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Imunologia e Inflamação

Imunologia e Inflamação

Os inibidores de imunologia e inflamação são compostos que modulam a resposta imunológica e os processos inflamatórios. Esses inibidores são cruciais para estudar os mecanismos de regulação imunológica, autoimunidade e inflamação crônica, bem como para desenvolver tratamentos para doenças inflamatórias, alergias e distúrbios relacionados ao sistema imunológico. Ao direcionar vias-chave no sistema imunológico, esses inibidores podem ajudar a reduzir respostas imunológicas excessivas ou inadequadas. Na CymitQuimica, oferecemos uma ampla seleção de inibidores de alta qualidade para apoiar sua pesquisa em imunologia, inflamação e desenvolvimento terapêutico.

Subcategorias de "Imunologia e Inflamação"

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Foram encontrados 3055 produtos de "Imunologia e Inflamação"

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  • Lunsekimig


    <p>Lunsekimig (SAR443765) is an IL-13/TSLP bis-antibody that links a nano-antibody targeting IL-13 and a variable region of the heavy chain (VHH) targeting TSLP for use in asthma research.</p>
    Cor e Forma:Odour Liquid
  • Tucotuzumab

    CAS:
    <p>Tucotuzumab: IgG1 monoclonal antibody targeting EpCAM, fused with IL-2, used as an immunosuppressant and antineoplastic.</p>
    Pureza:95%
    Cor e Forma:Liquid
  • CC-90002

    CAS:
    <p>CC-90002: humanized anti-CD47 mAb, high affinity, subnanomolar Kd. For hematologic and solid tumor research.</p>
    Cor e Forma:Liquid
  • Inolimomab

    CAS:
    <p>Inolimomab is a monoclonal antibody targeting CD25 (IL-2R α chain) for studying acute graft-versus-host disease (aGVHD).</p>
    Pureza:95% - 95%
    Cor e Forma:Liquid
  • Serotonin Creatinine Sulfate Monohydrate

    CAS:
    Fórmula:C14H19N5O2·H2SO4·H2O
    Pureza:>98.0%(T)
    Cor e Forma:White to Light yellow powder to crystal
    Peso molecular:405.43

    Ref: 3B-S0036

    1g
    69,00€
  • Indometacin Farnesil

    CAS:
    Fórmula:C34H40ClNO4
    Pureza:>98.0%(HPLC)
    Cor e Forma:Light yellow to Yellow to Orange clear liquid
    Peso molecular:562.15

    Ref: 3B-I0943

    100mg
    414,00€
  • Azathioprine

    CAS:
    Fórmula:C9H7N7O2S
    Pureza:>98.0%(T)(HPLC)
    Cor e Forma:Light yellow to Yellow to Green powder to crystal
    Peso molecular:277.26

    Ref: 3B-A2069

    5g
    229,00€
  • QNZ

    CAS:
    Fórmula:C22H20N4O
    Pureza:>98.0%(HPLC)
    Cor e Forma:White to Light yellow to Green powder to crystal
    Peso molecular:356.43

    Ref: 3B-Q0109

    5mg
    92,00€
    25mg
    314,00€
  • Ketorolac-d5

    CAS:
    <p>Ketorolac-d5 is a deuterated compound of ketorolac for isotope tracing. Ketorolac is a non-steroidal anti-inflammatory agent and inhibitor of COX-1 and COX-2.</p>
    Fórmula:C15H8D5NO3
    Pureza:98.99%
    Cor e Forma:Solid
    Peso molecular:260.3
  • Maresin 1

    CAS:
    Maresin 1 is biosynthesized by macrophages (MΦ) and possesses significant anti-inflammatory activity that attenuates LPS-induced lung injury in mice.
    Fórmula:C22H32O4
    Cor e Forma:Solid
    Peso molecular:360.49
  • Lusvertikimab

    CAS:
    <p>Lusvertikimab (OSE-127) is a humanized anti-IL7R antibody with anti-leukemic efficacy and can be used to study leukemia.</p>
    Pureza:95% - 98.4% (SDS-PAGE); 99% (SEC-HPLC)
    Cor e Forma:Liquid
  • Nepafenac-d5

    CAS:
    <p>Nepafenac D5 is the deuterium labeled Nepafenac, which is a selective inhibitor of COX-2 .</p>
    Fórmula:C15H14N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:259.31
  • D228

    CAS:
    <p>D228 is an oral anti-inflammatory,inhibi B and T lymphocytes, down-regulation of MyD88/TRAF6/p38 and up-regulation of IL-10,inflammatory bowel disease (IBD).</p>
    Fórmula:C22H28O12
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:484.45
  • BMS-378806

    CAS:
    BMS-378806 (BMS-806) selectively inhibits the binding of HIV-1 gp120 to the CD4 receptor with EC50 of 0.85-26.5 nM in virus.
    Fórmula:C22H22N4O4
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:406.43
  • FAPI-2

    CAS:
    <p>FAPI-2 is a specific inhibitor of fibroblast-activated protein based on the radiotracer FAP labeling, and has anticancer activity.</p>
    Fórmula:C40H56N10O10
    Pureza:98.76%
    Cor e Forma:Solid
    Peso molecular:836.93
  • 3,4-DAA

    CAS:
    3,4-DAA has anti-inflammatory activity and inhibits EOC20 cell-induced nitric oxide synthase (iNOS) induced by IFN-γ and lipopolysaccharide.
    Fórmula:C18H17NO6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:343.33
  • Amfenac

    CAS:
    <p>Amfenac promotes apoptosis in ARPE-19 cell culture.</p>
    Fórmula:C15H13NO3
    Cor e Forma:Solid
    Peso molecular:255.27
  • AHR-10037

    CAS:
    <p>AHR-10037, a NSAID, offers pain relief, fever reduction, safety, and low stomach risk, acting as a prodrug for COX inhibitors.</p>
    Fórmula:C15H13ClN2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:288.73
  • Vopikitug

    CAS:
    <p>Vopikitug is a humanized monoclonal antibody targeting IL-2RA with antitumor activity. It can be used to study cancer.</p>
    Pureza:99.1% (SDS-PAGE); 96.5% (SEC-HPLC) - 99.1% (SDS-PAGE); 96.5% (SEC-HPLC)
    Cor e Forma:Liquid
  • Azacyclonol hydrochloride

    CAS:
    <p>Azacyclonol hydrochloride can be used in the treatment of chronic schizophrenia.</p>
    Fórmula:C18H22ClNO
    Cor e Forma:Off White Crystalline Powder
    Peso molecular:303.83
  • Kamebakaurin

    CAS:
    <p>Kamebakaurin combats liver toxicity, cancer, inflammation, and neuroinflammation by blocking NF-κB, HIF-1α, and key signaling pathways.</p>
    Fórmula:C20H30O5
    Pureza:98.05%
    Cor e Forma:Solid
    Peso molecular:350.45
  • TMV-IN-9

    CAS:
    <p>TMV-IN-9 (compound A6) is an antiviral agent that exhibits exceptional inactivation effects against Tobacco Mosaic Virus (TMV), with an EC50 of 62.8 μg/mL. It demonstrates strong binding capabilities to the TMV capsid protein, with a binding affinity of 1.862 μM. Moreover, TMV-IN-9 significantly disrupts the integrity of TMV particles, thereby preventing the virus from infecting the host.</p>
    Fórmula:C20H20O8
    Cor e Forma:Solid
    Peso molecular:388.37
  • AZD4144

    CAS:
    <p>AZD4144 is a potent and selective NLRP3 inhibitor (IC50 = 54 nM) that reducs IL-1β and IL-18 production for immune disorders.</p>
    Fórmula:C18H16F3N3O3
    Pureza:99.02%
    Cor e Forma:Soild
    Peso molecular:379.33
  • (9α,13α,14α)-4-Hydroxy-3,7-dimethoxy-7,8-didehydromorphinan-6-one

    CAS:
    (9α,13α,14α)-4-Hydroxy-3,7-dimethoxy-7,8-didehydromorphinan-6-one is a major mechanism of Sinomenine.
    Fórmula:C18H21NO4
    Pureza:97.85%
    Cor e Forma:Soild
    Peso molecular:315.36
  • Etokimab

    CAS:
    <p>Etokimab (ANB-020) is a humanised monoclonal antibody targeting IL-33, neutrophil migration, atopic dermatitis, asthma, and sinusitis.</p>
    Pureza:95%
    Cor e Forma:Liquid
  • Avasopasem manganese

    CAS:
    <p>Avasopasem manganese is a drug candidate of superoxide dismutase mimetic.</p>
    Fórmula:C21H35Cl2MnN5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:483.38
  • Pelubiprofen

    CAS:
    <p>Pelubiprofen is a non-steroidal anti-inflammatory agent and a COX-2 inhibitor, which effectively reduces PGE(2) production by inhibiting COX activity.</p>
    Fórmula:C16H18O3
    Pureza:99.69%
    Cor e Forma:Solid
    Peso molecular:258.31
  • Catalase

    CAS:
    <p>Catalase, an enzyme, metabolizes H2O2 and ROS; its expression and localization change significantly in tumors.</p>
    Pureza:≥98%
    Cor e Forma:Small Colorless Crystals Or Powder At Room Temperature Almost Odourless Small Colourless Crystals Or A White Crystalline Powder
  • Allopurinol Sodium

    CAS:
    <p>Allopurinol Sodium is a xanthine oxidase inhibitor with an IC50 of 7.82±0.12 μM.</p>
    Fórmula:C5H4N4NaO
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:159.1
  • E3330

    CAS:
    <p>E3330 is a potent and selective APE1(Ref-1) inhibitor, which suppressed NF-kappa B DNA-binding activity.</p>
    Fórmula:C21H30O6
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:378.46
  • CB2 modulator 1

    CAS:
    <p>CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.</p>
    Fórmula:C18H19F3N4O2
    Pureza:99.6%
    Cor e Forma:Solid
    Peso molecular:380.36
  • HPN-01

    CAS:
    HPN-01 (IKK inhibitor XII) is an IKK inhibitor that inhibits IKK-α and IKK-ε, prolongs the lifespan of mice, and can be used to study immune disorders.
    Fórmula:C19H16ClN3O3S
    Pureza:98.07% - 98.17%
    Cor e Forma:Solid
    Peso molecular:401.87
  • Eltrombopag methyl ester

    CAS:
    <p>Eltrombopag methyl ester, a Tpo receptor agonist derivative, boosts platelet production for thrombocytopenia research.</p>
    Fórmula:C26H24N4O4
    Cor e Forma:Solid
    Peso molecular:456.49
  • RIP2 Kinase Inhibitor 3

    CAS:
    <p>RIP2 Kinase Inhibitor 3 is a potent and selective inhibitor of RIP2 with an IC50 of 1 nM.</p>
    Fórmula:C19H24N4O3S
    Pureza:99.32% - 99.52%
    Cor e Forma:Solid
    Peso molecular:388.48
  • hDDAH-1-IN-1

    CAS:
    hDDAH-1-IN-1 is a selective non-amino acid catalytic site inhibitor of human dimethylarginine dimethylaminohydrolase-1 (hDDAH-1) (Ki: 18 μM).
    Fórmula:C8H20N4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:188.27
  • MIP-1072

    CAS:
    <p>MIP-1072 is the prostate-specific membrane antigen inhibitor.</p>
    Fórmula:C19H26IN3O7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:535.33
  • GSK223

    CAS:
    GSK223 is an iE-DAP-stimulated IL-8 release inhibitor via the NOD1 signaling pathway.
    Fórmula:C21H18FN3O3S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:443.51
  • NCX1022

    CAS:
    <p>NCX1022 is a NO-releasing derivative of Hydrocortisone. It is the most widely used anti-inflammatory drug for the treatment of skin inflammation.</p>
    Fórmula:C29H35NO9
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:541.59
  • LC-R 505

    CAS:
    <p>LC-R 505 is an anti-inflammatory.</p>
    Fórmula:C20H26N2O5S
    Cor e Forma:Solid
    Peso molecular:406.5
  • FR20

    CAS:
    <p>FR20 is a human microsomal prostaglandin synthase 1 (mPGES 1) inhibitor.</p>
    Fórmula:C31H25Cl2N3O2
    Cor e Forma:Solid
    Peso molecular:542.46
  • Anisodine hydrobromide

    CAS:
    <p>Anisodine hydrobromide is an inhibitor of adenosine kinase.</p>
    Fórmula:C17H22BrNO5
    Cor e Forma:White Crystals Or Crystalline Powder
    Peso molecular:400.27
  • Oxyfenamate

    CAS:
    Oxyfenamate has anti-anxiety actions. It is also used in anxiety neuroses.
    Fórmula:C11H15NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:209.24
  • S-MTC

    CAS:
    <p>S-MTC is a selective inhibitor of type I nitric oxide synthase.</p>
    Fórmula:C7H15N3O2S
    Pureza:98%
    Cor e Forma:Off-White Powder / White Solid
    Peso molecular:205.28
  • RI-962

    CAS:
    <p>RI-962 is a potent and selective inhibitor of RIPK1 that protects cells from necrotic apoptosis by inhibiting RIPK1, RIPK3, and MLKL phosphorylation.</p>
    Fórmula:C28H28N6O2
    Pureza:99.39%
    Cor e Forma:Soild
    Peso molecular:480.56
  • L 748780

    CAS:
    <p>L 748780 is a selective inducible COX-2 inhibitor.</p>
    Fórmula:C19H14Cl3NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:426.68
  • Tiazotic acid

    CAS:
    <p>Tiazotic acid is an agent with the activity of antioxidant.</p>
    Fórmula:C5H7N3O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:173.19
  • ZXX2-77

    CAS:
    <p>ZXX2-77 is a cyclooxygenase-1 inhibitor.</p>
    Fórmula:C13H13ClN2O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:296.77
  • IRAK inhibitor 4

    CAS:
    <p>IRAK inhibitor 4 is an interleukin-1 receptor associated kinase 4 inhibitor.</p>
    Fórmula:C33H35F3N6O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:620.66
  • L-NIL hydrochloride

    CAS:
    <p>selective inhibitor of inducible nitric oxide synthase</p>
    Fórmula:C8H18ClN3O2
    Pureza:98%
    Cor e Forma:White To Off-White Solid
    Peso molecular:223.7
  • NCX-6560

    CAS:
    NCX-6560 is a novel NO-releasing derivative of atorvastatin, with those of atorvastatin.
    Fórmula:C37H42FN3O8
    Cor e Forma:Solid
    Peso molecular:675.74
  • Fagaramide

    CAS:
    <p>Fagaramide possesses Antiplasmodial activity.</p>
    Fórmula:C14H17NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:247.29
  • S-Isopropylisothiourea hydrobromide

    CAS:
    <p>S-Isopropylisothiourea hydrobromide is an iNOS inhibitor.</p>
    Fórmula:C4H11BrN2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:199.11
  • LY 150310

    CAS:
    <p>LY 150310, a histamine H1-receptor antagonist, can alter prostanoid concentrations in vitro and in vivo.</p>
    Fórmula:C13H14N2
    Cor e Forma:Solid
    Peso molecular:198.26
  • IRAK4-IN-16

    CAS:
    <p>IRAK4-IN-16 inhibits IRAK4 at 2.5nM; cytotoxic to OCI-LY10, TMD8, Ramos, HT cells with IC50s of 0.2, 0.2, 0.6, 2.7μM.</p>
    Fórmula:C17H20F2N8O
    Cor e Forma:Solid
    Peso molecular:390.39
  • Nω-Propyl-L-arginine hydrochloride

    CAS:
    <p>Highly selective and potent inhibitor of nNOS (Ki = 57 nM). Displays 3158-fold and 149-fold selectivity over iNOS and eNOS respectively. Hypotensive in vivo.</p>
    Fórmula:C9H21ClN4O2
    Cor e Forma:Solid
    Peso molecular:252.74
  • L 669083

    CAS:
    <p>L 669083 is two classes of potent leukotriene biosynthesis inhibitors photoaffinity analogue.</p>
    Fórmula:C29H29IN4O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:672.54
  • TYT-1

    CAS:
    <p>TYT-1 is a West Nile virus (WNV) inhibitor, antiviral (IC₅₀ = 0.7 mM) by blocking the pre-assembly replication step following viral entry into cells.</p>
    Fórmula:C21H17N3O2S3
    Pureza:98.49%
    Cor e Forma:Solid
    Peso molecular:439.57
  • SNAP 398299

    CAS:
    <p>SNAP 398299 is a Glycopeptide Receptor Type 3 (Gal3) antagonist with anxiolytic and antidepressant-like effects and is used in the study of mood disorders.</p>
    Fórmula:C27H24F3N3O2
    Pureza:97.16%
    Cor e Forma:Solid
    Peso molecular:479.49
  • APY0201

    CAS:
    <p>APY0201: potent, specific ATP-competitive PIKfyve inhibitor; IC50=5.2 nM; blocks PtdIns3P to PtdIns(3,5)P2 conversion.</p>
    Fórmula:C23H23N7O
    Pureza:98% - 99.74%
    Cor e Forma:Solid
    Peso molecular:413.48
  • T-5342126

    CAS:
    <p>T-5342126: TLR4 antagonist, lowers LPS-induced NO in cells (IC50=27.8 μM) &amp; cytokines in blood, cuts ethanol intake &amp; Iba1 in mice.</p>
    Fórmula:C25H32ClN3O3
    Cor e Forma:Solid
    Peso molecular:457.99
  • IRAK4-IN-17

    CAS:
    <p>IRAK4-IN-17 is a potent IRAK4 inhibitor with a 1.3 nM IC50, key for DLBCL research.</p>
    Fórmula:C17H20F2N8O
    Cor e Forma:Solid
    Peso molecular:390.39
  • HPGDS inhibitor 3

    CAS:
    <p>HPGDS inhibitor 3: oral, potent (IC50=9.4 nM; EC50=42 nM), selective, no CNS toxicity, good pharmacokinetics, anti-inflammatory.</p>
    Fórmula:C21H27N3O2
    Cor e Forma:Solid
    Peso molecular:353.46
  • OPC-163493

    CAS:
    <p>OPC-163493 is an orally active, liver-targeted mitochondrial uncoupling agent that diminishes Δψ (delta psi) and mitochondrial ROS (reactive oxygen species)</p>
    Fórmula:C14H8F3N5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:335.31
  • L-Kynurenine sulfate

    CAS:
    <p>L-Kynurenine sulfate activates AHR, leading naive T cells to anti-inflammatory Treg phenotype.</p>
    Fórmula:C10H14N2O7S
    Cor e Forma:Solid
    Peso molecular:306.29
  • STING modulator-4

    CAS:
    STING modulator-4: competitive, Ki=0.0933 μM (R232H STING), EC50 >10 μM (p-IRF3, THP-1 cells).
    Fórmula:C17H18N8O
    Cor e Forma:Solid
    Peso molecular:350.38
  • BC12-4

    CAS:
    <p>BC12-4 is a novel potent inhibitor of IL-2 secretion, it has potent immunomodulatory activity.</p>
    Fórmula:C19H14N2O3
    Cor e Forma:Solid
    Peso molecular:318.33
  • 3-Bromo-7-nitroindazole

    CAS:
    <p>3-Bromo-7-nitroindazole specifically inhibits nNOS, impacting NO synthesis in brain/body.</p>
    Fórmula:C7H4BrN3O2
    Pureza:98.2%
    Cor e Forma:Yellowish Solid
    Peso molecular:242.03
  • c-di-AMP

    CAS:
    <p>c-di-AMP (Cyclic diadenylate) is a STING agonist. It binds to the transmembrane protein STING thereby activating the TBK3-IRF3 signaling pathway.</p>
    Fórmula:C20H24N10O12P2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:658.41
  • Keap1-Nrf2-IN-13

    CAS:
    <p>Keap1-Nrf2-IN-13 is a PPI inhibitor (IC50: 0.15 μM) that binds Keap1 strongly, useful for oxidative stress and inflammation research.</p>
    Fórmula:C28H32N2O10S2
    Cor e Forma:Solid
    Peso molecular:620.69
  • AN3485 Hydrochloride

    CAS:
    <p>AN3485 Hydrochloride is an anti-inflammatory agent and a TLRs inhibitor, reducing ear swelling induced by PMA.</p>
    Fórmula:C14H14BCl2NO3
    Pureza:98.34%
    Cor e Forma:Solid
    Peso molecular:325.98
  • C5aR-IN-2

    CAS:
    <p>C5aR-IN-2, a potent C5aR inhibitor, shows promise for researching inflammatory diseases.</p>
    Fórmula:C36H40FN5O2
    Cor e Forma:Solid
    Peso molecular:593.73
  • Bay 65-1942 free base

    CAS:
    Bay 65-1942 free base is an inhibitor of ATP-competitive and selective IKKβ.
    Fórmula:C22H25N3O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:395.45
  • COX-2-IN-28

    CAS:
    <p>COX-2-IN-28 is a potent and selective COX-2 inhibitor capable of acting on COX-2 (IC50: 0.054 μM), 15-LOX (IC50: 2.14 μM) and COX-1 (IC50: 13.21 μM).</p>
    Fórmula:C30H27N7S3
    Cor e Forma:Solid
    Peso molecular:581.78
  • Enflicoxib

    CAS:
    <p>Enflicoxib is an effective treatment for canine osteoarthritis pain and inflammation, with faster onset than mavacoxib, improving veterinary outcomes.</p>
    Fórmula:C16H12F5N3O2S
    Pureza:99.88%
    Cor e Forma:Solid
    Peso molecular:405.34
  • AVE-9488

    CAS:
    <p>AVE-9488 is a novel endothelial NO synthase (eNOS) enhancer that upregulates eNOS expression, induces NO production, and may ameliorate portal hypertension.</p>
    Fórmula:C16H14FNO
    Pureza:99.87%
    Cor e Forma:Solid
    Peso molecular:255.29
  • AP-1/NF-κB activation inhibitor 1

    CAS:
    <p>AP-1/NF-κB activation inhibitor 1 is a potent inhibitor of AP-1 and NF-κB mediated transcriptional activation ( IC 50 =1 μM), does not blocking basal</p>
    Fórmula:C13H11F3N4O4
    Pureza:99.52% - 99.91%
    Cor e Forma:Solid
    Peso molecular:344.25
  • CD73-IN-8

    CAS:
    <p>CD73-IN-8 blocks CD73, hindering adenosine production that supports tumor growth, flagged as compound 57 in WO2022052886A1.</p>
    Fórmula:C17H13ClN4O2
    Cor e Forma:Solid
    Peso molecular:340.76
  • STING Agonist 12b

    CAS:
    <p>STING agonist 12b activates human/mouse STING, binds with Kd 26.4 μM, prompts interferon, and induces TNF-a, IL-6, IP-10, IL-1b in THP-1 cells.</p>
    Fórmula:C16H15NO2
    Cor e Forma:Solid
    Peso molecular:253.3
  • K-80001

    CAS:
    <p>K-80001 is a selective RXRα ligand and a COX-1/2 inhibitor, exhibiting IC50 values of 82.9μM for RXRα, 3.4μM for COX-1, and 1.2μM for COX-2, respectively [1].</p>
    Fórmula:C20H17FO2
    Cor e Forma:Solid
    Peso molecular:308.35
  • Bay 65-1942 hydrochloride

    CAS:
    <p>Bay 65-1942 hydrochloride is an inhibitor of ATP-competitive and selective IKKβ.</p>
    Fórmula:C22H26ClN3O4
    Cor e Forma:Solid
    Peso molecular:431.91
  • KIN1400

    CAS:
    <p>KIN1400 activates IRF3, boosts antiviral immunity, stimulates IFNbeta, and inhibits WNV, DV, and HCV.</p>
    Fórmula:C24H17F2N3O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:449.47
  • Emlenoflast sodium

    CAS:
    Emlenoflast sodium (MCC7840 sodium), a sulfonylurea, is a selective NLRP3 inflammasome inhibitor with an IC50 value of less than 100 nM for NLRP3 inflammasome,
    Fórmula:C19H24N4NaO3S
    Cor e Forma:Solid
    Peso molecular:411.47
  • Cyclic-di-GMP

    CAS:
    <p>Cyclic-di-GMP is a STING agonist and ubiquitous second messenger, which regulates the formation, motility and virulence of biofilms in various bacterial species</p>
    Fórmula:C20H24N10O14P2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:690.41
  • Edasalonexent

    CAS:
    Edasalonexent (CAT-1004) is an orally available NF-κB inhibitor for the improvement of Duchenne muscular dystrophy.
    Fórmula:C31H42N2O3
    Pureza:99.13% - >99.99%
    Cor e Forma:Solid
    Peso molecular:490.68
  • AMT hydrochloride

    CAS:
    <p>AMT hydrochloride is an iNOS inhibitor.</p>
    Fórmula:C5H11ClN2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:166.67
  • (R)-MALT1-IN-3

    CAS:
    <p>(R)-MALT1-IN-3 (121) inhibits MALT1 protease (IC50: 20 nM) and IL6/IL10 in OCI-LY3 (IC50: 60/40 nM).</p>
    Fórmula:C21H19F3N8O2
    Cor e Forma:Solid
    Peso molecular:472.42
  • COX-2-IN-20

    CAS:
    <p>COX-2-IN-20 (Compound 5d) is a selective and orally active inhibitor of COX-2 (IC 50 = 17.9 nM) with anti-inflammatory activity [1].</p>
    Fórmula:C11H9ClFN3O2
    Cor e Forma:Solid
    Peso molecular:269.66
  • APC-0576

    CAS:
    <p>APC-0576, an (S,S)-isomer, blocks NF-kappaB gene activation and may reduce inflammation in human cells.</p>
    Fórmula:C23H27N3O3
    Cor e Forma:Solid
    Peso molecular:393.48
  • ARV-393

    CAS:
    <p>ARV-393 is a PROTAC degrader targeting BCL6 orally available. ubiquitin proteasome for diffuse large b-cell lymphoma (DLBCL) and non-Hodgkin's lymphoma (NHL)</p>
    Fórmula:C46H53ClFN9O7
    Pureza:99.96%
    Cor e Forma:Soild
    Peso molecular:898.42
  • DDX3-IN-2

    CAS:
    <p>DDX3-IN-2 is a potent DDX3 inhibitor with an IC50 of 0.3 μM and shows broad antiviral effects, including against HIV resistance.</p>
    Fórmula:C20H23N5O
    Cor e Forma:Solid
    Peso molecular:349.43
  • Antiviral agent 14

    CAS:
    <p>Antiviral agent 14 is an antiviral agent that inhibits tobacco mosaic virus (TMV) (EC50: 135.5 μg/mL), and cucumber mosaic virus (CMV) (EC50: 178.6 μg/mL).</p>
    Fórmula:C24H26O7
    Cor e Forma:Solid
    Peso molecular:426.46
  • TRAF-STOP inhibitor 6877002

    CAS:
    <p>TRAF-STOP 6877002 inhibits CD40-TRAF6, curbing leukocyte recruitment and macrophage activation/proliferation in plaques.</p>
    Fórmula:C17H17NO
    Pureza:99.76%
    Cor e Forma:Solid
    Peso molecular:251.32
  • Mivotilate

    CAS:
    <p>Mivotilate, a potent, non-toxic aryl hydrocarbon receptor (AhR) activator, functions as a hepatoprotective agent.</p>
    Fórmula:C12H14N2O3S3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:330.45
  • Emlenoflast

    CAS:
    Emlenoflast (MCC7840) is a selective inhibitor of NLRP3 inflammasome.
    Fórmula:C19H24N4O3S
    Pureza:97.004% - 98.19%
    Cor e Forma:Solid
    Peso molecular:388.48
  • MIF-IN-2

    CAS:
    MIF-IN-2 is a MIF inhibitor with anticancer activity for the study of cancer and autoimmune diseases.
    Fórmula:C14H10ClN3O4
    Pureza:98.55%
    Cor e Forma:Solid
    Peso molecular:319.7
  • AZD8848

    CAS:
    AZD8848 is a selective antedrug agonist of toll-like receptor 7 (TLR7). It is developed for the research of asthma and allergic rhinitis.
    Fórmula:C29H43N7O5
    Cor e Forma:Solid
    Peso molecular:569.7
  • TLR7 agonist 1

    CAS:
    TLR7 agonist 1 is a selective and oral TLR7 agonist (IC50: 90 nM).
    Fórmula:C21H25N5O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:363.46
  • TLR7/8 agonist 6

    CAS:
    <p>Compound 4: Imidazoquinoline, potent TLR7/8 agonist, IC50: 0.18μM (TLR7), 5.34μM (TLR8).</p>
    Fórmula:C24H27N5O2
    Cor e Forma:Solid
    Peso molecular:417.5
  • TMV-IN-1

    CAS:
    <p>TMV-IN-1: a chalcone inhibits TMV with EC50s of 70.7 and 60.8 μg/mL, applicable in infection and tumor studies.</p>
    Fórmula:C28H26O4
    Cor e Forma:Solid
    Peso molecular:426.5
  • AR-C102222 hydrochloride

    CAS:
    AR-C102222 hydrochloride: oral iNOS inhibitor, selective, IC50=37 nM, with anti-inflammatory and pain relief effects.
    Fórmula:C19H17ClF2N6O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:418.83