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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5352 prodotti di "Proteina G/GPCR"

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  • CP-865569
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    CP-865569

    CAS:
    <p>CP-865569 is a CCR1 antagonist useful in the research of inflammatory and autoimmune diseases, including conditions such as rheumatoid arthritis and multiple sclerosis.</p>
    Formula:C22H26ClFN2O5S
    Colore e forma:Solid
    Peso molecolare:484.969

    Ref: TM-T206204

  • GPBAR1-IN-3
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    GPBAR1-IN-3

    CAS:
    <p>GPBAR1-IN-3 (Compound 14) is both a selective agonist for GPBAR1, with an EC50 value of 0.17 μM, and an antagonist for CysLT1R [1].</p>
    Formula:C21H23NO2
    Colore e forma:Solid
    Peso molecolare:321.41

    Ref: TM-T60863

  • (E/Z)-Ozagrel sodium
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    (E/Z)-Ozagrel sodium

    CAS:
    <p>(E/Z)-Ozagrel (sodium) [(E/Z)-OKY-046 (sodium)] is a mixture of the EZ isomers of Ozagrel (sodium). It acts as a thromboxane A2 (TXA2) synthase inhibitor. As an antiplatelet agent, Ozagrel (sodium) selectively inhibits human platelet aggregation, with an IC50 of 53.12 μM.</p>
    Formula:C13H11N2NaO2
    Colore e forma:Solid
    Peso molecolare:250.228

    Ref: TM-T204543

  • 2,3-dinor-11β-Prostaglandin F2α
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    2,3-dinor-11β-Prostaglandin F2α

    CAS:
    <p>2,3-dinor-11β-Prostaglandin F2α (2,3-dinor-11β-PGF2α) was recovered from the urine of both normal monkeys and humans when infused with radiolabeled PGD2, where</p>
    Formula:C18H30O5
    Colore e forma:Solid
    Peso molecolare:326.43

    Ref: TM-T37275

  • MRS2179 tetrasodium hydrate
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    MRS2179 tetrasodium hydrate

    <p>MRS2179 blocks turkey P2Y1 receptor (Kb 102 nM, pA2 6.99), affects platelet aggregation, and has varying IC50s on P2 receptors.</p>
    Formula:C11H15N5Na4O10P2
    Colore e forma:Solid
    Peso molecolare:576.21

    Ref: TM-T64078

  • Logo CymitQuimica
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    RF9 hydrochloride

    <p>RF9 hydrochloride is a potent and selective Neuropeptide FF receptor antagonist that acts on hNPFF1R (Ki: 58 nM) and hNPFF2R (Ki: 7 nM).</p>
    Formula:C26H39ClN6O3
    Colore e forma:Solid
    Peso molecolare:519.08

    Ref: TM-T63622

  • DA-302168S
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    DA-302168S

    CAS:
    <p>DA-302168S is an orally active, selective GLP-1R agonist with an EC50 value of 1.32 nM. It promotes insulin secretion and has a hypoglycemic effect. Additionally, DA-302168S reduces food intake. It primarily activates GLP-1R in humans and monkeys, with minimal effect on GLP-1R in rats, mice, and dogs. DA-302168S can be used for research in type 2 diabetes and obesity.</p>
    Formula:C33H24ClF2N3O5
    Colore e forma:Solid
    Peso molecolare:616.011

    Ref: TM-T206917

  • Logo CymitQuimica
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    SB 258741 hydrochloride

    <p>SB 258741 hydrochloride is a potent antagonist of the 5-HT 7 receptor, designed specifically for studying schizophrenia [1].</p>
    Formula:C19H31ClN2O2S
    Colore e forma:Solid
    Peso molecolare:386.98

    Ref: TM-T61724

  • Logo CymitQuimica
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    LJ-4517

    <p>LJ-4517 is an effective A2AAR antagonist (Ki=18.3 nM). LJ-4517 can effectively replace the binding of [3H] ZM241385 at WT A2AAR.</p>
    Formula:C19H21N5O3S
    Colore e forma:Solid
    Peso molecolare:399.47

    Ref: TM-T61914

  • Rivenprost
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    Rivenprost

    CAS:
    <p>Rivenprost, selective EP4 agonist (Ki: 0.7 nM), promotes bone growth, osteoblast differentiation, and aids wound healing.</p>
    Formula:C24H34O6S
    Colore e forma:Solid
    Peso molecolare:450.59

    Ref: TM-T36080

  • Taprostene
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    Taprostene

    CAS:
    <p>Taprostene (CG-4203), a stable Prostacyclin analogue, protects endothelium and myocardium post-ischemia in cats, with minimal hemodynamic impact.</p>
    Formula:C24H30O5
    Colore e forma:Solid
    Peso molecolare:398.49

    Ref: TM-T41251

  • Logo CymitQuimica
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    H3R antagonist 2

    <p>Compound 23: H3R antagonist with 170 nM Ki; inhibits AChE, BChE, hMAO B; IC50s: 180, 880, 775 nM; anti-pain, memory boost; crosses BBB. [1]</p>
    Formula:C24H29NO3
    Colore e forma:Solid
    Peso molecolare:379.49

    Ref: TM-T61603

  • Merigolix
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    Merigolix

    CAS:
    <p>Merigolix is a potent gonadotrophin releasing hormone (GnRH) antagonist .</p>
    Formula:C36H35F7N4O6
    Colore e forma:Solid
    Peso molecolare:752.68

    Ref: TM-T73327

  • CB2 receptor antagonist 1
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    CB2 receptor antagonist 1

    CAS:
    <p>Compound 29 is a potent, CB2-selective antagonist/reverse agonist. Derivatives 23 &amp; 24 offer antinociception; 24 activates cannabinoid/TRPV1 receptors.</p>
    Formula:C28H47NO3
    Colore e forma:Solid
    Peso molecolare:445.68

    Ref: TM-T62631

  • R-96544 hydrochloride
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    R-96544 hydrochloride

    CAS:
    <p>5-HT2 receptor antagonist</p>
    Formula:C22H29NO3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:355.47

    Ref: TM-T23219

  • CCR4 antagonist 2
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    CCR4 antagonist 2

    CAS:
    <p>CCR4 antagonist 2 (Compound 31) is a novel potent, orally bioavailable small molecule antagonists of CC chemokine receptor 4 (CCR4) that inhibits Treg</p>
    Formula:C26H28Cl2N6O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:511.45

    Ref: TM-T10713

  • 8-iso Prostaglandin F3α
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    8-iso Prostaglandin F3α

    CAS:
    <p>8-iso PGF3α is an isoprostane produced from the free-radical peroxidation of EPA.</p>
    Formula:C20H32O5
    Colore e forma:Solid
    Peso molecolare:352.47

    Ref: TM-T36164

  • Fasitibant
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    Fasitibant

    CAS:
    <p>Fasitibant is a potent and selective nonpeptide kinin B2 receptor antagonist.</p>
    Formula:C36H49Cl2N6O6S
    Colore e forma:Solid
    Peso molecolare:764.78

    Ref: TM-T68486

  • DMPX
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    DMPX

    CAS:
    <p>DMPX (3,7-Dimethyl-1-propargylxanthine) is a caffeine-like compound capable of crossing the blood-brain barrier. It serves as an A2-selective adenosine receptor (AR) antagonist, effectively and selectively blocking the hypothermia and behavioral inhibition induced by A2 adenosine receptor agonists, such as NECA. DMPX is utilized in research on diseases like Parkinson's disease.</p>
    Formula:C10H10N4O2
    Colore e forma:Solid
    Peso molecolare:218.212

    Ref: TM-T204595

  • BI-685509
    Targetmol
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    BI-685509

    CAS:
    <p>BI-685509: potent, oral sGC activator, boosts cGMP, enhances NO pathways, for CKD/DKD research.</p>
    Formula:C34H38N4O5
    Colore e forma:Solid
    Peso molecolare:582.69

    Ref: TM-T73332