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Transportador de Membranas/Canal Iónico

Transportador de Membranas/Canal Iónico

Os inibidores de transportadores de membrana e canais iônicos são compostos que bloqueiam a função de proteínas responsáveis pelo transporte de íons, nutrientes e outras moléculas através das membranas celulares. Esses inibidores são cruciais para o estudo da regulação da homeostase celular, transdução de sinais e neurotransmissão. Os inibidores de transportadores de membrana e canais iônicos também são importantes no desenvolvimento de tratamentos para distúrbios como epilepsia, doenças cardiovasculares e síndromes metabólicas. Na CymitQuimica, oferecemos uma ampla seleção de inibidores de alta qualidade de transportadores de membrana e canais iônicos para apoiar sua pesquisa em fisiologia, neurociência e farmacologia.

Subcategorias de "Transportador de Membranas/Canal Iónico"

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Foram encontrados 2277 produtos de "Transportador de Membranas/Canal Iónico"

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  • TRPC3/6-IN-1

    CAS:
    <p>TRPC3/6-IN-1 selectively inhibits hTRPC3/6 with IC50 of 1260/500 nM, useful in heart failure research.</p>
    Fórmula:C20H19N3O2S
    Cor e Forma:Solid
    Peso molecular:365.45
  • Ivacaftor-D9

    CAS:
    <p>CTP-656, a cystic fibrosis transmembrane conductance regulator (CFTR) channel activator, is used potentially for the treatment of cystic fibrosis.</p>
    Fórmula:C24H19D9N2O3
    Cor e Forma:Solid
    Peso molecular:401.55
  • RG100204

    CAS:
    <p>RG100204 is an orally active AQP9 inhibitor with anti-inflammatory properties. It alleviates cardiac dysfunction (systolic and diastolic) induced by sepsis, improves renal dysfunction, and reduces the elevation of the cellular damage marker LDH.</p>
    Fórmula:C20H26N6O2S2
    Cor e Forma:Solid
    Peso molecular:446.59
  • P-gp inhibitor 17

    CAS:
    <p>P-gp Inhibitor 17 (compound 2g), a potent inhibitor, directly interacts with the transmembrane domain of P-gp. This compound is useful for studying P-gp-mediated multidrug resistance in tumor cells [1].</p>
    Fórmula:C36H49N3O3
    Cor e Forma:Solid
    Peso molecular:571.79
  • CW0134

    CAS:
    <p>CW0134 (Compound 12) serves as a modulator for exportin1 (XPO1), disrupting chromatin binding and inhibiting NFAT transcription factors and T cell activation [1].</p>
    Fórmula:C11H7ClF3N3O2
    Cor e Forma:Solid
    Peso molecular:305.64
  • DPI 201-106

    CAS:
    <p>DPI 201-106: cardioselective h1 Na channel inhibitor, enhances heart contraction, blocks potassium and calcium currents.</p>
    Fórmula:C29H30N4O2
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:466.57
  • (+)-Nipecotic acid

    CAS:
    <p>(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.</p>
    Fórmula:C6H11NO2
    Pureza:99.38%
    Cor e Forma:Solid
    Peso molecular:129.16
  • Anxiolytic/nonsedative agent-1

    CAS:
    <p>TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.</p>
    Fórmula:C18H15N3O4
    Pureza:98.61%
    Cor e Forma:Solid
    Peso molecular:337.33
  • (S)-SNAP5114

    CAS:
    <p>(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.</p>
    Fórmula:C30H35NO6
    Pureza:97%
    Cor e Forma:Solid
    Peso molecular:505.6
  • Psora 4

    CAS:
    <p>Psora 4 (5-(4-Phenylbutoxy)psoralen) is a Kv1.3 blocker and a caloric restriction mimetic.</p>
    Fórmula:C21H18O4
    Cor e Forma:Solid
    Peso molecular:334.37
  • 3α,21-Dihydroxy-5α-pregnan-20-one

    CAS:
    <p>3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.</p>
    Fórmula:C21H34O3
    Pureza:98.00%
    Cor e Forma:Solid
    Peso molecular:334.49
  • AVE-0118

    CAS:
    <p>AVE-0118 is a potassium channel blocker and suppresses persistent atrial fibrillation.</p>
    Fórmula:C30H29N3O3
    Pureza:97.04% - 98.93%
    Cor e Forma:Solid
    Peso molecular:479.57
  • L589-420

    CAS:
    <p>L589-420 is a sodium pump inhibitor in human erythrocytes.</p>
    Fórmula:C14H14Cl2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:317.16
  • YM928

    CAS:
    <p>YM928 is an orally active antagonist of the AMPA receptor.</p>
    Fórmula:C14H10ClN3OS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:303.77
  • CCMQ

    CAS:
    <p>inhibits [3H]-homoquinolinic acid binding to non-NMDA sensitive sites</p>
    Fórmula:C12H9NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:231.2
  • Bms 188107

    CAS:
    <p>Bms 188107 is a calcium antagonist, it has cardioprotective effects.</p>
    Fórmula:C25H26N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:418.48
  • Caramiphen

    CAS:
    <p>Caramiphen is an antimuscarinic and anticholinergic agent that acts as an antagonist of the NMDA receptor.</p>
    Fórmula:C18H27NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:289.41
  • Viquidil

    CAS:
    <p>Viquidil is an agent with the activity of a vasodilator.</p>
    Fórmula:C20H24N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:324.42
  • (R)-Licarbazepine Acetate

    CAS:
    <p>(R)-Licarbazepine Acetate is a hopeful antiepileptic drug structurally related to Carbamazepine and Oxcarbazepine.</p>
    Fórmula:C17H16N2O3
    Cor e Forma:Solid
    Peso molecular:296.32
  • COR628

    CAS:
    <p>COR628 is the GABA(B) receptor positive allosteric modulator.</p>
    Fórmula:C16H23NO3S
    Cor e Forma:Solid
    Peso molecular:309.42
  • AZD 2066

    CAS:
    <p>AZD 2066 is a selective, orally active, and brain-penetrant mGluR5 antagonist with analgesic activity.</p>
    Fórmula:C19H16ClN5O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:381.82
  • BBR 2160

    CAS:
    <p>BBR 2160: a calcium-antagonist dihydropyridine derivative, reduces heart tissue contractility and shortens action potentials.</p>
    Fórmula:C21H25N3O7S
    Cor e Forma:Solid
    Peso molecular:463.5
  • LY-395153

    CAS:
    <p>LY-395153 is a novel potentiator of AMPA receptor.</p>
    Fórmula:C19H24N2O3S
    Cor e Forma:Solid
    Peso molecular:360.47
  • Tolperisone free base

    CAS:
    Tolperisone free base, a centrally acting muscle relaxant, has been used for the symptomatic treatment of spasticity and muscle spasm.
    Fórmula:C16H23NO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:245.36
  • Lercanidipine, (S)-

    CAS:
    <p>(S)-Lercanidipine: a dihydropyridine calcium blocker with prolonged antihypertensive and kidney-protective properties.</p>
    Fórmula:C36H41N3O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:611.73
  • Ensaculin HCl

    CAS:
    <p>Ensaculin: NMDA antagonist, 5HT1A agonist, may treat Alzheimer's, enhances memory, neuroprotective, binds multiple receptors.</p>
    Fórmula:C26H33ClN2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:489
  • Naftazone

    CAS:
    <p>Naftazone: vasoprotectant for hemostasis; boosts vein cell growth in vitro without affecting clotting.</p>
    Fórmula:C11H9N3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:215.21
  • Tiropramide

    CAS:
    <p>Tiropramide is an antispasmodic drug. It also useful to inhibit the contractile response of the urinary bladder and in managing abdominal pain in IBS.</p>
    Fórmula:C28H41N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:467.64
  • Riodipine

    CAS:
    <p>Riodipine, a calcium channel blocker, is used as cardiovascular drugs.</p>
    Fórmula:C18H19F2NO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:367.34
  • DS28120313

    CAS:
    <p>DS28120313 is an oral inhibitor of hepcidin production (IC50: 0.093 μM).</p>
    Fórmula:C16H17N5O2
    Cor e Forma:Solid
    Peso molecular:311.34
  • CPP-115

    CAS:
    <p>CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.</p>
    Fórmula:C7H9F2NO2
    Cor e Forma:Solid
    Peso molecular:177.15
  • Ethopropazine Hydrochloride

    CAS:
    <p>Ethopropazine Hydrochloride is the salt form of Profenamine,anticholinergic, antihistamine, and anti-adrenergic,Parkinson's disease,an AChE inhibitor</p>
    Fórmula:C19H25ClN2S
    Pureza:98.25%
    Cor e Forma:Solid
    Peso molecular:348.93
  • DHP-218

    CAS:
    <p>DHP-218, a calcium channel blocker, inhibits rat aorta contractions; pA2: 9.11, IC50: 6.3 nmol/L (high K+) &amp; 66 nmol/L (phenylephrine).</p>
    Fórmula:C18H21N2O7P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:408.34
  • BCTP

    CAS:
    <p>BCTP is a polymodal inhibitor of TRPV1. It has a reduced liability for hyperthermia.</p>
    Fórmula:C17H16ClN3OS
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:345.85
  • Chlormethiazole edisylate

    CAS:
    <p>Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.</p>
    Fórmula:C8H14ClNO6S3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:351.85
  • Talopram hydrochloride

    CAS:
    <p>noradrenalin transporter (NET) inhibitor</p>
    Fórmula:C20H26ClNO
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:331.88
  • IAA-94

    CAS:
    <p>IAA-94 is an inhibitor of chloride channels, it binds channels in bovine kidney cortex microsomes with a Ki value of 1 µM.</p>
    Fórmula:C17H18Cl2O4
    Cor e Forma:Solid
    Peso molecular:357.23
  • A 39355

    CAS:
    <p>A 39355 may specifically overcome multidrug resistance without the serious hypotensive effects associated with calcium antagonists.</p>
    Fórmula:C28H39Cl2N3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:504.54
  • UBP512

    CAS:
    <p>UBP512 is a NMDA receptor modulator.</p>
    Fórmula:C15H9IO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:348.14
  • Ronipamil

    CAS:
    <p>Ronipamil is an analogue of verapamil that used as a calcium entry blocker.</p>
    Fórmula:C32H48N2
    Cor e Forma:Solid
    Peso molecular:460.74
  • L 644711

    CAS:
    <p>L 644711 is an antagonist of HCO3(-)/Cl(-) antiporter.</p>
    Fórmula:C18H18Cl2O4
    Cor e Forma:Solid
    Peso molecular:369.24
  • N12N

    CAS:
    <p>N12N is a polyamine inverse NMDA receptor agonist.</p>
    Fórmula:C12H28N2
    Pureza:98%
    Cor e Forma:White Solid
    Peso molecular:200.36
  • Bromotetrandrine

    CAS:
    <p>Bromotetrandrine enhances chemo by inhibiting P-glycoprotein, countering efflux pumps.</p>
    Fórmula:C38H41BrN2O6
    Cor e Forma:Solid
    Peso molecular:701.65
  • Tedisamil

    CAS:
    <p>Tedisamil blocks cardiac K+ currents, slows heart rate, is a class III antiarrhythmic, and treats angina.</p>
    Fórmula:C19H32N2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:288.47
  • NP-252

    CAS:
    <p>NP-252 is a calcium channel antagonist potentially for the treatment of angina pectoris and congestive heart failure.</p>
    Fórmula:C26H35N3O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:469.57
  • UBP684

    CAS:
    <p>UBP684 enhances NMDAR responses, boosts l-glutamate/glycine, and mildly affects subunit agonist potency.</p>
    Fórmula:C17H20O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:256.34
  • Fenazinel Dihydrochloride

    CAS:
    <p>Fenazinel Dihydrochloride, a N-methyl-D-aspartate (NMDA) receptor antagonist, is used potentially for the treatment of ischemic stroke.</p>
    Fórmula:C21H27Cl2N3O2
    Cor e Forma:Solid
    Peso molecular:424.36
  • β-Neuroprotectin

    CAS:
    <p>beta-Neuroprotectin is a (3H)TCP binding inhibitor and provides protection against NMDA mediated neuronal cell death at low concentration.</p>
    Fórmula:C37H60N8O10
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:776.92
  • U 90042

    CAS:
    <p>GABAA receptor ligand</p>
    Fórmula:C17H13ClN6O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:352.78
  • MRS 2219

    CAS:
    <p>P2X1 receptor potentiator</p>
    Fórmula:C8H10NO5P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:231.14
  • COR627

    CAS:
    <p>COR627 is the GABA receptor positive allosteric modulator.</p>
    Fórmula:C20H27NO3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:361.5
  • trans-4-Hydroxycrotonic acid

    CAS:
    <p>ligand of γ-hydroxybutyric acid (GHB) receptor</p>
    Fórmula:C4H6O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:102.09
  • LY 81067

    CAS:
    <p>LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.</p>
    Fórmula:C22H24N4O
    Cor e Forma:Solid
    Peso molecular:360.45
  • AMG8163

    CAS:
    <p>AMG8163 is an antagonist of vanilloid receptor TRPV1.</p>
    Fórmula:C25H22F3N5O4S
    Cor e Forma:Solid
    Peso molecular:545.53
  • AH-1058 HCl

    CAS:
    <p>AH-1058 HCl is a lipophilic antiarrhythmic calcium channel blocker.</p>
    Fórmula:C30H29ClN2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:501.02
  • Watanidipine dihydrochloride

    CAS:
    <p>Watanidipine dihydrochloride is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.</p>
    Fórmula:C41H44Cl2N4O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:759.73
  • Kv1.5-IN-IIII

    CAS:
    <p>Kv1.5-IN-IIII is a potent inhibitor of Kv1.5.</p>
    Fórmula:C25H23ClN4O4S
    Cor e Forma:Solid
    Peso molecular:510.99
  • Evenamide HCl

    CAS:
    <p>Evenamide, a nav sodium channel blocker, is used potentially for the treatment of schizophrenia.</p>
    Fórmula:C16H27ClN2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:314.85
  • Gallopamil, (-)-

    CAS:
    <p>Gallopamil, (-)- is an L-type calcium channel blocker. It is used in the treatment of abnormal heart rhythms.</p>
    Fórmula:C28H40N2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:484.63
  • Pradigastat sodium

    CAS:
    <p>Pradigastat sodium is a novel inhibitor of DGAT-1.</p>
    Fórmula:C25H24F3N3NaO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:478.471
  • KR-31378

    CAS:
    <p>KR-31378, a K(ATP) channel activator, is used potentially for the treatment of ocular hypertension and glaucoma.</p>
    Fórmula:C22H27N5O4
    Cor e Forma:Solid
    Peso molecular:425.48
  • MCC1189

    CAS:
    <p>MCC1189 is a first-in-class MFS efflux pump CaMdr1p inhibitor.</p>
    Fórmula:C22H20N2O2
    Cor e Forma:Solid
    Peso molecular:344.41
  • AK-2-38

    CAS:
    <p>AK-2-38 is a nifedipine analogue with potent smooth muscle calcium antagonist action and partial agonist effects on isolated guinea pig left atrium.</p>
    Fórmula:C26H30N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:434.53
  • Azeloprazole

    CAS:
    <p>Azeloprazole, a proton pump inhibitor, is used potentially for the treatment of gastroesophageal reflux disease (GERD).</p>
    Fórmula:C22H27N3O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:429.53
  • Falipamil

    CAS:
    <p>Falipamil, a verapamil derivative, is a calcium channel blocker with antitachycardic and potential antianginal effects.</p>
    Fórmula:C24H32N2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:428.52
  • SGE-201

    CAS:
    <p>SGE-201 is an NMDA receptor allosteric modulator, revealing blocker differences via activity suppression and neuroprotection.</p>
    Fórmula:C26H44O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:388.63
  • Pentisomide

    CAS:
    <p>Pentisomide: class-I antiarrhythmic, affects depolarization &amp; repolarization, inhibits ischemia-reperfusion arrhythmias, in phase II trials.</p>
    Fórmula:C19H33N3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:319.48
  • NSC339614 potassium

    CAS:
    <p>NSC339614 potassium is a selective GluN1/GluN2C and GluN1/GluN2D receptors potentiator.</p>
    Fórmula:C10H5KN3O6S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:334.32
  • JY-XHe-053

    CAS:
    <p>JY-XHe-053 is a selective modulator of GABAA receptors.</p>
    Fórmula:C22H16FN3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:373.38
  • HIE-124

    CAS:
    <p>HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.</p>
    Fórmula:C10H12N2O3S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:240.28
  • Gallopamil HCl, (-)-

    CAS:
    <p>Gallopamil HCl, (-)- is an L-type calcium channel blocker. It is used in the treatment of abnormal heart rhythms.</p>
    Fórmula:C28H41ClN2O5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:521.09
  • Suclofenide

    CAS:
    <p>Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.</p>
    Fórmula:C16H13ClN2O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:364.8
  • Oe-9000

    CAS:
    <p>Oe-9000 blocks voltage-gated Na(+) currents in neurons at low µM, affecting both TTX-S and TTX-R types.</p>
    Fórmula:C21H29NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:343.46
  • A778317

    CAS:
    <p>A778317 is a stereoselective, high-affinity antagonist.</p>
    Fórmula:C23H25N3O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:359.46
  • AF-2785

    CAS:
    <p>In epididymal epithelial cells, AF-2785 inhibits cystic fibrosis transmembrane conductance regulator Cl(-) channels.</p>
    Fórmula:C17H12Cl2N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:347.2
  • A 80b

    CAS:
    <p>A-80b: synthetic pyridazinoindole; potent, lasting antihypertensive; lowers diastolic more; no change in heart rate; inhibits Ca2+-induced contraction.</p>
    Fórmula:C16H17N7
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:307.35
  • ABP-700

    CAS:
    <p>ABP-700 is a positive allosteric modulator of the GABAA receptor.</p>
    Fórmula:C17H18N2O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:314.34
  • NS4591

    CAS:
    <p>NS4591 is a modulator of SK-IK channels.</p>
    Fórmula:C11H12Cl2N2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:259.13
  • Methsuximide

    CAS:
    <p>Methsuximide is an anticonvulsant agent which appeared to be effective in petit mal, psychomotor and focal motor attacks [1].</p>
    Fórmula:C12H13NO2
    Cor e Forma:Crystals From Dilute Alcohol Solid
    Peso molecular:203.24
  • Carabersat

    CAS:
    <p>Carabersat(SB 204269) is a novel and effective anticonvulsant and antiepileptic agent.</p>
    Fórmula:C20H20FNO4
    Pureza:>99.99%
    Cor e Forma:Solid
    Peso molecular:357.38
  • Synthalin dihydrochloride

    CAS:
    <p>Synthalin dihydrochloride is a channel blocker of K+.</p>
    Fórmula:C12H30Cl2N6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:329.31
  • 3',4'-Dichlorobenzamil HCl

    CAS:
    <p>3',4'-Dichlorobenzamil HCl is an inhibitor of Na+ transport, Na+/Ca2+ exchanger, sarcoplasmic reticulum Ca2+ release channels.</p>
    Fórmula:C13H12Cl3N7O
    Pureza:98%
    Cor e Forma:Yellow Solid
    Peso molecular:388.64
  • BAY-Y-5959

    CAS:
    <p>BAY-Y-5959, a calcium channel agonist, is used potentially for the treatment of arrhythmia, heart failure and myocardial.</p>
    Fórmula:C26H24N4O2
    Cor e Forma:Solid
    Peso molecular:424.49
  • VU0183254

    CAS:
    <p>VU0183254, an insect OR agonist, inhibits odor-driven OR complex activation by targeting the Orco subunit.</p>
    Fórmula:C22H18N4O2S2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:434.53
  • AHR-9294

    CAS:
    <p>AHR-9294 is a novel inhibitor of H, K-ATPase. It also antagonizes gastric HCl secretion in vivo.</p>
    Fórmula:C22H24N2O3
    Cor e Forma:Solid
    Peso molecular:364.44
  • NSC103054

    CAS:
    <p>NSC103054 is an ABCG2 transporter function inhibitor.</p>
    Fórmula:C18H22Br2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:430.17
  • AHR-10718

    CAS:
    <p>AHR-10718 has an antiarrhythmic effect.</p>
    Fórmula:C22H35N3O7S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:485.6
  • Lubeluzole

    CAS:
    <p>Lubeluzole, a well-known neuroprotective agent, is recently proved useful to potentiate the activity of anti-cancer drugs.</p>
    Fórmula:C22H25F2N3O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:433.51
  • HENA

    CAS:
    <p>HENA is a novel activator of large conductance, voltage- and Ca2+-gated K+ (BK) channels.</p>
    Fórmula:C30H48NaO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:479.701
  • Lanceotoxin A

    CAS:
    <p>Lanceotoxin A is a potent Ip blocker.</p>
    Fórmula:C32H44O12
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:620.68
  • Dopropidil hydrochloride

    CAS:
    <p>Dopropidil, a calcium channel antagonist, is used potentially for the treatment of arrhymia and angina pectoris.</p>
    Fórmula:C20H36ClNO2
    Cor e Forma:Solid
    Peso molecular:357.96
  • SCH00013

    CAS:
    <p>SCH00013 is a cardiotonic that enhances myofibrillar Ca++ sensitivity, with notable effects at pH 7.2-7.4.</p>
    Fórmula:C18H20N4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:324.38
  • GZ4

    CAS:
    <p>GZ4 is a Ca2+ currents inhibitor, acting on cell surface channels.</p>
    Fórmula:C11H17NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:195.26
  • AFD-21

    CAS:
    <p>AFD-21 is a class I antiarrhythmic that inhibits sodium channels with moderate kinetics.</p>
    Fórmula:C28H39NO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:469.61
  • Hexadecylphosphoserine

    CAS:
    <p>Hexadecylphosphoserine is a representative growth inhibitor.</p>
    Fórmula:C19H40NO6P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:409.5
  • Metaphit

    CAS:
    <p>Acylator of PCP and σ-receptors</p>
    Fórmula:C18H24N2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:300.46
  • (S)-Baclofen

    CAS:
    <p>(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.</p>
    Fórmula:C10H12ClNO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:213.66
  • AMG7905

    CAS:
    <p>AMG7905 is a modulator of transient receptor potential vanilloid type 1.</p>
    Fórmula:C25H24F3N5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:483.55
  • Ro18-5362

    CAS:
    <p>Ro18-5362 is the less active prodrug of Ro 18-5364.</p>
    Fórmula:C22H25N3O2S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:395.52
  • Ceefourin-2

    CAS:
    <p>Ceefourin-2 is a highly selective multidrug resistance protein 4 inhibitor.</p>
    Fórmula:C15H9ClF3N3O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:355.7
  • BDF 9148

    CAS:
    <p>BDF 9148, a Na(+)-channel modulator, increases the contractile force of guinea-pig atria and papillary muscles.</p>
    Fórmula:C28H27N3O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:453.53
  • EO-122

    CAS:
    <p>EO-122, a calcium channel antagonist and sodium channel antagonist, is used potentially for the treatment of arrhythmia.</p>
    Fórmula:C16H23ClN2O
    Cor e Forma:Solid
    Peso molecular:294.82
  • DAA-1097

    CAS:
    <p>DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.</p>
    Fórmula:C24H24ClNO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:409.91
  • Levamlodipine gentisate

    CAS:
    <p>Levamlodipine gentisate, an active amlodipine enantiomer, is a dihydropyridine calcium channel blocker for treating hypertension and angina.</p>
    Fórmula:C27H31ClN2O9
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:563
  • JTT-552

    CAS:
    <p>JTT-552, a uric acid transporter 1 (URAT1) inhibitor, is used potentially for the treatment of hyperuricemia.</p>
    Fórmula:C15H12ClNO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:289.71
  • (S)-3-Carboxy-4-hydroxyphenylglycine

    CAS:
    <p>group I metabotropic glutamate receptor antagonist and group II mGlu agonist</p>
    Fórmula:C9H9NO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:211.17
  • TAS-4

    CAS:
    <p>TAS-4 is a modulator of metabotropic glutamate receptor 4-positive allosteric.</p>
    Fórmula:C12H8Cl2N2O
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:267.11
  • Hydroflumethiazide

    CAS:
    <p>Hydroflumethiazide is a thiazide diuretic. It has also shown the activity of anti-hypertensive.</p>
    Fórmula:C8H8F3N3O4S2
    Cor e Forma:Crystals Solid
    Peso molecular:331.29
  • Lombazole

    CAS:
    <p>Lombazole is an antimicrobial agent in the class of imidazole.</p>
    Fórmula:C22H17ClN2
    Cor e Forma:Solid
    Peso molecular:344.84
  • Aladorian

    CAS:
    <p>Aladorian (ARM036), a benzothiazepine, has anti-arrhythmic properties for heart failure and CPVT research.</p>
    Fórmula:C12H13NO4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:267.3
  • Arginylproline

    CAS:
    <p>Arginylproline is a dipeptide composed of arginine and proline. It is an incomplete breakdown product of protein digestion or protein catabolism.</p>
    Fórmula:C11H21N5O3
    Cor e Forma:Solid
    Peso molecular:271.32
  • Ro 8-4304

    CAS:
    <p>Ro 8-4304 Hydrochloride is an antagonist of NMDA receptor with IC50 of 0.4 μM</p>
    Fórmula:C21H23FN2O3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:370.42
  • CS476

    CAS:
    <p>CS476 is a potent drug of hypoglycaemic.</p>
    Fórmula:C24H29N3O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:471.57
  • Fluzinamide

    CAS:
    <p>Fluzinamide (AHR-8559) has anticonvulsant effects on ignited amygdala seizures.</p>
    Fórmula:C12H13F3N2O2
    Pureza:99.38% - >99.99%
    Cor e Forma:Solid
    Peso molecular:274.24
  • Laurinterol

    CAS:
    <p>Laurinterol is an antimicrobial from the marine alga Laurencia okamurai.</p>
    Fórmula:C15H19BrO
    Cor e Forma:Solid
    Peso molecular:295.21
  • BRL 55834

    CAS:
    <p>BRL 55834, a potassium channel activator, has shown to relax airways and vasculature in vivo.</p>
    Fórmula:C18H20F5NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:393.35
  • S-312-d

    CAS:
    <p>S-312d is a calcium channel antagonist. S-312-d can offer marked neuronal protective effects against ischemic injury.</p>
    Fórmula:C20H22N2O4S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:386.46
  • Niguldipine Free Base

    CAS:
    <p>Niguldipine Free Base is a calcium channel blocker and a₁-adrenergic receptor antagonist and a clinical modulator of multidrug resistance.</p>
    Fórmula:C36H39N3O6
    Pureza:98.97%
    Cor e Forma:Solid
    Peso molecular:609.71
  • CGP 28392

    CAS:
    <p>CGP 28392 is used as a partial calcium channel agonist.</p>
    Fórmula:C18H17F2NO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:365.33
  • RH01617

    CAS:
    <p>RH01617 possesses potent inhibitory activities against Kv1.5.</p>
    Fórmula:C22H26N2O5S
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:430.52
  • Glypromate

    CAS:
    <p>Glypromate (Gly-Pro-Glu) is a neuroprotective agent, is a weak NMDA receptor agonist</p>
    Fórmula:C12H19N3O6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:301.3
  • SR57227A

    CAS:
    <p>SR 57227A: Selective 5-HT3 receptor inhibitor, affects NMDA responses, has anti-depressant effects and reduces aggression in rats.</p>
    Fórmula:C10H14ClN3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:211.69
  • PNU-107484A

    CAS:
    <p>PNU-107484A is a unique GABA(A) receptor ligand.</p>
    Fórmula:C18H23ClN6
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:358.87
  • Dicirenone

    CAS:
    <p>Dicirenone (SC26304) inhibits the Mineralocorticoid receptor (MR), aldosterone regulation of the urinary K+:Na+ ratio, and aldosterone binding to renal</p>
    Fórmula:C26H36O5
    Pureza:99.1%
    Cor e Forma:Solid
    Peso molecular:428.56
  • Guanosine 5'-diphosphate ditromethamine

    CAS:
    Guanosine 5'-diphosphate ditromethamine (GDP ditromethamine) is a nucleoside diphosphate that activates ATP-sensitive K+ channels. It acts as a potential iron mobilizer, inhibiting the interaction between hepcidin and ferroportin, and modulating the IL-6/STAT-3 pathway. This compound finds application in inflammation research, such as studying anemia of inflammation (AI).
    Fórmula:C18H37N7O17P2
    Peso molecular:685.47
  • GSK1702934A

    CAS:
    <p>GSK1702934A is a TRPC3 agonist with pro-arrhythmic and positive inotropic effects and is used in the study of diabetes mellitus.</p>
    Fórmula:C22H25N3O2S
    Pureza:98.15%
    Cor e Forma:Solid
    Peso molecular:395.52
  • N-Oleoyl Valine

    CAS:
    N-Oleoyl valine, an N-acyl amine, antagonizes TRPV3 for thermoregulation; rises post-cold exposure; elevates in mouse lung injury.
    Fórmula:C23H43NO3
    Peso molecular:381.59
  • GS 39783

    CAS:
    <p>GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement and</p>
    Fórmula:C15H23N5O2S
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:337.44
  • SM-6586

    CAS:
    <p>SM-6586 is a potent calcium channel antagonist with inhibitory effects on Na+/H+ and Na+/Ca2+ exchange channels, and can be used in the study of cerebrovascular</p>
    Fórmula:C26H27N5O5
    Pureza:99.43%
    Cor e Forma:Solid
    Peso molecular:489.52
  • (5R)-BW-4030W92

    CAS:
    <p>(5R)-BW-4030W92 is the R-type of BW-4030W92, the active enantiomer.</p>
    Fórmula:C11H9Cl2FN4
    Pureza:98.27%
    Cor e Forma:Solid
    Peso molecular:287.12
  • AM12

    CAS:
    <p>AM12 inhibits Lanthanide-evoked TRPC5 activity (IC50: 0.28 μM).</p>
    Fórmula:C15H9BrO5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:349.13
  • ML402

    CAS:
    <p>ML402 (ZINC3671497) is an activator of TREK-1 and TREK-2 with EC50s of 13.7 μM and 5.9 μM.</p>
    Fórmula:C14H14ClNO2S
    Pureza:99.71%
    Cor e Forma:Solid
    Peso molecular:295.78
  • Zatebradine hydrochloride

    CAS:
    <p>Zatebradine hydrochloride (UL-FS-49CL) inhibits HCN channels (IC50: ~1.9 µM) blocking human HCN1-4 currents effectively.</p>
    Fórmula:C26H37ClN2O5
    Pureza:97%
    Cor e Forma:Solid
    Peso molecular:493.04
  • Cyclic ADP-ribose

    CAS:
    <p>cADPR, made from NAD+, boosts calcium in cells via Ryanodine receptors and TRPM2 channels.</p>
    Fórmula:C15H21N5O13P2
    Pureza:98%
    Cor e Forma:Lyophilized Powder
    Peso molecular:541.3
  • Bifenazate

    CAS:
    <p>Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.</p>
    Fórmula:C17H20N2O3
    Pureza:99.62%
    Cor e Forma:Solid Crystalline
    Peso molecular:300.35
  • BMS-919373

    CAS:
    <p>BMS-919373 is a potassium channel Kv1.5 (KCNA5) inhibitor for atrial fibrillation and acute coronary syndrome.</p>
    Fórmula:C25H20N6O2S
    Pureza:98.51% - 99.01%
    Cor e Forma:Solid
    Peso molecular:468.53
  • McN5691

    CAS:
    <p>McN5691 is a voltage sensitive calcium channel blocker.</p>
    Fórmula:C30H35NO3
    Pureza:98.93% - 99.38%
    Cor e Forma:Solid
    Peso molecular:457.6
  • Levosemotiadil

    CAS:
    <p>Levosemotiadil(SA 3212) is a novel calcium antagonist and a very potent inhibitor of low-density lipoprotein oxidation.Levosemotiadil may be used to prevent</p>
    Fórmula:C29H32N2O6S
    Pureza:98.53% - 99.47%
    Cor e Forma:Solid
    Peso molecular:536.64
  • (R)-Baclofen hydrochloride

    CAS:
    <p>Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.</p>
    Fórmula:C10H13Cl2NO2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:250.12
  • Vernakalant

    CAS:
    <p>Vernakalant (RSD-1235) is a mixed ion channel blocker.</p>
    Fórmula:C20H31NO4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:349.46
  • Amsacrine

    CAS:
    <p>Amsacrine (AMSA) (mAMSA) an antineoplastic agent which can intercalate into the DNA of tumor cells.</p>
    Fórmula:C21H19N3O3S
    Pureza:99.2%
    Cor e Forma:Yellow Crystalline Powder Solid
    Peso molecular:393.46
  • SCH 50911

    CAS:
    <p>SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.</p>
    Fórmula:C8H15NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:173.21
  • Phenamil

    CAS:
    <p>Phenamil is an inhibitor of epithelial sodium channels, activates the osteomorphin protein pathway to promote bone repair and induces significant fat formation.</p>
    Fórmula:C12H12ClN7O
    Pureza:99.07%
    Cor e Forma:Solid
    Peso molecular:305.72
  • B-TPMF

    CAS:
    <p>B-TPMF is a highly efficient and selective KCa2.1 channel inhibitor with an IC50 of 31 nM, interacting with serine residue at position 293 to inhibit KCa2.1.</p>
    Fórmula:C19H24N6O2
    Pureza:99.82%
    Cor e Forma:Solid
    Peso molecular:368.43
  • CM-TPMF

    CAS:
    <p>CM-TPMF is a highly efficient and potent activator of the K(Ca)2.1 channel, Ser293 in the transmembrane segment 5, neurological disorders.</p>
    Fórmula:C16H17ClN6O2
    Pureza:99.94%
    Cor e Forma:Solid
    Peso molecular:360.8
  • TTA-Q6

    CAS:
    <p>TTA-Q6 is a T-type Ca2+ channel antagonist that inhibits the uptake of extracellular calcium ions by tumour cells for the treatment of neurological diseases.</p>
    Fórmula:C20H15ClF3N3O
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:405.8
  • 18:0 LYSO-PE

    CAS:
    <p>18:0 LYSO-PE is a compound that induces an increase in [Ca2+]i and can be used as a phospholipid (PL) standard for lipid analysis by electrospray mass spectrometry (ESI-MS)/MS.</p>
    Fórmula:C23H48NO7P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:481.6
  • ABCG2-IN-1

    CAS:
    <p>ABCG2-IN-1 (compound K2), an analog of Ko143, constitutes an orally active inhibitor targeting ABCG2 with an inhibitory concentration (IC50) of 0.13 μM.</p>
    Fórmula:C26H36N4O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:468.59
  • E2730

    CAS:
    <p>E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.</p>
    Fórmula:C9H8F4N2O2S
    Pureza:98.22% - 98.54%
    Cor e Forma:Solid
    Peso molecular:284.23
  • TWIK-1/TREK-1-IN-2

    CAS:
    <p>TWIK-1/TREK-1-IN-2 (Compound 2g) serves as an inhibitor of both TWIK-1 and TREK-1, targeting the TREK-1 homodimer and TWIK-1/TREK-1 heterodimer with IC50 values</p>
    Fórmula:C20H29F3N2O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:386.45
  • ABCG2-IN-2

    CAS:
    <p>ABCG2-IN-2 is a potent inhibitor of ABCG2, exhibiting favorable oral pharmacokinetic profiles in mice, and is applicable for investigating tumor multidrug</p>
    Fórmula:C25H34N4O4
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:454.56
  • U-89843A

    CAS:
    <p>U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].</p>
    Fórmula:C16H24ClN5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:321.85
  • TWIK-1/TREK-1-IN-1

    CAS:
    <p>Compound 2a, identified as TWIK-1/TREK-1-IN-1, acts as an inhibitor of the TREK-1, a two-pore domain potassium channel (K2p) that forms TREK-1 homodimers and</p>
    Fórmula:C21H24F3NO3
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:395.42
  • D-3263 hydrochloride

    CAS:
    <p>D-3263 hydrochloride (D3263 HCl salt) is enteric-coated, orally bioavailable transient receptor potential melatonin member 8 (TRPM8) agonist.</p>
    Fórmula:C21H32ClN3O3
    Pureza:99.93%
    Cor e Forma:Solid
    Peso molecular:409.95
  • Vernakalant Hydrochloride

    CAS:
    <p>Vernakalant Hydrochloride (RSD1235 hydrochloride) is a mixed voltage- and frequency-dependent Na+ and atria-preferred K+ channel blocker.</p>
    Fórmula:C20H32ClNO4
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:385.93
  • YHO-13351 free base

    CAS:
    <p>YHO-13351 free base is the water-soluble prodrug of YHO-13177 which is an inhibitor of BCRP .</p>
    Fórmula:C26H33N3O4S
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:483.62
  • Pinacidil

    CAS:
    <p>Pinacidil (P 1134) is a guanidine that opens potassium channels and directly dilates peripheral blood vessels in small arteries, lowering blood pressure and</p>
    Fórmula:C13H19N5
    Pureza:99.9%
    Cor e Forma:Solid
    Peso molecular:245.32
  • TRPV4 agonist-1

    CAS:
    <p>TRPV4 agonist-1 is an agonist of TRPV4 (EC50: 60 nM in the hTRPV4 Ca2+ assay).</p>
    Fórmula:C25H23ClF2N4O2
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:484.93
  • PF 05089771 tosylate

    CAS:
    <p>PF-05089771 inhibits Nav1.7 channels (IC50: 11-33 nM), selective over Nav1.1-1.6/1.8, Ca+, K+ channels, TRPV1; 1000x affinity for half-inactivated state.</p>
    Fórmula:C18H12Cl2FN5O3S2·C7H8O3S
    Pureza:98.55%
    Cor e Forma:Solid
    Peso molecular:672.56
  • Lesogaberan

    CAS:
    <p>Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).</p>
    Fórmula:C3H9FNO2P
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:141.08
  • UK 78282 hydrochloride

    CAS:
    <p>UK-78282 hydrochloride, a Kv1.3 blocker.UK-78282 hydrochloride inhibits Kv1.3 voltage-gated potassium channels and suppresses human T cell activation.</p>
    Fórmula:C29H36ClNO2
    Pureza:99.68%
    Cor e Forma:Solid
    Peso molecular:466.05
  • Puliginurad

    CAS:
    <p>Puliginurad (YL-90148) is a urate transporter protein inhibitor that inhibits the reabsorption of uric acid.Puliginurad is used in the treatment of gout.</p>
    Fórmula:C19H16N2O2S
    Pureza:99.96% - 99.96%
    Cor e Forma:Solid
    Peso molecular:336.41
  • GX-674

    CAS:
    <p>GX-674 is a highly potent and selective voltage-gated sodium channel 1.7 (Nav1.7) antagonist with an IC50 value of 0.1 nM measured at -40 mV for the study of</p>
    Fórmula:C21H13ClF2N6O3S2
    Pureza:98.60%
    Cor e Forma:Solid
    Peso molecular:534.95
  • TRAM 39

    CAS:
    <p>TRAM 39 (2-Chloro-α,α-diphenylbenzeneacetonitrile) is a selective blocker of intermediate-conductance Ca2+-activated K+channels.</p>
    Fórmula:C20H14ClN
    Pureza:99.97%
    Cor e Forma:Solid
    Peso molecular:303.78
  • Tracazolate hydrochloride

    CAS:
    <p>Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.</p>
    Fórmula:C16H25ClN4O2
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:340.85
  • TRPM4-IN-2

    CAS:
    <p>NBA, or TRPM4-IN-2, is a potent TRPM4 inhibitor with IC50 of 0.16 μM, used in prostate and colorectal cancer research.</p>
    Fórmula:C19H14ClNO4
    Pureza:99.21%
    Cor e Forma:Solid
    Peso molecular:355.77
  • RO 4938581

    CAS:
    <p>RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).</p>
    Fórmula:C13H8BrF2N5
    Pureza:98%
    Cor e Forma:Solid
    Peso molecular:352.14
  • JYL 1421

    CAS:
    <p>JYL 1421 (SC 0030) is an antagonist of TRPV1 receptor (IC50 = 8 nM).</p>
    Fórmula:C20H26FN3O2S2
    Pureza:98.83%
    Cor e Forma:Solid
    Peso molecular:423.57
  • GDC-0276

    CAS:
    <p>GDC-0276 is an orally active, selective, and potent NaV1.7 inhibitor that can be used for the study of pain-related diseases.</p>
    Fórmula:C24H31FN2O4S
    Pureza:99.77%
    Cor e Forma:Solid
    Peso molecular:462.58
  • RY796

    CAS:
    <p>RY796 is a selective voltage-gated potassium (KV2) channel inhibitor that inhibits KV2.1 and KV2.2, used in research on neurological disorders.</p>
    Fórmula:C21H27N3O2
    Pureza:98.59%
    Cor e Forma:Solid
    Peso molecular:353.46
  • RN9893

    CAS:
    <p>RN9893 is a selective and potent TRPV4 receptor antagonist with IC50 values of 320, 420 and 660 nM for TRPV4 receptors in mouse, human and rat, respectively.</p>
    Fórmula:C21H23F3N4O5S
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:500.49
  • ATX-II TFA


    <p>ATX-II TFA, a specific Na+ channel modulator toxin, is derived from the venom of the sea anemone (Anemonia sulcata).</p>
    Pureza:98%
    Cor e Forma:Odour Solid
  • AZD 3043

    CAS:
    <p>AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.</p>
    Fórmula:C19H29NO5
    Pureza:98.19% - 99.55%
    Cor e Forma:Solid
    Peso molecular:351.44
  • E 0747

    CAS:
    <p>E 0747 is an antiarrhythmic agent of class 1C type. E-0747 suppresses arrhythmia by inhibiting the Na channels of cardiac cells.</p>
    Fórmula:C21H28ClN3O4
    Pureza:95.17%
    Cor e Forma:Solid
    Peso molecular:421.92
  • TRPV3 antagonist 74a

    CAS:
    <p>TRPV3 antagonist 74a (TRPV3 74a) is a specific TRPV3 antagonist for the study of neurological disorders.</p>
    Fórmula:C17H17F3N2O2
    Pureza:≥98.0%
    Cor e Forma:Solid
    Peso molecular:338.32
  • AVE1231

    CAS:
    <p>AVE1231 is a TASK-1 channel blocker that inhibits TASK-1 and can be used in the study of atrial fibrillation.</p>
    Fórmula:C20H27N3O4S
    Pureza:98.03%
    Cor e Forma:Solid
    Peso molecular:405.51
  • Phaclofen

    CAS:
    <p>GABAB antagonist</p>
    Fórmula:C9H13ClNO3P
    Pureza:99.32%
    Cor e Forma:White Solid
    Peso molecular:249.63
  • GAL-021 sulfate

    CAS:
    <p>GAL-021 sulfate is a BKCa channel blocker that inhibits the analgesic effects of opioids and is used in the study of respiratory control diseases.</p>
    Fórmula:C11H24N6O5S
    Pureza:99.92%
    Cor e Forma:Solid
    Peso molecular:352.41
  • Istaroxime hydrochloride

    CAS:
    <p>Istaroxime hydrochloride (PST2744 hydrochloride) is a Na+/K+-ATPase inhibitor and SERCA 2 activator, and is a novel positive inotropic compound.</p>
    Fórmula:C21H33ClN2O3
    Cor e Forma:Solid
    Peso molecular:396.95
  • GX-585

    CAS:
    <p>GX-585 is a novel potent inhibitor of NaV1.7 and highly selective against NaV1.5, having limited selectivity against NaV1.1 and NaV1.2.</p>
    Fórmula:C24H25Cl2FN4O3S
    Pureza:99.02% - 99.03%
    Cor e Forma:Solid
    Peso molecular:539.45
  • SRI-37240

    CAS:
    <p>SRI-37240 suppresses CFTR nonsense mutations, aids in fixing premature termination codons, works with G418.</p>
    Fórmula:C24H23N3O2
    Pureza:98.73%
    Cor e Forma:Solid
    Peso molecular:385.46
  • Aprikalim

    CAS:
    <p>Aprikalim opens KATP channels, protects the heart, and at high doses, dilates blood vessels.</p>
    Fórmula:C12H16N2OS2
    Pureza:99.42% - 99.90%
    Cor e Forma:Solid
    Peso molecular:268.4
  • Suriclone

    CAS:
    <p>Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.</p>
    Fórmula:C20H20ClN5O3S2
    Pureza:99.21% - 99.73%
    Cor e Forma:Solid
    Peso molecular:477.99
  • KT-362 fumarate

    CAS:
    <p>KT-362 fumarate, a novel antagonist of Ca, K, and Na channels, induces vasodilation and relaxes rabbit arterial strips.</p>
    Fórmula:C26H32N2O7S
    Pureza:99.75% - 99.98%
    Cor e Forma:Solid
    Peso molecular:516.61
  • AGN-201904

    CAS:
    AGN-201904 is a proton pump inhibitor, an omeprazole prodrug, which delays aging and may be used for the prevention and treatment of peptic ulcers.
    Fórmula:C25H25N3O8S2
    Pureza:97.32%
    Cor e Forma:Solid
    Peso molecular:559.61
  • DMT1 blocker 1

    CAS:
    <p>DMT1 blocker 1 inhibits DMT1; IC50=0.64μM; may prevent intestinal iron absorption.</p>
    Fórmula:C16H14N4O2
    Pureza:99.73%
    Cor e Forma:Solid
    Peso molecular:294.31
  • Trombodipine

    CAS:
    <p>Trombodipine (PCA-4230) is a platelet aggregation inhibitor with antithrombotic activity and protection against Listeria monocytogenes.</p>
    Fórmula:C21H24N2O7S
    Pureza:98.73% - 99.14%
    Cor e Forma:Solid
    Peso molecular:448.49
  • Elismetrep

    CAS:
    <p>Elismetrep (MT-8554) is an orally available TRPM8 inhibitor with potential analgesic activity for the study of vasomotor symptoms in postmenopausal women.</p>
    Fórmula:C27H21F3N2O5S
    Pureza:99.37% - 99.93%
    Cor e Forma:Solid
    Peso molecular:542.53
  • R 56865

    CAS:
    <p>R 56865 is a weak potential-operated channel inhibitor that inhibits the late sodium current in human isolated cardiomyocytes.</p>
    Fórmula:C23H28FN3OS
    Pureza:99.52%
    Cor e Forma:Solid
    Peso molecular:413.55
  • Riluzole hydrochloride

    CAS:
    <p>Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).</p>
    Fórmula:C8H6ClF3N2OS
    Pureza:99.76%
    Cor e Forma:Solid
    Peso molecular:270.66
  • SKF96067

    CAS:
    <p>SKF96067 is a reversible gastric H+/K+-ATPase inhibitor that can induce relaxation of human airway smooth muscle in vitro.</p>
    Fórmula:C21H22N2O2
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:334.41
  • Losigamone

    CAS:
    <p>Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about the treatment of partial seizures.</p>
    Fórmula:C12H11ClO4
    Pureza:99.98%
    Cor e Forma:Solid
    Peso molecular:254.67
  • TASK-1-IN-1

    CAS:
    <p>TASK-1-IN-1: Potent, selective TASK-1 blocker (IC50: 148 nM), weaker on TASK-3 (IC50: 1750 nM), anticancer properties.</p>
    Fórmula:C22H20N2O2
    Pureza:99.57%
    Cor e Forma:Soild
    Peso molecular:344.41
  • Nerisopam

    CAS:
    <p>Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.</p>
    Fórmula:C18H19N3O2
    Pureza:97.07%
    Cor e Forma:Solid
    Peso molecular:309.36
  • Fengabine

    CAS:
    <p>Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.</p>
    Fórmula:C17H17Cl2NO
    Pureza:99%
    Cor e Forma:Solid
    Peso molecular:322.23
  • TAK-653

    CAS:
    <p>TAK-653 is a selective AMPA receptor PAM with minimal agonist activity, showing antidepressant-like effects and safety in rats.</p>
    Fórmula:C19H23N3O3S
    Pureza:99.89%
    Cor e Forma:Solid
    Peso molecular:373.47
  • Neboglamine hydrochloride

    CAS:
    <p>Neboglamine (CR-2249, XY-2401) hydrochloride boosts NMDA receptor, aids schizophrenia research, and is orally active.</p>
    Fórmula:C13H25ClN2O3
    Pureza:99.19%
    Cor e Forma:Solid
    Peso molecular:292.8
  • DSP-0565

    CAS:
    <p>DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.</p>
    Fórmula:C14H12FNO
    Pureza:99.51% - 99.56%
    Cor e Forma:Solid
    Peso molecular:229.25
  • Alpidem

    CAS:
    <p>Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.</p>
    Fórmula:C21H23Cl2N3O
    Pureza:99.56% - 99.97%
    Cor e Forma:White To Off-White Solid
    Peso molecular:404.33
  • Muscimol HBr

    CAS:
    <p>Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.</p>
    Fórmula:C4H7BrN2O2
    Pureza:98.13%
    Cor e Forma:Off-White Powder
    Peso molecular:195.01