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Transportador de Membranas/Canal Iónico

Transportador de Membranas/Canal Iónico

Os inibidores de transportadores de membrana e canais iônicos são compostos que bloqueiam a função de proteínas responsáveis pelo transporte de íons, nutrientes e outras moléculas através das membranas celulares. Esses inibidores são cruciais para o estudo da regulação da homeostase celular, transdução de sinais e neurotransmissão. Os inibidores de transportadores de membrana e canais iônicos também são importantes no desenvolvimento de tratamentos para distúrbios como epilepsia, doenças cardiovasculares e síndromes metabólicas. Na CymitQuimica, oferecemos uma ampla seleção de inibidores de alta qualidade de transportadores de membrana e canais iônicos para apoiar sua pesquisa em fisiologia, neurociência e farmacologia.

Subcategorias de "Transportador de Membranas/Canal Iónico"

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Foram encontrados 2280 produtos de "Transportador de Membranas/Canal Iónico"

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  • BeKm-1
    Targetmol
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    BeKm-1

    CAS:
    <p>Potent, selective hERG (KV11.1) blocker; doesn't affect 14 other K+ channels; extends QTc in rabbit heart dose-dependently.</p>
    Fórmula:C174H261N51O52S6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:4091.65

    Ref: TM-TP2072

  • Pinacidil monohydrate
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    Pinacidil monohydrate

    CAS:
    <p>Pinacidil monohydrate is a potassium channel activator, antihypertensive drug.</p>
    Fórmula:C13H21N5O
    Pureza:99.94% - 99.98%
    Cor e Forma:Powder
    Peso molecular:263.34

    Ref: TM-T12478

  • Carbonic anhydrase inhibitor 32
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    Carbonic anhydrase inhibitor 32

    <p>Carbonic anhydrase inhibitor32 (compound 5B) is an orally active, selective inhibitor of hCA (carbonic anhydrase) II/VII, with Ki values of 6.3 nM for hCA II, 10.1 nM for hCA VII, and 681 nM for hCA I. It shows potential for neuroprotection and anticonvulsant effects by reducing mTOR activation and increasing hippocampal KCC2 levels.</p>
    Fórmula:C17H16N6O3S
    Cor e Forma:Solid
    Peso molecular:384.41

    Ref: TM-T207684

  • Logotipo do CymitQuimica
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    Huwentoxin I

    CAS:
    <p>Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.</p>
    Fórmula:C161H246N48O44S6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:3750.36

    Ref: TM-T80185

  • FD 12-9
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    FD 12-9

    CAS:
    <p>FD 12-9, Anti-glioblastoma activity. is a flavonoid dimer, acts as a dual inhibitor of P-gp and BCRP, with EC50s of 285 nM and 0.9 nM, respectively.</p>
    Fórmula:C51H47N3O11
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:877.93

    Ref: TM-T11268

  • UK-59811 hydrochloride
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    UK-59811 hydrochloride

    CAS:
    <p>UK-59811 hydrochloride, Br-dihydropyridine derivative, blocks Ca V Ab channels in bacteria, IC50: 194 nM.</p>
    Fórmula:C22H30BrClN2O5
    Cor e Forma:Solid
    Peso molecular:517.85

    Ref: TM-T39770

  • NAADP tetrasodium salt
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    NAADP tetrasodium salt

    CAS:
    <p>Ca2+ mobilizing agent</p>
    Fórmula:C21H27N6O18P3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:744.39

    Ref: TM-T23049

  • Conantokin G
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    Conantokin G

    CAS:
    <p>GluN2B-specific NMDA receptor blocker; IC50=480 nM in neurons, ~300 nM in oocytes; neuroprotective.</p>
    Fórmula:C88H138N26O44
    Pureza:98%
    Cor e Forma:White Lyophilised Solid
    Peso molecular:2264.21

    Ref: TM-TP2060

  • CP-628006
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    CP-628006

    CAS:
    <p>CP-628006 is a small molecule CFTR potentiator that effectively restores ATP-dependent channel gating to G551D-CFTR, the mutant form found in cystic fibrosis.</p>
    Fórmula:C32H35F3N2O2
    Cor e Forma:Solid
    Peso molecular:536.639

    Ref: TM-T40386

  • Logotipo do CymitQuimica
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    SLC6A8 corrector 1

    <p>SLC6A8 Corrector 1 is an orally active corrector for mutant SLC6A8 variants, capable of crossing the blood-brain barrier. It is utilized in the study of creatine transporter deficiency (CTD).</p>
    Fórmula:C21H25N3O2
    Cor e Forma:Solid
    Peso molecular:351.44

    Ref: TM-T201220

  • Dofetilide N-oxide
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    Dofetilide N-oxide

    CAS:
    Dofetilide N-oxide (UK-116856) is a metabolite of dofetilide. Dofetilide can block potassium channels and is a tertiary antiarrhythmic drug.
    Fórmula:C19H27N3O6S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:457.56

    Ref: TM-T11073

  • Logotipo do CymitQuimica
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    AQP4 (205-215) TFA

    <p>AQP4 (205-215) TFA is a fragment of the water channel protein-4 (AQP4). AQP4 acts as an autoimmune antigen in neuromyelitis optica, upregulating and presenting in B cells upon binding with CD40. AQP4 is associated with neuromyelitis optica (NMO), an autoimmune inflammatory disease of the central nervous system (CNS).</p>
    Cor e Forma:Odour Solid

    Ref: TM-TP3237

  • Chlorocresol
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    Chlorocresol

    CAS:
    <p>Chlorocresol (4-Chloro-3-methylphenol) is an antiseptic medication.</p>
    Fórmula:C7H7ClO
    Cor e Forma:Solid
    Peso molecular:142.58

    Ref: TM-T75311

  • L-R4W2
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    L-R4W2

    CAS:
    <p>Vanilloid TRPV1 (VR1) receptor antagonist peptide (IC50 ~ 0.1 μM); blocks Ca2+ currents in dorsal root ganglion neurons. Analgesic in vivo.</p>
    Fórmula:C46H71N21O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:1014.2

    Ref: TM-TP1934

  • N-hydroxy Riluzole
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    N-hydroxy Riluzole

    CAS:
    <p>N-hydroxy Riluzole, a metabolite of riluzole, is mainly produced by CYP1A2 in human liver.</p>
    Fórmula:C8H5F3N2O2S
    Cor e Forma:Solid
    Peso molecular:250.20

    Ref: TM-T35919

  • 8-Azido-ATP
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    8-Azido-ATP

    CAS:
    <p>8-Azido-ATP is a nucleotide analog that demonstrates photo-reactivity properties.</p>
    Fórmula:C10H15N8O13P3
    Cor e Forma:Solid
    Peso molecular:548.19

    Ref: TM-T40616

  • (±)17-HETE
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    (±)17-HETE

    CAS:
    <p>Electrolyte and fluid transport in the kidney are regulated in part by arachidonic acid and its metabolites.</p>
    Fórmula:C20H32O3
    Cor e Forma:Solid
    Peso molecular:320.473

    Ref: TM-T35523

  • Logotipo do CymitQuimica
    Targetmol
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    MS7710

    <p>MS7710 is a brain-penetrant inhibitor of hyperpolarization-activated cyclic nucleotide-gated (HCN) channels. It reduces Ih current by inhibiting HCN channels, thereby decreasing the activity of dopamine neurons in the ventral tegmental area (VTA). MS7710 effectively improves social interaction deficits and reward-related cognitive flexibility in mouse models of chronic social defeat stress (CSDS) and shows promise for depression research.</p>
    Cor e Forma:Odour Solid

    Ref: TM-T207039

  • Logotipo do CymitQuimica
    Targetmol
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    ω-Conotoxin MVIIC TFA

    <p>ω-Conotoxin MVIIC TFA is a peptide and neurotoxin blocks P-type and q-type voltage-sensitive neuronal Ca ++ channels (VGCCs) radiolabel immunoprecipitation.</p>
    Fórmula:C106H178N40O32S7·C2HF3O2
    Cor e Forma:Solid
    Peso molecular:2863.27

    Ref: TM-T75726

  • G-Glu-Ser
    Targetmol
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    G-Glu-Ser

    CAS:
    <p>G-Glu-Ser is a calcium receptor activator and Flavor-enriching agent.</p>
    Fórmula:C8H14N2O6
    Cor e Forma:Solid
    Peso molecular:234.21

    Ref: TM-T27411