N45O39SPurezza:98%Colore e forma:SolidPeso molecolare:3018.25Substance P (1-9)
CAS:<p>Substance P (1-9), a nonapeptide, slows its own inactivation and stimulates neurons.</p>Formula:C52H77N15O12Purezza:98%Colore e forma:SolidPeso molecolare:1104.26Albiglutide fragment TFA
<p>Albiglutide fragment (GLP-1 (7-36) analog) TFA represents a biologically active segment of Albiglutide, resistant to DPP-4 degradation due to its structure as a</p>Formula:C148H224N40O45·xC2HF3O2Colore e forma:SolidDETQ
CAS:<p>DETQ enhances human D1 dopamine receptor signaling, EC50=5.8 nM, less effective in rats/mice, inactive on D5.</p>Formula:C22H25Cl2NO3Colore e forma:SolidPeso molecolare:422.34Galanin Receptor Ligand M35
CAS:<p>M35, a galanin(1-13)-bradykinin(2-9) amide, acts as a galanin antagonist in rats and inhibits mouse pancreatic islets.</p>Formula:C107H153N27O26Purezza:98%Colore e forma:SolidPeso molecolare:2233.6GLP-1R agonist 16
CAS:<p>Compound 115a, a GLP-1R agonist, effectively activates the GLP-1 receptor with an EC50 of 0.15 nM [1].</p>Formula:C50H58FN10O6PColore e forma:SolidPeso molecolare:945.03Upacicalcet HCl
<p>Upacicalcet HCl, a calcium mimetic, reduces blood PTH by targeting parathyroid receptors; treats secondary hyperparathyroidism.</p>Formula:C11H15Cl2N3O6SPurezza:98.56%Colore e forma:SoildPeso molecolare:388.22exo-Tetrahydrocannabivarin
CAS:<p>exo-Tetrahydrocannabivarin (Compound 12) is an analog of Δ9,11-THC. It weakly binds to cannabinoid receptors (CB) with an IC50 of 1.4 μM. In mice, exo-Tetrahydrocannabivarin exhibits activity related to both motor function and analgesia.</p>Formula:C19H26O2Colore e forma:SolidPeso molecolare:286.415-HT2A receptor agonist-6
CAS:<p>5-HT2A receptor agonist-6 (compound 47) is a selective agonist of the 5-HT2A receptor with a pEC50 value of 6.58.</p>Formula:C18H19N3O3Colore e forma:SolidPeso molecolare:325.36MLS1082
CAS:<p>MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.</p>Formula:C24H23N3O2Purezza:99.53%Colore e forma:SolidPeso molecolare:385.46HAEGTFTSD
CAS:<p>HAEGTFTSD is GLP-1's initial segment; GLP-1 (7-36) amide, tied to food intake, stems from preproglucagon in L-cells.</p>Formula:C40H57N11O17Purezza:98%Colore e forma:SolidPeso molecolare:963.94FFN246
CAS:<p>FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation and</p>Formula:C15H13FN2OPurezza:98%Colore e forma:SolidPeso molecolare:256.27S1PR1 modulator 1
CAS:<p>S1PR1 modulator 1 is a selective inhibitor of S1PR1 with a pIC50 of 7.6.</p>Formula:C23H24N2O3SPurezza:99.69%Colore e forma:SolidPeso molecolare:408.51α-CGRP (mouse, rat) TFA
<p>α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is predominantly located at neuromuscular junctions and</p>Formula:C162H262N50O52S2·C2HF3O2Purezza:98%Colore e forma:SolidBA 1
CAS:<p>Potent BB1, BB2, and BB3 agonist; IC50: 0.26, 1.55, 2.52 nM. Boosts glucose transport in myocytes, promotes cancer cell growth in vitro.</p>Formula:C57H76N14O11Purezza:98%Colore e forma:SolidPeso molecolare:1133.32Hemokinin 1, human TFA
<p>Hemokinin-1 is a human TFA and selective NK1 agonist; also activates NK2 & NK3 and induces opioid-independent analgesia.</p>Formula:C56H85F3N14O16SColore e forma:SolidPeso molecolare:1299.425-HT6 agonist 1
Compound 19, a 5-HT6 agonist with an affinity (K i : 5 nM), exhibits antidepressant-like effects and enhances cognitive function while also inhibiting plateletFormula:C17H22Cl2N6SPurezza:98%Colore e forma:SolidPeso molecolare:413.37AB21 oxalate
<p>AB21 oxalate, a potent and selective S1R antagonist, exhibits binding affinities (Kis) of 13 nM and 102 nM for S1R and S2R, respectively.</p>Formula:C25H30N2O5Purezza:98%Colore e forma:SolidPeso molecolare:438.52Plecanatide acetate
CAS:<p>Plecanatide acetate: GC-C receptor agonist, EC50=190 nM (T84 cells), anti-inflammatory in murine colitis.</p>Formula:C67H108N18O28S4Purezza:98%Colore e forma:SolidPeso molecolare:1741.94PF-232798
CAS:<p>PF-232798 is a second generation oral CCR5 antagonist with potent broad-spectrum anti-HIV-1 activity.</p>Formula:C29H40FN5O2Colore e forma:SolidPeso molecolare:509.66LHRH
CAS:<p>Luteinizing hormone-releasing hormone (LHRH) is a neuropeptide produced in the hypothalamus that plays a pivotal role in regulating reproduction and has</p>Formula:C55H74N16O14Purezza:98%Colore e forma:SolidPeso molecolare:1183.27FGH31
<p>FGH31 (Compound 24), a dopamine D4 agonist, exhibits potent and selective GRK2-dependency with a K i of 1.6 nM and partially activates β-arrestin [1].</p>Formula:C33H36N4O2Purezza:98%Colore e forma:SolidPeso molecolare:520.66SR142948A
CAS:<p>SR142948A is a selective and reversible non-peptide neurotensin receptor antagonist blocking hypothermia and analgesic effects, NMDA-induced dopamine release.</p>Formula:C39H52ClN5O6Purezza:98%Colore e forma:SolidPeso molecolare:722.31ACT-1016-0707
CAS:<p>ACT-1016-0707 is a selective, insurmountable LPA1 antagonist with antifibrotic and anti-inflammatory activity in lung fibrosis models</p>Formula:C19H23ClN4O4SPurezza:99.905%Colore e forma:SolidPeso molecolare:438.93(Ala13)-Apelin-13 acetate
<p>(Ala13)-Apelin-13 acetate, an APJ antagonist, modulates CRF-induced enhanced colonic motility, visceral sensation, and gut barrier.</p>Formula:C65H111N23O18SPurezza:98%Colore e forma:SolidPeso molecolare:1534.79D3R ligand 1
<p>D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template.</p>Formula:C27H37NO5Purezza:98%Colore e forma:SolidPeso molecolare:455.59(-)-Eseroline fumarate
CAS:<p>(-)-Eseroline fumarate, a Physostigmine metabolite and AChE inhibitor, triggers cancer cell LDH release and neuronal cell death.</p>Formula:C17H22N2O5Colore e forma:SolidPeso molecolare:334.37V-0219 hydrochloride
<p>V-0219 hydrochloride: oral GLP-1R PAM for obesity-linked diabetes study.</p>Formula:C20H26ClF3N4O2Purezza:99.97%Colore e forma:SoildPeso molecolare:446.89(+)-Oxypeucedanin methanolate
CAS:<p>(+)-Oxypeucedanin methanolate (compound 9) is a natural compound that inhibits prostaglandin E2 production [1].</p>Formula:C17H18O6Colore e forma:SolidPeso molecolare:318.32Conopeptide rho-TIA
CAS:<p>Conopeptide rho-TIA, a peptide from Conus tulipa venom, acts as a selective, noncompetitive inhibitor at the human α1B-Adrenergic Receptor and as a competitive</p>Formula:C105H160N36O21S4Purezza:98%Colore e forma:SolidPeso molecolare:2390.88Lys-[Des-Arg9]Bradykinin
CAS:Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.Formula:C50H73N13O11Purezza:98%Colore e forma:SolidPeso molecolare:1032.21Paynantheine
CAS:<p>Paynantheine is an alkaloid with antinociceptive properties, found in Mitragyna speciosa. It also acts as an agonist at 5-HT1AR and 5-HT2BR receptors, inducing lower lip contraction and providing antinociception in rats.</p>Formula:C23H28N2O4Colore e forma:SolidPeso molecolare:396.48HAEGT
CAS:<p>HAEGT is the first N-terminal 1-5 residues of GLP-1 peptide.</p>Formula:C20H31N7O9Purezza:98%Colore e forma:SolidPeso molecolare:513.5PACAP (1-38) free acid
CAS:<p>PACAP (1-38) free acid, an endogenous neuropeptide, potently modulates gastrointestinal and neuroendocrine functions.</p>Colore e forma:SolidMAO-B-IN-3
<p>MAO-B-IN-3 is a reversible, selective inhibitor of monoamine oxidase B (MAO-B) with an IC50 of 96 nM and demonstrates affinity for the 5-HT6 receptor with a Ki</p>Formula:C24H25N3O2Purezza:98%Colore e forma:SolidPeso molecolare:387.47Neuropeptide W-30 (human)
CAS:<p>Neuropeptide W-30 (human) serves as a crucial stress mediator within the central nervous system, influencing the hypothalamus-pituitary-adrenal (HPA) axis and sympathetic outflow. It acts as an endogenous ligand for the two related orphan G-protein-coupled receptors (GPCRs), GPR7 and GPR8, binding and activating them at comparable effective doses [1] [2] [3].</p>Formula:C165H249N49O37SColore e forma:SolidPeso molecolare:3543.11GRP (14-27) (human, porcine, canine)
CAS:<p>GRP (14-27) (human, porcine, canine) functions as a ligand for bombesin receptors, with its specific binding being inhibited by GTP and GDP, while GMP does not</p>Formula:C75H110N24O16S2Purezza:98%Colore e forma:SolidPeso molecolare:1667.96Minesapride
CAS:<p>Minesapride: novel 5-HT4 partial agonist, may treat constipation-predominant IBS.</p>Formula:C21H31ClN4O5Purezza:99.85% - 99.88%Colore e forma:SolidPeso molecolare:454.95γ-1-Melanocyte Stimulating Hormone (MSH), amide
<p>γ-1-Melanocyte Stimulating Hormone (MSH), amide, a peptide consisting of 11 amino acids, plays a critical role in regulating sodium (Na+) balance and blood</p>Formula:C72H97N21O14SColore e forma:SolidPeso molecolare:1512.9PACAP (1-38) free acid TFA
<p>PACAP (1-38) free acid TFA, an endogenous neuropeptide, effectively enhances antral motility and somatostatin secretion, while concurrently suppressing gastrin</p>Colore e forma:Odour SolidPentagastrin meglumine
CAS:<p>Pentagastrin meglumine is a synthetic pentapeptide that has effects like gastrin when given parenterally.</p>Formula:C44H66N8O14SColore e forma:SolidPeso molecolare:963.11Ecnoglutide
CAS:<p>Ecnoglutide (XW003) is a glucagon-like peptide 1 (GLP-1) receptor agonist [1] .</p>Formula:C194H304N48O61Colore e forma:SolidPeso molecolare:4284.76Cenicriviroc Mesylate
CAS:<p>Cenicriviroc Mesylate (TBR-652 Mesylate) is an oral dual CCR2/CCR5 antagonist exhibiting anti-inflammatory and anti-fibrotic effects for liver fibrosis.</p>Formula:C42H56N4O7S2Purezza:98.819%Colore e forma:SolidPeso molecolare:793.05Neuropeptide Y (18-36) (porcine)
CAS:<p>"Neuropeptide Y (18-36) (porcine) is a NPY heart receptor blocker, halts I-NPY binding, aids in heart failure research."</p>Formula:C112H174N36O27Colore e forma:SolidPeso molecolare:2456.8Upidosin
CAS:<p>Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.</p>Formula:C31H33N3O4Purezza:99.66%Colore e forma:SolidPeso molecolare:511.61MLGFFQQPKPR-NH2
CAS:<p>MLGFFQQPKPR-NH2 is a reversed Substance P peptide. Substance P is a neuropeptide [1] .</p>Formula:C63H98N18O13SColore e forma:SolidPeso molecolare:1347.63Brexpiprazole S-oxide D8
CAS:<p>Brexpiprazole S-oxide D8 (DM-3411 D8) is a deuterium-labeled metabolite of Brexpiprazole, a partial agonist at 5-HT1A and dopamine receptors.</p>Formula:C25H19D8N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:457.61Bay 55-9837 TFA
<p>Bay 55-9837 TFA is a VPAC2 agonist with a 0.65 nM Kd, potential for type 2 diabetes research.</p>Formula:C150H240F3ClN44O44Colore e forma:SolidPeso molecolare:3456.22LTB4-IN-2
<p>LTB4-IN-2 (Compound 6x) is a selective inhibitor of Leukotriene B4 (LTB4), acting by specifically targeting the 5-Lipoxygenase-activating protein (FLAP) with an</p>Formula:C24H17N5S2Purezza:98%Colore e forma:SolidPeso molecolare:439.56KB-5492 FA
<p>KB-5492 FA is a selective sigma receptor inhibitor with antiulcerogenic effects.CAS 번호128-52-56-8</p>Formula:C24H32N2O8Purezza:98.12%Colore e forma:SolidPeso molecolare:476.52S 16474
CAS:<p>S 16474 is an antagonist of Neurokinin-1 Receptor.</p>Formula:C44H48N6NaO8Purezza:98%Colore e forma:SolidPeso molecolare:811.892(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
CAS:<p>Analog of LHRH, stimulates LH and FSH release, controls reproduction.</p>Formula:C59H84N18O14Colore e forma:SolidPeso molecolare:1269.41AY 254
CAS:<p>AY 254: Potent PAR2 agonist, ERK1/2 activation (EC50=2 nM), limits caspase 3/8, aids HT29 cell healing, boosts IL-8.</p>Formula:C30H49N9O6Colore e forma:SolidPeso molecolare:631.779GRPP (human)
CAS:<p>GRPP (human), a 30-amino-acid peptide derived from Gcg, modestly elevates plasma insulin levels while reducing plasma glucagon concentrations.</p>Formula:C136H215N41O58SColore e forma:SolidPeso molecolare:3384.47APJ receptor agonist 4
CAS:<p>Potent, orally active APJ receptor agonist 4; EC50: 0.06 nM, Ki: 0.07 nM; good pharmacokinetics in rodent HF model; safe in studies; boosts cardiac function.</p>Formula:C28H28ClFN6O3Colore e forma:SolidPeso molecolare:551.02Cortistatin-8
CAS:<p>ghrelin receptor antagonist</p>Formula:C47H68N12O9S2Purezza:98%Colore e forma:SolidPeso molecolare:1009.25Kisspeptin-54(human) TFA
<p>Endogenous kisspeptin-54(human) TFA targets KISS1/GPR54 receptors; Ki: 1.81 nM (rat), 1.45 nM (human); inhibits metastasis, boosts gonadotropin.</p>Formula:C258H401N79O78·C2HF3O2Colore e forma:SolidPeso molecolare:5971.45Cyclic SSTR agonist octreotide
<p>Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .</p>Formula:C53H71N11O14S2Colore e forma:SolidPeso molecolare:1150.33Amylin (8-37) (human)
CAS:Amylin (8-37) (human) is a fragment of human IAPP with a hairpin structure.Formula:C138H215N41O46Colore e forma:SolidPeso molecolare:3184.43Eletriptan
CAS:<p>Eletriptan, second-generation triptans used to treat migraines, is used as an abortion drug.</p>Formula:C22H26N2O2SColore e forma:SolidPeso molecolare:382.52(Trp7,β-Ala8)-Neurokinin A (4-10)
CAS:<p>(Trp7,β-Ala8)-Neurokinin A (4-10) is a potent neurokinin-3 (NK3) antagonist [1] .</p>Formula:C41H57N9O10SColore e forma:SolidPeso molecolare:868.01(D-Phe12,Nle21,38,α-Me-Leu37)-CRF (12-41) (human, rat)
CAS:<p>(D-Phe12,Nle21,38,α-Me-Leu37)-CRF (12-41) (human, rat) is a corticotropin-releasing factor (CRF) antagonist known to counteract the inhibitory effects of IL-1a</p>Formula:C159H267N49O43Colore e forma:SolidPeso molecolare:3553.12Vortioxetine D8
CAS:<p>Vortioxetine D8 is a deuterium-labeled antidepressant inhibiting 5-HT1A/B, 5-HT3A, 5-HT7 receptors & SERT (Ki: 15-1.6 nM).</p>Formula:C18H22N2SPurezza:98%Colore e forma:SolidPeso molecolare:306.5
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