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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

Mostrare 19 più sottocategorie

Trovati 5838 prodotti di "Proteina G/GPCR"

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  • U91356
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    U91356

    CAS:
    U91356 is an agonist of the dopamine receptors.
    Formula:C13H17N3O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:231.29

    Ref: TM-T13240

  • Vibegron
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    Vibegron

    CAS:
    Vibegron (MK-4618) is an effective and selective Beta 3 adrenergic receptor agonist, used to treat overactive bladder (OAB).
    Formula:C26H28N4O3
    Colore e forma:Solid
    Peso molecolare:444.53

    Ref: TM-T35052

  • AH22921
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    AH22921

    CAS:
    <p>AH22921 is an EP4 prostaglandin receptor antagonist with the ability to antagonize the activation of adenylyl cyclase by prostaglandins in CHO cells. It induces a rightward shift in the PGE? concentration-response curve in these cells, functioning as a non-competitive antagonist. AH22921 is selective for the EP4 receptor, inhibiting its activity in CHO cells without affecting the PGE? concentration-response curve in NPE cells that contain the EP2 receptor.</p>
    Formula:C29H35NO5
    Colore e forma:Solid
    Peso molecolare:477.59

    Ref: TM-T200553

  • LK 11
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    LK 11

    CAS:
    LK-11, an alkaloid derivative, inhibits the passive uptake of norepinephrine (NA) by synaptic vesicles in the thalamus, similarly to cocaine.
    Formula:C15H26N2O3
    Colore e forma:Solid
    Peso molecolare:282.38

    Ref: TM-T200284

  • Beloxepin
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    Beloxepin

    CAS:
    Beloxepin is an oral dual selective inhibitor of serotonin and norepinephrine uptake.
    Formula:C19H21NO2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:295.38

    Ref: TM-T26765

  • CCR5 antagonist 1
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    CCR5 antagonist 1

    CAS:
    CCR5 antagonist 1 is a CCR5 antagonist extracted from WO 2004054974 A2. It can inhibit HIV replication.
    Formula:C39H46ClF2N5O3S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:738.33

    Ref: TM-T10714

  • BI 639667
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    BI 639667

    CAS:
    BI 639667, an azaindazole-class compound, potently inhibits CCR1 (IC50=1.8 nM in calcium flux assays).
    Formula:C22H18FN5O3S
    Purezza:99.86%
    Colore e forma:Solid
    Peso molecolare:451.47

    Ref: TM-T14899

  • NK-1 Antagonist 1
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    NK-1 Antagonist 1

    CAS:
    NK-1 Antagonist 1 is a NK-1 receptor antagonist.
    Formula:C25H23F6N5O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:539.47

    Ref: TM-T12233

  • Logo CymitQuimica
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    CB1/2 agonist 1

    Potent CB1/2 agonist 1; crosses blood-brain barrier; anti-inflammatory, analgesic; for multiple sclerosis research.
    Formula:C21H24BrFN2O2
    Colore e forma:Solid
    Peso molecolare:435.33

    Ref: TM-T62468

  • Orvepitant
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    Orvepitant

    CAS:
    Orvepitant is a potent and selective NK1 antagonist, which may be potentially useful for patients with major depressive disorder (MDD), anxiety and insomnia.
    Formula:C31H35F7N4O2
    Colore e forma:Solid
    Peso molecolare:628.62

    Ref: TM-T69063

  • Toladryl
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    Toladryl

    CAS:
    <p>Toladryl is a derivative of Diphenhydramine that can cross the blood-brain barrier and exhibits oral activity, with antihistamine and anticholinergic properties. Its anticholinergic effects are approximately a tenth of those seen with Diphenhydramine, yet it offers 2-4 times the protection against lethal doses of histamine in guinea pigs. The side effects of Toladryl are fewer and milder compared to Diphenhydramine; however, at higher doses, it may cause symptoms such as insomnia, agitation, and disorientation related to the central nervous system. Toladryl is utilized in the research of allergic diseases.</p>
    Formula:C18H23NO
    Colore e forma:Solid
    Peso molecolare:269.38

    Ref: TM-T200797

  • MRGPRX2 modulator-3
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    MRGPRX2 modulator-3

    CAS:
    MRGPRX2 modulator-3 (Compound 4-400) is a quinoline derivative and an MRGPRX2 regulator. It is utilized in the investigation of MRGPRX2-related conditions, including allergies, itching, pain, inflammation, and autoimmune diseases.
    Formula:C21H21ClF3N5O
    Colore e forma:Solid
    Peso molecolare:451.87

    Ref: TM-T211385

  • SGL5213
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    SGL5213

    CAS:
    <p>SGL5213 is a potent oral SGLT1 inhibitor (IC50: 29 nM) with potential for treating type 2 diabetes.</p>
    Formula:C37H55N3O8
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:669.85

    Ref: TM-T12892

  • Hoe 892
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    Hoe 892

    CAS:
    Hoe 892 is a stable thia-thimo-analogue of prostacyclin and acts as a platelet aggregation inhibitor.
    Formula:C20H33NO4S
    Colore e forma:Solid
    Peso molecolare:383.55

    Ref: TM-T68751

  • Rocavorexant
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    Rocavorexant

    CAS:
    Rocavorexant is an antagonist of the orexin-1 receptor (orexin-1 receptor), exhibiting a pIC50 value of 9.1 for human OX1 and a pIC50 of 6.0 for human OX2.
    Formula:C18H19F3N8O
    Colore e forma:Solid
    Peso molecolare:420.392

    Ref: TM-T206374

  • L-796778 acetate
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    L-796778 acetate

    CAS:
    L-796778 acetate is a selective sst3 receptor agonist. In CHO-K1 cells expressing hsst3 receptors, it acts as a partial agonist that inhibits Forskolin-induced cAMP production, with an IC50 value of 18 nM. Additionally, L-796778 acetate exhibits anticonvulsant properties.
    Formula:C31H44N6O9
    Colore e forma:Solid
    Peso molecolare:644.716

    Ref: TM-T206311

  • GRK6-IN-4
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    GRK6-IN-4

    CAS:
    <p>GRK6-IN-4 is an inhibitor of G protein-coupled receptor kinase 6 (GRK6) with an IC50 value of 1.56 μM. GRK6-IN-4 is applicable for research related to hematological malignancies, inflammatory diseases, and autoimmune disorders.</p>
    Formula:C15H15N5
    Colore e forma:Solid
    Peso molecolare:265.313

    Ref: TM-T204959

  • Logo CymitQuimica
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    Meluadrine

    CAS:
    Meluadrine, a potent agonist of the β2 adrenergic receptor, is one of the metabolites of Tulobuterol [1].
    Formula:C12H18ClNO2
    Peso molecolare:243.73

    Ref: TM-T86882

  • Ersentilide
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    Ersentilide

    CAS:
    <p>Ersentilide, a benzamide derivative, functions as both a β1-adrenergic receptor antagonist and an Ikr blocker. It has demonstrated efficacy in animal models of cardiac arrhythmias.</p>
    Formula:C21H26N4O5S
    Colore e forma:Solid
    Peso molecolare:446.52

    Ref: TM-T201538

  • Arpromidine
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    Arpromidine

    CAS:
    <p>Arpromidine (BU-E-50) acts as an agonist for the histamine H2 receptor and an antagonist for the histamine H1 receptor. It demonstrates positive inotropic effects with a lower risk of inducing arrhythmias. Arpromidine can be utilized in studies related to congestive heart failure.</p>
    Formula:C21H25FN6
    Colore e forma:Solid
    Peso molecolare:380.462

    Ref: TM-T204236