
Ciclo celular/Ponto de verificação
Os inibidores do ciclo celular/ponto de verificação são compostos que interrompem a progressão normal do ciclo celular, particularmente em pontos de verificação regulatórios chave. Esses inibidores são cruciais para estudar a divisão celular, entender a proliferação de células cancerígenas e desenvolver terapias anticâncer. Ao direcionar fases específicas do ciclo celular, esses inibidores podem induzir a parada do ciclo celular, levando à apoptose ou senescência em células de divisão rápida. Na CymitQuimica, oferecemos uma ampla gama de inibidores de alta qualidade do ciclo celular/ponto de verificação para apoiar sua pesquisa em biologia do câncer, biologia celular e desenvolvimento de medicamentos.
Subcategorias de "Ciclo celular/Ponto de verificação"
- Aurora Quinase(94 produtos)
- CDK(500 produtos)
- Ciclo celular/Parada(4 produtos)
- Chk(42 produtos)
- DYRK(48 produtos)
- Dinamina(23 produtos)
- Ferroptose(215 produtos)
- HSP(169 produtos)
- Integrinas(224 produtos)
- Cinesina(66 produtos)
- LIM Quinase(19 produtos)
- Microtúbulo associado(261 produtos)
- PKC(102 produtos)
- PLK(28 produtos)
- ROCK(70 produtos)
- Rho(2 produtos)
- Wee1(15 produtos)
- c-Myc(69 produtos)
Exibir 10 mais subcategorias
Foram encontrados 3477 produtos de "Ciclo celular/Ponto de verificação"
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Arabinosylhypoxanthine
CAS:<p>Arabinosylhypoxanthine inhibits Ns5b polymerase in hepatitis C virus and can be used in biochemical experiments and organic synthesis.</p>Fórmula:C10H12N4O5Pureza:99.71%Cor e Forma:SolidPeso molecular:268.232'-Deoxy-2'-fluoro-3-Deaza-arabinouridine
CAS:<p>Nucleoside Derivatives - Fluoro-modified nucleosides, Arabino-nucleosides, Pyridine nucleosides, 3-Deazauridines, 2’-Modified nucleosides</p>Fórmula:C10H12FNO5Cor e Forma:SolidPeso molecular:245.22'-O-MOE-5MeU-3'-phosphoramidite
CAS:<p>2'-O-MOE-5MeU-3'-phosphoramidite is a Nucleoside Phosphoramidite.</p>Fórmula:C43H55N4O10PCor e Forma:SolidPeso molecular:818.899-(3-Deoxy-3-fluoro-β-D-ribofuranosyl)-6-(pyridine-4-yl)purine
CAS:<p>9-(3-Deoxy-3-fluoro-β-D-ribofuranosyl)-6-(pyridine-4-yl)purine is a Nucleoside Derivative - Fluoro-modified nucleoside, 6-Modified purine nucleoside, 3'-</p>Fórmula:C15H14FN5O3Cor e Forma:SolidPeso molecular:331.35'-O-DMTr-2',2'-difluoro-dC(Bz)-3'-CED-phosphoramidite
CAS:<p>Nucleoside Derivatives - Fluoro-modified nucleosides; 2’-Modified nucleosides; Nucleoside Phosphoramidites</p>Fórmula:C46H50F2N5O8PCor e Forma:SolidPeso molecular:869.895-(1-Hydroxy)(methoxycarbonyl)methyl uridine
CAS:<p>5-(1-Hydroxy)(methoxycarbonyl)methyl uridine is a Nucleoside Derivative - 5-Modified pyrimidine nucleoside; Naturally modified ribo-nucleoside.</p>Fórmula:C12H16N2O9Cor e Forma:SolidPeso molecular:332.261-O-Acetyl-2-O-benzoyl-3-O-tert-butyldiphenylsilyl-L-threofuranose
CAS:<p>1-O-Acetyl-2-O-benzoyl-3-O-tert-butyldiphenylsilyl-L-threofuranose is a Carbohydrate Derivative.</p>Fórmula:C29H32O6SiCor e Forma:SolidPeso molecular:504.65N1,N3-Bis(cyanomethyl)pseudouridine
<p>N1,N3-Bis(cyanomethyl)pseudouridine is a Nucleoside Derivative - C-nucleoside;N-Alkylated nucleoside.</p>Cor e Forma:Soild4',5'-Didehydro-5'-deoxy-5-methyluridine
CAS:<p>4',5'-Didehydro-5'-deoxy-5-methyluridine is a Nucleoside Derivative - 5'-Modified nucleoside, Didehydro-nucleoside.</p>Fórmula:C10H12N2O5Cor e Forma:SolidPeso molecular:240.213'-β-C-Methyl-5-trifluoromethyluridine
<p>3'-beta-C-Methyl-5-trifluoromethyluridine is a Nucleoside Derivative - 3'-Modified nucleoside, 5-Modified pyrimidine nucleoside, Fluoro-modified nucleoside.</p>Cor e Forma:SoildN6-(2-Propynyl)adenosine
CAS:<p>N6-(2-Propynyl)adenosine is a Nucleoside Derivative - 6-Modified purine nucleoside.</p>Fórmula:C13H15N5O4Cor e Forma:SolidPeso molecular:305.296-(2-O-Methyl-β-D-ribofuranosyl)-3-(2-oxo-propyl)-6H-imidazo[1,2-c]pyrimidin-5-one
CAS:<p>Nucleoside Derivatives - 2’-Modified nucleosides; Scaffolds and Templates;Bi-Tricyclic nucleosides</p>Fórmula:C15H19N3O6Cor e Forma:SolidPeso molecular:337.33α-5-Methyluridine
CAS:<p>Alpha-5-Methyluridine is a useful organic compound for research related to life sciences. The catalog number is TNU1643 and the CAS number is 3258-09-1.</p>Fórmula:C10H14N2O6Cor e Forma:SolidPeso molecular:258.23Methyl 2-deoxy-3,5-di-O-benzoyl-2-fluoro-4-thio-D-arabinopentofuranoside
CAS:<p>Methyl 2-deoxy-3,5-di-O-benzoyl-2-fluoro-4-thio-D-arabinopentofuranoside is a useful organic compound for research related to life sciences.</p>Fórmula:C20H19FO5SCor e Forma:SolidPeso molecular:390.437-TFA-ap-7-Deaza-dG
CAS:<p>5'-O-TBDMS-dG, a modified nucleoside, is utilized in the synthesis of deoxyribonucleic acid or nucleic acid.</p>Fórmula:C16H16F3N5O5Cor e Forma:SolidPeso molecular:415.3292-Thiopseudouridine
CAS:<p>Nucleoside Derivatives - C-nucleosides; Thio-nucleosides</p>Fórmula:C9H12N2O5SCor e Forma:SolidPeso molecular:260.275'-homocytidine
CAS:<p>5'-homocytidine is a useful organic compound for research related to life sciences. The catalog number is TNU1672 and the CAS number is 55085-34-2.</p>Fórmula:C10H15N3O5Cor e Forma:SolidPeso molecular:257.242'-O-Methyl-5-methylcytidine
CAS:<p>2'-O-Methyl-5-methylcytidine is a 2'-O-Methyl nucleoside.</p>Fórmula:C11H17N3O5Cor e Forma:SolidPeso molecular:271.275-Ethyl-4-thiouridine
CAS:<p>5-Ethyl-4-thiouridine is a Nucleoside Derivative - Thio-nucleoside, 5-Modified pyrimidine nucleoside.</p>Fórmula:C11H16N2O5SCor e Forma:SolidPeso molecular:288.322'-O-MOE-5-Me-C(Bz)
CAS:<p>Nucleoside Phosphoramidites; Ready for phosphorylation</p>Fórmula:C50H60N5O10PCor e Forma:SolidPeso molecular:922.012'-Chloro-N6-(4-methoxy)benzyl adenosine
CAS:<p>2'-Chloro-N6-(4-methoxy)benzyl adenosine is a Nucleoside Derivative - Halo-nucleoside;2-Modified purine nucleoside; 6-Modified purine nucleoside;.</p>Fórmula:C18H20ClN5O5Cor e Forma:SolidPeso molecular:421.836-Chloropurine -9-β-D-(3',5'-di-O-benzoyl-2'-deoxy-2'-fluoro)arabinoriboside
CAS:<p>6-Chloropurine -9-beta-D-(3',5'-di-O-benzoyl-2'-deoxy-2'-fluoro)arabinoriboside is a Fluoro-modified nucleoside; Halo-nucleoside; Arabino-nucleoside.</p>Fórmula:C24H18ClFN4O5Cor e Forma:SolidPeso molecular:496.877-Deazaguanosine
CAS:<p>Nucleoside Derivatives - 7-Deaza-purine nucleosides; Drugs and Inhibitors; Antiviral agent, anti-HCV</p>Fórmula:C11H14N4O5Cor e Forma:SolidPeso molecular:282.252'-O-(2-Azidoethyl)adenosine
CAS:<p>2'-O-(2-azidoethyl)adenosine is a purine nucleoside analog with potential antitumor activity.</p>Fórmula:C12H16N8O4Pureza:95%Cor e Forma:SolidPeso molecular:336.315-(3-Azidopropyl)cytidine
<p>5-(3-Azidopropyl)cytidine is a Nucleoside Derivative - 5-Modified pyrimidine nucleoside; Azido nucleoside.</p>Cor e Forma:Soild9-(2,3-Di-O-acetyl-6-O-benzoyl-5-deoxy-D-ribo-exofuranoyl)-6-chloropurine
<p>9-(2,3-Di-O-acetyl-6-O-benzoyl-5-deoxy-D-ribo-exofuranoyl)-6-chloropurine is a useful organic compound for research related to life sciences and the catalog</p>Cor e Forma:Soild1-(b-D-Xylofuranosyl)-6-azauracil
CAS:<p>1-(b-D-Xylofuranosyl)-6-azauracil is a Nucleoside Derivative - Xylo-nucleoside; 6-Aza-uridine.</p>Fórmula:C8H11N3O6Cor e Forma:SolidPeso molecular:245.195'-O-DMTr-3'-deoxyuridine 2'-CED phosphoramidite
CAS:<p>Nucleoside Derivatives –3’-Deoxy nucleosides;Nucleoside Phosphoramidites</p>Fórmula:C39H47N4O8PCor e Forma:SolidPeso molecular:730.79Adenosine-2-carboxamide
CAS:<p>Adenosine-2-carboxamide is a Nucleoside Derivative - 2-Modified purine nucleoside.</p>Fórmula:C11H14N6O5Cor e Forma:SolidPeso molecular:310.275'-O-Acetyl-2',3'-dideoxy-2',3'-didehydro-5-fluoro-uridine
CAS:<p>5'-O-Acetyl-2',3'-dideoxy-2',3'-didehydro-5-fluoro-uridine is a Nucleoside Derivative - Didehydro-nucleoside; Fluoro-modified nucleoside.</p>Fórmula:C11H11FN2O5Cor e Forma:SolidPeso molecular:270.212'-Amino-2'-deoxy-5-methyluridine
CAS:<p>Nucleoside Derivatives - Amino-nucleosides, 2’-Modified nucleosides, 5-Modified pyrimidine nucleosides</p>Fórmula:C10H15N3O5Cor e Forma:SolidPeso molecular:257.245-Aminomethyl uridine hydrochloride
CAS:<p>Nucleoside Derivatives - 5-Modified pyrimidine nucleosides; Amino nucleosides; Naturally modified ribo-nucleosides</p>Fórmula:C10H15N3O6Cor e Forma:SolidPeso molecular:273.245-Amino-2'-deoxyuridine hydrochloride
CAS:<p>5-Amino-2'-deoxyuridine hydrochloride is a Nucleoside Derivative - 5-Modified pyrimidine nucleoside; Amino nucleoside.</p>Fórmula:C9H14ClN3O5Cor e Forma:SolidPeso molecular:279.685-Methoxycarbonylmethyl-2-thiouridine
CAS:<p>5-Methoxycarbonylmethyl-2-thiouridine is a Nucleoside Derivative - Thio-nucleoside, 5-Modified pyrimidine nucleoside;Naturally modified ribo-nucleoside.</p>Fórmula:C12H16N2O7SCor e Forma:SolidPeso molecular:332.335'-O-TBDPS-5-methyl-2,2'-anhydrouridine
CAS:<p>5'-O-TBDPS-5-methyl-2,2'-anhydrouridine is a Nucleoside Derivative - Protected nucleoside with NH2/OH open.</p>Fórmula:C26H30N2O5SiCor e Forma:SolidPeso molecular:478.611-(b-D-Xylofuranosyl)uracil
CAS:<p>1-(b-D-Xylofuranosyl)uracil is a Nucleoside Derivative - Xylo-nucleoside.</p>Fórmula:C9H12N2O6Cor e Forma:SolidPeso molecular:244.22'-Deoxy-isoguanosine
CAS:<p>2'-Deoxy-isoguanosine is a Nucleoside Derivative - Iso-guanosine Derivative.</p>Fórmula:C10H13N5O4Cor e Forma:SolidPeso molecular:267.244'-Azido-3'-O-benzoyl-5'-O-(m-chlorobenzoyl)-2'-deoxy-2'-fluoro-β-D-arabinouridine
CAS:<p>Nucleoside Derivatives - Fluoro-modified nucleosides; Azido-nucleosides; 4’-Modified nucleosides</p>Fórmula:C23H17ClFN5O7Cor e Forma:SolidPeso molecular:529.863-Deoxy-1,2-O-isopropylidene-5-O-(p-toluoyl)- α-D-glycero-pent-3-enofuranose
CAS:<p>3-Deoxy-1,2-O-isopropylidene-5-O-(p-toluoyl)- α-D-glycero-pent-3-enofuranose is a useful organic compound for research related to life sciences.</p>Fórmula:C16H18O5Cor e Forma:SolidPeso molecular:290.31DMTr-dH2U-amidite
CAS:<p>Nucleoside Phosphoramidites; Nucleoside Derivatives - 2-Deoxy uridines</p>Fórmula:C39H47N4O7PCor e Forma:SolidPeso molecular:714.794-Amino-5-cyano-1-(β-D-ribofuranosyl)-7H-pyrrolo[2,3-d] pyrimidine
CAS:<p>Nucleoside Derivatives - 7-Deaza-purine nucleosides; Scaffolds and Templates</p>Fórmula:C12H13N5O4Cor e Forma:SolidPeso molecular:291.264-Deoxy-xylo-uridine
CAS:<p>Nucleoside Derivatives - Xylo-nucleosides; 4-Deoxy pyrimidine nucleosides</p>Fórmula:C9H12N2O5Cor e Forma:SolidPeso molecular:228.22'-Deoxy-2'-fluoro-3',5'-bis-O-TBDMS-uridine
CAS:<p>Nucleoside Derivatives –Fluoro-modified nucleosides;</p>Fórmula:C21H39FN2O5Si2Cor e Forma:SolidPeso molecular:474.714-Chloro-5-iodo-7-(2-deoxy-b-D-ribofuranosyl)-7H-pyrrolo[2,3-d]pyrimidine
CAS:<p>4-Chloro-5-iodo-7-(2-deoxy-b-D-ribofuranosyl)-7H-pyrrolo[2,3-d]pyrimidine is a Nucleoside Derivative - Halo-nucleoside, 7-Deaza-purine nucleoside.</p>Fórmula:C11H11ClIN3O3Cor e Forma:SolidPeso molecular:395.58N4-Desmethyl-N5-Methyl wyosine
CAS:<p>N4-Desmethyl-N5-Methyl wyosine is a Nucleoside Derivative - Bi-/Tri-cyclic nucleoside; naturally modified ribo-nucleoside.</p>Fórmula:C14H17N5O5Cor e Forma:SolidPeso molecular:335.321-[6-(Diethoxyphosphinyl)-2-O-(2-methoxyethyl)-β-D-ribo-hexofuranosyl]uracil
<p>Nucleoside Derivatives - Phosphorus-containing nucleosides; 2’-Modified nucleosides; 5’-Modified nucleosides</p>Cor e Forma:Soild1,2'-O-Dimethyl guanosine
CAS:<p>1,2'-O-Dimethyl guanosine is a Nucleoside Derivative - 3'-Modified nucleoside, N-Methylated/ alkylated nucleoside.</p>Fórmula:C12H17N5O5Cor e Forma:SolidPeso molecular:311.29Isocytidine
CAS:<p>Nucleosides - isocytidine derivative</p>Fórmula:C9H13N3O5Cor e Forma:SolidPeso molecular:243.222',3',5'-Tri-O-benzoyl-5-methoxyuridine
CAS:<p>2',3',5'-Tri-O-benzoyl-5-methoxyuridine is a 5-Modified Pyrimidine Nucleoside.</p>Fórmula:C31H26N2O10Cor e Forma:SolidPeso molecular:586.552-Methoxy-9-(β-D-ribofuranosyl)purine
CAS:<p>Nucleoside Derivatives - 6-De-aminopurine nucleosides, 2-Modified purine nucleosides</p>Fórmula:C11H14N4O5Cor e Forma:SolidPeso molecular:282.252'-Deoxy-2'-fluoro-N1-methyl inosine
CAS:<p>Nucleoside Derivatives - 2’-Modified nucleosides, Fluoro-modified nucleosides, N-Methylated /alkylated nucleosides</p>Fórmula:C11H13FN4O4Cor e Forma:SolidPeso molecular:284.242'-Chloro-2'-deoxyuridine
CAS:<p>2'-Chloro-2'-deoxyuridine is a Halo-nucleoside.</p>Fórmula:C9H11ClN2O5Cor e Forma:SolidPeso molecular:262.652'-Deoxy-N6,N6-dimethyladenosine
CAS:<p>2'-Deoxy-N6,N6-dimethyladenosine is a Nucleoside Derivative - 6-Modified purine nucleoside.</p>Fórmula:C12H17N5O3Cor e Forma:SolidPeso molecular:279.31-(b-D-Xylofuranosyl)-5-methylcytosine
CAS:<p>Nucleoside Derivatives –5-Modified pyrimidine nucleosides;Xylo-nucleosides</p>Fórmula:C10H15N3O5Cor e Forma:SolidPeso molecular:257.243'-O-Methyl-5-methyluridine
CAS:<p>3'-O-Methyl-5-methyluridine is a Nucleoside Derivative - 3'-Modified nucleoside.</p>Fórmula:C11H16N2O6Cor e Forma:SolidPeso molecular:272.251-Amino-7-cyclopropylmethyl-7,8-dihydro-8-oxo-9-(b-D-xylofuranosyl)guanine
CAS:<p>Nucleoside Derivatives - Xylo-nucleosides; 8-Modified purine nucleosides; Amino nucleosides; N-Methylated alkylated nucleosides</p>Fórmula:C14H20N6O6Cor e Forma:SolidPeso molecular:368.356-Chloro-9-(2,3,5-tri-O-benzoyl-2-C-methyl-β-D-ribofuranosyl)-9H-purine
CAS:<p>6-Chloro-9-(2,3,5-tri-O-benzoyl-2-C-methyl-β-D-ribofuranosyl)-9H-purine is a 2'-C-Methyl nucleoside; Halo-nucleoside.</p>Fórmula:C32H25ClN4O7Cor e Forma:SolidPeso molecular:613.021-(b-D-Xylofuranosyl)-5-trifluoromethyluracil
<p>1-(b-D-Xylofuranosyl)-5-trifluoromethyluracil is a Nucleoside Derivative - Xylo-nucleoside, Fluoro-modified nucleoside, 5-Modified pyrimidine nucleoside.</p>Cor e Forma:Soild2-Cyanoadenosine
CAS:<p>Nucleoside Derivatives - 2’-Modified purine nucleosides</p>Fórmula:C11H12N6O4Cor e Forma:SolidPeso molecular:292.255-Iodoarabinouridine
CAS:<p>5-Iodoarabinouridine is a Halo-nucleoside; Arabino-nucleoside.</p>Fórmula:C9H11IN2O6Cor e Forma:SolidPeso molecular:370.1N1-Ethylpseudouridine
CAS:<p>N1-Ethylpseudouridine is a Nucleoside Derivative - C-nucleoside; N-Methylated nucleoside.</p>Fórmula:C11H16N2O6Cor e Forma:SolidPeso molecular:272.252'-Deoxy-O6-[2-(4-nitrophenylethyl)]guanosine
CAS:<p>2'-Deoxy-O6-[2-(4-nitrophenylethyl)]guanosine is a Nucleoside Derivative - 6-Modified purine nucleoside.</p>Fórmula:C18H20N6O6Cor e Forma:SolidPeso molecular:416.39KS15
CAS:<p>KS15 is a cryptochrome (CRY) inhibitor that promotes G1 cell cycle arrest, enhances drug sensitivity in MCF-7 cells, antitumour against human breast cancer.</p>Fórmula:C20H22BrNO4Cor e Forma:SolidPeso molecular:420.33'-O-DMTr-thymidine 5'-CE phosphoramidite
CAS:<p>3'-O-DMTr-thymidine 5'-CE phosphoramidite (2'-OMe-U Phosphoramidite) is a purine nucleoside analog and phosphoramidite derivative .</p>Fórmula:C40H49N4O8PPureza:99.42%Cor e Forma:SolidPeso molecular:744.81Lifitegrast sodium
CAS:<p>Lifitegrast sodium (SAR-1118-023 sodium) is an integrin antagonist that reduces ocular surface inflammation and can be used to study dry eye.</p>Fórmula:C29H23Cl2N2NaO7SPureza:99.33%Cor e Forma:SolidPeso molecular:637.46GP-82996
CAS:<p>GP-82996 (CINK4) inhibits CDK4/6; IC50s: 1.5 μM (CDK4/D1), 5.6 μM (CDK6/D1), 25 μM (Cdk5/p35); triggers U2OS cancer cell apoptosis.</p>Fórmula:C27H32N6OPureza:99.94%Cor e Forma:SolidPeso molecular:456.58HDGFRP2/PSIP1-IN-1
CAS:<p>Compound BPP (HDGFRP2/PSIP1-IN-1) is a dual inhibitor targeting the PWWP domains of Hepatoma-derived Growth Factor Related Protein 2 (HDGFRP2) and its homologue PSIP1. This compound effectively hinders the occurrence and progression of Diffuse Intrinsic Pontine Glioma (DIPG). It demonstrates binding affinity with a Kd value of 7 μM for HDGFRP2, indicative of its efficient ligand efficacy at 0.47. Additionally, Compound BPP exhibits a Kd value of 27 μM when binding to the PSIP1 PWWP domain, and a Kd value of 14 μM against HDGFRP3, confirming its potency as an inhibitor within the HDGFRP2 PWWP subfamily.</p>Fórmula:C8H6BrN3Cor e Forma:SolidPeso molecular:224.06Napropamide
CAS:<p>Napropamide is an acetamide herbicide that inhibits root growth to control annual grasses and broadleaf weeds.</p>Fórmula:C17H21NO2Pureza:99.14%Cor e Forma:Colorless Crystals; (Tech Brown Solid) White-Like CrystalPeso molecular:271.35N-6-Furfurylguanosine
CAS:<p>N-6-Furfurylguanosine (kinetin riboside) is a purine nucleoside analog with cytotoxicity, inhibiting the growth of cancer cells.</p>Fórmula:C15H18N6O5Pureza:99.58%Cor e Forma:SolidPeso molecular:362.345,6-Dihydrothymidine
CAS:<p>2'-Deoxy-N2-methylguanosine is a purine nucleoside analog that can be used as a chemical probe to study DNA-protein interactions.</p>Fórmula:C10H16N2O5Pureza:99.90%Cor e Forma:SolidPeso molecular:244.24(S)-GNA-T-phosphoramidite
CAS:<p>(S)-GNA-T-phosphoramidite is a nucleoside analog commonly used in the synthesis of other active compounds.</p>Fórmula:C38H47N4O7PPureza:99.35%Cor e Forma:SolidPeso molecular:702.785-Aza-7-deazaguanine
CAS:<p>5-Aza-7-deazaguanine is a non-natural substituted nucleobase with potential antiviral activity, used in cancer and bacterial infection research.</p>Fórmula:C5H5N5OPureza:98.87%Cor e Forma:SolidPeso molecular:151.13DTP3
CAS:<p>DTP3 is a selective MKK7/GADD45β inhibitor, which inhibits cancer-selective NF-κB survival pathway.</p>Fórmula:C26H35N7O5Cor e Forma:SolidPeso molecular:525.62'-Amino-2'-deoxy-b-D-arabino-5-methyl uridine
CAS:<p>2'-Amino-2'-deoxy-b-D-arabino-5-methyl uridine is a purine nucleoside analog with potential antitumor activity.</p>Fórmula:C10H15N3O5Pureza:96.76%Cor e Forma:SolidPeso molecular:257.24A-674563
CAS:<p>A-674563 is an Akt1 inhibitor with Ki of 11 nM, modest potent to PKA and >30-fold selective for Akt1 over PKC.</p>Fórmula:C22H22N4OPureza:99.21%Cor e Forma:SolidPeso molecular:358.44GPRP
CAS:<p>GPRP (Gly-Pro-Arg-Pro) is a fibrin polymerization inhibitor.</p>Fórmula:C18H31N7O5Cor e Forma:White To Off-White PowderPeso molecular:425.48Maleic hydrazide
CAS:<p>Maleic hydrazide is a plant germination inhibitor that participates in nucleic acid metabolism pathways ,inhibiting cell division in the apical meristem.</p>Fórmula:C4H4N2O2Pureza:98.4%Cor e Forma:Crystals From Water Maleic Hydrazide Is An Odorless White Solid Sinks In Water (Uscg 1999)Peso molecular:112.09N6-Bz-5'-O-DMTr-3'-deoxyadenosine-2'-O-CED-phosphoramidite
CAS:<p>N6-Bz-5'-O-DMTr-3'-deoxyadenosine-2'-O-CED-phosphoramidite is an adenine nucleoside analog with potential vasodilator activity and anticancer activity.</p>Fórmula:C47H52N7O7PPureza:98.59%Cor e Forma:SolidPeso molecular:857.932'-O-Methylinosine
CAS:<p>2'-O-Methylinosine (2'-(o-Methyl)-inosine) is an orally bioavailable purine nucleoside analog with antihypertensive activity.</p>Fórmula:C11H14N4O5Pureza:99.88%Cor e Forma:SolidPeso molecular:282.252',5-Difluoro-2'-deoxy-1-arabinosyluracil
CAS:<p>2',5-Difluoro-2'-deoxy-1-arabinosyluracil (2'-Deoxy-2'-fluoro-5-fluoro-arabinouridine) is a urinary pyrimidine nucleoside analogue with potential antiepileptic</p>Fórmula:C9H10F2N2O5Pureza:99.94%Cor e Forma:SolidPeso molecular:264.18NU6102
CAS:<p>NU6102 is a CDK2 inhibitor with antitumor activity against CDK1/cyclinB, CDK1/CDK2, CDK4, DYRK1A , PDK1, and ROCKII, and it can be used to study rectal cancer.</p>Fórmula:C18H22N6O3SPureza:99.76%Cor e Forma:SolidPeso molecular:402.47LDC4297
CAS:<p>LDC4297 (LDC044297) is a potent and selective CDK7 inhibitor.</p>Fórmula:C23H28N8OPureza:98.25%Cor e Forma:SolidPeso molecular:432.52GW406108X
CAS:<p>GW406108X is a Kif15 and ULK1 inhibitor; IC50: 0.82 µM (ATPase), pIC50: 6.37; blocks autophagy.</p>Fórmula:C20H11Cl2NO4Pureza:98%Cor e Forma:SolidPeso molecular:400.21IRES-C11
CAS:<p>IRES-C11 is a specific inhibitor of translation that targets the internal ribosome entry site (IRES) of the c-MYC gene. It functions by blocking the interaction between heterogeneous nuclear ribonucleoprotein A1, a trans-acting factor required for c-MYC IRES activity, and its corresponding IRES. Notably, IRES-C11 does not inhibit the IRES activity of BAG-1, XIAP, and p53.</p>Fórmula:C13H11Cl2NO4Pureza:99.89%Cor e Forma:SolidPeso molecular:316.14Poloxime
CAS:<p>Poloxime is a hydrolysis product of poloxin and is a non-ATP-competitive Plk1 inhibitor. It also has moderate Plk1 inhibitory activity.</p>Fórmula:C10H13NO2Pureza:98%Cor e Forma:SolidPeso molecular:179.22TAME
CAS:<p>Tosyl-L-Arginine Methyl Ester (TAME (N-4-Tosyl-L-arginine methyl ester)) is an APC inhibitor.</p>Fórmula:C14H22N4O4SPureza:98%Cor e Forma:SolidPeso molecular:342.41Cilengitide TFA
CAS:<p>Cilengitide, αvβ3/αvβ5 inhibitor, IC50: 4.1/79 nM in vitro. 10x selectivity vs. gpIIbIIIa. Phase 2.</p>Fórmula:C29H41F3N8O9Cor e Forma:SolidPeso molecular:702.68Nolatrexed dihydrochloride
CAS:<p>Nolatrexed dihydrochloride (Thymitaq) is a soluble, lipophilic cancer drug that inhibits DNA replication, causing cell cycle arrest and apoptosis.</p>Fórmula:C14H14Cl2N4OSPureza:97.02%Cor e Forma:Tan SolidPeso molecular:357.26CCT244747
CAS:<p>CCT244747 is a potent and selective CHK1 inhibitor oral, ATP-competitive, and cytotoxic, abrogating drug-induced S and G2 blockade and inducing apoptosis .</p>Fórmula:C20H24N8O2Pureza:99.17%Cor e Forma:SolidPeso molecular:408.46Ribociclib hydrochloride
CAS:<p>Ribociclib hydrochloride is a highly specific CDK4/6 inhibitor (IC50: 10 nM and 39 nM, respectively).</p>Fórmula:C23H31ClN8OPureza:98%Cor e Forma:SolidPeso molecular:471sAJM589
CAS:<p>sAJM589 is a Myc inhibitor that dose-dependently disrupts Myc-Max heterodimers, thereby decreasing Myc protein levels and inhibiting the cellular proliferation.</p>Fórmula:C16H10N2OPureza:98%Cor e Forma:SolidPeso molecular:246.26Synucleozid hydrochloride
CAS:<p>Synucleozid hydrochloride inhibits the translation of the intrinsically disordered protein α-synuclein by targeting its structured mRNA.</p>Fórmula:C22H21ClN6Pureza:98.13%Cor e Forma:SolidPeso molecular:404.9N,N-Dimethyl-2'-O-methylcytidine
CAS:<p>N,N-Dimethyl-2'-O-methylcytidine (N4, N4, 2'-O-Trimethylcytidine) is a purine nucleoside analogue with anti-cancer activity.</p>Fórmula:C12H19N3O5Pureza:99.62%Cor e Forma:SolidPeso molecular:285.38-Chloroinosine
CAS:<p>8-Chloroinosine is a purine nucleoside analog and a metabolite of the anticancer compound 8-chloro-adenosine.</p>Fórmula:C10H11ClN4O5Pureza:99.37% - 99.56%Cor e Forma:SolidPeso molecular:302.67Kinesore
CAS:<p>Kinesore is a cell-permeable modulator that binds to the microtubule motor protein kinesin-1, thereby inhibiting the interaction between KLC2 and SKIP.</p>Fórmula:C20H16Br2N4O4Pureza:97.24%Cor e Forma:SolidPeso molecular:536.175'-O-DMT-N2-ibu-dG
CAS:<p>5'-O-DMT-N2-ibu-dG is a deoxynucleoside served as a building block in oligonucleotide synthesis, with protecting groups to prevent unwanted reactions.</p>Fórmula:C35H37N5O7Pureza:98.71%Cor e Forma:SolidPeso molecular:639.78-Bromoadenosine
CAS:<p>8-Bromoadenosine is an adenosine derivative. 8-Br-Adenosine inhibitis mitochondrial membrane potential, cytoplasmic Ca²⁺ levels, and RNA and protein synthesis.</p>Fórmula:C10H12BrN5O4Pureza:99.11%Cor e Forma:SolidPeso molecular:346.14NSC 23766
CAS:<p>NSC 23766 is a Rac1 GTPase inhibitor by targeting GEFs, inhibiting cell proliferation.NSC23766 competitively inhibits M2 mAChR-induced Rac1 activation.</p>Fórmula:C24H35N7Pureza:99.49%Cor e Forma:SolidPeso molecular:421.58N2-Isobutyryl-2-deoxyguanosine
CAS:<p>N2-Isobutyryl-2-deoxyguanosine(iBu-dG) is a nucleoside analog that can be used to synthesize oligonucleotides.</p>Fórmula:C14H19N5O5Pureza:97.03%Cor e Forma:SolidPeso molecular:337.33APE1-IN-1
CAS:<p>APE1-IN-1 is a purine/pyrimidine-free endonuclease 1 inhibitor with potential antitumor activity that enhances the toxicity of alkylating agents on cancer cells</p>Fórmula:C19H21N3OS2Pureza:98.5%Cor e Forma:SolidPeso molecular:371.52
