Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(942 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.949 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(149 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(410 prodotti)
- Recettore dell'endotelina(75 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(32 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(166 prodotti)
- Proteina Hedgehog/Smoothened(45 prodotti)
- Recettore dell'istamina(359 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(298 prodotti)
- PAFR(11 prodotti)
- PKA(49 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5378 prodotti di "Proteina G/GPCR"
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Setiptiline
CAS:Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.Formula:C19H19NPurezza:98.05% - 98.07%Colore e forma:SolidPeso molecolare:261.36CGP 20712 A
CAS:<p>CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that reverses RKT-induced gastric relaxation.</p>Formula:C24H29F3N4O8SPurezza:99.37%Colore e forma:SolidPeso molecolare:590.57UCM 608
CAS:<p>UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces an increase in GDP-GTP exchange.</p>Formula:C19H20N2O2Purezza:98.88%Colore e forma:SolidPeso molecolare:308.37Trabodenoson
CAS:<p>Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.</p>Formula:C15H20N6O6Purezza:99.94%Colore e forma:SolidPeso molecolare:380.36Pentoxyverine
CAS:Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.Formula:C20H31NO3Purezza:97.11%Colore e forma:SolidPeso molecolare:333.47Levocetirizine Dihydrochloride
CAS:<p>Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.</p>Formula:C21H27Cl3N2O3Purezza:99.89%Colore e forma:White Or Off-White Crystalline PowderPeso molecolare:461.81Bucindolol
CAS:<p>Bucindolol (BMY 13105) is a novel and potent β1-adrenergic receptor blocker that mediates vasodilation and can be used to study chronic heart failure.</p>Formula:C22H25N3O2Purezza:99.9%Colore e forma:SolidPeso molecolare:363.45WAY-100635 maleate
CAS:<p>WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).</p>Formula:C25H34N4O2·xC4H4O4Purezza:>99.99%Colore e forma:White SolidPeso molecolare:538.645GRK6-IN-2
CAS:<p>GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 has been studied in multiple myeloma.</p>Formula:C21H21FN6Purezza:98.94%Colore e forma:SolidPeso molecolare:376.43SID 7969543
CAS:<p>SID 7969543 is a selective SF-1 inhibitor with potential anticancer activity, inhibits SF-1-triggered luciferase expression and can be used for cancer research.</p>Formula:C24H24N2O7Purezza:98.94%Colore e forma:SolidPeso molecolare:452.46Clopidogrel thiolactone
CAS:Clopidogrel thiolactone (2-oxoclopidogrel), a P2Y12 receptor inhibitor, is an antiplatelet aggregation compound.Formula:C16H16ClNO3SPurezza:98.79%Colore e forma:SolidPeso molecolare:337.82(R)-Mirtazapine
CAS:<p>(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.</p>Formula:C17H19N3Purezza:99.75%Colore e forma:SolidPeso molecolare:265.35Ketanserin tartrate
CAS:Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.Formula:C26H28FN3O9Purezza:99.68%Colore e forma:SolidPeso molecolare:545.51Tandospirone
CAS:<p>Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.</p>Formula:C21H29N5O2Purezza:99.94%Colore e forma:SolidPeso molecolare:383.49Alfuzosin
CAS:<p>Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and urethral dysfunction.</p>Formula:C19H27N5O4Purezza:99.64%Colore e forma:White Crystaline PowderPeso molecolare:389.45Syk Inhibitor II
CAS:<p>Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).</p>Formula:C14H15F3N6OPurezza:97.63%Colore e forma:SolidPeso molecolare:340.3L-745870
CAS:<p>L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.</p>Formula:C18H19ClN4Purezza:98%Colore e forma:SolidPeso molecolare:326.82SR59230A hydrochloride
CAS:<p>SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue thermogenesis.</p>Formula:C21H28ClNO2Purezza:99.49%Colore e forma:SolidPeso molecolare:361.91Ropinirole
CAS:<p>Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.</p>Formula:C16H24N2OPurezza:99.68%Colore e forma:SolidPeso molecolare:260.38R 59-022
CAS:<p>R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.</p>Formula:C27H26FN3OSPurezza:98.55%Colore e forma:SolidPeso molecolare:459.58Cyproheptadine hydrochloride
CAS:<p>Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.</p>Formula:C21H21N·HClPurezza:99.88% - 99.97%Colore e forma:SolidPeso molecolare:323.86Travoprost
CAS:<p>Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.</p>Formula:C26H35F3O6Purezza:97.39% - 99.58%Colore e forma:Colorless OilPeso molecolare:500.55PACAP (1-38), human, ovine, rat
CAS:PACAP (1-38), human, ovine, rat (Pituitary Adenylate Cyclase Activating Polypeptide 38) is a neuropeptide with 38 amino acid residues.Formula:C203H331N63O53SPurezza:96.93% - 98.16%Colore e forma:SolidPeso molecolare:4534.26Risperidone Mesylate
CAS:<p>Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.</p>Formula:C24H31FN4O5SPurezza:98%Colore e forma:SolidPeso molecolare:506.59P2Y14R antagonist 1
CAS:<p>P2Y14R antagonist 1 (compound I-17) is a selective oral that inhibits inflammatory response in acute gouty arthritis the NLRP3/GSDMD y and cellular pyroptosis.</p>Formula:C15H12BrN3O2Purezza:98.88%Colore e forma:SolidPeso molecolare:346.18Olopatadine
CAS:<p>Olopatadine is an antihistamine and anti-allergy medication for itchy eyes, also possibly treats red skin syndrome.</p>Formula:C21H23NO3Purezza:98%Colore e forma:White Or Off-White Crystalline PowderPeso molecolare:337.4117-phenyl trinor Prostaglandin F2α isopropyl ester
CAS:<p>17-phenyl trinor PGF2α N-ethyl amide is an F-series prostaglandin analog which has been approved for use as an ocular hypotensive drug, sold under the Allergan</p>Formula:C26H38O5Colore e forma:SolidPeso molecolare:430.58Metoxibutropate
CAS:<p>Metoxibutropate is a biochemical.</p>Formula:C20H24O3Colore e forma:SolidPeso molecolare:312.4Blontuvetmab
CAS:<p>Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].</p>Colore e forma:LiquidGPR183-IN-1
CAS:<p>GPR183-IN-1 (compound 15) is an effective orally active inhibitor of GPR183. It inhibits Ca2+ mobilization with an IC50 value of 39.97 nM. GPR183-IN-1 holds potential for research in cancer, autoimmune diseases, pain, and osteoporosis.</p>Formula:C16H19BrN2O2Colore e forma:SolidPeso molecolare:351.24Uliledlimab
CAS:<p>Uliledlimab, a humanized monoclonal antibody against CD73, reduces extracellular adenosine production and modulates immunosuppressive pathways.</p>Purezza:95% - 95%Colore e forma:LiquidN-Methyl amisulpride
CAS:<p>N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.</p>Formula:C18H29N3O4SColore e forma:SolidPeso molecolare:383.51DL-Phenylephrine HCl
CAS:DL-Phenylephrine HCl is a selective agonist of the alpha1-adrenergic receptor.Formula:C9H14ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:203.67Methaphenilene hydrochloride
CAS:<p>Methaphenilene hydrochloride is an H1 receptor antagonist with antihistaminic and anticholinergic activity, in allergic inflammation and autonomic research.</p>Formula:C15H21ClN2SPurezza:99.84%Colore e forma:SolidPeso molecolare:296.86Mibavademab
CAS:<p>Mibavademab is a humanized anti-leptin receptor (LEPR) mAb under investigation for treating congenital leptin deficiency.</p>Purezza:95%Colore e forma:LiquidKeto Ziprasidone
CAS:<p>Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors.</p>Formula:C21H19ClN4O2SPurezza:98%Colore e forma:SolidPeso molecolare:426.92Triflupromazine
CAS:<p>Triflupromazine is a dopamine receptor D1/D2 antagonist and LHDA inhibitor that suppresses dopamine activity in (CNS)mental disorders, sedation, and antiemesis.</p>Formula:C18H19F3N2SColore e forma:SolidPeso molecolare:352.42Buflomedil
CAS:<p>Buflomedil is a vasoactive compound. Buflomedil has been used for peripheral arterial diseases.</p>Formula:C17H25NO4Purezza:98%Colore e forma:SolidPeso molecolare:307.38Meticillin
CAS:<p>Methicillin: Narrow-spectrum beta-lactam, penicillin-type antibiotic for certain gram-positive bacterial infections.</p>Formula:C17H20N2O6SColore e forma:SolidPeso molecolare:380.42Fremanezumab
CAS:<p>Fremanezumab (TEV-48125) is a humanised monoclonal antibody targeting CGRP, capable of neutralising human, mouse and rat CGRP, migraine.</p>Purezza:95% - 95%Colore e forma:LiquidEptinezumab
CAS:<p>Eptinezumab is a humanised monoclonal antibody targeting CGRP (calcitonin gene-related peptide), which prevents CGRP binding to its receptor, migraine.</p>Purezza:95% - 95%Colore e forma:LiquidPF-610355
CAS:<p>PF-610355 is a long-acting and potent β2-adrenergic receptor agonist (EC50: 0.26 nM).PF-610355 can be used to study asthma and COPD.</p>Formula:C34H39N3O6SPurezza:99.73%Colore e forma:SolidPeso molecolare:617.76Arazasetron HCl
CAS:<p>Arazasetron is an antiemetic which acts as a 5-HT3 receptor antagonist, pKi = 9.27.</p>Formula:C17H20ClN3O3Purezza:98%Colore e forma:SolidPeso molecolare:349.81Tulobuterol
CAS:<p>Tulobuterol is mainly used for the prevention and treatment of bronchial asthma, asthmatic bronchitis and chronic bronchitis. Research shows that it could inhibit rhinovirus infection in primary cultures of human tracheal epithelial cells.</p>Formula:C12H18ClNOColore e forma:Crystalline SolidPeso molecolare:227.73Escitalopram
CAS:<p>Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.</p>Formula:C20H21FN2OPurezza:99.82%Colore e forma:White Or White Crystalline PowderPeso molecolare:324.39Carlumab
CAS:<p>Carlumab is a high-affinity human monoclonal antibody that targets CCL2, suppressing the recruitment of monocytes/macrophages in the tumour microenvironment.</p>Purezza:95%Colore e forma:Liquid15-keto Prostaglandin F2α
CAS:<p>15-keto Prostaglandin F2α is a metabolite of Prostaglandin F2α that lowers intraocular pressure in rabbits.</p>Formula:C20H32O5Purezza:98%Colore e forma:SolidPeso molecolare:352.47Mirtazapine D3
CAS:Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .Formula:C17H19N3Purezza:98%Colore e forma:SolidPeso molecolare:268.37Dapagliflozin-d5
CAS:Dapagliflozin D5 (BMS-512148 D5) is deuterated Dapagliflozin. Dapagliflozin is a competitive SGLT2 inhibitor.Formula:C21H25ClO6Purezza:98%Colore e forma:SolidPeso molecolare:413.9Amitriptyline-d6 Hydrochloride
CAS:<p>Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.</p>Formula:C20H18D6ClNColore e forma:SolidPeso molecolare:319.90
