Transportador de Membranas/Canal Iónico
Os inibidores de transportadores de membrana e canais iônicos são compostos que bloqueiam a função de proteínas responsáveis pelo transporte de íons, nutrientes e outras moléculas através das membranas celulares. Esses inibidores são cruciais para o estudo da regulação da homeostase celular, transdução de sinais e neurotransmissão. Os inibidores de transportadores de membrana e canais iônicos também são importantes no desenvolvimento de tratamentos para distúrbios como epilepsia, doenças cardiovasculares e síndromes metabólicas. Na CymitQuimica, oferecemos uma ampla seleção de inibidores de alta qualidade de transportadores de membrana e canais iônicos para apoiar sua pesquisa em fisiologia, neurociência e farmacologia.
Subcategorias de "Transportador de Membranas/Canal Iónico"
- ABC(3 produtos)
- ATPase(93 produtos)
- Receptor de adiponectina(5 produtos)
- CFTR(64 produtos)
- Receptor CGRP(51 produtos)
- Canais de Cálcio(493 produtos)
- Canal de cloreto(49 produtos)
- Receptor GABA(336 produtos)
- Transportador de monoamina(23 produtos)
- Transportador de monocarboxilato(17 produtos)
- NKCC(2 produtos)
- NPC1L1(3 produtos)
- Cotransportador Na-K-Cl(8 produtos)
- OAT(27 produtos)
- OCT(7 produtos)
- P-gp(53 produtos)
- Canal de Potássio(276 produtos)
- Bomba de prótons(39 produtos)
- SGLT(30 produtos)
- Canal de Sódio(202 produtos)
- Canal TRP/TRPV(93 produtos)
Exibir 13 mais subcategorias
Foram encontrados 2277 produtos de "Transportador de Membranas/Canal Iónico"
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Lansoprazole sulfone
CAS:<p>Lansoprazole sulfone is a metabolite of the gastric pump inhibitor Lansoprazole.</p>Fórmula:C16H14F3N3O3SPureza:99.67%Cor e Forma:SolidPeso molecular:385.36Levosimendan
CAS:<p>Levosimendan (OR1259) is a calcium sensitizer for acute heart failure, enhancing cardiac contractility without raising calcium levels.</p>Fórmula:C14H12N6OPureza:99.37% - 99.91%Cor e Forma:Yellow Crystalline PowderPeso molecular:280.28Ocinaplon
CAS:<p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>Fórmula:C17H11N5OPureza:99.81%Cor e Forma:SolidPeso molecular:301.3Esomeprazole
CAS:<p>Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis.</p>Fórmula:C17H19N3O3SPureza:97.3%Cor e Forma:SolidPeso molecular:345.42Transdermal Peptide Disulfide Acetate
<p>Transdermal Peptide acetate(888486-23-5 free base) (TD 1 (peptide) acetate) is a 11-amino acid peptide, binds toNa+/K+-ATPase beta-subunit (ATP1B1), and mainly</p>Fórmula:C42H68N14O18S2Pureza:99.97%Cor e Forma:SolidPeso molecular:1121.2FGH10019
CAS:<p>FGH10019 is a novel inhibitor of sterol regulatory element-binding protein (SREBP) ( IC50 :1 μM).</p>Fórmula:C18H19N3O2S2Pureza:98.93%Cor e Forma:SolidPeso molecular:373.49KPT185
CAS:<p>KPT185 (KPT 185) is a selective CRM1 inhibitor, inducing apoptosis, cell-cycle arrest.</p>Fórmula:C16H16F3N3O3Pureza:98%Cor e Forma:SolidPeso molecular:355.31(R)-Lansoprazole
CAS:<p>(R)-Lansoprazole (T 168390) is the R-isomer of lansoprazole and a substituted benzimidazole prodrug with selective and irreversible proton pump inhibitor</p>Fórmula:C16H14F3N3O2SPureza:98.09% - 98.99%Cor e Forma:Brown SolidPeso molecular:369.36Budipine
CAS:<p>Budipine is a low affinity, N-methyl-D-aspartate receptor antagonist,is an antiparkinsonian agent.</p>Fórmula:C21H27NPureza:99.64%Cor e Forma:SolidPeso molecular:293.45PF-05186462
CAS:<p>PF-05186462 (PF-05150122) is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5.</p>Fórmula:C19H10ClF4N5O3S2Pureza:99.10% - 99.37%Cor e Forma:SolidPeso molecular:531.89VK-II-36
CAS:<p>VK-II-36, a carvedilol analog, suppresses sarcoplasmic reticulum (SR) Ca(2+) release but does not block the β-receptor.</p>Fórmula:C26H26N2O5Pureza:99.12%Cor e Forma:SolidPeso molecular:446.49α-Asarone
CAS:<p>alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.</p>Fórmula:C12H16O3Pureza:99.64% - 99.64%Cor e Forma:Monoclinic Needles From Water Monoclinic Needles From WaterPeso molecular:208.25Ralfinamide mesylate
CAS:<p>Ralfinamide mesylate (FCE-26742A (mesylate)) is an orally available Na+ channel blocker.</p>Fórmula:C18H23FN2O5SPureza:99.83%Cor e Forma:SolidPeso molecular:398.45Neboglamine
CAS:<p>Neboglamine, a glycine NMDA-associated agonist, is used potentially for the treatment of schizophrenia.</p>Fórmula:C13H24N2O3Pureza:98%Cor e Forma:SolidPeso molecular:256.34LY 303511 hydrochloride
CAS:<p>LY 303511 hydrochloride is a potent mTOR inhibitor</p>Fórmula:C19H19ClN2O2Pureza:98.47%Cor e Forma:SolidPeso molecular:342.82(-)-Blebbistatin
CAS:<p>(-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin II inhibitor with IC50 ranging from 0.5 to 5 μM.</p>Fórmula:C18H16N2O2Pureza:99.38% - 99.61%Cor e Forma:SolidPeso molecular:292.33AER-271
CAS:<p>AER-271 is an inhibitor of aquaporin-4.</p>Fórmula:C15H9ClF6NO5PPureza:97.45%Cor e Forma:SolidPeso molecular:463.65PF-06869206
CAS:<p>PF-06869206 is an oral selective inhibitor of the sodium-phosphate cotransporter NaPi2a (SLC34A1, IC50: 380 nM).</p>Fórmula:C15H14ClF3N4O2Pureza:99.79% - 99.88%Cor e Forma:SolidPeso molecular:374.75TKIM
CAS:<p>TKIM is a TWIK-related potassium channel 1 (TREK-1) inhibitor, binding to the pocket of the intermediate (IM) state of TREK-1.</p>Fórmula:C18H14ClN3O2SPureza:99.47%Cor e Forma:SolidPeso molecular:371.84ICA-069673
CAS:<p>ICA-069673 is an activator of KCNQ2/Q3 potassium channel (IC50: 0.69 μM).</p>Fórmula:C11H6ClF2N3OPureza:99.04% - 99.68%Cor e Forma:SolidPeso molecular:269.63HC-056456
CAS:<p>HC-056456 (3,4-Bis(2-thienoyl)-1,2,5-oxadiazole-N-oxide) is a CatSper channel modulator.</p>Fórmula:C12H6N2O4S2Pureza:99.62% - 99.65%Cor e Forma:SolidPeso molecular:306.32N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride
CAS:<p>N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride is an inhibitor of TRPC4.</p>Fórmula:C16H17ClN4Pureza:99.25%Cor e Forma:SolidPeso molecular:300.79L-DABA
CAS:<p>L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).</p>Fórmula:C4H10N2O2Pureza:99.32%Cor e Forma:SolidPeso molecular:118.13SB-705498
CAS:<p>SB705498 is a TRPV1 antagonist for hTRPV1. SB-705498 has been investigated for the treatment of Rhinitis, Chronic Cough, and Non-allergic Rhinitis.</p>Fórmula:C17H16BrF3N4OPureza:99.57% - ≥95%Cor e Forma:SolidPeso molecular:429.23CFTR corrector 2
CAS:<p>CFTR corrector 2 (FDL169) is a novel and potent CFTR corrector for treating cystic fibrosis (CF) patients who carry the F508del mutation.</p>Fórmula:C27H23FN4O4Pureza:99.66%Cor e Forma:SolidPeso molecular:486.49Lorediplon
CAS:<p>Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.</p>Fórmula:C20H15FN4O2SPureza:99.12% - 99.19%Cor e Forma:SolidPeso molecular:394.42TRPM8 antagonist 2
CAS:<p>TRPM8 antagonist 2 is a potent and selective TRPM8 antagonist with an IC50 of 0.2 nM. TRPM8 antagonist 2 is used in the research of neuropathic pain syndromes.</p>Fórmula:C26H26N2O2Pureza:98.1%Cor e Forma:SolidPeso molecular:398.5Tenatoprazole sodium
CAS:<p>Tenatoprazole sodium is a potent proton pump inhibitor with an IC50 of 6.2 μM against hog gastric H+/K+-ATPase.</p>Fórmula:C16H17N4NaO3SCor e Forma:SolidPeso molecular:368.39CLP290
CAS:<p>CLP290 is an activator of the neuron-specific K+-Cl cotransporter KCC2 and displays potential for the treatment of a wide range of neurological and psychiatric</p>Fórmula:C19H21FN4O3SPureza:99.93% - >99.99%Cor e Forma:SolidPeso molecular:404.46O4I2
CAS:<p>O4I2 is an effective Oct3/4 inducer in various human cell lines including human fibroblasts.</p>Fórmula:C12H11ClN2O2SPureza:97.97% - 99.84%Cor e Forma:SolidPeso molecular:282.75QO-40
CAS:<p>QO-40 is a KCNQ2/3 potassium channels activator.</p>Fórmula:C18H11ClF3N3OPureza:99.57%Cor e Forma:SolidPeso molecular:377.75Elacridar
CAS:<p>Elacridar (GG918) is a potent inhibitor of P-glycoprotein and BCRP.Cost-effective and quality-assured.</p>Fórmula:C34H33N3O5Pureza:98.12% - >99.99%Cor e Forma:SolidPeso molecular:563.64Phenyl benzoate
CAS:<p>Phenyl benzoate is a benzoate ester obtained by the formal condensation of phenol with benzoic acid.It is an important organic synthesis intermediate.</p>Fórmula:C13H10O2Pureza:99.63%Cor e Forma:White Crystalline PowderPeso molecular:198.22Guanosine 5'-diphosphate
CAS:<p>Guanosine 5'-diphosphate (GDP) as Potential Iron Mobilizer, Preventing the Hepcidin-Ferroportin Interaction and Modulating the Interleukin-6/Stat-3 Pathway.</p>Fórmula:C10H15N5O11P2Pureza:98.46% - 99.52%Cor e Forma:SolidPeso molecular:443.26-Aminonicotinic acid
CAS:<p>6-Aminonicotinic acid is a natural product.</p>Fórmula:C6H6N2O2Pureza:99.94%Cor e Forma:SoildPeso molecular:138.1238M8-B Hydrochloride
CAS:<p>M8-B Hydrochloride is a selective transient receptor potential melastatin-8 (TRPM8) channel antagonist.</p>Fórmula:C22H25ClN2O3SPureza:99.33%Cor e Forma:SolidPeso molecular:432.96Tetrabenazine Racemate
CAS:<p>Tetrabenazine Racemate (Rubigen) is a selective and reversible inhibitor of vesicular monoamine transporter-2 (VMAT-2).</p>Fórmula:C19H27NO3Pureza:98.65% - 98.86%Cor e Forma:SolidPeso molecular:317.42BZAD01
CAS:<p>BZAD01 is a selective NMDA NR1A/2B receptor antagonist.</p>Fórmula:C16H12F6N2OPureza:99.61% - 99.70%Cor e Forma:SolidPeso molecular:362.27DHQ
CAS:<p>DHQ (2,3-dihydroxy-quinoxalin) is an inducer of ATPase activity that of Herpes Simplex Virus thymidine kinase.</p>Fórmula:C8H6N2O2Pureza:99.89%Cor e Forma:SolidPeso molecular:162.15CL 218872
CAS:<p>CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.</p>Fórmula:C13H9F3N4Pureza:99.92%Cor e Forma:SolidPeso molecular:278.23Vonoprazan fumarate
CAS:<p>Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.</p>Fórmula:C17H16FN3O2S·C4H4O4Pureza:99.16% - 99.98%Cor e Forma:SolidPeso molecular:461.46Org 25543
CAS:<p>Org 25543 is the development of an N-Acyl amino acid that selectively inhibits the glycine transporter 2 to produce analgesia in a rat model of chronic pain.</p>Fórmula:C24H32N2O4Pureza:99.13%Cor e Forma:SolidPeso molecular:412.52HBT1
CAS:<p>HBT1 is an AMPA receptor potentiator that induces production of brain-derived neurotrophic factor (BDNF) and exhibits little agonistic effect in primary neurons</p>Fórmula:C16H17F3N4O2SPureza:99.52%Cor e Forma:SolidPeso molecular:386.39L-Phenylalanine-15N
CAS:L-Phenylalanine-15N, essential amino acid, Ca+ channel and NMDARs antagonist, used in food flavors and pharmaceuticals.Fórmula:C9H11NO2Pureza:98.98%Cor e Forma:SolidPeso molecular:166.18Pirmenol
CAS:<p>Pirmenol is a new antiarrhythmic drug</p>Fórmula:C22H30N2OPureza:97.24%Cor e Forma:SolidPeso molecular:338.49Nav1.8-IN-1
CAS:<p>Nav1.8-IN-1 (CHEMBL1270208) is an inhibitor of human NaV1.8</p>Fórmula:C20H15ClF3N3O2Pureza:97.59%Cor e Forma:SolidPeso molecular:421.8JNJ 303
CAS:<p>JNJ 303 is a potent blocker of IKs (IC50 : 64 nM).</p>Fórmula:C21H29ClN2O4SPureza:99.28%Cor e Forma:SolidPeso molecular:440.98Thonzonium Bromide
CAS:<p>Thonzonium bromide: antimicrobial surfactant, similar to Farnesol, blocks proton transport, inhibits bone loss (EC50=69 μM).</p>Fórmula:C32H55BrN4OPureza:98.48% - 99.94%Cor e Forma:SolidPeso molecular:591.71OAC3
CAS:<p>OAC3 (4-fluoro-N-(1H-indol-5-yl)benzamide) is an activator of octamer-bound transcription factor 4.</p>Fórmula:C15H11FN2OPureza:97.13%Cor e Forma:SolidPeso molecular:254.26Zoniporide hydrochloride hydrate
CAS:<p>Zoniporide HCl hydrate: selective NHE-1 inhibitor with a 14 nM IC50.</p>Fórmula:C17H19ClN6O2Pureza:98%Cor e Forma:SolidPeso molecular:374.83AMTB hydrochloride
CAS:<p>AMTB HCl: Novel TRPM8 blocker, relieves pain, treats urinary issues, moderates bladder reflexes in rats.</p>Fórmula:C23H27ClN2O2SPureza:99.08%Cor e Forma:SolidPeso molecular:430.99ML365
CAS:<p>ML365 is a novel selective small molecule inhibitor of TASK1(KCNK3).</p>Fórmula:C22H20N2O3Pureza:98.78%Cor e Forma:SolidPeso molecular:360.41AM-92016 hydrochloride
CAS:AM-92016 is a specific blocker of rectifier potassium current.Fórmula:C19H24Cl2N2O4S·HClPureza:98.68%Cor e Forma:SolidPeso molecular:483.84ASP2905
CAS:<p>ASP-2905 is a potent and selective inhibitor of potassium channel Kv12.2 encoded by the Kcnh3/BEC1 gene.</p>Fórmula:C20H17FN8Pureza:97.29%Cor e Forma:SolidPeso molecular:388.4Baclofen hydrochloride
CAS:<p>Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.</p>Fórmula:C10H13Cl2NO2Pureza:99.55%Cor e Forma:SolidPeso molecular:250.122Minoxidil sulfate
CAS:<p>Minoxidil sulfate (U-58838) is the active metabolite required to exert the vasodilatory and hair growing effects of minoxidil.</p>Fórmula:C9H15N5O4SPureza:99.01% - 99.72%Cor e Forma:White Crystalline SolidPeso molecular:289.31A-803467
CAS:<p>A-803467 is a selective NaV1.8 channel blocker.</p>Fórmula:C19H16ClNO4Pureza:96.94% - 98%Cor e Forma:SolidPeso molecular:357.79Prilocaine
CAS:<p>Prilocaine (NSC-40027) is a local anesthetic of the amino amide type, which acts on the sodium channel on the neuronal membrane and limits the spread of</p>Fórmula:C13H20N2OPureza:98.49%Cor e Forma:Needles SolidPeso molecular:220.31GlyH-101
CAS:<p>GlyH-101 is a cell-permeable glycinyl hydrazone compound that blocks CFTR with Ki of 1.4 uM.</p>Fórmula:C19H15Br2N3O3Pureza:98.71% - 98.78%Cor e Forma:SolidPeso molecular:493.15RY785
CAS:<p>RY785 is a potent and selective inhibitor of voltage-gated potassium channel such as KV2.2 (IC50 = 50 nM). RY785 may be used in pain relief studies.</p>Fórmula:C21H20N4O2SPureza:99.78%Cor e Forma:SolidPeso molecular:392.47Flupirtine maleate
CAS:<p>Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.</p>Fórmula:C15H17FN4O2·C4H4O4Pureza:99.5% - 99.9%Cor e Forma:Off-White Crystalline PowderPeso molecular:420.39Selinexor (KPT-330)
CAS:<p>Selinexor (KPT-330) is an orally available, small molecule inhibitor of CRM1 (exportin 1 or XPO1), with potential antineoplastic activity.</p>Fórmula:C17H11F6N7OPureza:98% - 99.97%Cor e Forma:SolidPeso molecular:443.31Quinine hydrobromide
CAS:<p>Quinidine: oral, selective P450db inhibitor, K+ channel blocker (IC50=19.9μM), antiarrhythmic, used in malaria research.</p>Fórmula:C20H25BrN2O2Cor e Forma:SolidPeso molecular:405.336ICA-121431
CAS:<p>ICA-121431: a potent Nav1.7 inhibitor (IC50=19 nM for rat), minimal effect on human Nav1.5/Nav1.7.</p>Fórmula:C23H19N3O3S2Pureza:98.06%Cor e Forma:SolidPeso molecular:449.55Vonoprazan
CAS:<p>Vonoprazan (TAK-438 (free base)) is an orally active potassium-competitive acid blocker.Vonoprazan can be used for the treatment of gastroduodenal ulcer and</p>Fórmula:C17H16FN3O2SPureza:99.87% - 99.92%Cor e Forma:SolidPeso molecular:345.39Eniporide hydrochloride
CAS:<p>Eniporide hydrochloride (EMD-96785 hydrochloride) serves as a robust inhibitor of the sodium/hydrogen (Na+/H+) exchange process.</p>Fórmula:C14H17ClN4O3SCor e Forma:SolidPeso molecular:356.83Esomeprazole hemistrontium
CAS:<p>Esomeprazole hemistrontium, potent oral proton pump inhibitor, reduces gastric acid by blocking H+, K+-ATPase.</p>Fórmula:C34H36N6O6S2SrCor e Forma:SolidPeso molecular:776.44Ononetin
CAS:<p>Ononetin (2',4'-Dihydroxy-2-(4-methoxyphenyl)acetophenone) is a TRPM3 channel blocker(IC50: 0.3 μM).</p>Fórmula:C15H14O4Pureza:98.06%Cor e Forma:SolidPeso molecular:258.27NPPB
CAS:<p>NPPB is a chloride channel blocker with IC50 of 80 nM .</p>Fórmula:C16H16N2O4Pureza:99.95%Cor e Forma:Light Yellow To Yellow SolidPeso molecular:300.31Ivacaftor
CAS:<p>Ivacaftor (VX-770) (VX-770) is a potentiator of CFTR targeting G551D-CFTR (EC50: 100 nM) and F508del-CFTR (EC50: 25 nM) in Fisher rat thyroid cells,</p>Fórmula:C24H28N2O3Pureza:99% - 99.98%Cor e Forma:SolidPeso molecular:392.49Myomodulin acetate(110570-93-9 free base)
<p>Myomodulin acetate is present in two identified aplysia neurons that contain myomodulin A the ARC motor neuron B16 and the abdominal neuron L10.</p>Fórmula:C38H71N11O10S2Pureza:99.24%Cor e Forma:SolidPeso molecular:906.17NS6180
CAS:<p>NS6180 is a potent and selective KCa3.1 channel inhibitor(IC50= 9 nM). It prevents T-cell activation and inflammation.</p>Fórmula:C16H12F3NOSPureza:99.83% - ≥95%Cor e Forma:SolidPeso molecular:323.33Jujuboside A
CAS:<p>Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.</p>Fórmula:C58H94O26Pureza:98% - >99.99%Cor e Forma:SolidPeso molecular:1207.35Flecainide hydrochloride
CAS:<p>Flecainide is a medication used to prevent and treat abnormally fast heart rates. This includes ventricular and supraventricular tachycardias.</p>Fórmula:C17H21ClF6N2O3Pureza:97.79%Cor e Forma:SolidPeso molecular:450.81BAY-8002
CAS:<p>BAY-8002 is a potent dual MCT1/2 inhibitor (IC50 values are 3, 8, and 12 nM at rat (C6), human (DLD-1) and mouse (4T1) MCT1 respectively).</p>Fórmula:C20H14ClNO5SPureza:98.7% - 99.13%Cor e Forma:SolidPeso molecular:415.85Tetraethylammonium chloride
CAS:<p>Tetraethylammonium chloride is a quaternary ammonium compound.</p>Fórmula:C8H20ClNPureza:≥95%Cor e Forma:White Solid Solid Particulate/PowderPeso molecular:165.7SAR7334 hydrochloride
CAS:<p>SAR7334 hydrochloride is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).</p>Fórmula:C21H24Cl3N3OPureza:98%Cor e Forma:SolidPeso molecular:440.79Pikamilone
CAS:<p>Pikamilone (Picamilon) is an intelligent medicine.</p>Fórmula:C10H12N2O3Pureza:99.38%Cor e Forma:White Crystalline PowderPeso molecular:208.21Raxatrigine
CAS:<p>Raxatrigine (CNV 1014802) has been investigated for the treatment of Bipolar Disorder and Bipolar Depression.</p>Fórmula:C18H19FN2O2Pureza:98% - 99.43%Cor e Forma:SolidPeso molecular:314.35ML329
CAS:<p>ML329 is a small molecule inhibitor of MITF, inhibiting TRPM-1 promoter activity.</p>Fórmula:C16H12N2O4SPureza:98.96%Cor e Forma:SolidPeso molecular:328.34UBP551
CAS:<p>UBP551 is a potent and selective NMDA receptors modulator.</p>Fórmula:C11H8O4Pureza:98.69%Cor e Forma:SolidPeso molecular:204.18Omecamtiv mecarbil
CAS:<p>Omecamtiv mecarbil (CK-1827452) has been used in trials studying the treatment and basic science of Heart Failure, Echocardiogram, Pharmacokinetics, Chronic</p>Fórmula:C20H24FN5O3Pureza:98% - 99.23%Cor e Forma:SolidPeso molecular:401.43VU0134992
CAS:<p>VU0134992 is an Kir4.1 blocker with an IC50 value of 0.97 μM</p>Fórmula:C20H31BrN2O2Pureza:99.86%Cor e Forma:SolidPeso molecular:411.38ML204
CAS:<p>ML204 is a novel potent antagonist that selectively modulates native TRPC4/C5 ion channels.</p>Fórmula:C15H18N2Pureza:98.1% - 99.72%Cor e Forma:SolidPeso molecular:226.32CCTA-1523
CAS:<p>CCTA-1523 is an efflux function of ABCG2 inhibitor. CCTA-1523 selectively reverses ABCG2-mediated MDR in cancer cells.</p>Fórmula:C16H15Cl2NO3Pureza:99.71%Cor e Forma:SolidPeso molecular:340.2Evifacotrep
CAS:<p>Evifacotrep: TRPC5 antagonist for neurological disease research (WO2020061162, compound 100).</p>Fórmula:C18H12ClF4N5O2Pureza:98.6%Cor e Forma:SolidPeso molecular:441.77RN-1734
CAS:<p>RN-1734 is selective TRPV4 channel antagonist(IC50 of 2.3 μM,5.9 μM,3.2 μM for hTRPV4, mTRPV4 and rTRPV4,respectively)</p>Fórmula:C14H22Cl2N2O2SPureza:99.1% - 99.3%Cor e Forma:SolidPeso molecular:353.31BPU-11
CAS:<p>BPU-11 (Biphenyl Urea 11) is an HCN4 CLP ligand that acts by modulating channel function and completely abolishing the cAMP-induced shift in V1/2.</p>Fórmula:C32H31N5OPureza:99.16%Cor e Forma:SolidPeso molecular:501.62ONO-8590580
CAS:<p>ONO-8590580 (CS-2894) is a negative allosteric modulator of GABAA α5.</p>Fórmula:C21H21FN6Pureza:99.43%Cor e Forma:SolidPeso molecular:376.43AMG9810
CAS:<p>AMG 9810 blocks capsaicin's action on TRPV1; human IC50=24.5 nM, rat IC50=85.6 nM.</p>Fórmula:C21H23NO3Pureza:99.79% - 99.95%Cor e Forma:SolidPeso molecular:337.41Levamlodipine hydrochloride
CAS:<p>Levamlodipine hydrochloride is a medication used to lower blood pressure and prevent chest pain.</p>Fórmula:C20H26Cl2N2O5Cor e Forma:SolidPeso molecular:445.34S0859
CAS:<p>S0859 is an N-cyanosulphonamide that blocks the sodium/bicarbonate cotransporter (NBC, also known as SLC4A7), which regulates intracellular pH.</p>Fórmula:C29H24ClN3O3SPureza:98% - 99.53%Cor e Forma:SolidPeso molecular:530.04GsMTx4 TFA (1209500-46-8 free base)
<p>GsMTx4 TFA is a spider venom peptide that selectively inhibits cationic permeable mechanically-sensitive channels (MSCs). Cost-effective and quality-assured.</p>Fórmula:C187H279N48O48S6F3Pureza:98% - 99.81%Cor e Forma:SolidPeso molecular:4216.93Efonidipine hydrochloride
CAS:<p>Efonidipine HCl (NZ-105) blocks T-type/L-type calcium channels; used in hypertension treatment.</p>Fórmula:C34H39ClN3O7PCor e Forma:SolidPeso molecular:668.12Tipepidine
CAS:<p>Tipepidine: non-narcotic cough suppressant, has antidepressant effects, inhibits DA D2 receptors (IC50=7.0 μM), activates VTA dopamine neurons.</p>Fórmula:C15H17NS2Cor e Forma:SolidPeso molecular:275.43NS11394
CAS:<p>NS11394 is a effective and subtype-selective GABA(A) receptor-positive modulator; possesses a functional efficacy selectivity profile of α(5) > α(3) > α(2) > α(</p>Fórmula:C23H19N3OPureza:99.44% - 99.86%Cor e Forma:SolidPeso molecular:353.42Aptiganel hydrochloride
CAS:<p>Aptiganel hydrochloride（Cerestat） is the salt form of Aptiganel.Aptiganel is a non-competitive NMDA antagonist with neuroprotective effects used in the treatment of stroke and focal cerebral ischemia.</p>Fórmula:C20H22ClN3Pureza:99.89%Cor e Forma:SolidPeso molecular:339.86Ginsenoside Rc
CAS:<p>Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.</p>Fórmula:C53H90O22Pureza:98.83% - 99.56%Cor e Forma:White PowderPeso molecular:1079.27Chloroprocaine
CAS:<p>Chloroprocaine: Na,K-ATPase inhibitor, IC50=13 mM, local anesthetic.</p>Fórmula:C13H19ClN2O2Cor e Forma:SolidPeso molecular:270.76AZD7325
CAS:<p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>Fórmula:C19H19FN4O2Pureza:99.83%Cor e Forma:SolidPeso molecular:354.38ABT-639 hydrochloride
CAS:<p>ABT-639 hydrochloride is a selective, novel T-type Ca2+ channel blocker.</p>Fórmula:C20H21Cl2F2N3O3SCor e Forma:SolidPeso molecular:492.36PF 429242
CAS:<p>PF-429242 inhibits SREBP site 1 protease selectively (IC50: 0.175 μM); reduces cholesterol synthesis in CHO cells (IC50: 0.53 μM).</p>Fórmula:C25H35N3O2Pureza:99.27%Cor e Forma:SolidPeso molecular:409.56Loreclezole hydrochloride
CAS:<p>Loreclezole hydrochloride is an antiepileptic, enhancing GABA A receptors with β2/β3 subunits.</p>Fórmula:C10H7Cl4N3Cor e Forma:SolidPeso molecular:310.99Bepridil free base
CAS:<p>Bepridil: Class IV anti-arrhythmic, calcium blocker, dilates coronary arteries.</p>Fórmula:C24H34N2OCor e Forma:SolidPeso molecular:366.54Ibutilide
CAS:<p>Ibutilide (U70226E) is an antiarrhythmic that prolongs action potential by blocking I Kr in AT-1 cells.</p>Fórmula:C20H36N2O3SCor e Forma:SolidPeso molecular:384.58BTS
CAS:<p>BTS (N-Tosylbenzylamine) is a potent inhibitor of Ca2+-stimulated myosin S1 ATPase (IC50 : 5 μM) .</p>Fórmula:C14H15NO2SPureza:99.45%Cor e Forma:White Crystalline SolidPeso molecular:261.34Fluralaner
CAS:<p>Fluralaner (A1443) is an isoxazoline ectoparasiticide.</p>Fórmula:C22H17Cl2F6N3O3Pureza:99.72% - 99.90%Cor e Forma:Solid PowderPeso molecular:556.29Nelonemdaz potassium
CAS:<p>Nelonemdaz potassium (Salfaprodil) is a potent NR2B-selective NMDA antagonist with neuroprotective properties.</p>Fórmula:C15H7F7KNO3Cor e Forma:SolidPeso molecular:421.31ICA-105574
CAS:<p>ICA-105574 activates hERG, enhancing peak current and shortening action potential, while modulating activation kinetics.</p>Fórmula:C19H14N2O4Pureza:98.89%Cor e Forma:SolidPeso molecular:334.33AZD7507
CAS:<p>AZD7507 is a CSF-1R inhibitor with an IC50 of 32 nM. AZD7507 has antitumor activity.</p>Fórmula:C23H27FN6O3Pureza:99.55% - 99.78%Cor e Forma:SolidPeso molecular:454.5Optovin
CAS:<p>Optovin is a TRPA1 activator, which is reversibly photoactivated.</p>Fórmula:C15H13N3OS2Pureza:99.47% - 99.67%Cor e Forma:SolidPeso molecular:315.41Bifemelane
CAS:<p>Bifemelane, a nootropic, releases Ca2+ from stores and enables its entry via channels for astrocyte research.</p>Fórmula:C18H23NOCor e Forma:SolidPeso molecular:269.38Rbin-1
CAS:<p>Rbin-1 (Ribozinoindole-1) is a potent,specific inhibitor of eukaryotic ribosome biogenesis.</p>Fórmula:C13H12N4SPureza:99.83%Cor e Forma:SolidPeso molecular:256.33Sepimostat dimethanesulfonate
CAS:<p>Sepimostat dimethanesulfonate (FUT-187) is a neuroprotective NR2B receptor antagonist with an inhibition Ki of 27.7 μM.</p>Fórmula:C23H27N5O8S2Cor e Forma:SolidPeso molecular:565.62Azumolene sodium anhydrous
CAS:<p>Azumolene sodium, a muscle relaxant, blocks calcium release from muscles and halts SOCE linked to RyR1 except when induced by thapsigargin.</p>Fórmula:C13H8BrN4NaO3Cor e Forma:SolidPeso molecular:371.13TRAM-34
CAS:<p>TRAM-34 (Triarylmethane-34), an effective and specific inhibitor of the intermediate-conductance Ca2+-activated K+ channel, does not block cytochrome P450.</p>Fórmula:C22H17ClN2Pureza:99.01% - 99.91%Cor e Forma:SolidPeso molecular:344.84Esomeprazole potassium salt
CAS:<p>Esomeprazole potassium, a potent oral proton pump inhibitor, curbs acid secretion in stomach cells, aiding GERD research.</p>Fórmula:C17H18KN3O3SCor e Forma:SolidPeso molecular:383.51Benzamil
CAS:<p>Benzamil blocks ENaC, inhibiting sodium transport (IC50=4 nM) and binds with Kd=5 nM to bovine kidney membranes.</p>Fórmula:C13H14ClN7OPureza:99.79%Cor e Forma:SolidPeso molecular:319.75BRITE-338733
CAS:<p>BRITE-338733 is a novel inhibitor of ATPase. BRITE 338733 inhibits the expression of RecA in bacteria (IC50=4.7 μM) for the bacterial infections treatment.</p>Fórmula:C27H35N3O2Pureza:99.85%Cor e Forma:SolidPeso molecular:433.59AM92016
CAS:<p>AM92016 is a specific blocker of the time dependent delayed rectifier potassium current. AM92016 does not show any β-adrenoceptor blocking activity.</p>Fórmula:C26H30Cl2N2O6SCor e Forma:SolidPeso molecular:569.49Tiagabine hydrochloride hydrate
CAS:<p>Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.</p>Fórmula:C20H28ClNO3S2Cor e Forma:SolidPeso molecular:430.02TC-I2000
CAS:<p>TC-I2000 is an TRPM8 channel blocker. Inhibits icilin-induced TRPM8 channel activation in rTRPM8-expressing CHO cells with IC50 of 53 nM.</p>Fórmula:C23H18F4N2OPureza:99.778%Cor e Forma:SolidPeso molecular:414.4Tezacaftor
CAS:<p>Tezacaftor (VX661) is a small molecule that can be used as a corrector of the cystic fibrosis transmembrane conductance regulator (CFTR) gene function.</p>Fórmula:C26H27F3N2O6Pureza:98.84% - >99.99%Cor e Forma:SolidPeso molecular:520.5CX614
CAS:<p>CX614 is a positive allosteric modulator of the AMPA receptor concerning AMPA.</p>Fórmula:C13H13NO4Pureza:97.37%Cor e Forma:SolidPeso molecular:247.25Tariquidar dihydrochloride
CAS:<p>Tariquidar dihydrochloride, also known as XR9576 dihydrochloride, is a potent, specific P-glycoprotein (P-gp) inhibitor exhibiting high affinity (Kd = 5.1 nM).</p>Fórmula:C38H40Cl2N4O6Cor e Forma:SolidPeso molecular:719.65GAL-021
CAS:<p>GAL-021 an intravenous BKCa-channel blocker.</p>Fórmula:C11H22N6OPureza:97.71% - 99.66%Cor e Forma:SolidPeso molecular:254.33Acecainide hydrochloride
CAS:<p>Acecainide hydrochloride (NAPA) is the major hepatic metabolite of procainamide.Cost-effective and quality-assured.</p>Fórmula:C15H24ClN3O2Pureza:98.023% - 99.81%Cor e Forma:SolidPeso molecular:313.836-(4-Methoxyphenyl)-3-pyridazinamine
CAS:<p>6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist</p>Fórmula:C11H11N3OPureza:99.03%Cor e Forma:SolidPeso molecular:201.22Cinacalcet metabolite M4
CAS:<p>Cinacalcet metabolite M4 (Rarechem AL BW 1078) is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.</p>Fórmula:C10H12F3NPureza:97.13%Cor e Forma:SolidPeso molecular:203.2Glibenclamide potassium
CAS:<p>Glibenclamide potassium, a more soluble form of Glibenclamide, exists as anhydrous and hydrate salts.</p>Fórmula:C23H27ClKN3O5SCor e Forma:SolidPeso molecular:532.09ZD7288
CAS:<p>ZD7288 (ICI D7288), a selective hyperpolarization-activated cyclic nucleotide-gated channel blocker, inhibits hippocampal synaptic plasticity.</p>Fórmula:C15H21ClN4Pureza:99.99%Cor e Forma:SolidPeso molecular:292.81ML 297
CAS:<p>ML 297 is a selective Kir3.1/3.2 (GIRK1/2) channel activator (IC50 values are 160, 887 and 914 nM for GIRK1/2, GIRK1/4 and GIRK1/3 respectively).</p>Fórmula:C17H14F2N4OPureza:97.85%Cor e Forma:SolidPeso molecular:328.32ML335
CAS:<p>ML335 is a selective activator of TREK-1 and TREK-2.</p>Fórmula:C15H14Cl2N2O3SPureza:99.73% - 99.79%Cor e Forma:SolidPeso molecular:373.25XEN907
CAS:<p>XEN907 is a novel spiro oxindole NaV1.7 blocker. XEN907 also inhibits hNaV1.7 (IC50: 3 nM).</p>Fórmula:C21H21NO4Pureza:99.92%Cor e Forma:SolidPeso molecular:351.4(S)-(-)-5-Fluorowillardiine hydrochloride
CAS:<p>(S)-(-)-5-Fluorowillardiine hydrochloride is a potent and specific agonist of AMPAR.</p>Fórmula:C7H9ClFN3O4Cor e Forma:SolidPeso molecular:253.62Amifampridine phosphate
CAS:<p>Amifampridine treats rare muscle diseases like LEMS and congenital myasthenias, targeting specific enzyme defects.</p>Fórmula:C5H10N3O4PCor e Forma:SolidPeso molecular:207.12Pipequaline hydrochloride
CAS:<p>Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.</p>Fórmula:C22H25ClN2Pureza:99.46%Cor e Forma:SolidPeso molecular:352.9Piperazine
CAS:<p>Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.</p>Fórmula:C4H10N2Cor e Forma:SolidPeso molecular:86.14Tiludronate
CAS:<p>Tiludronate, an oral bisphosphonate, treats metabolic bone disorders and inhibits osteoclasts.</p>Fórmula:C7H9ClO6P2SCor e Forma:SolidPeso molecular:318.61PF-4840154
CAS:<p>PF-4840154: potent TrpA1 agonist; EC50 of 97 nM (rat) & 23 nM (human); triggers nociception in mice.</p>Fórmula:C26H38N6O2Pureza:>99.99%Cor e Forma:SolidPeso molecular:466.62Enflurane
CAS:<p>Enflurane (Efrane), a volatile anaesthetic, inhibits Ca2+-activated K+ channels and is used to gauge anesthesia levels in gas chromatography.</p>Fórmula:C3H2ClF5OPureza:99.64%Cor e Forma:Clear Colorless Liquid Ordinary Temperature And Pressure Bp 56 8°C Density 1 50 G Cm-3 At Room Temperature Used As AnPeso molecular:184.49Elobixibat hydrate
CAS:<p>Elobixibat hydrate, an IBAT inhibitor, IC50: 0.53 nM (human), 0.13 nM (mouse), 5.8 nM (canine); for CIC research.</p>Fórmula:C36H47N3O8S2Cor e Forma:SolidPeso molecular:713.9JNJ-26990990
CAS:<p>"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."</p>Fórmula:C9H10N2O2S2Pureza:97.37%Cor e Forma:SolidPeso molecular:242.32Esomeprazole Magnesium
CAS:<p>Esomeprazole Magnesium (NEXIUM) is the S-isomer of omeprazole, can reduce gastric acid secretion with selective and irreversible proton pump inhibitor activity.</p>Fórmula:C34H36MgN6O6S2Pureza:98.76% - 99.73%Cor e Forma:SolidPeso molecular:713.12Epaminurad
CAS:<p>Epaminurad (UR-1102) is an oral URAT1 inhibitor for gout research with a Ki of 0.057 μM, modestly affects OAT1/3.</p>Fórmula:C14H10Br2N2O3Cor e Forma:SolidPeso molecular:414.054-Acetamidobutanoic acid
CAS:<p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>Fórmula:C6H11NO3Pureza:98.51%Cor e Forma:SolidPeso molecular:145.16Ropivacaine hydrochloride monohydrate
CAS:<p>Ropivacaine hydrochloride monohydrate (LEA-103 HCl) is an anaesthetic agent and blocks impulse conduction through inhibiting sodium ion influx reversibly.</p>Fórmula:C17H29ClN2O2Pureza:99.94% - 99.95%Cor e Forma:White SolidPeso molecular:328.88Pilsicainide
CAS:<p>Pilsicainide (SUN 1165 free acid) is a potent class Ic antiarrhythmic agent. Pilsicainide is a potent sodium channel blocker[1][2].</p>Fórmula:C17H24N2OCor e Forma:SolidPeso molecular:272.39Tiagabine
CAS:<p>Tiagabine (NO050328) is an Anti-epileptic Agent.</p>Fórmula:C20H25NO2S2Pureza:99.25%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:375.55Tetrabenazine methanesulfonate
CAS:<p>Tetrabenazine methanesulfonate: ex-antipsychotic/therapy for movement disorders, blocks neurotransmitter uptake, labels vesicle transport.</p>Fórmula:C20H31NO6SPureza:98%Cor e Forma:SolidPeso molecular:413.53Disopyramide phosphate
CAS:<p>Disopyramide: Class 1a anti-arrhythmic, treats Ventricular Tachycardia, reduces heart muscle contractility.</p>Fórmula:C21H32N3O5PCor e Forma:SolidPeso molecular:437.47QX-222 chloride
CAS:<p>QX-222 chloride (Lidocaine N-Methyl Hydrochloride) is a sodium channel blocker.</p>Fórmula:C13H21ClN2OPureza:97.37%Cor e Forma:SolidPeso molecular:256.77Safinamide
CAS:<p>Safinamide: reversible MAO-B inhibitor, enhances dopamine, blocks glutamate release, sodium, calcium channels; may treat Parkinson's, RLS, epilepsy.</p>Fórmula:C17H19FN2O2Pureza:99.92%Cor e Forma:SolidPeso molecular:302.34VU590
CAS:<p>VU590 is an inhibitor of extrarenal medullary potassium ROMK.VU590 inhibits Kir7.1 and modulates uterine myometrial contractility and melanocortin signalling.</p>Fórmula:C24H32N4O7Pureza:98.06%Cor e Forma:SolidPeso molecular:488.53JNJ-28583113
CAS:<p>JNJ-28583113 is a TRPM2 antagonist, inducing phosphorylation of GSK3α and β subunits, protecting cells from oxidative stress-induced cell death.</p>Fórmula:C19H21F3N2O2Pureza:98.57%Cor e Forma:SolidPeso molecular:366.38Apinocaltamide
CAS:<p>Apinocaltamide (ACT-709478) is an orally available and selective T-type calcium channel blocker that cross BBB for Cav3.1, Cav3.2, and Cav3.3,epilepsy.</p>Fórmula:C22H18F3N5OPureza:99.80%Cor e Forma:SolidPeso molecular:425.41CX717
CAS:<p>CX 717 is a positive allosteric modulator of AMPA receptor which has an antidepressant-like effect.</p>Fórmula:C11H11N3O3Pureza:99.81%Cor e Forma:SoildPeso molecular:233.23Riluzole
CAS:<p>Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.</p>Fórmula:C8H5F3N2OSPureza:99.71% - 99.88%Cor e Forma:PowderPeso molecular:234.2HUP30
CAS:<p>HUP30 is a potent vasodilating agent. HUP30 can stimulate soluble guanylyl cyclase, activate K+ channels, and block extracellular Ca2+ influx.</p>Fórmula:C14H15N3O3SPureza:99.96%Cor e Forma:SolidPeso molecular:305.35N-Methyl-L-leucin
CAS:<p>N-Methyl-L-leucine ((S)-4-Methyl-2-(methylamino)pentanoic acid) is a novel calcium channel antagonist used in pain research.</p>Fórmula:C7H15NO2Pureza:99.87%Cor e Forma:SolidPeso molecular:145.2SRI-41315
CAS:<p>SRI-41315 is an eRF1 degrader that acts as a molecular glue at the ribosomal decoding center.SRI-41315 induces extended pauses at the termination codon.</p>Fórmula:C22H19N3O2Pureza:99.87%Cor e Forma:SolidPeso molecular:357.41Dimiracetam
CAS:<p>Dimiracetam, a NMDA-receptor antagonist, is used potentially for the treatment of neuropathic pain.</p>Fórmula:C6H8N2O2Pureza:>99.99% - >99.99%Cor e Forma:SolidPeso molecular:140.14ZT-1a
CAS:<p>ZT-1a is a SPAK inhibitor.ZT-1a inhibits SPAK.ZT-1a can be used for the prevention and treatment of neurodegenerative and neurocognitive disorders.</p>Fórmula:C22H15Cl3N2O2Pureza:99.77%Cor e Forma:SolidPeso molecular:445.73Ro 25-6981 Maleate
CAS:<p>Ro 25-6981 Maleate is an NMDA receptor antagonist used in the study of neurological disorders such as Parkinson's and epilepsy.</p>Fórmula:C26H33NO6Pureza:99.42%Cor e Forma:SolidPeso molecular:455.54Doxapram
CAS:<p>Doxapram (Dopram) is a respiratory stimulant that inhibits TASK-1, TASK-3, and TASK-1/TASK-3 heterodimer channels.</p>Fórmula:C24H30N2O2Pureza:99.42%Cor e Forma:SolidPeso molecular:378.51VB124
CAS:<p>VB124 is an orally active, potent and selective MCT4 inhibitor. VB124 blocked lactate importand expor in MDA-MB-231 cells.Cost-effective and quality-assured.</p>Fórmula:C23H23ClN2O4Pureza:99.21% - 99.57%Cor e Forma:SoildPeso molecular:426.89Darigabat
CAS:<p>Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.</p>Fórmula:C22H21FN4O3SPureza:98.42% - 99.29%Cor e Forma:SolidPeso molecular:440.49Mtb ATP synthase-IN-1
CAS:<p>Mtb ATP synthase-IN-1 is a potent, low-toxicity M. tuberculosis inhibitor with good oral bioavailability and metabolic stability.</p>Fórmula:C17H13N3O4Pureza:98.28%Cor e Forma:SolidPeso molecular:323.30Methionine
CAS:<p>Methionine (D-Methionine) (MRX-1024; D-Methionine) is an effective chemoprotective agent which can also inhibit the neuronal activity through GABAA receptor</p>Fórmula:C5H11NO2SPureza:99.13% - 99.62%Cor e Forma:SolidPeso molecular:149.21PF 03716556
CAS:<p>PF 03716556 (PF-3716556) , an effective and specific P-CAB (potassium-competitive acid blocker), is utilized for the treatment of gastroesophageal reflux</p>Fórmula:C22H26N4O3Pureza:99.79% - 99.85%Cor e Forma:SolidPeso molecular:394.47Lanicemine dihydrochloride
CAS:<p>Lanicemine dihydrochloride (AZD-6765 dihydrochloride) is an NMDA channel blocker with antidepressant activity and can be used to study neurological diseases.</p>Fórmula:C13H16Cl2N2Pureza:98.37%Cor e Forma:SolidPeso molecular:271.19Bupivacaine
CAS:<p>Bupivacaine (AH-250) is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channels</p>Fórmula:C18H28N2OPureza:99.83%Cor e Forma:SolidPeso molecular:288.43Propoxycaine hydrochloride
CAS:<p>Propoxycaine hydrochloride is an ester local anesthetic that inhibits voltage-gated sodium channels, modulates nerve impulses, and induces loss of sensation.</p>Fórmula:C16H27ClN2O3Pureza:97.25%Cor e Forma:SolidPeso molecular:330.85BL-1249
CAS:<p>BL-1249 is a selective and potent non-steroidal potassium channel activator with anti-inflammatory activity that activates K2P2.1 (TREK-1) and K2P10.1 (TREK-2).</p>Fórmula:C17H17N5Pureza:98% - 98.25%Cor e Forma:SolidPeso molecular:291.35Bupivacaine-d9
CAS:Bupivacaine-d9 is a deuterated compound of Bupivacaine. Bupivacaine has a CAS number of 38396-39-3. Bupivacaine is a NMDA receptor inhibitor.Bupivacaine can block sodium, L-calcium, and potassium channels.Bupivacaine potently blocks SCN5A channels with the IC50 of 69.5 μM. Bupivacaine can be used for the research of chronic pain.Fórmula:C18H19D9N2OCor e Forma:SolidPeso molecular:297.48SAR7334
CAS:<p>SAR7334 (TRCP6-IN-1) is a potent and specific inhibitor of TRPC6(IC50 of 7.9 nM).</p>Fórmula:C21H22ClN3OPureza:99.62% - 99.71%Cor e Forma:SolidPeso molecular:367.87Eleclazine
CAS:<p>Eleclazine (GS-6615) is a novel and selective voltage-gated sodium channel inhibitor with antiarrhythmic properties that reduces peak sodium current (INaP).</p>Fórmula:C21H16F3N3O3Pureza:98.67%Cor e Forma:SolidPeso molecular:415.37Amlodipine besilate impurity G
CAS:<p>Amlodipine besilate impurity G is a Calcium Channel antagonist with potential application in the study of neurological diseases and is an impurity in the</p>Fórmula:C17H18ClNO4Pureza:98%Cor e Forma:SolidPeso molecular:335.78Amlodipine hydrochloride
CAS:<p>Amlodipine hydrochloride is a salt of Amlodipine --- a medication used to lower blood pressure and prevent chest pain.</p>Fórmula:C20H26Cl2N2O5Cor e Forma:SolidPeso molecular:445.34FSC231
CAS:<p>FSC231 is a PICK1 inhibitor with analgesic activity, activating GSK-3β and ERK1/2.</p>Fórmula:C13H10Cl2N2O3Pureza:99.66%Cor e Forma:SolidPeso molecular:313.14VGSC blocker-1
CAS:<p>VGSC blocker-1 inhibits 34.9% INa in nNav1.5 at 1 μM, reduces MDA-MB-231 invasion by 0.3%, non-toxic.</p>Fórmula:C24H32F2N2Cor e Forma:SolidPeso molecular:386.52Eperisone
CAS:<p>Eperisone: a muscle relaxant for stiffness and pain, relaxes muscles, improves circulation, and mitigates pain by inhibiting reflexes and vasodilation.</p>Fórmula:C17H25NOCor e Forma:SolidPeso molecular:259.39MCT-IN-1
CAS:<p>MCT-IN-1 (compound 2) acts as a potent inhibitor of the monocarboxylate transporter (MCT), demonstrating IC50 values of 9 nM for MCT1 and 14 nM for MCT4.</p>Fórmula:C19H26N2O3Cor e Forma:SolidPeso molecular:330.42Flavoxate
CAS:<p>Flavoxate is an anticholinergic with antimuscarinic effects.</p>Fórmula:C24H25NO4Cor e Forma:SolidPeso molecular:391.46Cinepazide
CAS:<p>Cinepazide: a vasodilator targeting adenosine A2 receptors, treats various vascular diseases.</p>Fórmula:C22H31N3O5Cor e Forma:White PowderPeso molecular:417.5BAY-390
CAS:<p>BAY-390, a selective TRPA1 inhibitor, crosses species, penetrates brains, with IC50s: 16-82 nM. Used in inflammation research.</p>Fórmula:C13H15F4NOCor e Forma:SolidPeso molecular:277.26Propafenone D7 hydrochloride
CAS:<p>Propafenone D7 hydrochloride is the deuterium labeled Propafenone, and is a classic anti-arrhythmic medication.</p>Fórmula:C21H28ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:384.95Methocarbamol D5
CAS:<p>Methocarbamol is a central muscle relaxant. Methocarbamol D5 is deuterium labeled Methocarbamol.</p>Fórmula:C11H15NO5Pureza:98%Cor e Forma:SolidPeso molecular:246.27PBFI-AM
CAS:<p>PBFI-AM is a useful tool to determine intracellular K + content [1] .</p>Fórmula:C58H62N2O24Cor e Forma:SolidPeso molecular:1171.11Nifedipine-d6
CAS:<p>Nifedipine D6 is deuterium labeled nifedipine which is a potent blocker of calcium channel.</p>Fórmula:C17H18N2O6Pureza:98%Cor e Forma:SolidPeso molecular:352.37Repaglinide D5
CAS:<p>Repaglinide D5 is deuterium labeled Repaglinide. Repaglinide is an insulin secretagogue for treatment type-2 diabetes mellitus.</p>Fórmula:C27H36N2O4Pureza:98%Cor e Forma:SolidPeso molecular:457.62Dofetilide D4
CAS:<p>Dofetilide D4 (UK 68789 D4), a deuterium-labeled version of Dofetilide, is categorized as a Class III antiarrhythmic medication.</p>Fórmula:C19H27N3O5S2Pureza:98%Cor e Forma:SolidPeso molecular:445.59Topiramate D12
CAS:<p>Topiramate D12 is a deuterium labeled Topiramate. Topiramate is an agent of broad-spectrum antiepileptic. Topiramate is an antagonist of GluR5 receptor.</p>Fórmula:C12H21NO8SPureza:98%Cor e Forma:SolidPeso molecular:351.44Bumetanide-d5
CAS:<p>Bumetanide D5 is a deuterium-labeled Bumetanide. Bumetanide is a Na+-K+-Cl- (NKCC1) inhibitor (IC50s: 0.68 and 4.0 μM for hNKCC1A and hNKCC2A).</p>Fórmula:C17H20N2O5SPureza:98%Cor e Forma:SolidPeso molecular:369.45A-317491 sodium salt hydrate
<p>A-317491 sodium salt hydrate is a non-nucleotide P2X3 and P2X2/3 receptor antagonist, which inhibits calcium flux mediated by the receptors.</p>Fórmula:C33H29NNaO9Pureza:98%Cor e Forma:SolidPeso molecular:606.57N-Acetylglycyl-D-glutamic acid
CAS:<p>Excitatory peptide that induces seizures</p>Fórmula:C9H14N2O6Pureza:98%Cor e Forma:SolidPeso molecular:246.22R-(-)-Niguldipine hydrochloride
CAS:<p>R-(-)-Niguldipine HCl: L-type Ca2+ blocker, K+ agonist, α1A antagonist; lowers blood pressure; weaker enantiomer.</p>Fórmula:C36H40ClN3O6Cor e Forma:SolidPeso molecular:646.178-Pcpt-cGMP sodium
CAS:<p>8-Pcpt-cGMP sodium, with an EC50 of 0.5 μM, acts as an agonist for cyclic nucleotide-gated (CNG) channels and demonstrates effective membrane permeability. This compound is utilized in research focused on the role of CNG channels in visual and olfactory signal transduction.</p>Fórmula:C16H14ClN5NaO7PSCor e Forma:SolidPeso molecular:509.79MNI-caged-NMDA
CAS:<p>NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group</p>Fórmula:C14H17N3O6Pureza:98%Cor e Forma:SolidPeso molecular:323.30Pradigastat
CAS:Pradigastat (LCQ-908) is a diacylglycerol acyltransferase 1 (DGAT1) inhibitor for the treatment of constipation and can be used in the study of obesityFórmula:C25H24F3N3O2Pureza:95.21% - 95.21%Cor e Forma:SolidPeso molecular:455.47
