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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

Mostrare 18 più sottocategorie

Trovati 5337 prodotti di "Proteina G/GPCR"

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  • D1R antagonist 1
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    D1R antagonist 1

    CAS:
    <p>Compound 12a (D1R antagonist 1) is a D1R antagonist that participates in both G-protein-coupled and β-arrestin-mediated signaling pathways [1].</p>
    Formula:C22H26BrNO4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:448.35

    Ref: TM-T78735

  • MRS4833
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    MRS4833

    CAS:
    <p>MRS4833 (compound 15) is an orally active, potent, competitive antagonist of P2Y14R, exhibiting IC50 values of 5.92 nM for hP2Y14R and 4.8 nM for mP2Y14R. It reduces airway eosinophilia in protease-mediated asthma models and reverses chronic neuropathic pain in mouse CCI models.</p>
    Formula:C30H24F3NO3
    Colore e forma:Solid
    Peso molecolare:503.51

    Ref: TM-T200837

  • Cendifensine
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    Cendifensine

    CAS:
    <p>Cendifensine functions as a monoamine reuptake inhibitor, targeting the serotonin transporter (SERT), norepinephrine transporter (NET), and dopamine transporter (DAT).</p>
    Formula:C14H17Cl2NO
    Colore e forma:Solid
    Peso molecolare:286.197

    Ref: TM-T206480

  • VGD071
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    VGD071

    CAS:
    <p>VGD071, a compound that targets sortilin, presents a promising avenue for forthcoming research utilizing mouse models of breast cancer.</p>
    Formula:C32H41N3O4S2
    Colore e forma:Solid
    Peso molecolare:595.82

    Ref: TM-T64206

  • GHSR-1a agonist-1
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    GHSR-1a agonist-1

    CAS:
    <p>GHSR-1a agonist-1 (Compound 4b) is an orally active agonist of the human growth hormone secretagogue receptor 1a (GHSR-1a) with an EC50 of 0.49 nM. It effectively stimulates the release of endogenous growth hormone by activating GHSR-1a. Doses as low as 0.1 mg/kg (administered orally) can increase body weight and length in 4-week-old rats. GHSR-1a agonist-1 is applicable in research on pediatric growth and developmental delays.</p>
    Formula:C30H37N5O4
    Colore e forma:Solid
    Peso molecolare:531.646

    Ref: TM-T206698

  • SCH-900822
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    SCH-900822

    CAS:
    <p>SCH-900822 is a potent and selective glucagon receptor antagonist.</p>
    Formula:C34H43Cl2N7O2
    Colore e forma:Solid
    Peso molecolare:652.66

    Ref: TM-T71201

  • Fosrolapitant
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    Fosrolapitant

    CAS:
    <p>Fosrolapitant is an antagonist of the neurokinin 1 (NK1) receptor.</p>
    Formula:C27H29F6N2O8P
    Colore e forma:Solid
    Peso molecolare:654.49

    Ref: TM-T201161

  • U91356
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    U91356

    CAS:
    <p>U91356 is an agonist of the dopamine receptors.</p>
    Formula:C13H17N3O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:231.29

    Ref: TM-T13240

  • Rodatristat
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    Rodatristat

    CAS:
    <p>Rodatristat is an effective tryptophan hydroxylase 1 and TPH2 inhibitor (IC50s: 33 nM and 7 nM, respectively).</p>
    Formula:C27H27ClF3N5O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:561.98

    Ref: TM-T16780

  • ADORA2A/PDE4D-IN-1
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    ADORA2A/PDE4D-IN-1

    CAS:
    <p>ADORA2A/PDE4D-IN-1 (Compound 9) is a dual inhibitor of the adenosine A2a receptor (ADORA2A) and phosphodiesterase 4D (PDE4D). This compound is applicable for research in bronchial asthma.</p>
    Formula:C14H11N5
    Colore e forma:Solid
    Peso molecolare:249.271

    Ref: TM-T204528

  • Bometolol Hydrochloride
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    Bometolol Hydrochloride

    CAS:
    <p>Bometolol Hydrochloride is a beta-adrenergic blocking compound used for the treatment of cardiovascular disease.</p>
    Formula:C25H33ClN2O7
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:508.99

    Ref: TM-T13585

  • PF-07258669
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    PF-07258669

    CAS:
    <p>PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.</p>
    Formula:C25H27FN6O2
    Purezza:99.9%
    Colore e forma:Solid
    Peso molecolare:462.52

    Ref: TM-T69526

  • BQ-788
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    BQ-788

    CAS:
    <p>BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation of coronary perfusion pressure.</p>
    Formula:C34H51N5O7
    Purezza:98.81%
    Colore e forma:Solid
    Peso molecolare:641.8

    Ref: TM-T10595

  • BMS-986141
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    BMS-986141

    CAS:
    <p>BMS-986141(UDM-003183) is a selective and potent protease-activated receptor-4 (PAR-4) antagonist with oral activity and an IC50 value of 0.4 nM.BMS-98614</p>
    Formula:C27H23N5O5S2
    Purezza:98.43% - 99.26%
    Colore e forma:Solid
    Peso molecolare:561.63

    Ref: TM-T63966

  • Dersimelagon
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    Dersimelagon

    CAS:
    <p>Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist.Cost-effective and quality-assured.</p>
    Formula:C36H45F4N3O5
    Purezza:97.35% - 98.23%
    Colore e forma:Solid
    Peso molecolare:675.75

    Ref: TM-T25310

  • SB-423562
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    SB-423562

    CAS:
    <p>SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.</p>
    Formula:C26H32N2O4
    Purezza:99.22%
    Colore e forma:Solid
    Peso molecolare:436.54

    Ref: TM-T12846

  • SB-224289 hydrochloride
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    SB-224289 hydrochloride

    CAS:
    <p>SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.</p>
    Formula:C32H33ClN4O3
    Purezza:97.82% - 98.99%
    Colore e forma:Solid
    Peso molecolare:557.08

    Ref: TM-T12841

  • AZD5462
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    AZD5462

    CAS:
    <p>AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart failure and cancer.</p>
    Formula:C30H41FN2O6
    Purezza:98.32% - 99.63%
    Colore e forma:Solid
    Peso molecolare:544.65

    Ref: TM-T63838

  • AZD-5672
    Targetmol
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    AZD-5672

    CAS:
    <p>AZD-5672 is an antagonist of CCR5 with an IC50 of 0.32 nM.</p>
    Formula:C32H38F2N2O5S2
    Purezza:98.1%
    Colore e forma:Solid
    Peso molecolare:632.78

    Ref: TM-T30260

  • LSN3318839
    Targetmol
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    LSN3318839

    CAS:
    <p>LSN3318839 is a potent and orally available glucagon-like peptide-1 receptor (GLP-1R) modulator.LSN3318839 enhances GLP-1R G-protein-coupled signaling and can</p>
    Formula:C26H23Cl2N3O2
    Purezza:99.21%
    Colore e forma:Solid
    Peso molecolare:480.39

    Ref: TM-T63166