Product Information
- 6-Bromo-N-(3,4,5-trimethoxyphenyl)-4-quinolinamine
A potent and selective inhibitor of cyclin G-associated kinase (GAK) with Ki of 3.1 nM. The compound has more than 50-fold selectivity over the closest off-target kinase RIPK2, making it a potent tool for the study of GAK biology. SGC-GAK-1 was tested in vitro in human prostate carcinoma cell lines and showed strong growth inhibition in cell lines with androgen-dependent growth.
Chemical properties
Technical inquiry about: 3D-FB166265 SGC GAK 1
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