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Transportador de Membranas/Canal Iónico

Transportador de Membranas/Canal Iónico

Os inibidores de transportadores de membrana e canais iônicos são compostos que bloqueiam a função de proteínas responsáveis pelo transporte de íons, nutrientes e outras moléculas através das membranas celulares. Esses inibidores são cruciais para o estudo da regulação da homeostase celular, transdução de sinais e neurotransmissão. Os inibidores de transportadores de membrana e canais iônicos também são importantes no desenvolvimento de tratamentos para distúrbios como epilepsia, doenças cardiovasculares e síndromes metabólicas. Na CymitQuimica, oferecemos uma ampla seleção de inibidores de alta qualidade de transportadores de membrana e canais iônicos para apoiar sua pesquisa em fisiologia, neurociência e farmacologia.

Subcategorias de "Transportador de Membranas/Canal Iónico"

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Foram encontrados 2280 produtos de "Transportador de Membranas/Canal Iónico"

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  • Glisoxepide

    CAS:
    <p>Glisoxepide: sulphonamide, oral K(ATP) blocker, antihyperglycemic, affects heart.</p>
    Fórmula:C20H27N5O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:449.52
  • Tedisamil

    CAS:
    <p>Tedisamil blocks cardiac K+ currents, slows heart rate, is a class III antiarrhythmic, and treats angina.</p>
    Fórmula:C19H32N2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:288.47
  • NP-252

    CAS:
    <p>NP-252 is a calcium channel antagonist potentially for the treatment of angina pectoris and congestive heart failure.</p>
    Fórmula:C26H35N3O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:469.57
  • UBP684

    CAS:
    <p>UBP684 enhances NMDAR responses, boosts l-glutamate/glycine, and mildly affects subunit agonist potency.</p>
    Fórmula:C17H20O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:256.34
  • Fenazinel Dihydrochloride

    CAS:
    <p>Fenazinel Dihydrochloride, a N-methyl-D-aspartate (NMDA) receptor antagonist, is used potentially for the treatment of ischemic stroke.</p>
    Fórmula:C21H27Cl2N3O2
    Cor e Forma:Solid
    Peso molecular:424.36
  • β-Neuroprotectin

    CAS:
    <p>beta-Neuroprotectin is a (3H)TCP binding inhibitor and provides protection against NMDA mediated neuronal cell death at low concentration.</p>
    Fórmula:C37H60N8O10
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:776.92
  • U 90042

    CAS:
    <p>GABAA receptor ligand</p>
    Fórmula:C17H13ClN6O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:352.78
  • MRS 2219

    CAS:
    <p>P2X1 receptor potentiator</p>
    Fórmula:C8H10NO5P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:231.14
  • COR627

    CAS:
    <p>COR627 is the GABA receptor positive allosteric modulator.</p>
    Fórmula:C20H27NO3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:361.5
  • trans-4-Hydroxycrotonic acid

    CAS:
    <p>ligand of γ-hydroxybutyric acid (GHB) receptor</p>
    Fórmula:C4H6O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:102.09
  • LY 81067

    CAS:
    <p>LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.</p>
    Fórmula:C22H24N4O
    Cor e Forma:Solid
    Peso molecular:360.45
  • AMG8163

    CAS:
    <p>AMG8163 is an antagonist of vanilloid receptor TRPV1.</p>
    Fórmula:C25H22F3N5O4S
    Cor e Forma:Solid
    Peso molecular:545.53
  • AH-1058 HCl

    CAS:
    <p>AH-1058 HCl is a lipophilic antiarrhythmic calcium channel blocker.</p>
    Fórmula:C30H29ClN2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:501.02
  • Watanidipine dihydrochloride

    CAS:
    <p>Watanidipine dihydrochloride is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.</p>
    Fórmula:C41H44Cl2N4O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:759.73
  • Kv1.5-IN-IIII

    CAS:
    <p>Kv1.5-IN-IIII is a potent inhibitor of Kv1.5.</p>
    Fórmula:C25H23ClN4O4S
    Cor e Forma:Solid
    Peso molecular:510.99
  • TPMPA

    CAS:
    <p>GABAA-ρ antagonist</p>
    Fórmula:C6H12NO2P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:161.14
  • Evenamide HCl

    CAS:
    <p>Evenamide, a nav sodium channel blocker, is used potentially for the treatment of schizophrenia.</p>
    Fórmula:C16H27ClN2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:314.85
  • Gallopamil, (-)-

    CAS:
    <p>Gallopamil, (-)- is an L-type calcium channel blocker. It is used in the treatment of abnormal heart rhythms.</p>
    Fórmula:C28H40N2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:484.63
  • DS1

    CAS:
    <p>DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.</p>
    Fórmula:C18H10Br2ClN3OS
    Cor e Forma:Solid
    Peso molecular:511.62
  • Pradigastat sodium

    CAS:
    <p>Pradigastat sodium is a novel inhibitor of DGAT-1.</p>
    Fórmula:C25H24F3N3NaO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:478.471
  • KR-31378

    CAS:
    <p>KR-31378, a K(ATP) channel activator, is used potentially for the treatment of ocular hypertension and glaucoma.</p>
    Fórmula:C22H27N5O4
    Cor e Forma:Solid
    Peso molecular:425.48
  • MCC1189

    CAS:
    <p>MCC1189 is a first-in-class MFS efflux pump CaMdr1p inhibitor.</p>
    Fórmula:C22H20N2O2
    Cor e Forma:Solid
    Peso molecular:344.41
  • AK-2-38

    CAS:
    <p>AK-2-38 is a nifedipine analogue with potent smooth muscle calcium antagonist action and partial agonist effects on isolated guinea pig left atrium.</p>
    Fórmula:C26H30N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:434.53
  • Azeloprazole

    CAS:
    <p>Azeloprazole, a proton pump inhibitor, is used potentially for the treatment of gastroesophageal reflux disease (GERD).</p>
    Fórmula:C22H27N3O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:429.53
  • Falipamil

    CAS:
    <p>Falipamil, a verapamil derivative, is a calcium channel blocker with antitachycardic and potential antianginal effects.</p>
    Fórmula:C24H32N2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:428.52
  • SGE-201

    CAS:
    <p>SGE-201 is an NMDA receptor allosteric modulator, revealing blocker differences via activity suppression and neuroprotection.</p>
    Fórmula:C26H44O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:388.63
  • Pentisomide

    CAS:
    <p>Pentisomide: class-I antiarrhythmic, affects depolarization &amp; repolarization, inhibits ischemia-reperfusion arrhythmias, in phase II trials.</p>
    Fórmula:C19H33N3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:319.48
  • NSC339614 potassium

    CAS:
    <p>NSC339614 potassium is a selective GluN1/GluN2C and GluN1/GluN2D receptors potentiator.</p>
    Fórmula:C10H5KN3O6S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:334.32
  • JY-XHe-053

    CAS:
    <p>JY-XHe-053 is a selective modulator of GABAA receptors.</p>
    Fórmula:C22H16FN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:373.38
  • HIE-124

    CAS:
    <p>HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.</p>
    Fórmula:C10H12N2O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:240.28
  • Gallopamil HCl, (-)-

    CAS:
    <p>Gallopamil HCl, (-)- is an L-type calcium channel blocker. It is used in the treatment of abnormal heart rhythms.</p>
    Fórmula:C28H41ClN2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:521.09
  • Suclofenide

    CAS:
    <p>Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.</p>
    Fórmula:C16H13ClN2O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:364.8
  • PD 122860

    CAS:
    <p>PD 122860 is a dihydropyridine enhancing heart contractility, altering ECG, and relaxing aortic rings.</p>
    Fórmula:C23H20F3N3O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:491.48
  • Oe-9000

    CAS:
    <p>Oe-9000 blocks voltage-gated Na(+) currents in neurons at low µM, affecting both TTX-S and TTX-R types.</p>
    Fórmula:C21H29NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:343.46
  • A778317

    CAS:
    <p>A778317 is a stereoselective, high-affinity antagonist.</p>
    Fórmula:C23H25N3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:359.46
  • AF-2785

    CAS:
    <p>In epididymal epithelial cells, AF-2785 inhibits cystic fibrosis transmembrane conductance regulator Cl(-) channels.</p>
    Fórmula:C17H12Cl2N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:347.2
  • A 80b

    CAS:
    <p>A-80b: synthetic pyridazinoindole; potent, lasting antihypertensive; lowers diastolic more; no change in heart rate; inhibits Ca2+-induced contraction.</p>
    Fórmula:C16H17N7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:307.35
  • ABP-700

    CAS:
    <p>ABP-700 is a positive allosteric modulator of the GABAA receptor.</p>
    Fórmula:C17H18N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:314.34
  • NS4591

    CAS:
    <p>NS4591 is a modulator of SK-IK channels.</p>
    Fórmula:C11H12Cl2N2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:259.13
  • NMDA receptor modulator 5

    CAS:
    <p>NMDA receptor modulator 5 (Compound 195), a potent NMDA receptor modulator, exhibits potential for neurological disorder research [1].</p>
    Fórmula:C14H11F3N2O3S
    Cor e Forma:Solid
    Peso molecular:344.31
  • Methsuximide

    CAS:
    Methsuximide is an anticonvulsant agent which appeared to be effective in petit mal, psychomotor and focal motor attacks [1].
    Fórmula:C12H13NO2
    Cor e Forma:Crystals From Dilute Alcohol Solid
    Peso molecular:203.24
  • Carabersat

    CAS:
    <p>Carabersat(SB 204269) is a novel and effective anticonvulsant and antiepileptic agent.</p>
    Fórmula:C20H20FNO4
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:357.38
  • ZAPA sulfate

    CAS:
    <p>GABAA receptors agonist</p>
    Fórmula:C4H8N2O6S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:244.25
  • Synthalin dihydrochloride

    CAS:
    <p>Synthalin dihydrochloride is a channel blocker of K+.</p>
    Fórmula:C12H30Cl2N6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:329.31
  • 3',4'-Dichlorobenzamil HCl

    CAS:
    <p>3',4'-Dichlorobenzamil HCl is an inhibitor of Na+ transport, Na+/Ca2+ exchanger, sarcoplasmic reticulum Ca2+ release channels.</p>
    Fórmula:C13H12Cl3N7O
    Pureza:98%
    Cor e Forma:Yellow Solid
    Peso molecular:388.64
  • BAY-Y-5959

    CAS:
    <p>BAY-Y-5959, a calcium channel agonist, is used potentially for the treatment of arrhythmia, heart failure and myocardial.</p>
    Fórmula:C26H24N4O2
    Cor e Forma:Solid
    Peso molecular:424.49
  • VU0183254

    CAS:
    <p>VU0183254, an insect OR agonist, inhibits odor-driven OR complex activation by targeting the Orco subunit.</p>
    Fórmula:C22H18N4O2S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:434.53
  • AHR-9294

    CAS:
    <p>AHR-9294 is a novel inhibitor of H, K-ATPase. It also antagonizes gastric HCl secretion in vivo.</p>
    Fórmula:C22H24N2O3
    Cor e Forma:Solid
    Peso molecular:364.44
  • NSC103054

    CAS:
    <p>NSC103054 is an ABCG2 transporter function inhibitor.</p>
    Fórmula:C18H22Br2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:430.17
  • AHR-10718

    CAS:
    <p>AHR-10718 has an antiarrhythmic effect.</p>
    Fórmula:C22H35N3O7S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:485.6
  • SOCE inhibitor 1

    CAS:
    <p>SOCE inhibitor 1 is a inhibitor of store-operated calcium entry (SOCE)(IC50 of 4.4 μM).</p>
    Fórmula:C25H22F3N5O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:513.47
  • (RS)-3,4-DCPG

    CAS:
    <p>antagonist of AMPA receptors and agonist of mGluR8</p>
    Fórmula:C10H9NO6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:239.18
  • Lubeluzole

    CAS:
    <p>Lubeluzole, a well-known neuroprotective agent, is recently proved useful to potentiate the activity of anti-cancer drugs.</p>
    Fórmula:C22H25F2N3O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:433.51
  • HENA

    CAS:
    <p>HENA is a novel activator of large conductance, voltage- and Ca2+-gated K+ (BK) channels.</p>
    Fórmula:C30H48NaO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:479.701
  • NMDA receptor potentiator-1

    CAS:
    <p>Compound 1368 is a selective NMDA receptor enhancer; IC50s: 4 μM for NR2C, 5 μM for NR2D.</p>
    Fórmula:C26H26ClNO5
    Cor e Forma:Solid
    Peso molecular:467.94
  • KC 12291 hydrochloride

    CAS:
    <p>voltage-gated sodium channel blocker</p>
    Fórmula:C22H28ClN3O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:449.99
  • Lanceotoxin A

    CAS:
    <p>Lanceotoxin A is a potent Ip blocker.</p>
    Fórmula:C32H44O12
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:620.68
  • Dopropidil hydrochloride

    CAS:
    <p>Dopropidil, a calcium channel antagonist, is used potentially for the treatment of arrhymia and angina pectoris.</p>
    Fórmula:C20H36ClNO2
    Cor e Forma:Solid
    Peso molecular:357.96
  • MPO-IN-5

    CAS:
    <p>MPO-IN-5: strong, irreversible MPO blocker; IC50s: 0.22 μM for peroxidation, 2.8 μM for hERG.</p>
    Fórmula:C24H24N6O2
    Cor e Forma:Solid
    Peso molecular:428.49
  • SCH00013

    CAS:
    <p>SCH00013 is a cardiotonic that enhances myofibrillar Ca++ sensitivity, with notable effects at pH 7.2-7.4.</p>
    Fórmula:C18H20N4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:324.38
  • GZ4

    CAS:
    <p>GZ4 is a Ca2+ currents inhibitor, acting on cell surface channels.</p>
    Fórmula:C11H17NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:195.26
  • AFD-21

    CAS:
    <p>AFD-21 is a class I antiarrhythmic that inhibits sodium channels with moderate kinetics.</p>
    Fórmula:C28H39NO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:469.61
  • Hexadecylphosphoserine

    CAS:
    <p>Hexadecylphosphoserine is a representative growth inhibitor.</p>
    Fórmula:C19H40NO6P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:409.5
  • 4-(Phenyldiazenyl)benzoic acid

    CAS:
    <p>4-(Phenyldiazenyl)benzoic acid is a photosensitive and photoswitchable TRPA1 agonist that can be used as pharmacological tool to study pain signaling.</p>
    Fórmula:C13H10N2O2
    Cor e Forma:Solid
    Peso molecular:226.23
  • Metaphit

    CAS:
    <p>Acylator of PCP and σ-receptors</p>
    Fórmula:C18H24N2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:300.46
  • (S)-Baclofen

    CAS:
    <p>(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.</p>
    Fórmula:C10H12ClNO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:213.66
  • AMG7905

    CAS:
    <p>AMG7905 is a modulator of transient receptor potential vanilloid type 1.</p>
    Fórmula:C25H24F3N5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:483.55
  • Ro18-5362

    CAS:
    <p>Ro18-5362 is the less active prodrug of Ro 18-5364.</p>
    Fórmula:C22H25N3O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:395.52
  • Ceefourin-2

    CAS:
    <p>Ceefourin-2 is a highly selective multidrug resistance protein 4 inhibitor.</p>
    Fórmula:C15H9ClF3N3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:355.7
  • BDF 9148

    CAS:
    <p>BDF 9148, a Na(+)-channel modulator, increases the contractile force of guinea-pig atria and papillary muscles.</p>
    Fórmula:C28H27N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:453.53
  • JTV-519 fumarate

    CAS:
    <p>Ryanodine receptor (RyR) inhibitor; stabilizes RyR2 in a closed conformation. Exhibits antiarrhythmic and cardioprotective properties in vivo.</p>
    Fórmula:C29H36N2O6S
    Cor e Forma:Solid
    Peso molecular:540.67
  • EO-122

    CAS:
    <p>EO-122, a calcium channel antagonist and sodium channel antagonist, is used potentially for the treatment of arrhythmia.</p>
    Fórmula:C16H23ClN2O
    Cor e Forma:Solid
    Peso molecular:294.82
  • DAA-1097

    CAS:
    <p>DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.</p>
    Fórmula:C24H24ClNO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:409.91
  • Levamlodipine gentisate

    CAS:
    <p>Levamlodipine gentisate, an active amlodipine enantiomer, is a dihydropyridine calcium channel blocker for treating hypertension and angina.</p>
    Fórmula:C27H31ClN2O9
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:563
  • JTT-552

    CAS:
    <p>JTT-552, a uric acid transporter 1 (URAT1) inhibitor, is used potentially for the treatment of hyperuricemia.</p>
    Fórmula:C15H12ClNO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:289.71
  • TRPC5-IN-1

    CAS:
    <p>TRPC5-IN-1 is a TRPC5 inhibitor active in various animal models of chronic kidney disease.</p>
    Fórmula:C20H16N4O
    Cor e Forma:Solid
    Peso molecular:328.37
  • (S)-3-Carboxy-4-hydroxyphenylglycine

    CAS:
    <p>group I metabotropic glutamate receptor antagonist and group II mGlu agonist</p>
    Fórmula:C9H9NO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:211.17
  • PNU 37883 hydrochloride

    CAS:
    <p>Kir6 (KATP) channel antagonist</p>
    Fórmula:C21H36ClN3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:381.98
  • TAS-4

    CAS:
    <p>TAS-4 is a modulator of metabotropic glutamate receptor 4-positive allosteric.</p>
    Fórmula:C12H8Cl2N2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:267.11
  • N20C hydrochloride

    CAS:
    <p>N20C hydrochloride (2-((3,3-diphenylpropyl)amino)acetamide hydrochloride) is a non-competitive NMDA receptor open-channel blocker.</p>
    Fórmula:C17H21ClN2O
    Pureza:99.9%
    Cor e Forma:Solid
    Peso molecular:304.81
  • Hydroflumethiazide

    CAS:
    <p>Hydroflumethiazide is a thiazide diuretic. It has also shown the activity of anti-hypertensive.</p>
    Fórmula:C8H8F3N3O4S2
    Cor e Forma:Crystals Solid
    Peso molecular:331.29
  • Gea 857

    CAS:
    <p>Gea 857 is a potassium conductance putative blocker.</p>
    Fórmula:C15H22ClNO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:283.79
  • Lombazole

    CAS:
    <p>Lombazole is an antimicrobial agent in the class of imidazole.</p>
    Fórmula:C22H17ClN2
    Cor e Forma:Solid
    Peso molecular:344.84
  • D-3263

    CAS:
    <p>D-3263 is an agonist of transient receptor potential melatonin member 8 (TRPM8) with potential antitumor activity.</p>
    Fórmula:C21H31N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:373.49
  • TB 21007

    CAS:
    <p>GABAA receptor inverse agonist</p>
    Fórmula:C15H17NO2S3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:339.5
  • Aladorian

    CAS:
    <p>Aladorian (ARM036), a benzothiazepine, has anti-arrhythmic properties for heart failure and CPVT research.</p>
    Fórmula:C12H13NO4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:267.3
  • Arginylproline

    CAS:
    <p>Arginylproline is a dipeptide composed of arginine and proline. It is an incomplete breakdown product of protein digestion or protein catabolism.</p>
    Fórmula:C11H21N5O3
    Cor e Forma:Solid
    Peso molecular:271.32
  • GSK-5498A

    CAS:
    <p>GSK-5498A: Selective CARC blocker, inhibits release of mediators from mast cells and cytokines from T-cells (IC50, 1 μM).</p>
    Fórmula:C18H11F6N3O
    Cor e Forma:Solid
    Peso molecular:399.29
  • Ro 8-4304

    CAS:
    <p>Ro 8-4304 Hydrochloride is an antagonist of NMDA receptor with IC50 of 0.4 μM</p>
    Fórmula:C21H23FN2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:370.42
  • GABAA receptor agent 6

    CAS:
    <p>GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].</p>
    Fórmula:C18H25N3O2
    Cor e Forma:Solid
    Peso molecular:315.41
  • AMG8788

    CAS:
    <p>AMG8788 is a selective, potent and orally active TRPM8 antagonist (IC50: 63.2 nM).</p>
    Fórmula:C23H18F4N2O
    Cor e Forma:Solid
    Peso molecular:414.4
  • CS476

    CAS:
    <p>CS476 is a potent drug of hypoglycaemic.</p>
    Fórmula:C24H29N3O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:471.57
  • Fluzinamide

    CAS:
    <p>Fluzinamide (AHR-8559) has anticonvulsant effects on ignited amygdala seizures.</p>
    Fórmula:C12H13F3N2O2
    Pureza:99.38% - >99.99%
    Cor e Forma:Solid
    Peso molecular:274.24
  • Laurinterol

    CAS:
    <p>Laurinterol is an antimicrobial from the marine alga Laurencia okamurai.</p>
    Fórmula:C15H19BrO
    Cor e Forma:Solid
    Peso molecular:295.21
  • BRL 55834

    CAS:
    <p>BRL 55834, a potassium channel activator, has shown to relax airways and vasculature in vivo.</p>
    Fórmula:C18H20F5NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:393.35
  • S-312-d

    CAS:
    <p>S-312d is a calcium channel antagonist. S-312-d can offer marked neuronal protective effects against ischemic injury.</p>
    Fórmula:C20H22N2O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:386.46
  • FG8119

    CAS:
    <p>FG8119 is a novel benzodiazepine agonist with potential anticonvulsant and antiepileptic activity for the study of neurological disorders.</p>
    Fórmula:C17H15N5O2
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:321.33
  • PF-05214030

    CAS:
    <p>PF-05214030 is a novel potent TRPV4 antagonist (hTRPV4 IC50 4nM; rTRPV4 IC50 27nM).</p>
    Fórmula:C17H13Cl2FN2O4S
    Cor e Forma:Solid
    Peso molecular:431.27
  • (RS)-CPP

    CAS:
    <p>(RS)-CPP is a NMDA antagonist.</p>
    Fórmula:C8H17N2O5P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:252.2
  • V116517

    CAS:
    <p>V-116517, a TRPV1 antagonist, is used potentially for the treatment of severe pain due to osteoarthritis and chronic pain due postherpetic neuralgia (PHN).</p>
    Fórmula:C19H18ClF3N4O3
    Cor e Forma:Solid
    Peso molecular:442.82
  • Quinine hemisulfate

    CAS:
    <p>Quinidine: antiarrhythmic, orally active, inhibits cytochrome P450db, blocks K+ channels (IC50: 19.9μM), may aid in malaria research.</p>
    Fórmula:C40H50N4O8S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:746.92
  • Niguldipine Free Base

    CAS:
    <p>Niguldipine Free Base is a calcium channel blocker and a₁-adrenergic receptor antagonist and a clinical modulator of multidrug resistance.</p>
    Fórmula:C36H39N3O6
    Pureza:98.97%
    Cor e Forma:Solid
    Peso molecular:609.71
  • CGP 28392

    CAS:
    <p>CGP 28392 is used as a partial calcium channel agonist.</p>
    Fórmula:C18H17F2NO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:365.33
  • Almokalant

    CAS:
    <p>Almokalant: Class III antiarrhythmic, K+ channel blocker, inhibits Ikr current.</p>
    Fórmula:C18H28N2O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:352.49
  • UT-B-IN-1

    CAS:
    <p>UT-B-IN-1: reversible UT-B inhibitor, IC50: 10 nM (human), 25 nM (mouse), low toxicity, diuretic research tool.</p>
    Fórmula:C20H17N5O2S3
    Cor e Forma:Solid
    Peso molecular:455.58
  • RH01617

    CAS:
    <p>RH01617 possesses potent inhibitory activities against Kv1.5.</p>
    Fórmula:C22H26N2O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:430.52
  • GSK-5503A

    CAS:
    <p>GSK-5503A is a novel channel blocker of CRAC.</p>
    Fórmula:C23H17F2N3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:405.4
  • Glypromate

    CAS:
    <p>Glypromate (Gly-Pro-Glu) is a neuroprotective agent, is a weak NMDA receptor agonist</p>
    Fórmula:C12H19N3O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:301.3
  • D-AP4

    CAS:
    <p>broad spectrum excitatory amino acid receptor antagonist</p>
    Fórmula:C4H10NO5P
    Pureza:98%
    Cor e Forma:White Powder
    Peso molecular:183.1
  • SR57227A

    CAS:
    <p>SR 57227A: Selective 5-HT3 receptor inhibitor, affects NMDA responses, has anti-depressant effects and reduces aggression in rats.</p>
    Fórmula:C10H14ClN3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:211.69
  • L-701252

    CAS:
    <p>L-701252, a potent glycine site NMDA receptor antagonist, exhibits an inhibition concentration (IC50) of 420 nM.</p>
    Fórmula:C13H10ClNO3
    Pureza:97.7%
    Cor e Forma:White Crystalline Solid
    Peso molecular:263.68
  • PNU-107484A

    CAS:
    <p>PNU-107484A is a unique GABA(A) receptor ligand.</p>
    Fórmula:C18H23ClN6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:358.87
  • LY 233536

    CAS:
    <p>LY 233536 is a novel, competitive antagonist of NMDA receptor.</p>
    Fórmula:C12H19N5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:265.31
  • BK 129

    CAS:
    BK 129 is a local anesthetic with relaxant properties. BK 129 inhibits Ca2+ entry into the smooth muscle cell and Ca2+ release from sarcoplasmic reticulum.
    Fórmula:C22H36N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:392.53
  • H100

    CAS:
    <p>H100 inhibits Cl- transport, mildly affects NaK2Cl cotransporter and Band 3 anion exchanger, not KCl cotransporter.</p>
    Fórmula:C18H16N2O6S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:388.4
  • Dicirenone

    CAS:
    <p>Dicirenone (SC26304) inhibits the Mineralocorticoid receptor (MR), aldosterone regulation of the urinary K+:Na+ ratio, and aldosterone binding to renal</p>
    Fórmula:C26H36O5
    Pureza:99.1%
    Cor e Forma:Solid
    Peso molecular:428.56
  • Guanosine 5'-diphosphate ditromethamine

    CAS:
    Guanosine 5'-diphosphate ditromethamine (GDP ditromethamine) is a nucleoside diphosphate that activates ATP-sensitive K+ channels. It acts as a potential iron mobilizer, inhibiting the interaction between hepcidin and ferroportin, and modulating the IL-6/STAT-3 pathway. This compound finds application in inflammation research, such as studying anemia of inflammation (AI).
    Fórmula:C18H37N7O17P2
    Peso molecular:685.47
  • KMUP-4

    CAS:
    <p>Kmup-4 is an enhancer of cGMP activity and an aortic smooth muscle relaxant.</p>
    Fórmula:C19H23N7O4
    Cor e Forma:Solid
    Peso molecular:413.43
  • GSK1702934A

    CAS:
    <p>GSK1702934A is a TRPC3 agonist with pro-arrhythmic and positive inotropic effects and is used in the study of diabetes mellitus.</p>
    Fórmula:C22H25N3O2S
    Pureza:98.15%
    Cor e Forma:Solid
    Peso molecular:395.52
  • Eltanexor Z-isomer

    CAS:
    <p>Eltanexor Z-isomer, less active than KPT-8602, inhibits Z138, MM1S, and 3T3 cells with IC50s: 100 nM-50 μM, &lt;100 nM, &gt;30 μM.</p>
    Fórmula:C17H10F6N6O
    Cor e Forma:Solid
    Peso molecular:428.29
  • N-Oleoyl Valine

    CAS:
    N-Oleoyl valine, an N-acyl amine, antagonizes TRPV3 for thermoregulation; rises post-cold exposure; elevates in mouse lung injury.
    Fórmula:C23H43NO3
    Peso molecular:381.59
  • GS 39783

    CAS:
    <p>GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement and</p>
    Fórmula:C15H23N5O2S
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:337.44
  • 3-Chlorodiphenylamine

    CAS:
    3-Cl-DPA, a cardiac troponin activator, acts by a mechanism distinct from bepridil or TFP.
    Fórmula:C12H10ClN
    Cor e Forma:Solid
    Peso molecular:203.67
  • SM-6586

    CAS:
    <p>SM-6586 is a potent calcium channel antagonist with inhibitory effects on Na+/H+ and Na+/Ca2+ exchange channels, and can be used in the study of cerebrovascular</p>
    Fórmula:C26H27N5O5
    Pureza:99.43%
    Cor e Forma:Solid
    Peso molecular:489.52
  • (5R)-BW-4030W92

    CAS:
    <p>(5R)-BW-4030W92 is the R-type of BW-4030W92, the active enantiomer.</p>
    Fórmula:C11H9Cl2FN4
    Pureza:98.27%
    Cor e Forma:Solid
    Peso molecular:287.12
  • NHE3-IN-3

    CAS:
    <p>NHE3-IN-3 inhibits human/rat NHE3 with pIC50s 6.2/6.6; 98% oral bioavailability in rats.</p>
    Fórmula:C16H16Cl2N2O2S
    Cor e Forma:Solid
    Peso molecular:371.28
  • Bamaluzole

    CAS:
    <p>Bamaluzole is an agonist of GABA receptor.</p>
    Fórmula:C14H12ClN3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:273.72
  • UBP141

    CAS:
    <p>UBP141 is a antagonist of N-methyl-D-aspartate (NMDA) receptor.</p>
    Fórmula:C21H18N2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:378.38
  • Aprindine hydrochloride

    CAS:
    <p>Aprindine HCl, a Class 1b antiarrhythmic, treats heart arrhythmias, outperforming digoxin in delaying atrial fibrillation. It's effective orally.</p>
    Fórmula:C22H31ClN2
    Cor e Forma:Solid
    Peso molecular:358.95
  • TC-AQP1-1

    CAS:
    <p>TC-AQP1-1 blocks aquaporin 1; found via virtual screening; hinders water flux in Xenopus oocytes at low µM.</p>
    Fórmula:C12H10O4
    Pureza:97.59%
    Cor e Forma:Solid
    Peso molecular:218.21
  • GABAA receptor agent 8

    CAS:
    <p>Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.</p>
    Fórmula:C19H16N4O
    Cor e Forma:Solid
    Peso molecular:316.36
  • AM12

    CAS:
    <p>AM12 inhibits Lanthanide-evoked TRPC5 activity (IC50: 0.28 μM).</p>
    Fórmula:C15H9BrO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:349.13
  • KRP-199

    CAS:
    <p>KRP-199, a highly potent and selective antagonist for the AMPA receptors, exhibits good neuroprotective effects in vivo.</p>
    Fórmula:C22H14F3N5O7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:517.37
  • Nav1.7-IN-2

    CAS:
    <p>Nav1.7-IN-2 is avoltage-gated sodium channels (Nav) inhibitor in particular Nav 1.7(IC50 of 80 nM).</p>
    Fórmula:C22H22FN5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:407.44
  • Cilobradine hydrochloride

    CAS:
    <p>Cilobradine hydrochloride (DK-AH 269) is an HCN Channel blocker and an open channel blocker of neuronal Ih and related cardiac If channels.</p>
    Fórmula:C28H39ClN2O5
    Pureza:98.40%
    Cor e Forma:Solid
    Peso molecular:519.07
  • (S)-(-)-HA 966

    CAS:
    <p>(S)-(-)-HA 966 is a NMDA receptor antagonist.</p>
    Fórmula:C4H8N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:116.12
  • Sodium Channel inhibitor 2

    CAS:
    <p>Sodium Channel inhibitor 2 is a blocker of sodium channel.</p>
    Fórmula:C26H25Cl2N3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:466.4
  • NMDA receptor antagonist 5

    CAS:
    <p>Compound 10e: potent, non-toxic, brain-permeable NMDA receptor antagonist; key for neurological research.</p>
    Fórmula:C19H16BrNO2
    Cor e Forma:Solid
    Peso molecular:370.24
  • Nav1.1 activator 1

    CAS:
    <p>Nav1.1 activator 1 is a highly potent activator of Nav1.1 with BBB penetration.</p>
    Fórmula:C24H23F3N4O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:440.46
  • Diproteverine

    CAS:
    <p>Diproteverine is a calcium antagonist, it has antianginal property.</p>
    Fórmula:C26H35NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:425.56
  • FSBA hydrochloride

    CAS:
    <p>FSBA hydrochloride(5'-p-Fluorosulfonylbenzoyladenosine) is an ATP analogue serving as an affinity probe for the ATP site of Na/K-ATPase.</p>
    Fórmula:C17H17ClFN5O7S
    Pureza:97.96%
    Cor e Forma:Solid
    Peso molecular:489.86
  • GNE-6901

    CAS:
    <p>GNE-6901 is a selective GluN2A PAM.</p>
    Fórmula:C18H17FN2O3S
    Cor e Forma:Solid
    Peso molecular:360.4
  • TC-T 6000

    CAS:
    <p>TC-T 6000 (hENT4-IN-1) is an ENT4 inhibitor with vasodilator activity that inhibits hENT1 and hENT2 for the study of cancer and cardiovascular damage.</p>
    Fórmula:C26H48N8O2
    Pureza:98.14%
    Cor e Forma:Solid
    Peso molecular:504.71
  • CP-465022 (maleate)

    CAS:
    <p>CP-465022 Maleate: A selective noncompetitive AMPA antagonist with IC50 of 25 nM, showing anticonvulsant effects and useful for AMPA-related studies.</p>
    Fórmula:C30H28ClFN4O5
    Cor e Forma:Solid
    Peso molecular:579.02
  • CGP 36216 hydrochloride

    CAS:
    <p>CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).</p>
    Fórmula:C5H14NO2P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:151.14
  • CP-457920

    CAS:
    <p>CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.</p>
    Fórmula:C18H17N3O3
    Pureza:99.06% - 99.74%
    Cor e Forma:Solid
    Peso molecular:323.35
  • ML402

    CAS:
    <p>ML402 (ZINC3671497) is an activator of TREK-1 and TREK-2 with EC50s of 13.7 μM and 5.9 μM.</p>
    Fórmula:C14H14ClNO2S
    Pureza:99.71%
    Cor e Forma:Solid
    Peso molecular:295.78
  • ATX-II TFA


    <p>ATX-II TFA, a specific Na+ channel modulator toxin, is derived from the venom of the sea anemone (Anemonia sulcata).</p>
    Pureza:98%
    Cor e Forma:Odour Solid
  • Lemildipine

    CAS:
    <p>Lemildipine is a new blocker of dihydropyridine calcium entry.</p>
    Fórmula:C20H22Cl2N2O6
    Cor e Forma:Solid
    Peso molecular:457.3
  • Zatebradine hydrochloride

    CAS:
    <p>Zatebradine hydrochloride (UL-FS-49CL) inhibits HCN channels (IC50: ~1.9 µM) blocking human HCN1-4 currents effectively.</p>
    Fórmula:C26H37ClN2O5
    Pureza:97%
    Cor e Forma:Solid
    Peso molecular:493.04
  • Nav1.7 inhibitor

    CAS:
    <p>Nav1.7 inhibitor is a Nav1.7 inhibitor for research in the field of pain and anesthesia.</p>
    Fórmula:C15H11Cl3FNO4S
    Pureza:97.52%
    Cor e Forma:Solid
    Peso molecular:426.68
  • CP-100356 hydrochloride

    CAS:
    <p>CP-100356 hydrochloride is an MDR1 (P-gp) and BCRP inhibitor, a nucleotide-derived substrate analog that induces stomatal opening in the dark.</p>
    Fórmula:C31H37ClN4O6
    Pureza:99.19%
    Cor e Forma:Solid
    Peso molecular:597.1
  • Cyclic ADP-ribose

    CAS:
    <p>cADPR, made from NAD+, boosts calcium in cells via Ryanodine receptors and TRPM2 channels.</p>
    Fórmula:C15H21N5O13P2
    Pureza:98%
    Cor e Forma:Lyophilized Powder
    Peso molecular:541.3
  • Bifenazate

    CAS:
    <p>Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.</p>
    Fórmula:C17H20N2O3
    Pureza:99.62%
    Cor e Forma:Solid Crystalline
    Peso molecular:300.35
  • BMS-919373

    CAS:
    <p>BMS-919373 is a potassium channel Kv1.5 (KCNA5) inhibitor for atrial fibrillation and acute coronary syndrome.</p>
    Fórmula:C25H20N6O2S
    Pureza:98.51% - 99.01%
    Cor e Forma:Solid
    Peso molecular:468.53
  • PKF050-638

    CAS:
    <p>PKF050-638 disrupts CRM1-NES, inhibits HIV-1 Rev export; selective with IC50=0.04 μM.</p>
    Fórmula:C13H13ClN4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:292.72
  • Nav1.7-IN-6

    CAS:
    <p>Nav1.7-IN-6, a selective inhibitor of Nav1.7.</p>
    Fórmula:C25H25ClF6N2O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:598.99
  • Terodiline hydrochloride

    CAS:
    <p>Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2),</p>
    Fórmula:C20H28ClN
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:317.9
  • Istaroxime oxalate

    CAS:
    <p>Istaroxime (PST-2744) is a positive inotrope that inhibits Na+/K+ ATPase, raising intracellular sodium and calcium levels.</p>
    Fórmula:C23H34N2O7
    Cor e Forma:Solid
    Peso molecular:450.53
  • FR-168888 mesylate

    CAS:
    <p>FR-168888, a new Na+/H+ exchange inhibitor, can protect the heart from arrhythmia and myocardial cell death in ischemic and reperfused situations.</p>
    Fórmula:C14H18N4O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:354.38
  • TRPC6-PAM-C20

    CAS:
    <p>TRPC6-PAM-C20, a selective enhancer for TRPC6, boosts calcium in HEK cells and OAG-related platelet clumping, EC50: 2.37μM.</p>
    Fórmula:C22H21NO4
    Pureza:98.16%
    Cor e Forma:Solid
    Peso molecular:363.41
  • Nav1.8-IN-2

    CAS:
    <p>Nav1.8-IN-2 (compound 35A) strongly inhibits Nav1.8 (IC50: 0.4 nM), useful for researching pain, cough, and pruritus.</p>
    Fórmula:C18H13Cl2F3N2O3
    Cor e Forma:Solid
    Peso molecular:433.21
  • McN5691

    CAS:
    <p>McN5691 is a voltage sensitive calcium channel blocker.</p>
    Fórmula:C30H35NO3
    Pureza:98.93% - 99.38%
    Cor e Forma:Solid
    Peso molecular:457.6
  • Levosemotiadil

    CAS:
    <p>Levosemotiadil(SA 3212) is a novel calcium antagonist and a very potent inhibitor of low-density lipoprotein oxidation.Levosemotiadil may be used to prevent</p>
    Fórmula:C29H32N2O6S
    Pureza:98.53% - 99.47%
    Cor e Forma:Solid
    Peso molecular:536.64
  • Picoprazole

    CAS:
    <p>Picoprazole is a specific H+/K+-ATPase inhibitor (IC50 of 3.1±0.4 μM).</p>
    Fórmula:C17H17N3O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:343.4
  • Farnesyl pyrophosphate

    CAS:
    <p>Farnesyl pyrophosphate: 15-C isoprenoid, TRPM2 agonist, crucial for cholesterol, ubiquinones, protein farnesylation, and GGPP synthesis.</p>
    Fórmula:C15H28O7P2
    Cor e Forma:Solid
    Peso molecular:382.33
  • (R)-Baclofen hydrochloride

    CAS:
    <p>Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.</p>
    Fórmula:C10H13Cl2NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:250.12
  • KRN4884

    CAS:
    <p>KRN 4884 activates KATP channels (EC50=0.55 μM) at 0.1-3 μM with 1 mM ATP.</p>
    Fórmula:C15H14ClN5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:299.76
  • Vernakalant

    CAS:
    <p>Vernakalant (RSD-1235) is a mixed ion channel blocker.</p>
    Fórmula:C20H31NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:349.46
  • GABA-AT-IN-1

    CAS:
    <p>GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.</p>
    Fórmula:C23H18N2O6
    Cor e Forma:Solid
    Peso molecular:418.4
  • CCD-3693

    CAS:
    <p>CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.</p>
    Fórmula:C21H31F3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:372.46
  • L-4FPG

    CAS:
    <p>L-4FPG is a Glycine derivative, inhibits the neutral amino acid transporters ASCT1 and ASCT2.</p>
    Fórmula:C8H8FNO2
    Pureza:99.26%
    Cor e Forma:Solid
    Peso molecular:169.15
  • Amsacrine

    CAS:
    <p>Amsacrine (AMSA) (mAMSA) an antineoplastic agent which can intercalate into the DNA of tumor cells.</p>
    Fórmula:C21H19N3O3S
    Pureza:99.2%
    Cor e Forma:Yellow Crystalline Powder Solid
    Peso molecular:393.46
  • CFTR corrector 9

    CAS:
    <p>CFTR corrector 9 is a CF modulator used to research cystic fibrosis and related disorders.</p>
    Fórmula:C16H14N2O4
    Pureza:98.24%
    Cor e Forma:Solid
    Peso molecular:298.29
  • Nifekalant hydrochloride

    CAS:
    <p>Nifekalant hydrochloride is an IKr potassium channel blocker with an IC50 of 10 µM.</p>
    Fórmula:C19H28ClN5O5
    Pureza:99.91%
    Cor e Forma:Solid
    Peso molecular:441.91
  • V-9302

    CAS:
    <p>V-9302 (V9302) is a competitive antagonist of transmembrane glutamine flux that selectively and potently targets the amino acid transporter ASCT2 (IC50: 9.6 uM</p>
    Fórmula:C34H38N2O4
    Pureza:98% - 99.54%
    Cor e Forma:Solid
    Peso molecular:538.68
  • Benzamil hydrochloride

    CAS:
    <p>Benzamil hydrochloride is a specific and potent sodium channel (ENaC) blocker.</p>
    Fórmula:C13H15Cl2N7O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:356.21
  • Homoquinolinic acid

    CAS:
    <p>NMDA receptor agonist</p>
    Fórmula:C8H7NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:181.15
  • SCH 50911

    CAS:
    <p>SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.</p>
    Fórmula:C8H15NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:173.21
  • Abeprazan

    CAS:
    <p>Abeprazan is a potassium-competitive acid blocker targeting acid-related diseases without acid activation.</p>
    Fórmula:C19H17F3N2O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:410.41
  • ICA

    CAS:
    <p>ICA (N-[4-(2-Pyridinyl)-2-thiazolyl]-2-pyridinamine) is a SK channel inhibitor and exhibits antileishmanial activity (IC50: 2.1 µM).</p>
    Fórmula:C13H10N4S
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:254.31
  • LY339434

    CAS:
    <p>LY339434 is a potent and selective agonist of the kainate receptor GluK1, GluR5.</p>
    Fórmula:C18H19NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:313.35
  • Sabiporide

    CAS:
    <p>Sabiporide is a NHE-1 inhibitor and a cardioprotective agent.</p>
    Fórmula:C18H20ClF3N6O2
    Cor e Forma:Solid
    Peso molecular:444.84
  • Biricodar dicitrate

    CAS:
    <p>Biricodar dicitrate (VX-710) is a potent MDR inhibitor with no anticancer activity and can be used to study prostate cancer.</p>
    Fórmula:C46H57N3O21
    Pureza:97.78% - 99.78%
    Cor e Forma:Solid
    Peso molecular:987.95
  • Ro 25-6981 HCl

    CAS:
    <p>Ro 25-6981 HCl is an effective and selective NMDA glutamate receptors containing the NR2B subunit antagonist.</p>
    Fórmula:C22H30ClNO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:375.93
  • RH 3421

    CAS:
    <p>RH 3421 is used as a neuroactive dihydropyrazole insecticide.</p>
    Fórmula:C20H17ClF3N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:439.82
  • Phenamil

    CAS:
    <p>Phenamil is an inhibitor of epithelial sodium channels, activates the osteomorphin protein pathway to promote bone repair and induces significant fat formation.</p>
    Fórmula:C12H12ClN7O
    Pureza:99.07%
    Cor e Forma:Solid
    Peso molecular:305.72
  • B-TPMF

    CAS:
    <p>B-TPMF is a highly efficient and selective KCa2.1 channel inhibitor with an IC50 of 31 nM, interacting with serine residue at position 293 to inhibit KCa2.1.</p>
    Fórmula:C19H24N6O2
    Pureza:99.82%
    Cor e Forma:Solid
    Peso molecular:368.43
  • WX-081

    CAS:
    <p>WX-081 is an anti-TB drug effective against DS-TB (MIC: 0.083 μg/ml) and MDR-TB strains (MIC: 0.11 μg/ml) with hERG inhibition (IC50: 1.89 μM).</p>
    Fórmula:C34H33ClN2O2
    Cor e Forma:Solid
    Peso molecular:537.09
  • CM-TPMF

    CAS:
    <p>CM-TPMF is a highly efficient and potent activator of the K(Ca)2.1 channel, Ser293 in the transmembrane segment 5, neurological disorders.</p>
    Fórmula:C16H17ClN6O2
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:360.8
  • YM 244769 hydrochloride

    CAS:
    <p>inhibitor of the reverse mode of Na+/Ca2+ exchange (NCX)</p>
    Fórmula:C26H23ClFN3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:479.93
  • Ro 8-4304 hydrochloride

    CAS:
    <p>Ro 8-4304 hydrochloride is a NMDA receptor antagonist.</p>
    Fórmula:C21H24ClFN2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:406.88
  • ZD-9379

    CAS:
    <p>ZD-9379 is a NMDA receptor antagonist.</p>
    Fórmula:C19H14ClN3O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:383.79
  • UBP714

    CAS:
    <p>UBP714, derived from UBP608, boosts NMDAR in CA1 hippocampus, promising for schizophrenia and cognitive deficits treatment.</p>
    Fórmula:C11H7BrO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:283.07
  • TTA-Q6

    CAS:
    <p>TTA-Q6 is a T-type Ca2+ channel antagonist that inhibits the uptake of extracellular calcium ions by tumour cells for the treatment of neurological diseases.</p>
    Fórmula:C20H15ClF3N3O
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:405.8
  • 18:0 LYSO-PE

    CAS:
    <p>18:0 LYSO-PE is a compound that induces an increase in [Ca2+]i and can be used as a phospholipid (PL) standard for lipid analysis by electrospray mass spectrometry (ESI-MS)/MS.</p>
    Fórmula:C23H48NO7P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:481.6
  • ABCG2-IN-1

    CAS:
    <p>ABCG2-IN-1 (compound K2), an analog of Ko143, constitutes an orally active inhibitor targeting ABCG2 with an inhibitory concentration (IC50) of 0.13 μM.</p>
    Fórmula:C26H36N4O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:468.59
  • UCL-1848 trifluoroacetate salt

    CAS:
    <p>UCL-1848 trifluoroacetate salt is a selective Ca2+-activated, SK potassium channel blocker.</p>
    Fórmula:C32H34F6N4O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:652.638
  • E2730

    CAS:
    <p>E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.</p>
    Fórmula:C9H8F4N2O2S
    Pureza:98.22% - 98.54%
    Cor e Forma:Solid
    Peso molecular:284.23
  • TWIK-1/TREK-1-IN-2

    CAS:
    <p>TWIK-1/TREK-1-IN-2 (Compound 2g) serves as an inhibitor of both TWIK-1 and TREK-1, targeting the TREK-1 homodimer and TWIK-1/TREK-1 heterodimer with IC50 values</p>
    Fórmula:C20H29F3N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:386.45