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Transportador de Membranas/Canal Iónico

Transportador de Membranas/Canal Iónico

Os inibidores de transportadores de membrana e canais iônicos são compostos que bloqueiam a função de proteínas responsáveis pelo transporte de íons, nutrientes e outras moléculas através das membranas celulares. Esses inibidores são cruciais para o estudo da regulação da homeostase celular, transdução de sinais e neurotransmissão. Os inibidores de transportadores de membrana e canais iônicos também são importantes no desenvolvimento de tratamentos para distúrbios como epilepsia, doenças cardiovasculares e síndromes metabólicas. Na CymitQuimica, oferecemos uma ampla seleção de inibidores de alta qualidade de transportadores de membrana e canais iônicos para apoiar sua pesquisa em fisiologia, neurociência e farmacologia.

Subcategorias de "Transportador de Membranas/Canal Iónico"

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Foram encontrados 2277 produtos de "Transportador de Membranas/Canal Iónico"

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  • 5-Tridecanol
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    5-Tridecanol

    CAS:
    <p>5-Tridecanol blocks ion flux in sodium channels.</p>
    Fórmula:C13H28O
    Pureza:97.87%
    Cor e Forma:Solid
    Peso molecular:200.36

    Ref: TM-T84115

  • LY-368975 hydrochloride
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    LY-368975 hydrochloride

    CAS:
    <p>LY-368975 hydrochloride is a bioactive chemical.</p>
    Fórmula:C17H22ClNOS
    Cor e Forma:Solid
    Peso molecular:323.88

    Ref: TM-T33015

  • Withaphysalin D
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    Withaphysalin D

    CAS:
    <p>Withaphysalin D, from water lilies, blocks GluN2B NMDARs and is neuroprotective, crossing the blood-brain barrier.</p>
    Fórmula:C28H34O6
    Cor e Forma:Solid
    Peso molecular:466.57

    Ref: TM-T75571

  • WAY-326766
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    WAY-326766

    CAS:
    <p>WAY-326766 increases ion transport through mutant CFTR and can be used to alter the lifespan of eukaryotes.WAY-326766 can be used to treat cystic fibrosis (CF).</p>
    Fórmula:C21H23N3O5
    Pureza:98.76%
    Cor e Forma:Solid
    Peso molecular:397.42

    Ref: TM-T77604

  • Logotipo do CymitQuimica
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    ATP Synthesis-IN-1

    <p>ATP Synthesis-IN-1 (Compound 4), a quinoline derivative, potently inhibits PA ATP synthesis with an IC50 of 11.1μg/mL and exhibits antibacterial properties.</p>
    Cor e Forma:Odour Solid

    Ref: TM-T82945

  • Logotipo do CymitQuimica
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    Anticancer agent 108

    <p>Anticancer Agent 108 (Compound 3.10) serves as a potent P-gp inhibitor exhibiting considerable antitumor properties while maintaining reduced toxicity to both</p>
    Fórmula:C18H9NO5S2
    Cor e Forma:Solid
    Peso molecular:383.4

    Ref: TM-T78693

  • Na2+ - Ca2+ Exchanger inhibitory peptide
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    Na2+ - Ca2+ Exchanger inhibitory peptide

    <p>Na+-Ca2+Exchanger inhibitory peptide (XIP) is an inhibitor of the Na+-Ca2+ exchanger with a Ki of 200 nM. It acts non-competitively to inhibit Na+-dependent Ca2+ uptake and Na+-dependent Ca2+ efflux in sarcolemmal vesicles.</p>
    Fórmula:C112H161N27O33
    Cor e Forma:Solid
    Peso molecular:2413.64

    Ref: TM-TP3107

  • Logotipo do CymitQuimica
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    Anticonvulsant agent 9

    <p>Anticonvulsant agent 9 (compound 4f) is an activator of the α1β2γ2GABA_A receptor, with an EC50 value of 1.24 μM. It inhibits the inactivation of Nav1.2 channels and exhibits significant anticonvulsant activity.</p>
    Fórmula:C22H24N4O2
    Cor e Forma:Solid
    Peso molecular:376.45

    Ref: TM-T205256

  • Logotipo do CymitQuimica
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    GpTx-1 TFA

    <p>GpTx-1 TFA is a polypeptide NaV1.7 sodium channel antagonist isolated from the venom of the Chilean spider Grammostola porter. It exhibits potent inhibitory activity on the NaV1.7 channel with an IC50 value of 10 nM, demonstrating excellent selectivity over NaV1.4 (IC50 = 0.301 μM) and NaV1.5 (IC50 = 4.20 μM) with &gt;20-fold and &gt;950-fold selectivity, respectively.</p>
    Cor e Forma:Odour Solid

    Ref: TM-TP3232

  • Logotipo do CymitQuimica
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    EVT-401

    <p>EVT-401 (P2X7 receptor antagonist-1), a purinergic P2X7 receptor antagonist, demonstrates efficacy in combating neuroinflammation [1].</p>
    Fórmula:C22H20F4N2O3
    Cor e Forma:Solid
    Peso molecular:436.4

    Ref: TM-T74409

  • Ampullosporin A
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    Ampullosporin A

    CAS:
    <p>Ampullosporin A is a peptaibol-type polypeptide isolated from the fungus Sepedonium ampullosporum (HKI-0053), exhibiting neuromodulatory activity. It inhibits hyperactivity induced by the NMDA receptor antagonist MK-801 and ameliorates social behavior abnormalities caused by subchronic ketamine treatment. Ampullosporin A modulates glutamate receptor activity without affecting dopamine D1 and D2 receptors.</p>
    Fórmula:C77H127N19O19
    Cor e Forma:Solid
    Peso molecular:1622.95

    Ref: TM-TN9041

  • Logotipo do CymitQuimica
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    Astressin 2B

    CAS:
    <p>CRF2 antagonist with IC50 of 1.3 nM; &gt;500 nM for CRF1. Aids gastric emptying.</p>
    Fórmula:C183H307N49O53
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:4041.69

    Ref: TM-TP2095

  • (Iso)-Atagabalin HCl
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    (Iso)-Atagabalin HCl

    CAS:
    <p>(Iso)-Atagabalin HCl(isomer-Atagabalin HCl) is an alpha -2- delta ligand that can be used to treat non-restorative sleep.</p>
    Fórmula:C10H20ClNO2
    Pureza:99.26% - >99.99%
    Cor e Forma:Soild
    Peso molecular:221.72

    Ref: TM-T30188L1

  • Imagabalin
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    Imagabalin

    CAS:
    <p>Imagabalin is an active compound used in the study of neurological diseases.</p>
    Fórmula:C9H19NO2
    Cor e Forma:Solid
    Peso molecular:173.25

    Ref: TM-T32143

  • 6,7-dimethylisatin
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    6,7-dimethylisatin

    CAS:
    <p>6,7-Dimethylisatin (6,7-dimethyl-1H-indole-2,3-dione) inhibits hGAT3 with IC50 of 108 μM. 6,7-Dimethylisatin also inhibits hBGT1, hGAT2.</p>
    Fórmula:C10H9NO2
    Pureza:98.98%
    Cor e Forma:Solid
    Peso molecular:175.18

    Ref: TM-T77568

  • Logotipo do CymitQuimica
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    Antidepressant agent 4

    <p>Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.</p>
    Fórmula:C19H38ClN5O2S
    Cor e Forma:Solid
    Peso molecular:436.06

    Ref: TM-T75003

  • (2R,3S,11bS)-Dihydrotetrabenazine
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    (2R,3S,11bS)-Dihydrotetrabenazine

    CAS:
    <p>(2R,3S,11bS)-Tetrabenazine impurity, VMAT inhibitor for movement disorders.</p>
    Fórmula:C19H29NO3
    Pureza:99.29%
    Cor e Forma:Solid
    Peso molecular:319.44

    Ref: TM-T67882

  • Levamlodipine besylate Hemipentahydrate
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    Levamlodipine besylate Hemipentahydrate

    CAS:
    <p>Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.</p>
    Fórmula:C20H25ClN2O5·C6H6O3SH2O
    Cor e Forma:Solid
    Peso molecular:1224.18

    Ref: TM-T204904

  • RU-TRAAK-2
    Targetmol
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    RU-TRAAK-2

    CAS:
    <p>RU-TRAAK-2 reversibly inhibits TWIK-related K+ channel, inactive on Kv1.2, GIRK2, Slo1.</p>
    Fórmula:C19H17N3OS
    Pureza:99.81%
    Cor e Forma:Solid
    Peso molecular:335.42

    Ref: TM-T60061

  • (±)16-HETE
    Targetmol
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    (±)16-HETE

    CAS:
    <p>Electrolyte and fluid transport in the kidney are regulated in part by arachidonic acid and its metabolites.</p>
    Fórmula:C20H32O3
    Cor e Forma:Solid
    Peso molecular:320.473

    Ref: TM-T35465