Estimated delivery in United States, on Tuesday 21 Jan 2025
Product Information
Name:
SGC GAK 1
Synonyms:
- 6-Bromo-N-(3,4,5-trimethoxyphenyl)-4-quinolinamine
Description:
A potent and selective inhibitor of cyclin G-associated kinase (GAK) with Ki of 3.1 nM. The compound has more than 50-fold selectivity over the closest off-target kinase RIPK2, making it a potent tool for the study of GAK biology. SGC-GAK-1 was tested in vitro in human prostate carcinoma cell lines and showed strong growth inhibition in cell lines with androgen-dependent growth.
Notice:
Our products are intended for lab use only. For any other use, please contact us.
Brand:
Biosynth
Long term storage:
Notes:
Chemical properties
Molecular weight:
388.04226
Formula:
C18H17BrN2O3
Purity:
Min. 95%
Color/Form:
Solid
InChI:
InChI=1S/C18H17BrN2O3/c1-22-16-9-12(10-17(23-2)18(16)24-3)21-15-6-7-20-14-5-4-11(19)8-13(14)15/h4-10H,1-3H3,(H,20,21)
InChI key:
InChIKey=AUOSKLDNVNGKRR-UHFFFAOYSA-N
SMILES:
COc1cc(Nc2ccnc3ccc(Br)cc23)cc(OC)c1OC
MDL:
Melting point:
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Density:
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EINECS:
Merck:
HS code:
Technical inquiry about: 3D-FB166265 SGC GAK 1
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