Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(993 prodotti)
- Recettore dell'adenosina(246 prodotti)
- Recettore adrenergico(3.004 prodotti)
- Recettore della bombesina(33 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(153 prodotti)
- CaSR(33 prodotti)
- Recettore dei cannabinoidi(212 prodotti)
- Recettore della dopamina(433 prodotti)
- Recettore dell'endotelina(79 prodotti)
- Recettore GNRH(77 prodotti)
- GPCR19(32 prodotti)
- GRK(32 prodotti)
- GTPase(22 prodotti)
- Recettore del glucagone(182 prodotti)
- Proteina Hedgehog/Smoothened(47 prodotti)
- Recettore dell'istamina(381 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(26 prodotti)
- Recettore OX(41 prodotti)
- Recettore degli oppioidi(310 prodotti)
- PAFR(12 prodotti)
- PKA(51 prodotti)
- Recettore S1P(18 prodotti)
- SGLT(31 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5745 prodotti di "Proteina G/GPCR"
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Fenoldopam
CAS:Fenoldopam is a selective D1-like dopamine receptor partial agonist (EC50 = 57 nM).Formula:C16H16ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:305.76BIIE-0246
CAS:BIIE-0246 is a selective NPY2R antagonist, IC50=15 nM at the rat [125I]PYY3-36 site, reduces NPY-stimulated expression of p-AKT S473 and P-p44/42 MAPK.Formula:C49H57N11O6Purezza:98%Colore e forma:SolidPeso molecolare:896.05K-(D-1-Nal)-FwLL-NH2
CAS:<p>Potent ghrelin receptor inverse agonist with Ki of 4.9/31 nM in COS7/HEK293T; blocks Gq/G13 signaling.</p>Formula:C51H67N9O6Purezza:98%Colore e forma:SolidPeso molecolare:902.13REGN-7544
<p>REGN-7544 is a humanised monoclonal antibody targeting NPR1, which blocks and inhibits NPR1 to increase blood pressure, hypotensione.</p>Purezza:95%Colore e forma:Odour LiquidAdrenocorticotropic Hormone (ACTH) (1-39), rat TFA
Adrenocorticotropic Hormone (ACTH) (1-39), rat (TFA) is a potent melanocortin 2 receptor (MC2) agonist.Formula:C212H316F3N57O59SPurezza:98%Colore e forma:SolidPeso molecolare:4696.18GLP-1R agonist 19
CAS:GLP-1R agonist 19 (M3190) is a potent, selective GLP-1 receptor agonist that demonstrates excellent plasma and liver microsomal stability, along with low hERG toxicity [1].Formula:C94H136FN21O25Colore e forma:SolidPeso molecolare:1979.214-Butyl-α-agarofuran
CAS:4-Butyl-alpha-agarofuran, a Gharu-wood derivative, is an anxiolytic, antidepressant, and aids neurological research.Formula:C18H30OColore e forma:SolidPeso molecolare:262.43CAY10734
CAS:<p>CAY10734 has a wide range of applications in life science related research.</p>Formula:C23H25N3O3Colore e forma:SolidPeso molecolare:391.471BAM(8-22)
CAS:<p>Potent MRGPRX1 agonist peptide; first found in bovine adrenal glands. Non-opioid, lacking met-enkephalin motif. EC50: 8-150 nM.</p>Formula:C91H127N25O23SPurezza:98%Colore e forma:SolidPeso molecolare:1971.22Ivabradine-d3 hydrochloride
CAS:Ivabradine HCl: novel If blocker, IC50 2.9 μM, slows heart rate; D3 version is deuterium labeled.Formula:C27H37ClN2O5Purezza:98%Colore e forma:SolidPeso molecolare:508.07PACAP (1-27), human, ovine, rat TFA
PACAP (1-27) TFA is a pacap-38 fragment and PACAP receptor antagonist with IC50s: 3nm (rat PAC1), 2nm (rat VPAC1), 5nm (human VPAC2).Formula:C144H225F3N40O41SPurezza:98%Colore e forma:SolidPeso molecolare:3261.68Exendin-4 (3-39)
CAS:<p>Exendin-4 (3-39) is a truncated peptide missing first 2 amino acids of Exendin-4, a potent GLP-1r agonist used in diabetes and HPA axis research.</p>Formula:C176H272N46O58SColore e forma:SolidPeso molecolare:3992.44CCG258208 hydrochloride
<p>GRKs-IN-1 HCl (14as) strongly inhibits GRK2 (IC50=130nM) & GRK5 (IC50=7.1μM), is a paroxetine derivative with 100x cardiac boost.</p>Colore e forma:Solid(p-Iodo-Phe7)-ACTH (4-10)
CAS:<p>(p-Iodo-Phe7)-ACTH (4-10), an ACTH derivative and MC receptor antagonist, inhibits α-MSH-induced grooming in rats.</p>Formula:C44H58IN13O10SColore e forma:SolidPeso molecolare:1087.98Isobutyryl-L-carnitine
CAS:<p>Isobutyryl-L-carnitine is a member of the class of compounds known as acylcarnitines. Isobutyryl-L-carnitine is a product of the acyl-CoA dehydrogenases.</p>Formula:C11H21NO4Purezza:98%Colore e forma:SolidPeso molecolare:231.29Amisulpride hydrochloride
CAS:<p>Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.</p>Formula:C17H28ClN3O4SColore e forma:SolidPeso molecolare:405.94M617
CAS:Galanin GAL1 agonist, Ki: GAL1 0.23 nM, GAL2 5.71 nM; boosts rat appetite, lessens inflammation pain.Formula:C112H161N29O28Purezza:98%Colore e forma:SolidPeso molecolare:2361.6811-deoxy Prostaglandin E2
CAS:11-deoxy PGE2 is a synthetic PGE2 analog, a potent bronchoconstrictor, 5-30x stronger than PGF2α on human respiratory muscles.Formula:C20H32O4Colore e forma:SolidPeso molecolare:336.47GB-6
CAS:<p>GB-6, a short linear peptide that selectively binds to the gastrin releasing peptide receptor (GRPR), shows potential as a high-contrast imaging probe due to</p>Formula:C32H45N11O8Purezza:98%Colore e forma:SolidPeso molecolare:711.77Ceruletide Ammonium Salt
Ceruletide Ammonium Salt is a decapeptide, originating from the skin of tropical frogs, which is a potent cholecystokinin receptor agonist and a safe andFormula:C58H77N14O21S2Purezza:98.47% - 98.54%Colore e forma:SoildPeso molecolare:1370.44Nolomirole
CAS:Nolomirole is a dopamine receptor agonist that reduces symptoms of congestive heart failure caused by monoclinine.Formula:C19H27NO4Colore e forma:SolidPeso molecolare:333.42N6-Benzyl-5'-ethylcarboxamido adenosine
CAS:N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.Formula:C19H22N6O4Colore e forma:SolidPeso molecolare:398.42(+)-OSU 6162
CAS:(+)-OSU 6162 (Piperidine, 3-[3-(methylsulfonyl)phenyl]-1-propyl-, (3R)-) is an agonist of 5-HT Receptor with anti-Alzheimer and antidepressant activities.Formula:C15H23NO2SPurezza:98.19%Colore e forma:SoildPeso molecolare:281.41TT-OAD2
CAS:<p>TT-OAD2 is a non-peptide agonist of glucagon-like peptide-1 (GLP-1) receptor (EC50: 5 nM), with the potential for diabetes treatment.</p>Formula:C50H49Cl4N3O6Purezza:98%Colore e forma:SolidPeso molecolare:929.75GW-328267
CAS:GW-328267 is an agonist of the adenosine A2 receptor.Formula:C21H26N10O4Colore e forma:SolidPeso molecolare:482.5AZP-531
CAS:<p>Azp-531 is a disacylated ghrelin used to improve blood sugar control and weight loss.</p>Formula:C40H63N15O13Purezza:98%Colore e forma:SolidPeso molecolare:962.02Dapoxetine
CAS:<p>Dapoxetine (Dapoxetina) is a selective serotonin reuptake inhibitor, for the treatment of premature ejaculation.</p>Formula:C21H23NOPurezza:99.73%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:305.42Carazolol-d7
CAS:Carazolol-d7 is the deuterium-labeled isotope of Carazolol, commonly used in pharmacokinetic studies to investigate the metabolic pathways of Carazolol.Formula:C18H22N2O2Colore e forma:SolidPeso molecolare:305.42Obestatin(rat)
CAS:Endogenous peptide that suppresses food intake and body weight-gainFormula:C114H174N34O31Purezza:98%Colore e forma:SolidPeso molecolare:2516.81Labradimil
CAS:Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.Formula:C49H75N15O12SPurezza:98%Colore e forma:SolidPeso molecolare:1098.29GIP/GLP-1 dual receptor agonist-1
CAS:Compound 4: GIP/GLP-1 agonist for metabolic/fatty liver disease research.Colore e forma:SolidAntidepressant agent 3
Agent 3: orally active, antidepressant, anxiolytic, boosts performance and cognition.Formula:C17H30ClN5O2SColore e forma:SolidPeso molecolare:403.9717-trifluoromethylphenyl trinor Prostaglandin F2α ethyl amide
CAS:<p>Prostaglandin F2α (PGF2α), acting through the FP receptor, causes smooth muscle contraction and exhibits potent luteolytic activity.</p>Formula:C26H36F3NO4Colore e forma:SolidPeso molecolare:483.572Prosaptide TX14(A)
CAS:GPR37L1/GPR37 agonist with EC50 of 5/7 nM, activates G proteins, enhances ERK, myelin synthesis, neuro/glioprotection.Formula:C69H110N16O26Purezza:98%Colore e forma:SolidPeso molecolare:1579.72Ilatreotide
CAS:<p>Ilatreotide is a Amadori compound of octreotide.</p>Formula:C61H86N10O20S2Purezza:98%Colore e forma:SolidPeso molecolare:1343.53Motilin, canine
CAS:<p>Motilin canine, a 22-amino acid peptide, functions as a robust gastrointestinal smooth muscle contraction agonist.</p>Formula:C120H194N36O34Purezza:98%Colore e forma:SolidPeso molecolare:2685.05Vapreotide
CAS:Vapreotide is an antagonist of the neurokinin-1 (NK1) receptor (IC50: 330 nM).Formula:C57H70N12O9S2Purezza:98%Colore e forma:SolidPeso molecolare:1131.38S1P2 antagonist 1
CAS:S1P2 antagonist 1 is an orally bioavailable S1P2 antagonist against fibrotic diseases.Formula:C23H21ClN4O4Colore e forma:SolidPeso molecolare:452.9Galcanezumab
CAS:Galcanezumab: humanized IgG4 antibody that targets CGRP for migraine and cluster headache prevention/treatment.Purezza:> 95%Colore e forma:LiquidPeso molecolare:144.08 kDaBenzquinamide
CAS:<p>Benzquinamide (P2647), an antiemetic agent with anticancer activity, inhibits p-glycoprotein-mediated drug efflux and potentiates the cytotoxicity of anticancer</p>Formula:C22H32N2O5Purezza:94.86%Colore e forma:SolidPeso molecolare:404.5Guanylate cyclase-IN-1
CAS:<p>Guanylate cyclase-IN-1 (Example 46) is a specific inhibitor of guanylate cyclase, employed in research related to cardiovascular diseases.</p>Formula:C20H17FN8OColore e forma:SolidPeso molecolare:404.409Melanostatin, frog TFA
Melanostatin, frog TFA is an α-MSH release inhibitor, a 36 amino acid peptide isolated from the frog brain.Purezza:99.23%Colore e forma:Odour SolidTocrifluor T1117
CAS:Fluorescent form of AM 251, CB1 receptor antagonistFormula:C56H53Cl2N7O5Purezza:98%Colore e forma:SolidPeso molecolare:974.97IRL-1038
CAS:<p>ETB endothelin receptor antagonist</p>Formula:C68H92N14O15S2Purezza:98%Colore e forma:SolidPeso molecolare:1409.67Nafetolol
CAS:Nafetolol (K 5407) is a biochemical reagent that can be used to synthesize other compounds.Formula:C19H29NO3Purezza:98.91%Colore e forma:SolidPeso molecolare:319.44σ1 Receptor ligand 1
σ1 Receptor ligand 1 (compound 5I) is a σ1 receptor ligand with a Ki value of 3.9 nM. It demonstrates a high plasma protein binding rate (89%) and exhibits good metabolic stability in the presence of mouse liver microsomes and NADPH. σ1 Receptor ligand 1 is applicable in neuroscience and cancer research.Formula:C22H28N2O2Colore e forma:SolidPeso molecolare:352.47RS 18286
CAS:RS 18286 is a LHRH antagonist.Formula:C74H101Cl2N17O14Colore e forma:SolidPeso molecolare:1523.6ACTH (11-24)
CAS:ACTH (11-24) is an adrenocorticotrophin fragment, stimulates cortisol, and antagonizes ACTH (1-39)/(1-10) in adrenal cells.Formula:C77H134N24O16Purezza:98%Colore e forma:SolidPeso molecolare:1652.04[18F]-Labeled L-dopa precursor
CAS:[18F]-Labeled L-dopa precursor is a precursor for synthesis of 18F-labeled L-dopa[1].Formula:C35H36N2O7Colore e forma:SolidPeso molecolare:596.67Cortagine
<p>Potent CRF1 agonist, EC50 = 0.18 nM in rats. Exhibits in vivo anxiolytic and antidepressant effects; reduces mouse defensive behavior.</p>Formula:C192H323N55O63SPurezza:98%Colore e forma:SolidPeso molecolare:4442.06Bradykinin (1-3)
CAS:<p>Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.</p>Formula:C16H28N6O4Purezza:98%Colore e forma:SolidPeso molecolare:368.43Vapitadine
CAS:Vapitadine is a non-sedative antihistamine compound that relieves itching caused by atopic dermatitis.Formula:C17H20N4OPurezza:99.77% - 99.86%Colore e forma:SoildPeso molecolare:296.37d[Leu4,Lys8]-VP acetate
d[Leu4,Lys8]-VP acetate: Vasopressin V1b agonist. Ki: rat 0.16 nM, human 0.52 nM, mouse 1.38 nM. Low antidiuretic/vasopressor effects.Formula:C49H71N11O13S2Purezza:98.86%Colore e forma:SolidPeso molecolare:1086.28A-286501
CAS:<p>A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.</p>Formula:C11H14BrN5O2Purezza:98%Colore e forma:SolidPeso molecolare:328.175-methoxy-α-Ethyltryptamine
CAS:<p>5-Methoxy-alpha-ethyltryptamine is a psychoactive substance that can cause various effects. It belongs to the tryptamine chemical class and can be used for various psychoactive and stimulant effects. </p>Formula:C13H18N2OPurezza:98.25%Colore e forma:SolidPeso molecolare:218.29isomer-Cilansetron
CAS:isomer-Cilansetron is an isomer of Cilansetron.Formula:C20H21N3OPurezza:99.92% - 99.96%Colore e forma:SoildPeso molecolare:319.4Edg-2 receptor inhibitor 1
CAS:Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).Formula:C27H27NO5Purezza:99.47%Colore e forma:SolidPeso molecolare:445.51Sarafotoxin S6c
CAS:<p>Highly selective ETB endothelin receptor agonist (Ki values are 0.29 and 28000 nM at ETB and ETA receptors respectively).</p>Formula:C103H147N27O37S5Purezza:98%Colore e forma:SolidPeso molecolare:2516Pasireotide (diaspartate)
CAS:Pasireotide diaspartate (SOM230) has high agonist activity at sst1/2/3/5, less at sst4; it's antiproliferative and proapoptotic.Formula:C66H80N12O17Colore e forma:SolidPeso molecolare:1313.41JNJ-39933673
CAS:JNJ-39933673 is a bio-active chemical.Formula:C48H54F2N2O11Colore e forma:SolidPeso molecolare:872.96Corynanthine
CAS:Corynanthe is a plant alkaloid. Corynanthe also has an alpha-2-adrenergic blocking activity.Formula:C21H26N2O3Purezza:98%Colore e forma:SolidPeso molecolare:354.44Semaglutide TFA
<p>Semaglutide TFA is a glucagon-like peptide-1 congener that induces weight loss, lowers blood glucose levels and reduces cardiovascular risk in diabetic patients</p>Formula:C189H290F3N45O61Purezza:99.69%Colore e forma:SolidPeso molecolare:4225.6482CAY10597
CAS:<p>PGD2 effects via DP1/CRTH2/DP2 receptors; CAY10597 blocks CRTH2/DP2 (Ki=37nM), R enantiomer stronger (Ki=23-22nM), inhibits eosinophil migration (IC50=40nM).</p>Formula:C20H14ClFN2O5Colore e forma:SolidPeso molecolare:416.79Chir 2279
CAS:<p>CHIR 2279, a peptoid trimer, binds alpha 1-adrenoceptors, blocking epinephrine effects in dogs (pseudo pA2 6.86).</p>Formula:C34H36N4O4Colore e forma:SolidPeso molecolare:564.67Thiothixene
CAS:Thiothixene has a wide range of applications in life science related research.Formula:C23H29N3O2S2Colore e forma:SolidPeso molecolare:443.62Clomipramine D3
CAS:Clomipramine D3 is deuterium-labeled Clomipramine, blocking serotonin, norepinephrine, dopamine transporters (Ki: 0.14, 54, 3 nM).Formula:C19H23ClN2Purezza:98%Colore e forma:SolidPeso molecolare:317.87Amylin (IAPP), feline
Amylin (IAPP), feline is the peptide subunit of amyloid found in pancreatic islets of type 2 diabetic patients and in insulinomas.Formula:C165H270N52O54S2Purezza:98%Colore e forma:SolidPeso molecolare:3910.45L-770644
CAS:L-770644 is an agonist of B3 adrenergic receptor.Formula:C30H37N7O4SColore e forma:SolidPeso molecolare:591.72Tezusomant
CAS:Tezusomant is an antagonist of the growth hormone receptor (growth hormone receptor). It is being investigated for potential use in conditions like acromegaly, which are caused by excessive secretion of growth hormone.Formula:C120H171N23O32SColore e forma:SolidPeso molecolare:2479.84σ1R-IN-1
σ1R-IN-1 ((R,R)-1a) is an effective σ-1R inhibitor with an IC50 of 110 nM. It shows promising potential for use in research related to neuropsychiatric disorders.Formula:C15H22N2Colore e forma:SolidPeso molecolare:230.35ent-Prostaglandin E2
CAS:<p>Enzymatic PGE2 is optically pure; radical peroxidation makes it racemic. In oxidative stress, rac-PGE2 forms via 15-E2t-isoprostane.</p>Formula:C20H32O5Colore e forma:SolidPeso molecolare:352.471HAEGTFTSDVS
CAS:HAEGTFTSDVS is the first N-terminal 1-11 residues of GLP-1 peptide.Formula:C48H71N13O20Purezza:98%Colore e forma:SolidPeso molecolare:1150.18Flunarizine
CAS:<p>Flunarizine is an orally administered peripheral vasodilator, a dual blocker of voltage-gated Na+/Ca2+ channels and a D2 dopamine receptor antagonist.</p>Formula:C26H26F2N2Purezza:99.9%Colore e forma:SolidPeso molecolare:404.50Lysophosphatidic acid
CAS:Lysophosphatidic acid is a bioactive chemical.Formula:C21H41O7PColore e forma:SolidPeso molecolare:436.52FK 224
CAS:<p>FK 224 is an antagonist of tachykinin receptor.</p>Formula:C54H72N8O13Colore e forma:SolidPeso molecolare:1041.213V-0219 hydrochloride
<p>V-0219 hydrochloride: oral GLP-1R PAM for obesity-linked diabetes study.</p>Formula:C20H26ClF3N4O2Purezza:99.97%Colore e forma:SoildPeso molecolare:446.89Setmelanotide Acetate(920014-72-8 free base)
CAS:Setmelanotide Acetate(920014-72-8 free base) (RM-493 Acetate) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nMFormula:C51H72N18O11S2Purezza:99.71%Colore e forma:SolidPeso molecolare:1177.35D-Epinephrine
CAS:<p>D-Epinephrine: a hormone and drug, boosts heart rate, muscle blood flow, pupil size, and sugar levels in stress responses.</p>Formula:C9H13NO3Colore e forma:SolidPeso molecolare:183.2[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide
CAS:<p>Potent, selective NPY Y5 receptor agonist; IC50: 0.24 nM (Y5), >500 nM (Y2), 530 nM (Y1), 51 nM (Y4); Ki: 0.1-0.15 nM (Y5); increases food intake in vivo.</p>Formula:C183H281N57O54S2Purezza:98%Colore e forma:SolidPeso molecolare:4207.67Amitraz
CAS:<p>Amitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine demodectic mange.</p>Formula:C19H23N3Purezza:99.88%Colore e forma:White/Pale Yellow Crystalline SolidPeso molecolare:293.41Adenosine 3'-monophosphate (sodium salt hydrate)
Adenosine 3'-monophosphate (sodium salt hydrate) (3'-AMP) is a nucleotide and cAMP-generating agonist that elevates cAMP levels in NG108-15 cells.Formula:C10H15N5NaO8PColore e forma:SolidPeso molecolare:387.22HS014
CAS:Potent MC4 antagonist; Ki: 3.16 nM (MC4), 108 (MC1), 54.4 (MC3), 694 (MC5). Boosts rat appetite, mouse pain, blocks IL-1β Fos in hypothalamus.Formula:C71H94N20O17S2Purezza:98%Colore e forma:SolidPeso molecolare:1563.77KSK67
CAS:<p>KSK67 is a selective dual antagonist of sigma-2 and histamine H3 receptors with inhibitory effects on H3 receptors, sigma-1, and sigma-2 receptors, with Ki</p>Formula:C22H27N3O2Purezza:99.11%Colore e forma:SoildPeso molecolare:365.47Adrenomedullin (16-31), human
CAS:<p>Adrenomedullin (16-31), human is amino acid residues 16-31 fragment of human adrenomedullin (hADM).</p>Formula:C82H129N25O21S2Purezza:98%Colore e forma:SolidPeso molecolare:1865.19LMN-NKA acetate
LMN-NKA acetate is a modified Neurokinin A (4-10) and selective NK2R (Neurokinin 2 receptor) agonist induces bladder contraction smooth muscle contraction.Formula:C41H68N8O12Colore e forma:SolidPeso molecolare:865.03AdTx1
<p>Selective non-competitive α1A adrenoceptor antagonist with Ki of 0.35 nM; inactive on other GPCRs; affects phenylephrine actions.</p>Formula:C310H481N87O100S8Purezza:98%Colore e forma:SolidPeso molecolare:7283.22VU0453379 hydrochloride
VU0453379 hydrochloride: selective CNS-penetrant GLP-1R PAM, EC50 1.3 μM.Formula:C26H35ClN4O2Colore e forma:SolidPeso molecolare:471.03(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
CAS:V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.Formula:C52H74N14O12S2Purezza:98%Colore e forma:White Lyophilized PowderPeso molecolare:1151.38ACTH (1-17)
CAS:<p>ACTH (1-17), a potent MC1 receptor agonist with a Ki of 0.21 nM, is a variant of corticotropin from the pituitary gland.</p>Formula:C95H145N29O23SPurezza:98%Colore e forma:SolidPeso molecolare:2093.41Atrial Natriuretic Peptide (ANP) (1-28), rat
CAS:Atrial Natriuretic Peptide (1-28), rat is the major circulating form of ANP in rats.Formula:C128H205N45O39S2Purezza:98%Colore e forma:SolidPeso molecolare:3062.41Mesoridazine Besylate
CAS:<p>Mesoridazine Besylate (Serentil), a piperidine antipsychotic and phenothiazine, treats schizophrenia; it's a thioridazine metabolite.</p>Formula:C27H32N2O4S3Purezza:99.58%Colore e forma:SolidPeso molecolare:544.75LCKLSL acetate
LCKLSL acetate is a potent AnxA2 inhibitor, blocking tPA binding and plasmin production, with anti-angiogenic effects.Formula:C32H61N7O10SPurezza:99.9%Colore e forma:SolidPeso molecolare:735.93Cholecystokinin Octapeptide, desulfated
CAS:Cholecystokinin Octapeptide, desulfated (CCK Octapeptide, non-sulfated) is an octapeptide composed of 8 amino acids from cholecystokinin-8.Formula:C49H62N10O13S2Purezza:97.12%Colore e forma:SolidPeso molecolare:1063.21FFN246
CAS:FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation andFormula:C15H13FN2OPurezza:98%Colore e forma:SolidPeso molecolare:256.27Human growth hormone-releasing factor
CAS:<p>GHRH from the hypothalamus prompts the pituitary to produce/release GH by attaching to the GHRHR.</p>Formula:C215H358N72O66SPurezza:98%Colore e forma:SolidPeso molecolare:5039.65Halometasone
CAS:<p>Halometasone: synthetic corticosteroid for psoriasis and eczema treatment.</p>Formula:C22H27ClF2O5Colore e forma:SolidPeso molecolare:444.9Mosapride citrate dihydrate
CAS:<p>Mosapride Citrate, a 5-HT4 agonist, boosts gut movement by enhancing acetylcholine release.</p>Formula:C27H35ClFN3O11Purezza:98%Colore e forma:SolidPeso molecolare:632.04Parstatin(human) TFA
<p>Parstatin(human) TFA, a cell-penetrating PAR-1 thrombin receptor agonist peptide, effectively inhibits angiogenesis, as indicated by studies [1] [2].</p>Formula:C193H331F3N64O55S3Colore e forma:SolidPeso molecolare:4581.28Alprostadil ethyl ester
CAS:<p>Alprostadil ethyl ester is a biochemical used in the treatment of scleroderma.</p>Formula:C22H38O5Colore e forma:SolidPeso molecolare:382.53MRS-1706
CAS:<p>MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.</p>Formula:C27H29N5O5Purezza:99.00%Colore e forma:SolidPeso molecolare:503.55Men 10208
CAS:<p>Men 10208 is an antagonist of the neurokinin A receptor.</p>Formula:C61H75N15O12Purezza:98%Colore e forma:SolidPeso molecolare:1210.36[Tyr3]Octreotate
CAS:<p>[Tyr3]Octreotate is a long peptide compound containing 8 amino acids and is a functional DOTA chelating agent with covalent bonds.</p>Formula:C49H64N10O12S2Purezza:98.21%Colore e forma:SoildPeso molecolare:1049.22ACTH (1-14)
CAS:ACTH (1-14) is a pituitary hormone fragment that controls cortisol and androgen levels.Formula:C77H109N21O20SPurezza:98%Colore e forma:SolidPeso molecolare:1680.88Adenosine receptor agonist 1
<p>Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.</p>Formula:C12H14ClN5O2SeColore e forma:SolidPeso molecolare:374.68Protease-Activated Receptor-1, PAR-1 Agonist
CAS:Selective peptide agonist that mimics thrombin to activate PAR-1 receptor, enabling targeted receptor activation.Formula:C35H58N10O9Colore e forma:SolidPeso molecolare:762.91Methionyl-Lysyl-Bradykinin
CAS:Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin [1] [2] .Formula:C61H94N18O13SColore e forma:SolidPeso molecolare:1319.58Y1 receptor antagonist 1 formic
<p>H 409-22 isomer formic, a formate salt of Y1 receptor antagonist 1, is an antagonist of the neuropeptide Y1 receptor (neuropeptide Y1 receptor). This compound effectively blocks the actions of the receptor, playing a crucial role in modulating physiological responses.</p>Formula:C29H35N5O5Colore e forma:SolidPeso molecolare:533.62INCB3344 R-isomer
<p>INCB3344 is a potent CCR2 antagonist. INCB3344 R-isomer is the R-isomer of INCB3344.</p>Formula:C29H34F3N3O6Purezza:98%Colore e forma:SolidPeso molecolare:577.59(Ala13)-Apelin-13 acetate
<p>(Ala13)-Apelin-13 acetate, an APJ antagonist, modulates CRF-induced enhanced colonic motility, visceral sensation, and gut barrier.</p>Formula:C65H111N23O18SPurezza:98%Colore e forma:SolidPeso molecolare:1534.79Neuropeptide AF (cattle)
CAS:Neuropeptide AF (cattle) is an RFamide that acts on MrgprA4 (~60 nM), MrgprC11 (~300 nM), NPFF1 (~25-325 nM), NPFF2 (~1-5 nM), and modulates pain.Formula:C89H130N24O24Colore e forma:SolidPeso molecolare:1920.13cAC 253 acetate
<p>cAC 253 acetate (TP2135 Free base) is an amylin antagonist. cAC 253 acetate inhibits 125I-adrenomedullin binding, with an IC50 of 25 nM.</p>Formula:C128H206N42O42S2Purezza:98.16% - 99.99%Colore e forma:SoildPeso molecolare:3069.39Fasitibant chloride
CAS:<p>Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.</p>Formula:C36H49Cl3N6O6SColore e forma:SolidPeso molecolare:800.23Fasitibant chloride hydrochloride
CAS:Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.Formula:C36H50Cl4N6O6SColore e forma:SolidPeso molecolare:836.7APJ receptor agonist 1
CAS:Potent APJ-R agonist 1, biphenyl acid, EC50: 0.093 nM (human), 0.12 nM (rat), targets apelin-13, promising for heart failure study.Formula:C31H26ClN3O3Colore e forma:SolidPeso molecolare:524.02Desmethyl Mirtazapine (hydrochloride)
CAS:<p>Desmethyl mirtazapine is a metabolite of the antidepressant mirtazapine.1It is formed from mirtazapine by the cytochrome P450 (CYP) isoform CYP3A4.</p>Formula:C16H18ClN3Colore e forma:SolidPeso molecolare:287.79Lys-Bradykinin
CAS:Endogenous bradykinin receptor agonistFormula:C56H85N17O12Purezza:98%Colore e forma:SolidPeso molecolare:1188.38Lys-[Des-Arg9]Bradykinin TFA
CAS:<p>Lys-[Des-Arg9]Bradykinin TFA: natural kinin, selective B1 agonist; Ki: 0.12 nM (human), 1.7 nM (mouse), 0.23 nM (rabbit); weak on B2 receptors.</p>Formula:C54H75F6N13O15Colore e forma:SolidPeso molecolare:1260.24CRF(6-33)(human)
CAS:<p>CRFBP inhibitor peptide; blocks CRF, reduces weight gain, boosts activity in obese rats.</p>Formula:C141H231N41O43SPurezza:98%Colore e forma:SolidPeso molecolare:3220.68Pasireotide pamoate
CAS:Pasireotide pamoate is a stable cyclohexapeptide somatostatin mimic. Pasireotide pamoate exhibits antisecretory, antiproliferative, and proapoptotic activity.Formula:C81H82N10O15Purezza:98%Colore e forma:SolidPeso molecolare:1435.58[Ala11,D-Leu15]-Orexin B(human)
CAS:OX2 receptor agonist with 400x selectivity vs OX1. EC50: 0.13 nM (OX2), 52 nM (OX1).Formula:C120H206N44O35SPurezza:98%Colore e forma:SolidPeso molecolare:2857.28Urocortin II, mouse
CAS:Mouse Urocortin II: Selective CRF2 agonist, Ki 0.66 nM for CRFR2, >100 nM for CRFR1, affects central neural circuits.Formula:C187H320N56O50Colore e forma:SolidPeso molecolare:4152.96HL2-m5
CAS:HL2-m5 is an inhibitor of the sonic hedgehog/patched (Shh/PTCH1) interaction, with a Kd for Shh of 170 nM. It effectively inhibits the activation of the Hedgehog signaling pathway and the transcription of Gli-controlled genes, with an IC50 of 230 nM.Formula:C70H101N15O24S3Colore e forma:SolidPeso molecolare:1632.835-hydroxy Propranolol
CAS:<p>5-hydroxy Propranolol, a propranolol metabolite, is formed in the liver via P450 2D6.</p>Formula:C16H21NO3Colore e forma:SolidPeso molecolare:275.348Apigenin 6,8-di-C-α-L-arabinopyranoside
CAS:Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.Formula:C25H26O13Colore e forma:SolidPeso molecolare:534.47H4R antagonist 3
CAS:<p>H4R antagonist 3 is a novel histamine-4 receptor (H4R) antagonist with an EC50 <10 mM.H4R antagonist 3 has potential inflammatory activity for the study of</p>Formula:C19H21ClN4SPurezza:98%Colore e forma:SolidPeso molecolare:372.92Stressin I
Potent CRF1 agonist; Ki: 1.5 nM (CRF1), 224 nM (CRF2). Boosts ACTH, enhances stool frequency after i.p. administration.Formula:C203H337N57O56Purezza:98%Colore e forma:SolidPeso molecolare:4472.24TGR5 agonist 4
<p>TGR5 agonist 4 (compound 19), a derivative of cholic acid, selectively activates the TGR5 receptor with an effective concentration (EC50) of 4 μM [1].</p>Formula:C24H38F2O5Colore e forma:SolidPeso molecolare:444.55Cortistatin-14 acetate
<p>Cortistatin-14 acetate, a neuropeptide have structural similarity to somatostatin-14, binds and exerts its function via the somatostatin receptors (sst1-sst5).</p>Formula:C83H118N20O20S2Purezza:98.24% - 99.63%Colore e forma:SoildPeso molecolare:1780.08Septide
CAS:<p>Septide is an NK1 receptor agonist acting at a site distinct from substance P.</p>Formula:C39H53N7O7SPurezza:98%Colore e forma:SolidPeso molecolare:763.95Xenopus orexin B
CAS:Xenopus orexin B, a neuropeptide identified as an endogenous ligand for an orphan G-protein-coupled receptor, acts as a potent agonist of OX2R [1].Formula:C130H219N45O40S2Colore e forma:SolidPeso molecolare:3116.54MCL0129
CAS:<p>MCL0129, a selective and non-peptidergic melanocortin 4 (MC4) receptor antagonist, is a potential treatment for cachexia.</p>Formula:C34H47FN4OPurezza:98%Colore e forma:SolidPeso molecolare:546.76MDL 19301
CAS:MDL 19301 is a nonsteroidal, anti-inflammatory agent.Formula:C15H21NS2Purezza:98%Colore e forma:SolidPeso molecolare:279.46TRAP-5 amide
CAS:TRAP-5 amide is a peptide agonist for protease-activated receptor 1 (PAR 1) [1].Formula:C30H51N9O6Colore e forma:SolidPeso molecolare:633.78Levocarnitine propionate hydrochloride
CAS:Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.Formula:C10H20ClNO4Purezza:90% - 99.77%Colore e forma:SolidPeso molecolare:253.72Alcaftadine carboxylic acid
CAS:Alcaftadine is a novel antihistamine for preventing allergic conjunctivitis.Formula:C19H21N3O2Colore e forma:SolidPeso molecolare:323.39Albenatide
CAS:<p>Albenatide is a modified analog of exendin 4 conjugated to recombinant human albumin.</p>Formula:C26H47N7O9SPurezza:98%Colore e forma:SolidPeso molecolare:633.76Galanin (1-29)(rat, mouse)
CAS:<p>Non-selective galanin agonist; Ki: GAL1-0.98, GAL2-1.48, GAL3-1.47 nM. Anticonvulsant, stops full seizures in rats.</p>Formula:C141H211N43O41Purezza:98%Colore e forma:White Lyophilized PowderPeso molecolare:3164.499TGR5 agonist 7
TGR5 agonist 7 (Compound 22-Na) is an intestine-restricted, orally active agonist of the G protein-coupled bile acid receptor TGR5 (GPBAR1 or GPR131) with an EC50 of less than 1 μM. In mouse models, it demonstrates blood glucose-lowering effects, making it useful for diabetes research.Formula:C37H59N2NaO9SColore e forma:SolidPeso molecolare:730.9315(S)-15-methyl Prostaglandin F2α methyl ester
CAS:15(S)-15-methyl Prostaglandin F2α methyl ester can be used in related research in the field of life sciences.Formula:C22H38O5Colore e forma:SolidPeso molecolare:382.5317-phenoxy trinor Prostaglandin F2α ethyl amide
CAS:Prostaglandin F2α (PGF2α), acting through the FP receptor, causes smooth muscle contraction and exhibits potent luteolytic activity.Formula:C25H37NO5Colore e forma:SolidPeso molecolare:431.573Calcitonin Gene Related Peptide (CGRP) II, rat
CAS:<p>CGRP II is a potent vasodilator that boosts pancreatic enzyme levels by activating β-cell receptors.</p>Formula:C163H267N51O50S2Purezza:98%Colore e forma:SolidPeso molecolare:3805.31AG 045572
CAS:<p>AG 045572 is a potent GnRH receptor antagonist that inhibits the GnRH receptor in humans and rats with Ki values of 6.0 nM and 3.8 nM, respectively.AG 045572 is</p>Formula:C30H37NO5Purezza:99.96%Colore e forma:SolidPeso molecolare:491.62CH 275
CAS:Potent sst1 agonist with 30.9 nM IC50; selective over sst2-5; inhibits somatostatin in rat nucleus accumbens.Formula:C74H96N14O15S2Purezza:98%Colore e forma:SolidPeso molecolare:1485.8Neuropeptide Y (22-36)
CAS:Neuropeptide Y (22-36) is a 15-amino acid fragment of NPY, which is abundant in the mammalian brain and involved in multiple physiological functions.Formula:C85H139N29O21Purezza:98%Colore e forma:SolidPeso molecolare:1903.19FR252384
CAS:FR252384 is an antagonist of the neuropeptide Y-Y5 receptor (IC50: 2.3 nM).Formula:C18H17N3Purezza:98%Colore e forma:SolidPeso molecolare:275.35MEN 11270
CAS:<p>B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.</p>Formula:C60H90N20O11SPurezza:98%Colore e forma:SolidPeso molecolare:1299.56Urocortin II, human TFA
<p>hUcn II, a CRF family member, targets CRF2 receptor, has time-linked stress regulation effects, showing mild motor suppression and delayed anxiolytic action.</p>Formula:C196H340F3N63O56SPurezza:98%Colore e forma:SolidPeso molecolare:4564.3Ethylnorepinephrine hydrochloride
CAS:<p>Ethylnorepinephrine hydrochloride is a unique bronchodilator.</p>Formula:C10H16ClNO3Purezza:98%Colore e forma:SolidPeso molecolare:233.69SB 258585
CAS:<p>SB 258585: Selective 5-HT6 antagonist, binds human receptors, used in cognitive and antipsychotic assays.</p>Formula:C18H22IN3O3SPurezza:99.8%Colore e forma:SoildPeso molecolare:487.36FR167344 free base
CAS:FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.Formula:C30H28BrCl2N5O4Purezza:98%Colore e forma:SolidPeso molecolare:673.38Ontazolast
CAS:<p>Ontazolast: a small-molecule LTB4R antagonist targeting asthma and immune disorders.</p>Formula:C21H25N3OPurezza:99.79%Colore e forma:SoildPeso molecolare:335.44Ro 25-1553
CAS:<p>Ro 25-1553 is a 31-amino acid analog of vasoactive intestinal peptide (VIP) that functions as an agonist for the VIP2 receptor (VPAC2 receptor). In guinea pig models, Ro 25-1553 exhibits bronchodilator effects on tracheal smooth muscle contraction induced by neural stimuli or Carbachol.</p>Formula:C160H258N46O46Colore e forma:SolidPeso molecolare:3562.04Antidepressant agent 4
Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.Formula:C19H38ClN5O2SColore e forma:SolidPeso molecolare:436.06Clotizolam
CAS:<p>Clotizolam is a thienotriazolodiazepine derivative with PAF antagonistic properties, exhibiting sedative, anxiolytic, anticonvulsant, and muscle relaxant effects.</p>Formula:C15H10Cl2N4SColore e forma:SolidPeso molecolare:349.24Phoenixin-14 TFA
Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.Formula:C75H110N18O20·xC2HF3O2Purezza:99.11%Colore e forma:SolidPeso molecolare:1583.78 (free base)Nebentan
CAS:<p>Nebentan (YM598) is an oral, selective ETA antagonist; Ki: 0.697 nM (ETA), 569 nM (ETB); may slow cor pulmonale, myocardial infarction.</p>Formula:C24H21N5O5SColore e forma:SolidPeso molecolare:491.52FSLLRY-NH2
CAS:<p>PAR2 antagonist; counters taxol effects, PKC in mice; inhibits ERK, collagen in fibroblasts; lessens dermatophyte itch in mice.</p>Formula:C39H60N10O8Purezza:98%Colore e forma:SolidPeso molecolare:796.97Somatostatin-28 (1-14)
CAS:<p>Somatostatin-28 (1-14) is a truncated neuropeptide from prosomatostatin cleavage.</p>Formula:C61H105N23O21SPurezza:98%Colore e forma:SolidPeso molecolare:1528.71Hemopressin(rat)
CAS:Peptide inhibitor for ep24.15, neurolysin & ACE with Ki 27.76, 3.43, 1.87 μM. Lowers blood pressure, modulates CB1 receptor, reduces pain & food intake.Formula:C53H77N13O12Purezza:98%Colore e forma:SolidPeso molecolare:1088.27TT 232
CAS:sst1/sst4 somatostatin receptors agonistFormula:C45H58N10O9S2Purezza:98%Colore e forma:SolidPeso molecolare:947.13RF9
CAS:RF9 is an effective and selective antagonist of the Neuropeptide FF receptor (Kis: 58±5 and 75±9 nM for hNPFF1R and hNPFF2R, respectively).Formula:C26H38N6O3Purezza:98%Colore e forma:SolidPeso molecolare:482.62Jmv 167
CAS:Jmv 167 is an antagonist of the Cholecystokinin receptor.Formula:C51H68N8O14SPurezza:98%Colore e forma:SolidPeso molecolare:1049.21APJ receptor agonist 10
CAS:<p>APJ receptor agonist 10 (Compound I choline salt) modulates the activity of the APJ receptor, making it useful for pulmonary hypertension research. Compared to its free form, this compound exhibits improved bioavailability.</p>Formula:C26H36N7O6SColore e forma:SolidPeso molecolare:574.67Plecanatide acetate
CAS:Plecanatide acetate: GC-C receptor agonist, EC50=190 nM (T84 cells), anti-inflammatory in murine colitis.Formula:C67H108N18O28S4Purezza:98%Colore e forma:SolidPeso molecolare:1741.9416,16-dimethyl Prostaglandin F2α
CAS:<p>16,16-dimethyl Prostaglandin F2α can be used in related research in the field of life sciences. Its product number is T37993 and CAS number is 39746-23-1.</p>Formula:C22H38O5Colore e forma:SolidPeso molecolare:382.541Calcitonin (8-32), salmon
CAS:Calcitonin (8-32), salmon: selective amylin receptor antagonist, regulates calcium/phosphorus, thyroid origin, 32-aa peptide.Formula:C119H198N36O37Purezza:98%Colore e forma:SolidPeso molecolare:2725.06SB 201146
CAS:<p>SB 201146 is a leukotriene B4 antagonist with high affinity.</p>Formula:C30H35LiN2O5SColore e forma:SolidPeso molecolare:542.61Maceneolignan H
CAS:Maceneolignan H, a neolignane from Myristica fragrans, selectively blocks CCR3 (EC50=1.4μM) with allergy research potential.Formula:C24H30O7Colore e forma:SolidPeso molecolare:430.49O-Desmethyl Mebeverine alcohol hydrochloride
CAS:<p>O-Desmethyl Mebeverine alcohol HCl, a metabolite of Mebeverine, is a strong α1 inhibitor, relaxing the GI tract.</p>Formula:C15H26ClNO2Colore e forma:SolidPeso molecolare:287.8317-phenyl trinor Prostaglandin F2α cyclopropyl methyl amide
CAS:Prostaglandin F2α (PGF2α) activates the FP receptor, promoting smooth muscle contraction and luteolysis.Formula:C27H39NO4Colore e forma:SolidPeso molecolare:441.612GLP-1(7-36), amide acetate
CAS:GLP-1(7-36), amide acetate is a derivative of GLP-1 peptide , activate the GLP-1 receptor, promote insulin secretion,Type 2 diabetes mellitus and obesity.Formula:C151H230N40O47Purezza:99.89%Colore e forma:SolidPeso molecolare:3357.68Hemopressin(human, mouse) TFA
CAS:Hemopressin TFA: nonapeptide from hemoglobin, oral CB1 inverse agonist, eases inflammatory pain.Formula:C52H80F3N13O14Purezza:98%Colore e forma:SolidPeso molecolare:1168.27Alosetron
CAS:Alosetron, a 5-HT3 antagonist, is used for the management of severe diarrhea-predominant irritable bowel syndrome (IBS) in women only.Formula:C17H18N4OPurezza:98%Colore e forma:Crystalline PowderPeso molecolare:294.36LRGILS-NH2
CAS:<p>LRGILS-NH2, reverse sequence of SLIGRL-NH2, is a control peptide for PAR2, affecting gut transit.</p>Formula:C29H56N10O7Purezza:98%Colore e forma:SolidPeso molecolare:656.82L-770644 dihydrochloride
CAS:L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.Formula:C30H38ClN7O4SColore e forma:SolidPeso molecolare:628.19GRK2i
CAS:GRK2 inhibitory polypeptide that specifically inhibits Gβγ activation of GRK2. Corresponds to the Gβγ-binding domain and acts as a cellular Gβγ antagonist.Formula:C153H256N50O41SPurezza:98%Colore e forma:SolidPeso molecolare:3484.08Eletriptan
CAS:<p>Eletriptan, second-generation triptans used to treat migraines, is used as an abortion drug.</p>Formula:C22H26N2O2SColore e forma:SolidPeso molecolare:382.52Thielavin A
CAS:Thielavin A, from T. terricola, inhibits COX and glucose-6-phosphatase; non-competitive α-glucosidase inhibitor.Formula:C29H30O10Colore e forma:SolidPeso molecolare:538.549GRL093-22
<p>GRL093-22 is an effective and selective inhibitor of G protein-coupled receptor kinases (GRK), with IC50 values of 60 nM for GRK5 and 40 nM for GRK6. It shows potential for research in heart failure and multiple myeloma.</p>Formula:C33H29FN6O3Colore e forma:SolidPeso molecolare:576.62BQ-123 TFA
BQ-123 TFA: Potent ETA antagonist, IC50 = 7.3 nM, Ki = 25 nM, inhibits ET-1 cell proliferation, lowers rat BP.Formula:C33H43F3N6O9Colore e forma:SolidPeso molecolare:724.72Besipirdine hydrochloride
CAS:<p>Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with cardiovascular activity that inhibits the uptake of biogenic amines.</p>Formula:C16H18ClN3Purezza:98.45%Colore e forma:SoildPeso molecolare:287.79Quetiapine-d4 fumarate
CAS:Deuterium-labeled Quetiapine fumarate; an antidepressant and anxiolytic 5-HT agonist, dopamine antagonist.Formula:C25H29N3O6SPurezza:98%Colore e forma:SolidPeso molecolare:503.61S1PR1 modulator 1
CAS:S1PR1 modulator 1 is a selective inhibitor of S1PR1 with a pIC50 of 7.6.Formula:C23H24N2O3SPurezza:99.69%Colore e forma:SolidPeso molecolare:408.5115(S)-15-methyl Prostaglandin D2
CAS:15(S)-15-methyl PGD2 is a stable PGD2 analog that induces vasoconstriction, raises blood pressure, and shows strong antifertility effects.Formula:C21H34O5Colore e forma:SolidPeso molecolare:366.49Tebufelone
CAS:<p>Tebufelone is a potent NSAID, inhibits CO, has anti-inflammatory and analgesic properties, and blocks lipoxygenase products (IC50 ~20-22 microM).</p>Formula:C20H28O2Purezza:99.32%Colore e forma:SolidPeso molecolare:300.44Cetirizine Impurity C dihydrochloride
CAS:Cetirizine Impurity C dihydrochloride is a Cetirizine metabolite and long-acting H1-antihistamine.Formula:C21H27Cl3N2O3Colore e forma:SolidPeso molecolare:461.81Apelin-12 acetate
Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.Formula:C66H107N21O16SPurezza:98.82%Colore e forma:SolidPeso molecolare:1482.75O-2172
CAS:<p>O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).</p>Formula:C14H16Cl2O2Colore e forma:SolidPeso molecolare:287.18Prostaglandin F2α isopropyl ester
CAS:PGF2α isopropyl ester is an ester prodrug of PGF2α with enhanced lipid solubility.Formula:C23H40O5Colore e forma:SolidPeso molecolare:396.568Tabernanthalog
CAS:<p>TBG is a 5-HT2A agonist reducing alcohol/heroin cravings and promoting neuroplasticity with antidepressant effects in rodents.</p>Formula:C14H18N2OPurezza:99.82% - 99.89%Colore e forma:SoildPeso molecolare:230.31Glucagon-like peptide 1 (1-37), human TFA
Human Glucagon-like peptide 1 (1-37) TFA is a potent GLP-1 receptor agonist derived from proglucagon.Formula:C188H276N51F3O61Purezza:98%Colore e forma:SolidPeso molecolare:4283.5Neuromedin N
CAS:<p>Neuromedin N is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct expression and effects.</p>Formula:C38H63N7O8Purezza:98%Colore e forma:SolidPeso molecolare:745.95PD 144418 oxalate
CAS:<p>PD 144418 oxalate: σ1 receptor ligand, Ki=0.08 nM; 1377 nM for σ2, minimal affinity elsewhere; potential antipsychotic.</p>Formula:C20H24N2O5Purezza:98.76%Colore e forma:SolidPeso molecolare:372.42β2AR/M-receptor agonist-1
CAS:β2AR/M-receptor agonist-1 (example 131), a muscarinic antagonist and β2 adrenoceptor agonist (MABA), exhibits dual potency towards β2 adrenoceptor andFormula:C43H56BrN3O7Colore e forma:SolidPeso molecolare:806.82PACAP-Related Peptide (PRP), human
PRP, human: 29-amino-acid PACAP precursor segment, synthesized for biological/structural research.Formula:C139H229N41O42Purezza:98%Colore e forma:SolidPeso molecolare:3146.5720-SOLA
<p>20-SOLA is the first water-soluble 20-HETE antagonist with oral bioavailability. It significantly improves blood pressure changes and kidney damage associated with the streptozotocin (STZ) diabetic mouse model. Additionally, 20-SOLA acts as a GPR75 receptor blocker. This compound is useful in research related to cardiovascular pathology.</p>Formula:C33H62O9Peso molecolare:602.43938Adrogolide HCl
CAS:Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.Formula:C22H26ClNO4SColore e forma:SolidPeso molecolare:435.96GLP-1R Antagonist 1
CAS:<p>GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).</p>Formula:C16H11ClF6N4O2Purezza:99.84%Colore e forma:SolidPeso molecolare:440.73Secretin, porcine
CAS:Porcine secretin: 27-amino acid peptide for diagnosing pancreatic dysfunction and gastrinoma, stimulates bicarbonate fluid.Formula:C130H220N44O41·xC2H4O2Purezza:98%Colore e forma:SolidPeso molecolare:N/AAlverine hydrochloride
CAS:<p>Alverine hydrochloride is a parasympatholytic.</p>Formula:C20H28ClNColore e forma:SolidPeso molecolare:317.9
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