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Transportador de Membranas/Canal Iónico

Transportador de Membranas/Canal Iónico

Os inibidores de transportadores de membrana e canais iônicos são compostos que bloqueiam a função de proteínas responsáveis pelo transporte de íons, nutrientes e outras moléculas através das membranas celulares. Esses inibidores são cruciais para o estudo da regulação da homeostase celular, transdução de sinais e neurotransmissão. Os inibidores de transportadores de membrana e canais iônicos também são importantes no desenvolvimento de tratamentos para distúrbios como epilepsia, doenças cardiovasculares e síndromes metabólicas. Na CymitQuimica, oferecemos uma ampla seleção de inibidores de alta qualidade de transportadores de membrana e canais iônicos para apoiar sua pesquisa em fisiologia, neurociência e farmacologia.

Subcategorias de "Transportador de Membranas/Canal Iónico"

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Foram encontrados 2277 produtos de "Transportador de Membranas/Canal Iónico"

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  • Huwentoxin I

    CAS:
    <p>Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.</p>
    Fórmula:C161H246N48O44S6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:3750.36
  • Oleoyl-D-lysine

    CAS:
    <p>Oleoyl-D-lysine: lipid-based GlyT2 inhibitor, eases neuropathic pain in mice, safe, non-sedative, no respiratory depression.</p>
    Fórmula:C24H46N2O3
    Cor e Forma:Solid
    Peso molecular:410.63
  • L-Palmitoylcarnitine TFA


    <p>L-Palmitoylcarnitine TFA: long-chain fat metabolite that disrupts membranes in ischaemia &amp; inhibits KATP channels via Kir6.2 interaction.</p>
    Fórmula:C25H46F3NO6
    Cor e Forma:Solid
    Peso molecular:513.63
  • PDDHV

    CAS:
    <p>PDDHV: a capsaicin-like vanilloid selective for rat TRPV1; induces Ca2+ uptake in neurons, EC50 of 70 nM.</p>
    Fórmula:C49H72O11
    Cor e Forma:Solid
    Peso molecular:837.09
  • Ziconotide

    CAS:
    <p>Ziconotide: analgesic from cone snail for severe, chronic pain; synthetic ω-conotoxin.</p>
    Fórmula:C102H172N36O32S7
    Pureza:98%
    Cor e Forma:White Powder
    Peso molecular:2639.13
  • Homocarnosine

    CAS:
    <p>Homocarnosine is an endogenous dipeptide in cerebral regions and cerebrospinal fluid.</p>
    Fórmula:C10H16N4O3
    Cor e Forma:Solid
    Peso molecular:240.26
  • (±)5(6)-DiHETE

    CAS:
    <p>Eicosapentaenoic acid is an ω-3 polyunsaturated fatty acid that is abundant in marine organisms and fish oils.</p>
    Fórmula:C20H32O4
    Cor e Forma:Solid
    Peso molecular:336.472
  • CHET3

    CAS:
    <p>CHET3 is a highly selective allosteric activator for TASK-3-containing K2P channels. CHET3 has shown potent in vivo analgesic effects. Cost-effective and quality-assured.</p>
    Fórmula:C21H21N5O3S
    Pureza:99.64% - >99.99%
    Cor e Forma:Soild
    Peso molecular:423.49
  • 17(S)-HETE

    CAS:
    <p>Arachidonic acid and its CYP450 metabolite, 17(S)-HETE, regulate kidney electrolytes; 17(S)-HETE reduces proximal tubule ATPase activity by 70% at 2 μM.</p>
    Fórmula:C20H32O3
    Cor e Forma:Solid
    Peso molecular:320.473
  • Resolvin D2 methyl ester

    CAS:
    <p>RvD2 is an anti-inflammatory lipid made from docosahexaenoic acid by 15- and 5-lipoxygenase. Its methyl ester may serve as a prodrug.</p>
    Fórmula:C23H34O5
    Cor e Forma:Solid
    Peso molecular:390.52
  • WAY-326766

    CAS:
    <p>WAY-326766 increases ion transport through mutant CFTR and can be used to alter the lifespan of eukaryotes.WAY-326766 can be used to treat cystic fibrosis (CF).</p>
    Fórmula:C21H23N3O5
    Pureza:98.76%
    Cor e Forma:Solid
    Peso molecular:397.42
  • ProTx II

    CAS:
    <p>Selective NaV1.7 inhibitor, alters activation, reduces current, 100x more selective for 1.7 over other Na+ channels.</p>
    Fórmula:C168H250N46O41S8
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:3826.59
  • Neurotransmitter Receptor Compound Library


    <p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>
    Cor e Forma:Odour Solid
  • GpTx-1 TFA


    <p>GpTx-1 TFA is a polypeptide NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. It exhibits potent inhibitory activity on the NaV1.7 channel with an IC50 value of 10 nM, demonstrating excellent selectivity over NaV1.4 (IC50 = 0.301 μM) and NaV1.5 (IC50 = 4.20 μM) with &gt;20-fold and &gt;950-fold selectivity, respectively.</p>
    Cor e Forma:Odour Solid
  • TRPV4 antagonist 4

    CAS:
    <p>Potent TRPV4 blocker with 22.65 nM IC50; inhibits current and aids acute lung injury.</p>
    Fórmula:C28H32Cl2N6O
    Cor e Forma:Solid
    Peso molecular:539.50
  • Chlorotoxin TFA


    <p>Chlorotoxin TFA, a scorpion venom peptide, blocks chloride channels and has anti-cancer properties.</p>
    Fórmula:C160H250F3N53O49S11
    Cor e Forma:Solid
    Peso molecular:4109.74
  • Trans (2,3)-Dihydrotetrabenazine

    CAS:
    <p>Trans (2,3)-Dihydrotetrabenazine is a Tetrabenazine metabolite, shows inhibition activity on vesicular monoamine transporter (VMAT2).</p>
    Fórmula:C19H29NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:319.44
  • TRPA1-IN-1

    CAS:
    <p>TRPA1-IN-1 is a potent, selective antagonist of the TRPA1 channel, demonstrating significant oral bioavailability as a small molecule.</p>
    Fórmula:C19H17ClN6O3
    Cor e Forma:Solid
    Peso molecular:412.83
  • Tiludronate disodium hemihydrate

    CAS:
    <p>Tiludronate: an oral bisphosphonate for bone disorder research; inhibits osteoclasts and reduces inflammation.</p>
    Fórmula:C14H16Cl2Na4O13P4S2
    Cor e Forma:Solid
    Peso molecular:743.16
  • Mambalgin 1

    CAS:
    <p>ASIC1a inhibitor; IC50: 192 nM (human), 72 nM (dimer); inactive channel binding; selective; pain response delay.</p>
    Fórmula:C272H429N85O84S10
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:6554.51