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Transportador de Membranas/Canal Iónico

Transportador de Membranas/Canal Iónico

Os inibidores de transportadores de membrana e canais iônicos são compostos que bloqueiam a função de proteínas responsáveis pelo transporte de íons, nutrientes e outras moléculas através das membranas celulares. Esses inibidores são cruciais para o estudo da regulação da homeostase celular, transdução de sinais e neurotransmissão. Os inibidores de transportadores de membrana e canais iônicos também são importantes no desenvolvimento de tratamentos para distúrbios como epilepsia, doenças cardiovasculares e síndromes metabólicas. Na CymitQuimica, oferecemos uma ampla seleção de inibidores de alta qualidade de transportadores de membrana e canais iônicos para apoiar sua pesquisa em fisiologia, neurociência e farmacologia.

Subcategorias de "Transportador de Membranas/Canal Iónico"

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Foram encontrados 2280 produtos de "Transportador de Membranas/Canal Iónico"

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  • Tetradifon

    CAS:
    <p>Tetradifon is a broad-spectrum organochlorine acaricide that inhibits mitochondrial OSCP, blocking energy production (IC50=4.5-27nmoL/mg) with oligomycin-like effects.</p>
    Fórmula:C12H6Cl4O2S
    Pureza:99.84%
    Cor e Forma:Yellowish Odorless Oil
    Peso molecular:356.05
  • Pradigastat

    CAS:
    Pradigastat (LCQ-908) is a diacylglycerol acyltransferase 1 (DGAT1) inhibitor for the treatment of constipation and can be used in the study of obesity
    Fórmula:C25H24F3N3O2
    Pureza:95.21% - 95.21%
    Cor e Forma:Solid
    Peso molecular:455.47
  • Diphenidol

    CAS:
    <p>Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.</p>
    Fórmula:C21H27NO
    Cor e Forma:Needles From Petroleum Ether Solid
    Peso molecular:309.45
  • N-Acetylglycyl-D-glutamic acid

    CAS:
    <p>Excitatory peptide that induces seizures</p>
    Fórmula:C9H14N2O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:246.22
  • S1647

    CAS:
    S1647 is a dual inhibitor targeting both ASBT and SOAT. It is utilized in research focused on intrahepatic cholestasis, cholestatic pruritus, and constipation.
    Fórmula:C19H13Cl2N3O5S
    Peso molecular:466.30
  • MNI-caged-NMDA

    CAS:
    <p>NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group</p>
    Fórmula:C14H17N3O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:323.30
  • DL-AP7

    CAS:
    <p>DL-AP7: competitive NMDA antagonist, anticonvulsant, inhibits NMDA convulsions, impairs mice learning.</p>
    Fórmula:C7H16NO5P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:225.18
  • Clopamide

    CAS:
    <p>Clopamide (Brinaldix) is a piperidine and sulfamoylbenzamide-based diuretic with thiazide-like diuretic activity.</p>
    Fórmula:C14H20ClN3O3S
    Pureza:99.71%
    Cor e Forma:White To Yellowish Crystalline Powder
    Peso molecular:345.84
  • IEM 1754 2HBr

    CAS:
    <p>IEM 1754 2HBr (IEM 1754 dihydrobromide) is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM.</p>
    Fórmula:C16H30N2·2HBr
    Pureza:99.71% - 99.72%
    Cor e Forma:Solid
    Peso molecular:412.25
  • Verapamil

    CAS:
    <p>Verapamil (CP-16533-1), an oral calcium channel blocker, inhibits P-gp and CYP3A4, used for hypertension, arrhythmias, and angina research.</p>
    Fórmula:C27H38N2O4
    Pureza:99.61% - 99.93%
    Cor e Forma:Oil
    Peso molecular:454.6
  • Otaplimastat

    CAS:
    <p>SP-8203 is a reactive oxygen species inhibitor and superoxide dismutase stimulant.</p>
    Fórmula:C28H34N6O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:534.61
  • DL-AP5 Sodium salt

    CAS:
    DL-AP5 Sodium salt is a NMDA receptor antagonist.
    Fórmula:C5H12NNaO5P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:220.12
  • JYL 1421

    CAS:
    <p>JYL 1421 (SC 0030) is an antagonist of TRPV1 receptor (IC50 = 8 nM).</p>
    Fórmula:C20H26FN3O2S2
    Pureza:98.83%
    Cor e Forma:Solid
    Peso molecular:423.57
  • Linopirdine dihydrochloride

    CAS:
    <p>KV7 (KCNQ) voltage-gated potassium channels blocker</p>
    Fórmula:C26H22ClN3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:427.93
  • TDN345

    CAS:
    <p>TDN345 is a antagonist of Ca2+, for the treatment of vascular and senile dementia including Alzheimer's disease.</p>
    Fórmula:C28H34F2N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:468.58
  • Lu AE98134

    CAS:
    <p>Lu AE98134 enhances Nav1.1, Nav1.2, and Nav1.5 sodium channels, but not Nav1.4/1.6/1.7; studied in CNS diseases like schizophrenia.</p>
    Fórmula:C21H23N5O3S
    Cor e Forma:Solid
    Peso molecular:425.5
  • PK-THPP

    CAS:
    <p>PK-THPP is a channel blocker of TASK-3.</p>
    Fórmula:C29H32N4O2
    Cor e Forma:Solid
    Peso molecular:468.59
  • MPX-007

    CAS:
    <p>MPX-007, a potent NMDA inhibitor, inhibits GluN2A-containing NMDA receptors expressed in HEK cells with IC50s of 27 nM.</p>
    Fórmula:C18H17F2N5O3S2
    Cor e Forma:Solid
    Peso molecular:453.49
  • LUF7346

    CAS:
    <p>LUF7346 is an allosteric modulator of hERG.</p>
    Fórmula:C20H15BrN2O3
    Cor e Forma:Solid
    Peso molecular:411.25
  • NS5818

    CAS:
    <p>NS5818 inhibits ClC.</p>
    Fórmula:C23H19Cl2N7O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:496.35
  • P-CAB agent 2

    CAS:
    <p>Potent P-CAB agent 2 blocks gastric acid secretion; H+/K+-ATPase IC50 &lt;100 nM, hERG IC50 18.69 μM; non-toxic.</p>
    Fórmula:C22H25FN2O4S
    Cor e Forma:Solid
    Peso molecular:432.51
  • RS 029

    CAS:
    <p>RS 029 is a nitroimidazole that has been exhibited to significantly inhibit (Na+K+) ATP-ase activity.</p>
    Fórmula:C13H16N6O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:352.3
  • CP 339818 hydrochloride

    CAS:
    <p>KV1.3 channel antagonist</p>
    Fórmula:C21H25ClN2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:340.89
  • Laniquidar

    CAS:
    <p>Laniquidar (R101933) inhibits P-glycoprotein (IC50: 0.51 μM), poor oral bioavailability, modulates drug resistance transporters.</p>
    Fórmula:C37H36N4O3
    Cor e Forma:Solid
    Peso molecular:584.71
  • Vincanol

    CAS:
    <p>Vincanol is a potent voltage-gated Na+ channels blocker.</p>
    Fórmula:C19H24N2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:296.41
  • NS004

    CAS:
    <p>NS004 is a large-conductance K+ channel opener, it inhibits mitochondrial function in glioma cells.</p>
    Fórmula:C14H8ClF3N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:328.67
  • BGT1-IN-9

    CAS:
    <p>BGT1-IN-9 is an M1 muscarinic agonist.</p>
    Fórmula:C5H10ClN3O2
    Cor e Forma:Solid
    Peso molecular:179.605
  • KCa2 channel modulator 1

    CAS:
    <p>Compound 2o, a selective K/Ca2 channel enhancer, boosts rat K Ca 2.2 (EC50: 0.99 μM) and human K Ca 2.3 (EC50: 0.19 μM).</p>
    Fórmula:C16H15ClFN5
    Cor e Forma:Solid
    Peso molecular:331.78
  • (S)-(-)-5-Iodowillardiine

    CAS:
    <p>hGluR5 kainate receptor agonist</p>
    Fórmula:C7H8IN3O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:325.06
  • Leconotide

    CAS:
    <p>Leconotide is a calcium channel blocker and antihyperalgesia agent; isolated from the venom of the cone snail, Conus catus.</p>
    Fórmula:C107H179N35O36S7
    Cor e Forma:Solid
    Peso molecular:2756.23
  • TTA-P2

    CAS:
    <p>TTA-P2: potent CNS-penetrating T-type Ca2+ channel blocker; eliminates Cav3.1 window currents.</p>
    Fórmula:C21H29Cl2FN2O2
    Cor e Forma:Solid
    Peso molecular:431.37
  • NAV26

    CAS:
    <p>NAV26 is a selective blocker of the Nav1.7 channel.</p>
    Fórmula:C22H21F3N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:434.41
  • GABAA receptor modulator-2

    CAS:
    <p>Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.</p>
    Fórmula:C22H22FN3O5S
    Cor e Forma:Solid
    Peso molecular:459.49
  • ANO1-IN-2

    CAS:
    <p>ANO1-IN-2: potent ANO1 blocker (IC50: 1.75 μM), less effective on ANO2 (IC50: 7.43 μM), inhibits glioblastoma cell growth.</p>
    Fórmula:C16H14ClN3O2S2
    Cor e Forma:Solid
    Peso molecular:379.88
  • BMS-284640

    CAS:
    <p>BMS-284640 is a NHE inhibitor that protects against MI in animal studies.</p>
    Fórmula:C15H19N3O2
    Cor e Forma:Solid
    Peso molecular:273.33
  • Lanicemine

    CAS:
    <p>Lanicemine is a low-trapping NMDA channel blocker. It also has a binding (Ki: 0.56-2.1 μM).</p>
    Fórmula:C13H14N2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:198.26
  • P2X2/3 modulator-1

    CAS:
    <p>Compound 46, a P2X2/3 modulator, could aid in research of pain, CNS disorders, and inflammation.</p>
    Fórmula:C26H21N5O
    Cor e Forma:Solid
    Peso molecular:419.48
  • RuBi-4AP

    CAS:
    <p>voltage-dependent K+ channel blocker</p>
    Fórmula:C30H28Cl2N8Ru
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:672.57
  • UTA1inh-C1

    CAS:
    <p>UTA1inh-C1 is a novel inhibitor of kidney urea transporter UT-A1.</p>
    Fórmula:C22H24N6O4S2
    Cor e Forma:Solid
    Peso molecular:500.59
  • BIIB-513

    CAS:
    <p>BIIB-513 is an inhibitor of Na+/H+ exchange.</p>
    Fórmula:C19H25N5O8S2
    Cor e Forma:Solid
    Peso molecular:515.56
  • GDC-0276

    CAS:
    <p>GDC-0276 is an orally active, selective, and potent NaV1.7 inhibitor that can be used for the study of pain-related diseases.</p>
    Fórmula:C24H31FN2O4S
    Pureza:99.77%
    Cor e Forma:Solid
    Peso molecular:462.58
  • Ro 41-3290

    CAS:
    <p>Ro 41-3290 is the desethylated derivative of Ro 41-3696, which is an agonist of nonbenzodiazepine partial at the benzodiazepine receptor.</p>
    Fórmula:C24H21ClN2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:420.89
  • TRPC6-IN-3

    CAS:
    <p>TRPC6-IN-3 is an oral TRPC6 ion channel inhibitor, regulating calcium levels and membrane potential.</p>
    Fórmula:C22H22FN5O3
    Cor e Forma:Solid
    Peso molecular:423.44
  • KR-30450

    CAS:
    <p>KR-30450, a potassium channel agonist, is used potentially for the treatment of hypertension.</p>
    Fórmula:C17H18N2O6
    Cor e Forma:Solid
    Peso molecular:346.33
  • CP-409092 hydrochloride

    CAS:
    <p>CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.</p>
    Fórmula:C17H20ClN3O2
    Cor e Forma:Solid
    Peso molecular:333.81
  • GABAA receptor agent 5

    CAS:
    <p>Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.</p>
    Fórmula:C21H25N3O2S
    Cor e Forma:Solid
    Peso molecular:383.51
  • GNE-0439

    CAS:
    <p>GNE-0439 is a Nav1.7-selective inhibitor (IC50 0.34 μM), also targeting Nav1.5 and mutant N1742K channels, valuable for ion channel research.</p>
    Fórmula:C21H31NO3
    Pureza:99.60%
    Cor e Forma:Solid
    Peso molecular:345.48
  • Taquidil

    CAS:
    <p>Tocainide hydrochloride: oral antiarrhythmic, sodium channel blocker, akin to lidocaine.</p>
    Fórmula:C11H17ClN2O
    Cor e Forma:Solid
    Peso molecular:228.718
  • Procyclidine

    CAS:
    <p>Procyclidine is an anticholinergic, muscarinic and NMDA antagonist used in Parkinson's and psychiatric disorder studies.</p>
    Fórmula:C19H29NO
    Cor e Forma:Solid
    Peso molecular:287.44
  • TMB 8 (hydrochloride)

    CAS:
    <p>TMB 8 blocks nAChRs (IC50: 390-480 nM), reduces Ca2+ in muscles, hinders rabbit aorta contraction at 50 μM, and inhibits PKC dose-dependently.</p>
    Fórmula:C22H38ClNO5
    Cor e Forma:White Solid
    Peso molecular:431.99
  • Etbicyphat

    CAS:
    <p>Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.</p>
    Fórmula:C6H11O4P
    Cor e Forma:Solid
    Peso molecular:178.12
  • CGP-78608

    CAS:
    <p>CGP-78608 is a glycine site-specific N-methyl-D-aspartate receptor antagonist prevents activation of the NMDA/NO/CGMP pathway by ammonia.</p>
    Fórmula:C11H13BrN3O5P
    Cor e Forma:Solid
    Peso molecular:378.12
  • TTT-28

    CAS:
    <p>TTT-28, a thiazole-valine peptidomimetic, selectively inhibits ABCB1 to reverse MDR with low toxicity.</p>
    Fórmula:C31H31N3O6S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:573.66
  • Radequinil

    CAS:
    <p>Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).</p>
    Fórmula:C18H14N4O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:334.33
  • PF-06649298

    CAS:
    <p>PF-06649298 inhibits NaCT, blocking citrate transport in hepatocytes, IC50: 16.2 μM, affects glucose and lipid metabolism.</p>
    Fórmula:C16H22O5
    Cor e Forma:Solid
    Peso molecular:294.34
  • Ro 19-4603

    CAS:
    <p>Benzodiazepine inverse agonist</p>
    Fórmula:C15H17N3O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:319.38
  • P2X3 antagonist 36

    CAS:
    <p>P2X3 antagonist 36 is a P2X3 antagonist.</p>
    Fórmula:C20H18ClF3N6O3
    Cor e Forma:Solid
    Peso molecular:482.84
  • UBP618

    CAS:
    <p>UBP618 is a GluN1/GluN2 receptors pan-inhibitor.</p>
    Fórmula:C17H11BrO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:343.17
  • LY 233053

    CAS:
    <p>LY 233053 is a Competitive NMDA receptor antagonist.</p>
    Fórmula:C8H13N5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:211.22
  • ATPA

    CAS:
    <p>ATPA activates GluR5 glutamate receptors; EC50s range 0.66-32 μM across GluR5 variants.</p>
    Fórmula:C10H16N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:228.24
  • GX-585

    CAS:
    <p>GX-585 is a novel potent inhibitor of NaV1.7 and highly selective against NaV1.5, having limited selectivity against NaV1.1 and NaV1.2.</p>
    Fórmula:C24H25Cl2FN4O3S
    Pureza:99.02% - 99.03%
    Cor e Forma:Solid
    Peso molecular:539.45
  • GS-462808

    CAS:
    <p>GS-462808: Cardiac Nav1.5 inhibitor, less brain penetration/activity.</p>
    Fórmula:C17H12F3N5O3
    Cor e Forma:Solid
    Peso molecular:391.3
  • Pipazethate

    CAS:
    <p>Pipipyrazine is a nonnarcotic oral cough suppressant, cough suppressant.</p>
    Fórmula:C21H25N3O3S
    Cor e Forma:Solid
    Peso molecular:399.51
  • Cavα2δ1&NET-IN-2

    CAS:
    <p>Cavα2δ1&amp;NET-IN-2 .</p>
    Fórmula:C22H26N6O2S
    Cor e Forma:Solid
    Peso molecular:438.55
  • Bliretrigine

    CAS:
    <p>Bliretrigine, a sodium channel blocker, effectively relieves pain [1] [2] [3].</p>
    Fórmula:C20H24N4O2
    Cor e Forma:Solid
    Peso molecular:352.43
  • DS2

    CAS:
    <p>Positive allosteric modulator of δ-subunit containing GABAA receptors</p>
    Fórmula:C18H12ClN3OS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:353.83
  • AJG-049 HCl

    CAS:
    <p>AJG-049 HCl is a calcium channel antagonist that inhibits L-type Ca2+ channels via diltiazem-binding site(s).</p>
    Fórmula:C27H31ClN2O2
    Cor e Forma:Solid
    Peso molecular:451.01
  • NNC052090

    CAS:
    <p>NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).</p>
    Fórmula:C27H30N2O2
    Cor e Forma:Solid
    Peso molecular:414.54
  • A 784168

    CAS:
    <p>A-784168: potent, oral TRPV1 inhibitor with good CNS penetration.</p>
    Fórmula:C19H15F6N3O3S
    Cor e Forma:Solid
    Peso molecular:479.4
  • Arachidonyl serotonin

    CAS:
    <p>Dual FAAH inhibitor/TRPV1 antagonist</p>
    Fórmula:C30H42N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:462.67
  • P-CAB agent 1

    CAS:
    <p>Compound B19, a P-CAB, inhibits H+/K+-ATPase with IC50 of 60.50 nM, useful in ARD research.</p>
    Fórmula:C26H23FN4O
    Cor e Forma:Solid
    Peso molecular:426.49
  • UR-MB108

    CAS:
    <p>UR-MB108 is a potent and selective inhibitor of ABCG2 (BCRP), displaying an IC50 value of 79 nM, and exhibits stability in blood plasma.</p>
    Fórmula:C40H38N6O4
    Cor e Forma:Solid
    Peso molecular:666.77
  • Cariporide Mesylate

    CAS:
    <p>Cariporide Mesylate is a selective inhibitor of the Na+/H+ exchanger isoform 1.</p>
    Fórmula:C13H21N3O6S2
    Cor e Forma:Solid
    Peso molecular:379.45
  • U89232

    CAS:
    <p>U-89232 is an opener of the cardioselective KATP channel.</p>
    Fórmula:C19H25N5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:355.43
  • UK-52831

    CAS:
    <p>UK-52831, a calcium channel antagonist, is used potentially for the treatment of hypertension and myocardia ischemia.</p>
    Fórmula:C22H26Cl2N6O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:525.39
  • URAT1 inhibitor 4

    CAS:
    <p>URAT1 inhibitor 4 is a potent, orally active Lesinurad derivative with a 7.56 μM IC50, showing greater in vivo efficacy.</p>
    Fórmula:C27H20BrN3O4S3
    Cor e Forma:Solid
    Peso molecular:626.56
  • TC-P 262

    CAS:
    <p>P2X3 and P2X2/3 receptor antagonist</p>
    Fórmula:C14H18N4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:258.32
  • Azimilide

    CAS:
    <p>class III anti-arrhythmic drug</p>
    Fórmula:C23H28ClN5O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:457.95
  • TRPM4-IN-2

    CAS:
    <p>NBA, or TRPM4-IN-2, is a potent TRPM4 inhibitor with IC50 of 0.16 μM, used in prostate and colorectal cancer research.</p>
    Fórmula:C19H14ClNO4
    Pureza:99.21%
    Cor e Forma:Solid
    Peso molecular:355.77
  • DDO-02001

    CAS:
    <p>DDO-02001 can be used in anti-arrhythmia research. DDO-02001 is a moderately potent inhibitor of Kv1.5 potassium channel with an IC50 value of 17.7 μM [1].</p>
    Fórmula:C20H24N2O2
    Cor e Forma:Solid
    Peso molecular:324.42
  • ASIC-IN-1

    CAS:
    <p>ASIC-IN-1 is a potent inhibitor of acid-sensing ion channels, demonstrating an IC 50 value of less than 10 μM.</p>
    Fórmula:C23H25N3O2
    Cor e Forma:Solid
    Peso molecular:375.46
  • TRPV antagonist 1

    CAS:
    <p>TRPV antagonist 1 is an antagonist of transient receptor potential vanilloid (TRPV; IC50 &lt; 250 nM).</p>
    Fórmula:C26H21F3N2O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:514.52
  • Becampanel

    CAS:
    <p>Becampanel (AMP397) is the first competitive AMPA antagonist. Becampanel (AMP397) also is an antiepileptic agent.</p>
    Fórmula:C10H11N4O7P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:330.19
  • Flordipine

    CAS:
    <p>Flordipine is used as a calcium channel blocker.</p>
    Fórmula:C26H33F3N2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:510.55
  • MRK-623

    CAS:
    <p>MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.</p>
    Fórmula:C20H17FN4O
    Cor e Forma:Solid
    Peso molecular:348.37
  • CAY10608

    CAS:
    <p>CAY10608 selectively blocks NR2B NMDA receptors (IC50 = 50 nM), is neuroprotective, and reduces brain infarct size in ischemia.</p>
    Fórmula:C18H22Cl2N2O4S
    Cor e Forma:Solid
    Peso molecular:433.35
  • 6'-Iodoresiniferatoxin

    CAS:
    <p>TRPV1 (VR1) vanilloid receptor partial agonist</p>
    Fórmula:C37H39IO9
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:754.6
  • Alilusem

    CAS:
    <p>Alilusem is a new diuretic that is beneficial to the clinical treatment of hypertension.</p>
    Fórmula:C17H15ClKN2O5S
    Cor e Forma:Solid
    Peso molecular:433.92
  • LUF7244

    CAS:
    <p>LUF7244 is a K v 11.1 channel modulator with anti-arrhythmia research potential, curbing early afterdepolarizations.</p>
    Fórmula:C20H15ClN2O3
    Cor e Forma:Solid
    Peso molecular:366.8
  • SRI-37240

    CAS:
    <p>SRI-37240 suppresses CFTR nonsense mutations, aids in fixing premature termination codons, works with G418.</p>
    Fórmula:C24H23N3O2
    Pureza:98.73%
    Cor e Forma:Solid
    Peso molecular:385.46
  • RO 4938581

    CAS:
    <p>RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).</p>
    Fórmula:C13H8BrF2N5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:352.14
  • Pregabalin arenacarbil

    CAS:
    <p>Pregabalin arenacarbil is a gabamimetic.</p>
    Fórmula:C15H27NO6
    Cor e Forma:Solid
    Peso molecular:317.38
  • ML67-33

    CAS:
    <p>ML67-33 selectively activates K2P channels; EC50: 36.3 μM (cell-free), 9.7 μM (HEK293). Reversible TREK-1 modulation.</p>
    Fórmula:C18H17Cl2N5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:374.27
  • PMPA (NMDA antagonist)

    CAS:
    <p>PMPA (NMDA antagonist) is a Competitive NMDA receptor antagonist.</p>
    Fórmula:C6H13N2O5P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:224.15
  • piCRAC-1

    CAS:
    <p>piCRAC-1 is a powerful inhibitor of the photoinducible Ca2+ release-activated Ca2+ (CRAC) channel.</p>
    Fórmula:C17H10F6N4
    Cor e Forma:Solid
    Peso molecular:384.28
  • AMP-PNP tetralithium

    CAS:
    <p>AMP analog that blocks Kir6 channels, inhibits axonal transport, and stabilizes organelle-microtubule interactions.</p>
    Fórmula:C10H13Li4N6O12P3
    Cor e Forma:Solid
    Peso molecular:529.93
  • Cyphenothrin

    CAS:
    <p>Cyphenothrin, a synthetic pyrethroid, combats carbamate-resistant cockroaches.</p>
    Fórmula:C24H25NO3
    Cor e Forma:Faint Yellow Sticky Liquid
    Peso molecular:375.46
  • RyRs activator 3

    CAS:
    <p>RyRs activator 3 (compound A4) serves as an insecticide highly effective against both the diamondback moths, M.</p>
    Fórmula:C23H19BrCl2N6O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:578.25
  • CGP11952

    CAS:
    <p>CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.</p>
    Fórmula:C21H21Cl2N5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:446.33
  • QAQ dichloride

    CAS:
    <p>QAQ dichloride is a photoswitchable blocker of Na v/K v channels, active in trans form, and a light-sensitive analgesic targeting pain neurons.</p>
    Fórmula:C28H44N6O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:496.69
  • Atomoxetine

    CAS:
    <p>Atomoxetine (HSDB 7352) is a selective norepinephrine inhibitor that may cause an increase in blood pressure by increasing norepinephrine concentrations in</p>
    Fórmula:C17H21NO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:255.35
  • VU0529331

    CAS:
    <p>VU0529331 activates non-GIRK1 potassium channels (EC50: ~5.1 μM GIRK2, 5.2 μM GIRK1/2) and GIRK4 channels.</p>
    Fórmula:C22H20N6O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:384.43
  • YS-035 hydrochloride

    CAS:
    <p>inhibitor of outward K+ currents</p>
    Fórmula:C21H30ClNO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:395.92
  • Ned-K

    CAS:
    <p>Ned-K blocks NAADP, reduces heart ischemia-reperfusion calcium waves.</p>
    Fórmula:C31H31N5O3
    Cor e Forma:Solid
    Peso molecular:521.61
  • Relutrigine

    CAS:
    <p>Relutrigine (PRAX-562) is an oral persistent sodium channel inhibitor with anticonvulsant properties, IC50 of 141 nM/75 nM for ATX-II/SCN8A-N1768D.</p>
    Fórmula:C15H11F6N5O2
    Cor e Forma:Solid
    Peso molecular:407.27
  • (R)-(+)-HA-966

    CAS:
    <p>(R)-(+)-HA-966 ((+)-HA-966) is a partial agonist/antagonist of glycine site of the N-methyl-D-aspartate (NMDA) receptor complex. (R)-(+)-HA-966 selectively blocks the activation of the mesolimbic dopamine system by amphetamine, has the potential for neuro</p>
    Fórmula:C4H8N2O2
    Cor e Forma:White Solid
    Peso molecular:116.12
  • RY796

    CAS:
    <p>RY796 is a selective voltage-gated potassium (KV2) channel inhibitor that inhibits KV2.1 and KV2.2, used in research on neurological disorders.</p>
    Fórmula:C21H27N3O2
    Pureza:98.59%
    Cor e Forma:Solid
    Peso molecular:353.46
  • P-gp inhibitor 4

    CAS:
    <p>P-gp inhibitor 4 is a selective P-glycoprotein modulator with an EC 50 of 94 nM.</p>
    Fórmula:C38H38N2O8S2
    Cor e Forma:Solid
    Peso molecular:714.85
  • NMDA-IN-2

    CAS:
    <p>NMDA-IN-2 (compound 6b) is a Procaine derivative that is an inhibitor of NMDA receptor 2B subtype [1].</p>
    Fórmula:C15H22N2O3
    Cor e Forma:Solid
    Peso molecular:278.35
  • PD-307243

    CAS:
    <p>PD-307243 is an activator of hERG channel.</p>
    Fórmula:C20H15Cl2N3O2
    Cor e Forma:Solid
    Peso molecular:400.26
  • RQ-00311651

    CAS:
    <p>RQ-00311651 is a novel T-type Ca2+ channel blocker. RQ-00311651 also inhibited high K-induced Ca signaling in those cells.</p>
    Fórmula:C19H18F3N5O2
    Cor e Forma:Solid
    Peso molecular:405.37
  • DDO-02005

    CAS:
    <p>DDO-02005, a Kv1.5 inhibitor (IC50: 0.72 μM), counters fibrillation and arrhythmias in rats.</p>
    Fórmula:C21H27Cl2N3O2
    Cor e Forma:Solid
    Peso molecular:424.37
  • (±)-C3001a

    CAS:
    <p>(RS)-C3001a is the racemic mixture of C3001a (CAS: 2415154-29-7). C3001a is a selective activator of the TREK channel.</p>
    Fórmula:C21H20N2O3S
    Pureza:99.13%
    Cor e Forma:Solid
    Peso molecular:380.46
  • TRPC3/6-IN-1

    CAS:
    <p>TRPC3/6-IN-1 selectively inhibits hTRPC3/6 with IC50 of 1260/500 nM, useful in heart failure research.</p>
    Fórmula:C20H19N3O2S
    Cor e Forma:Solid
    Peso molecular:365.45
  • UBP 302

    CAS:
    <p>UBP 302 is a selective GLUK5 kainate receptor antagonist with Kd 402 nM; low GluK2 affinity.</p>
    Fórmula:C15H15N3O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:333.3
  • GABAA receptor agent 4

    CAS:
    <p>Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.</p>
    Fórmula:C17H24N2O
    Cor e Forma:Solid
    Peso molecular:272.39
  • Ivacaftor-D9

    CAS:
    <p>CTP-656, a cystic fibrosis transmembrane conductance regulator (CFTR) channel activator, is used potentially for the treatment of cystic fibrosis.</p>
    Fórmula:C24H19D9N2O3
    Cor e Forma:Solid
    Peso molecular:401.55
  • Clathrodin

    CAS:
    <p>Clathrodin is a voltage-gated sodium (NaV) channels modulator.</p>
    Fórmula:C11H13N5O
    Cor e Forma:Solid
    Peso molecular:231.25
  • RG100204

    CAS:
    <p>RG100204 is an orally active AQP9 inhibitor with anti-inflammatory properties. It alleviates cardiac dysfunction (systolic and diastolic) induced by sepsis, improves renal dysfunction, and reduces the elevation of the cellular damage marker LDH.</p>
    Fórmula:C20H26N6O2S2
    Cor e Forma:Solid
    Peso molecular:446.59
  • MRS4719

    CAS:
    <p>MRS4719: potent P2X4 antagonist, IC50 0.503 μM. Reduces infarct, brain atrophy, Ca2+ influx. Used in ischemic stroke research.</p>
    Fórmula:C26H13N5O3S·C6H15N
    Cor e Forma:Solid
    Peso molecular:504.6
  • Dofequidar

    CAS:
    <p>Dofequidar (MS-209 free base) is a quinoline derivative that inhibits the efflux of chemotherapeutic agents.</p>
    Fórmula:C30H31N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:481.59
  • Neramexane Mesylate

    CAS:
    <p>Neramexane: NMDA &amp; nicotinic receptor blocker with neuroprotective, antidepressant, and cognitive-enhancing effects.</p>
    Fórmula:C12H27NO3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:265.41
  • P-gp inhibitor 17

    CAS:
    <p>P-gp Inhibitor 17 (compound 2g), a potent inhibitor, directly interacts with the transmembrane domain of P-gp. This compound is useful for studying P-gp-mediated multidrug resistance in tumor cells [1].</p>
    Fórmula:C36H49N3O3
    Cor e Forma:Solid
    Peso molecular:571.79
  • CW0134

    CAS:
    <p>CW0134 (Compound 12) serves as a modulator for exportin1 (XPO1), disrupting chromatin binding and inhibiting NFAT transcription factors and T cell activation [1].</p>
    Fórmula:C11H7ClF3N3O2
    Cor e Forma:Solid
    Peso molecular:305.64
  • Indantadol HCl

    CAS:
    <p>Indantadol HCl (CHF-3381) is a NMDA antagonist and nonselective MAO inhibitor.</p>
    Fórmula:C11H15ClN2O
    Pureza:98.24%
    Cor e Forma:Solid
    Peso molecular:226.7
  • Aprikalim

    CAS:
    <p>Aprikalim opens KATP channels, protects the heart, and at high doses, dilates blood vessels.</p>
    Fórmula:C12H16N2OS2
    Pureza:99.42% - 99.90%
    Cor e Forma:Solid
    Peso molecular:268.4
  • Norbormide

    CAS:
    <p>Norbormide is a toxic compound used as a rodenticide. It has several mechanisms of action, acting as a vasoconstrictor and calcium channel blocker.</p>
    Fórmula:C33H25N3O3
    Pureza:98%
    Cor e Forma:Crystals From Methylene Chloride + Ether Norbormide Is A Colorless To Off-White Crystalline Powder Used As A Selective Rat Poison (Epa 1998)
    Peso molecular:511.57
  • DPI 201-106

    CAS:
    <p>DPI 201-106: cardioselective h1 Na channel inhibitor, enhances heart contraction, blocks potassium and calcium currents.</p>
    Fórmula:C29H30N4O2
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:466.57
  • (S)-ML753286

    CAS:
    <p>(S)-ML753286 is a breast cancer resistance protein (BCRP) inhibitor (IC50: 0.6 μM on BCRP efflux transporter).</p>
    Fórmula:C20H25N3O3
    Cor e Forma:Solid
    Peso molecular:355.43
  • IEM 1460

    CAS:
    <p>AMPA receptors blocker</p>
    Fórmula:C19H38Br2N2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:454.33
  • YS-201

    CAS:
    <p>YS-201 is an antagonist of dihydropyridine-type calcium channel.</p>
    Fórmula:C24H31N3O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:457.52
  • (+)-Nipecotic acid

    CAS:
    <p>(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.</p>
    Fórmula:C6H11NO2
    Pureza:99.38%
    Cor e Forma:Solid
    Peso molecular:129.16
  • SL-651498

    CAS:
    <p>SL-651498, a GABAA receptor agonist, is used potentially for the treatment of anxiety.</p>
    Fórmula:C23H20FN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:389.42
  • CGP 46381

    CAS:
    <p>CGP 46381 is a GABAB receptor antagonist.</p>
    Fórmula:C10H22NO2P
    Pureza:98%
    Cor e Forma:White Solid
    Peso molecular:219.26
  • Anipamil

    CAS:
    <p>Anipamil is a long-acting blocker of calcium channel,and for the treatment of cardiovascular disease.</p>
    Fórmula:C34H52N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:520.79
  • Nav1.7-IN-3

    CAS:
    <p>Nav1.7-IN-3 is a selective and orally bioavailable inhibitor of voltage-gated sodium channel Nav1.7(IC50 of 8 nM).</p>
    Fórmula:C17H20ClFN4O2S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:430.95
  • Y 23684

    CAS:
    <p>Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.</p>
    Fórmula:C18H13ClN2O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:356.83
  • L-trans-2,4-PDC

    CAS:
    <p>L-trans-2,4-PDC is an EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor.</p>
    Fórmula:C6H9NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:159.14
  • UBP 296

    CAS:
    <p>GluR5-subunit containing kainate receptor antagonist</p>
    Fórmula:C15H15N3O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:333.3
  • Caldaret

    CAS:
    <p>Caldaret is an intracellular Ca2+ handling modulator that acts through reverse mode Na+/Ca2+ exchanger inhibition.</p>
    Fórmula:C11H16N2O3S
    Cor e Forma:Solid
    Peso molecular:256.32
  • ORM-10962

    CAS:
    <p>ORM-10962 is a potent, highly selective inhibitor of sodium-calcium exchanger (NCX) (for the reverse and forward mode inhibition with IC50 values of 67 and 55</p>
    Fórmula:C27H29N3O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:459.54
  • MC-70

    CAS:
    <p>MC-70 is a potent P-glycoprotein (P-gp) inhibitor (EC50 = 0.69 μM).</p>
    Fórmula:C24H25NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:375.46
  • Anxiolytic/nonsedative agent-1

    CAS:
    <p>TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.</p>
    Fórmula:C18H15N3O4
    Pureza:98.61%
    Cor e Forma:Solid
    Peso molecular:337.33
  • (S)-SNAP5114

    CAS:
    <p>(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.</p>
    Fórmula:C30H35NO6
    Pureza:97%
    Cor e Forma:Solid
    Peso molecular:505.6
  • NCS-382

    CAS:
    <p>γ-Hydroxybutyric acid antagonist</p>
    Fórmula:C13H14O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:218.25
  • Topiramate lithium

    CAS:
    <p>Topiramate lithium: antiepileptic, GluR5 antagonist, enhances GABA, inhibits kainate/AMPA, Na+/Ca2+ channels; ↑ K+ conductance; ↓ carbonic anhydrase.</p>
    Fórmula:C12H20LiNO8S
    Cor e Forma:Solid
    Peso molecular:345.29
  • RN9893

    CAS:
    <p>RN9893 is a selective and potent TRPV4 receptor antagonist with IC50 values of 320, 420 and 660 nM for TRPV4 receptors in mouse, human and rat, respectively.</p>
    Fórmula:C21H23F3N4O5S
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:500.49
  • HZ166

    CAS:
    <p>HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.</p>
    Fórmula:C21H16N4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:356.38
  • AMG9678

    CAS:
    <p>AMG9678 is a selective, potent, orally active TRPM8 antagonist (IC50: 31.2 nM).</p>
    Fórmula:C20H18F6N2O
    Cor e Forma:Solid
    Peso molecular:416.36
  • Psora 4

    CAS:
    <p>Psora 4 (5-(4-Phenylbutoxy)psoralen) is a Kv1.3 blocker and a caloric restriction mimetic.</p>
    Fórmula:C21H18O4
    Cor e Forma:Solid
    Peso molecular:334.37
  • Asivatrep

    CAS:
    <p>Asivatrep (PAC14028) is a selective and potent antagonist of transient receptor potential vanilloid subtype 1 (TRPV1) for the study of atopic dermatitis.</p>
    Fórmula:C21H22F5N3O3S
    Pureza:95.13%
    Cor e Forma:Solid
    Peso molecular:491.48
  • 3α,21-Dihydroxy-5α-pregnan-20-one

    CAS:
    <p>3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.</p>
    Fórmula:C21H34O3
    Pureza:98.00%
    Cor e Forma:Solid
    Peso molecular:334.49
  • Terodiline

    CAS:
    <p>Terodiline is an orally available selective muscarinic M1 receptor and calcium channel antagonist for the study of diseases caused by abnormal bladder function.</p>
    Fórmula:C20H27N
    Pureza:98.20% - 99.59%
    Cor e Forma:Solid
    Peso molecular:281.44
  • Kadethrin

    CAS:
    <p>Kadethrin is a synthetic pyrethroid. It was used as a pesticide.</p>
    Fórmula:C23H24O4S
    Pureza:98%
    Cor e Forma:Yellow-Brown Viscous Oil Solid
    Peso molecular:396.5
  • (S)-Lercanidipine hydrochloride

    CAS:
    <p>(S)-Lercanidipine hydrochloride is the S-enantiomer of Lercanidipine hydrochloride. (S)-lercanidipine hydrochloride is a potent blocker of calcium channel.</p>
    Fórmula:C36H42ClN3O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:648.19
  • AVE-0118

    CAS:
    <p>AVE-0118 is a potassium channel blocker and suppresses persistent atrial fibrillation.</p>
    Fórmula:C30H29N3O3
    Pureza:97.04% - 98.93%
    Cor e Forma:Solid
    Peso molecular:479.57
  • VU625

    CAS:
    <p>VU625 (VU007625) is an AeKir1 inhibitor (IC50: 96.8nM) that acts as a mosquito killer and inhibits AeKir1-mediated currents.</p>
    Fórmula:C19H22N2O4S
    Pureza:99.08%
    Cor e Forma:Solid
    Peso molecular:374.45
  • RN-9893 (hydrochloride)

    CAS:
    <p>RN-9893 is a TRPV4 antagonist with human/rat IC50s of 0.42/0.66 μM; selective over TRPV1, TRPV3, TRPM8. Reduces rat TRPV4 activity (IC50: 0.57-2.1 μM).</p>
    Fórmula:C21H24ClF3N4O5S
    Cor e Forma:Solid
    Peso molecular:536.95
  • MK-7145

    CAS:
    <p>MK-7145 is an inhibitor of ROMK(IC50 of 0.045 μM).</p>
    Fórmula:C26H30N2O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:466.53
  • TG41

    CAS:
    <p>TG41 is a GABAA receptors positive modulator.</p>
    Fórmula:C18H13BrCl2N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:440.12
  • CAY10719

    CAS:
    <p>CAY10719 selectively inhibits ABCG2 (IC50 = 0.23 μM), reverses SN 38 resistance, and inhibits ATPase, with low ABCG1 activity.</p>
    Fórmula:C25H20Cl2N2O2
    Cor e Forma:Solid
    Peso molecular:451.34
  • Sodium Channel inhibitor 1

    CAS:
    Sodium Channel inhibitor1 is a novel and selective voltage-gated sodium channel for pain treatment.
    Fórmula:C24H19F4N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:473.42
  • Corrector C4

    CAS:
    <p>Corrector C4, a corrector commonly used to study cystic fibrosis mutants, works by alleviating the interaction between CFTR transmembrane domain mutants and</p>
    Fórmula:C21H17ClN4O2S2
    Pureza:98.36%
    Cor e Forma:Solid
    Peso molecular:456.97
  • NMDA receptor modulator 3

    CAS:
    <p>NMDA receptor modulator 3 (Compound 99) is a potent modulator of NMDA receptor that can be used in the research of neurological disorder [1].</p>
    Fórmula:C12H9F3N2O2S
    Cor e Forma:Solid
    Peso molecular:302.27
  • Lidoflazine

    CAS:
    <p>Lidoflazine: antianginal, blocks HERG K+ &amp; Ca channels, risks QT prolongation &amp; arrhythmia.</p>
    Fórmula:C30H35F2N3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:491.62
  • PF-0713

    CAS:
    <p>PF 0713, a GABAA receptor agonist, is used as an intravenous sedative-hypnotic for general anaesthesia, ICU sedation, procedural sedation, chemotherapy.</p>
    Fórmula:C14H22O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:206.32
  • L589-420

    CAS:
    <p>L589-420 is a sodium pump inhibitor in human erythrocytes.</p>
    Fórmula:C14H14Cl2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:317.16
  • YM928

    CAS:
    <p>YM928 is an orally active antagonist of the AMPA receptor.</p>
    Fórmula:C14H10ClN3OS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:303.77
  • CCMQ

    CAS:
    inhibits [3H]-homoquinolinic acid binding to non-NMDA sensitive sites
    Fórmula:C12H9NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:231.2
  • Bms 188107

    CAS:
    <p>Bms 188107 is a calcium antagonist, it has cardioprotective effects.</p>
    Fórmula:C25H26N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:418.48
  • Caramiphen

    CAS:
    <p>Caramiphen is an antimuscarinic and anticholinergic agent that acts as an antagonist of the NMDA receptor.</p>
    Fórmula:C18H27NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:289.41
  • (2R,3S)-Chlorpheg

    CAS:
    <p>(2R,3S)-Chlorpheg is a NMDA receptor antagonist.</p>
    Fórmula:C11H12ClNO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:257.67
  • Viquidil

    CAS:
    <p>Viquidil is an agent with the activity of a vasodilator.</p>
    Fórmula:C20H24N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:324.42
  • (R)-Licarbazepine Acetate

    CAS:
    <p>(R)-Licarbazepine Acetate is a hopeful antiepileptic drug structurally related to Carbamazepine and Oxcarbazepine.</p>
    Fórmula:C17H16N2O3
    Cor e Forma:Solid
    Peso molecular:296.32
  • COR628

    CAS:
    <p>COR628 is the GABA(B) receptor positive allosteric modulator.</p>
    Fórmula:C16H23NO3S
    Cor e Forma:Solid
    Peso molecular:309.42
  • AZD 2066

    CAS:
    <p>AZD 2066 is a selective, orally active, and brain-penetrant mGluR5 antagonist with analgesic activity.</p>
    Fórmula:C19H16ClN5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:381.82
  • BBR 2160

    CAS:
    <p>BBR 2160: a calcium-antagonist dihydropyridine derivative, reduces heart tissue contractility and shortens action potentials.</p>
    Fórmula:C21H25N3O7S
    Cor e Forma:Solid
    Peso molecular:463.5
  • LY-395153

    CAS:
    <p>LY-395153 is a novel potentiator of AMPA receptor.</p>
    Fórmula:C19H24N2O3S
    Cor e Forma:Solid
    Peso molecular:360.47
  • Tolperisone free base

    CAS:
    Tolperisone free base, a centrally acting muscle relaxant, has been used for the symptomatic treatment of spasticity and muscle spasm.
    Fórmula:C16H23NO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:245.36
  • Lercanidipine, (S)-

    CAS:
    <p>(S)-Lercanidipine: a dihydropyridine calcium blocker with prolonged antihypertensive and kidney-protective properties.</p>
    Fórmula:C36H41N3O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:611.73
  • Ensaculin HCl

    CAS:
    <p>Ensaculin: NMDA antagonist, 5HT1A agonist, may treat Alzheimer's, enhances memory, neuroprotective, binds multiple receptors.</p>
    Fórmula:C26H33ClN2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:489
  • Naftazone

    CAS:
    <p>Naftazone: vasoprotectant for hemostasis; boosts vein cell growth in vitro without affecting clotting.</p>
    Fórmula:C11H9N3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:215.21
  • Tiropramide

    CAS:
    <p>Tiropramide is an antispasmodic drug. It also useful to inhibit the contractile response of the urinary bladder and in managing abdominal pain in IBS.</p>
    Fórmula:C28H41N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:467.64
  • Riodipine

    CAS:
    <p>Riodipine, a calcium channel blocker, is used as cardiovascular drugs.</p>
    Fórmula:C18H19F2NO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:367.34
  • DS28120313

    CAS:
    <p>DS28120313 is an oral inhibitor of hepcidin production (IC50: 0.093 μM).</p>
    Fórmula:C16H17N5O2
    Cor e Forma:Solid
    Peso molecular:311.34
  • CPP-115

    CAS:
    <p>CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.</p>
    Fórmula:C7H9F2NO2
    Cor e Forma:Solid
    Peso molecular:177.15
  • Ethopropazine Hydrochloride

    CAS:
    <p>Ethopropazine Hydrochloride is the salt form of Profenamine,anticholinergic, antihistamine, and anti-adrenergic,Parkinson's disease,an AChE inhibitor</p>
    Fórmula:C19H25ClN2S
    Pureza:98.25%
    Cor e Forma:Solid
    Peso molecular:348.93
  • DHP-218

    CAS:
    <p>DHP-218, a calcium channel blocker, inhibits rat aorta contractions; pA2: 9.11, IC50: 6.3 nmol/L (high K+) &amp; 66 nmol/L (phenylephrine).</p>
    Fórmula:C18H21N2O7P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:408.34
  • S3337

    CAS:
    <p>S3337 is an inhibitor of H+, K+-ATPase</p>
    Fórmula:C18H21N3O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:359.44
  • BCTP

    CAS:
    <p>BCTP is a polymodal inhibitor of TRPV1. It has a reduced liability for hyperthermia.</p>
    Fórmula:C17H16ClN3OS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:345.85
  • Chlormethiazole edisylate

    CAS:
    <p>Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.</p>
    Fórmula:C8H14ClNO6S3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:351.85
  • Talopram hydrochloride

    CAS:
    <p>noradrenalin transporter (NET) inhibitor</p>
    Fórmula:C20H26ClNO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:331.88
  • IAA-94

    CAS:
    <p>IAA-94 is an inhibitor of chloride channels, it binds channels in bovine kidney cortex microsomes with a Ki value of 1 µM.</p>
    Fórmula:C17H18Cl2O4
    Cor e Forma:Solid
    Peso molecular:357.23
  • JNJ-55511118

    CAS:
    <p>JNJ-55511118 is a TARP γ8 allosteric modulator with anticonvulsant activity, which can be used in research on chronic operant alcohol self-administration.</p>
    Fórmula:C14H8ClF3N2O2
    Cor e Forma:Solid
    Peso molecular:328.67
  • A 39355

    CAS:
    <p>A 39355 may specifically overcome multidrug resistance without the serious hypotensive effects associated with calcium antagonists.</p>
    Fórmula:C28H39Cl2N3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:504.54
  • UBP512

    CAS:
    <p>UBP512 is a NMDA receptor modulator.</p>
    Fórmula:C15H9IO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:348.14
  • Ronipamil

    CAS:
    <p>Ronipamil is an analogue of verapamil that used as a calcium entry blocker.</p>
    Fórmula:C32H48N2
    Cor e Forma:Solid
    Peso molecular:460.74
  • L 644711

    CAS:
    <p>L 644711 is an antagonist of HCO3(-)/Cl(-) antiporter.</p>
    Fórmula:C18H18Cl2O4
    Cor e Forma:Solid
    Peso molecular:369.24
  • N12N

    CAS:
    <p>N12N is a polyamine inverse NMDA receptor agonist.</p>
    Fórmula:C12H28N2
    Pureza:98%
    Cor e Forma:White Solid
    Peso molecular:200.36
  • Bromotetrandrine

    CAS:
    Bromotetrandrine enhances chemo by inhibiting P-glycoprotein, countering efflux pumps.
    Fórmula:C38H41BrN2O6
    Cor e Forma:Solid
    Peso molecular:701.65