
Transportador de Membranas/Canal Iónico
Os inibidores de transportadores de membrana e canais iônicos são compostos que bloqueiam a função de proteínas responsáveis pelo transporte de íons, nutrientes e outras moléculas através das membranas celulares. Esses inibidores são cruciais para o estudo da regulação da homeostase celular, transdução de sinais e neurotransmissão. Os inibidores de transportadores de membrana e canais iônicos também são importantes no desenvolvimento de tratamentos para distúrbios como epilepsia, doenças cardiovasculares e síndromes metabólicas. Na CymitQuimica, oferecemos uma ampla seleção de inibidores de alta qualidade de transportadores de membrana e canais iônicos para apoiar sua pesquisa em fisiologia, neurociência e farmacologia.
Subcategorias de "Transportador de Membranas/Canal Iónico"
- ABC(3 produtos)
- ATPase(93 produtos)
- Receptor de adiponectina(5 produtos)
- CFTR(64 produtos)
- Receptor CGRP(51 produtos)
- Canais de Cálcio(493 produtos)
- Canal de cloreto(49 produtos)
- Receptor GABA(336 produtos)
- Transportador de monoamina(23 produtos)
- Transportador de monocarboxilato(17 produtos)
- NKCC(2 produtos)
- NPC1L1(3 produtos)
- Cotransportador Na-K-Cl(8 produtos)
- OAT(27 produtos)
- OCT(7 produtos)
- P-gp(53 produtos)
- Canal de Potássio(276 produtos)
- Bomba de prótons(39 produtos)
- SGLT(30 produtos)
- Canal de Sódio(202 produtos)
- Canal TRP/TRPV(93 produtos)
Exibir 13 mais subcategorias
Foram encontrados 2277 produtos de "Transportador de Membranas/Canal Iónico"
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TRPC3/6-IN-1
CAS:<p>TRPC3/6-IN-1 selectively inhibits hTRPC3/6 with IC50 of 1260/500 nM, useful in heart failure research.</p>Fórmula:C20H19N3O2SCor e Forma:SolidPeso molecular:365.45Ivacaftor-D9
CAS:<p>CTP-656, a cystic fibrosis transmembrane conductance regulator (CFTR) channel activator, is used potentially for the treatment of cystic fibrosis.</p>Fórmula:C24H19D9N2O3Cor e Forma:SolidPeso molecular:401.55RG100204
CAS:<p>RG100204 is an orally active AQP9 inhibitor with anti-inflammatory properties. It alleviates cardiac dysfunction (systolic and diastolic) induced by sepsis, improves renal dysfunction, and reduces the elevation of the cellular damage marker LDH.</p>Fórmula:C20H26N6O2S2Cor e Forma:SolidPeso molecular:446.59P-gp inhibitor 17
CAS:<p>P-gp Inhibitor 17 (compound 2g), a potent inhibitor, directly interacts with the transmembrane domain of P-gp. This compound is useful for studying P-gp-mediated multidrug resistance in tumor cells [1].</p>Fórmula:C36H49N3O3Cor e Forma:SolidPeso molecular:571.79CW0134
CAS:<p>CW0134 (Compound 12) serves as a modulator for exportin1 (XPO1), disrupting chromatin binding and inhibiting NFAT transcription factors and T cell activation [1].</p>Fórmula:C11H7ClF3N3O2Cor e Forma:SolidPeso molecular:305.64DPI 201-106
CAS:<p>DPI 201-106: cardioselective h1 Na channel inhibitor, enhances heart contraction, blocks potassium and calcium currents.</p>Fórmula:C29H30N4O2Pureza:99.94%Cor e Forma:SolidPeso molecular:466.57(+)-Nipecotic acid
CAS:<p>(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.</p>Fórmula:C6H11NO2Pureza:99.38%Cor e Forma:SolidPeso molecular:129.16Anxiolytic/nonsedative agent-1
CAS:<p>TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.</p>Fórmula:C18H15N3O4Pureza:98.61%Cor e Forma:SolidPeso molecular:337.33(S)-SNAP5114
CAS:<p>(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.</p>Fórmula:C30H35NO6Pureza:97%Cor e Forma:SolidPeso molecular:505.6Psora 4
CAS:<p>Psora 4 (5-(4-Phenylbutoxy)psoralen) is a Kv1.3 blocker and a caloric restriction mimetic.</p>Fórmula:C21H18O4Cor e Forma:SolidPeso molecular:334.373α,21-Dihydroxy-5α-pregnan-20-one
CAS:<p>3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.</p>Fórmula:C21H34O3Pureza:98.00%Cor e Forma:SolidPeso molecular:334.49AVE-0118
CAS:<p>AVE-0118 is a potassium channel blocker and suppresses persistent atrial fibrillation.</p>Fórmula:C30H29N3O3Pureza:97.04% - 98.93%Cor e Forma:SolidPeso molecular:479.57L589-420
CAS:<p>L589-420 is a sodium pump inhibitor in human erythrocytes.</p>Fórmula:C14H14Cl2O4Pureza:98%Cor e Forma:SolidPeso molecular:317.16YM928
CAS:<p>YM928 is an orally active antagonist of the AMPA receptor.</p>Fórmula:C14H10ClN3OSPureza:98%Cor e Forma:SolidPeso molecular:303.77CCMQ
CAS:<p>inhibits [3H]-homoquinolinic acid binding to non-NMDA sensitive sites</p>Fórmula:C12H9NO4Pureza:98%Cor e Forma:SolidPeso molecular:231.2Bms 188107
CAS:<p>Bms 188107 is a calcium antagonist, it has cardioprotective effects.</p>Fórmula:C25H26N2O4Pureza:98%Cor e Forma:SolidPeso molecular:418.48Caramiphen
CAS:<p>Caramiphen is an antimuscarinic and anticholinergic agent that acts as an antagonist of the NMDA receptor.</p>Fórmula:C18H27NO2Pureza:98%Cor e Forma:SolidPeso molecular:289.41Viquidil
CAS:<p>Viquidil is an agent with the activity of a vasodilator.</p>Fórmula:C20H24N2O2Pureza:98%Cor e Forma:SolidPeso molecular:324.42(R)-Licarbazepine Acetate
CAS:<p>(R)-Licarbazepine Acetate is a hopeful antiepileptic drug structurally related to Carbamazepine and Oxcarbazepine.</p>Fórmula:C17H16N2O3Cor e Forma:SolidPeso molecular:296.32COR628
CAS:<p>COR628 is the GABA(B) receptor positive allosteric modulator.</p>Fórmula:C16H23NO3SCor e Forma:SolidPeso molecular:309.42AZD 2066
CAS:<p>AZD 2066 is a selective, orally active, and brain-penetrant mGluR5 antagonist with analgesic activity.</p>Fórmula:C19H16ClN5O2Pureza:98%Cor e Forma:SolidPeso molecular:381.82BBR 2160
CAS:<p>BBR 2160: a calcium-antagonist dihydropyridine derivative, reduces heart tissue contractility and shortens action potentials.</p>Fórmula:C21H25N3O7SCor e Forma:SolidPeso molecular:463.5LY-395153
CAS:<p>LY-395153 is a novel potentiator of AMPA receptor.</p>Fórmula:C19H24N2O3SCor e Forma:SolidPeso molecular:360.47Tolperisone free base
CAS:Tolperisone free base, a centrally acting muscle relaxant, has been used for the symptomatic treatment of spasticity and muscle spasm.Fórmula:C16H23NOPureza:98%Cor e Forma:SolidPeso molecular:245.36Lercanidipine, (S)-
CAS:<p>(S)-Lercanidipine: a dihydropyridine calcium blocker with prolonged antihypertensive and kidney-protective properties.</p>Fórmula:C36H41N3O6Pureza:98%Cor e Forma:SolidPeso molecular:611.73Ensaculin HCl
CAS:<p>Ensaculin: NMDA antagonist, 5HT1A agonist, may treat Alzheimer's, enhances memory, neuroprotective, binds multiple receptors.</p>Fórmula:C26H33ClN2O5Pureza:98%Cor e Forma:SolidPeso molecular:489Naftazone
CAS:<p>Naftazone: vasoprotectant for hemostasis; boosts vein cell growth in vitro without affecting clotting.</p>Fórmula:C11H9N3O2Pureza:98%Cor e Forma:SolidPeso molecular:215.21Tiropramide
CAS:<p>Tiropramide is an antispasmodic drug. It also useful to inhibit the contractile response of the urinary bladder and in managing abdominal pain in IBS.</p>Fórmula:C28H41N3O3Pureza:98%Cor e Forma:SolidPeso molecular:467.64Riodipine
CAS:<p>Riodipine, a calcium channel blocker, is used as cardiovascular drugs.</p>Fórmula:C18H19F2NO5Pureza:98%Cor e Forma:SolidPeso molecular:367.34DS28120313
CAS:<p>DS28120313 is an oral inhibitor of hepcidin production (IC50: 0.093 μM).</p>Fórmula:C16H17N5O2Cor e Forma:SolidPeso molecular:311.34CPP-115
CAS:<p>CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.</p>Fórmula:C7H9F2NO2Cor e Forma:SolidPeso molecular:177.15Ethopropazine Hydrochloride
CAS:<p>Ethopropazine Hydrochloride is the salt form of Profenamine,anticholinergic, antihistamine, and anti-adrenergic,Parkinson's disease,an AChE inhibitor</p>Fórmula:C19H25ClN2SPureza:98.25%Cor e Forma:SolidPeso molecular:348.93DHP-218
CAS:<p>DHP-218, a calcium channel blocker, inhibits rat aorta contractions; pA2: 9.11, IC50: 6.3 nmol/L (high K+) & 66 nmol/L (phenylephrine).</p>Fórmula:C18H21N2O7PPureza:98%Cor e Forma:SolidPeso molecular:408.34BCTP
CAS:<p>BCTP is a polymodal inhibitor of TRPV1. It has a reduced liability for hyperthermia.</p>Fórmula:C17H16ClN3OSPureza:98%Cor e Forma:SolidPeso molecular:345.85Chlormethiazole edisylate
CAS:<p>Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.</p>Fórmula:C8H14ClNO6S3Pureza:98%Cor e Forma:SolidPeso molecular:351.85Talopram hydrochloride
CAS:<p>noradrenalin transporter (NET) inhibitor</p>Fórmula:C20H26ClNOPureza:98%Cor e Forma:SolidPeso molecular:331.88IAA-94
CAS:<p>IAA-94 is an inhibitor of chloride channels, it binds channels in bovine kidney cortex microsomes with a Ki value of 1 µM.</p>Fórmula:C17H18Cl2O4Cor e Forma:SolidPeso molecular:357.23A 39355
CAS:<p>A 39355 may specifically overcome multidrug resistance without the serious hypotensive effects associated with calcium antagonists.</p>Fórmula:C28H39Cl2N3OPureza:98%Cor e Forma:SolidPeso molecular:504.54UBP512
CAS:<p>UBP512 is a NMDA receptor modulator.</p>Fórmula:C15H9IO2Pureza:98%Cor e Forma:SolidPeso molecular:348.14Ronipamil
CAS:<p>Ronipamil is an analogue of verapamil that used as a calcium entry blocker.</p>Fórmula:C32H48N2Cor e Forma:SolidPeso molecular:460.74L 644711
CAS:<p>L 644711 is an antagonist of HCO3(-)/Cl(-) antiporter.</p>Fórmula:C18H18Cl2O4Cor e Forma:SolidPeso molecular:369.24N12N
CAS:<p>N12N is a polyamine inverse NMDA receptor agonist.</p>Fórmula:C12H28N2Pureza:98%Cor e Forma:White SolidPeso molecular:200.36Bromotetrandrine
CAS:<p>Bromotetrandrine enhances chemo by inhibiting P-glycoprotein, countering efflux pumps.</p>Fórmula:C38H41BrN2O6Cor e Forma:SolidPeso molecular:701.65Tedisamil
CAS:<p>Tedisamil blocks cardiac K+ currents, slows heart rate, is a class III antiarrhythmic, and treats angina.</p>Fórmula:C19H32N2Pureza:98%Cor e Forma:SolidPeso molecular:288.47NP-252
CAS:<p>NP-252 is a calcium channel antagonist potentially for the treatment of angina pectoris and congestive heart failure.</p>Fórmula:C26H35N3O5Pureza:98%Cor e Forma:SolidPeso molecular:469.57UBP684
CAS:<p>UBP684 enhances NMDAR responses, boosts l-glutamate/glycine, and mildly affects subunit agonist potency.</p>Fórmula:C17H20O2Pureza:98%Cor e Forma:SolidPeso molecular:256.34Fenazinel Dihydrochloride
CAS:<p>Fenazinel Dihydrochloride, a N-methyl-D-aspartate (NMDA) receptor antagonist, is used potentially for the treatment of ischemic stroke.</p>Fórmula:C21H27Cl2N3O2Cor e Forma:SolidPeso molecular:424.36β-Neuroprotectin
CAS:<p>beta-Neuroprotectin is a (3H)TCP binding inhibitor and provides protection against NMDA mediated neuronal cell death at low concentration.</p>Fórmula:C37H60N8O10Pureza:98%Cor e Forma:SolidPeso molecular:776.92U 90042
CAS:<p>GABAA receptor ligand</p>Fórmula:C17H13ClN6OPureza:98%Cor e Forma:SolidPeso molecular:352.78MRS 2219
CAS:<p>P2X1 receptor potentiator</p>Fórmula:C8H10NO5PPureza:98%Cor e Forma:SolidPeso molecular:231.14COR627
CAS:<p>COR627 is the GABA receptor positive allosteric modulator.</p>Fórmula:C20H27NO3SPureza:98%Cor e Forma:SolidPeso molecular:361.5trans-4-Hydroxycrotonic acid
CAS:<p>ligand of γ-hydroxybutyric acid (GHB) receptor</p>Fórmula:C4H6O3Pureza:98%Cor e Forma:SolidPeso molecular:102.09LY 81067
CAS:<p>LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.</p>Fórmula:C22H24N4OCor e Forma:SolidPeso molecular:360.45AMG8163
CAS:<p>AMG8163 is an antagonist of vanilloid receptor TRPV1.</p>Fórmula:C25H22F3N5O4SCor e Forma:SolidPeso molecular:545.53AH-1058 HCl
CAS:<p>AH-1058 HCl is a lipophilic antiarrhythmic calcium channel blocker.</p>Fórmula:C30H29ClN2O3Pureza:98%Cor e Forma:SolidPeso molecular:501.02Watanidipine dihydrochloride
CAS:<p>Watanidipine dihydrochloride is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.</p>Fórmula:C41H44Cl2N4O6Pureza:98%Cor e Forma:SolidPeso molecular:759.73Kv1.5-IN-IIII
CAS:<p>Kv1.5-IN-IIII is a potent inhibitor of Kv1.5.</p>Fórmula:C25H23ClN4O4SCor e Forma:SolidPeso molecular:510.99Evenamide HCl
CAS:<p>Evenamide, a nav sodium channel blocker, is used potentially for the treatment of schizophrenia.</p>Fórmula:C16H27ClN2O2Pureza:98%Cor e Forma:SolidPeso molecular:314.85Gallopamil, (-)-
CAS:<p>Gallopamil, (-)- is an L-type calcium channel blocker. It is used in the treatment of abnormal heart rhythms.</p>Fórmula:C28H40N2O5Pureza:98%Cor e Forma:SolidPeso molecular:484.63Pradigastat sodium
CAS:<p>Pradigastat sodium is a novel inhibitor of DGAT-1.</p>Fórmula:C25H24F3N3NaO2Pureza:98%Cor e Forma:SolidPeso molecular:478.471KR-31378
CAS:<p>KR-31378, a K(ATP) channel activator, is used potentially for the treatment of ocular hypertension and glaucoma.</p>Fórmula:C22H27N5O4Cor e Forma:SolidPeso molecular:425.48MCC1189
CAS:<p>MCC1189 is a first-in-class MFS efflux pump CaMdr1p inhibitor.</p>Fórmula:C22H20N2O2Cor e Forma:SolidPeso molecular:344.41AK-2-38
CAS:<p>AK-2-38 is a nifedipine analogue with potent smooth muscle calcium antagonist action and partial agonist effects on isolated guinea pig left atrium.</p>Fórmula:C26H30N2O4Pureza:98%Cor e Forma:SolidPeso molecular:434.53Azeloprazole
CAS:<p>Azeloprazole, a proton pump inhibitor, is used potentially for the treatment of gastroesophageal reflux disease (GERD).</p>Fórmula:C22H27N3O4SPureza:98%Cor e Forma:SolidPeso molecular:429.53Falipamil
CAS:<p>Falipamil, a verapamil derivative, is a calcium channel blocker with antitachycardic and potential antianginal effects.</p>Fórmula:C24H32N2O5Pureza:98%Cor e Forma:SolidPeso molecular:428.52SGE-201
CAS:<p>SGE-201 is an NMDA receptor allosteric modulator, revealing blocker differences via activity suppression and neuroprotection.</p>Fórmula:C26H44O2Pureza:98%Cor e Forma:SolidPeso molecular:388.63Pentisomide
CAS:<p>Pentisomide: class-I antiarrhythmic, affects depolarization & repolarization, inhibits ischemia-reperfusion arrhythmias, in phase II trials.</p>Fórmula:C19H33N3OPureza:98%Cor e Forma:SolidPeso molecular:319.48NSC339614 potassium
CAS:<p>NSC339614 potassium is a selective GluN1/GluN2C and GluN1/GluN2D receptors potentiator.</p>Fórmula:C10H5KN3O6SPureza:98%Cor e Forma:SolidPeso molecular:334.32JY-XHe-053
CAS:<p>JY-XHe-053 is a selective modulator of GABAA receptors.</p>Fórmula:C22H16FN3O2Pureza:98%Cor e Forma:SolidPeso molecular:373.38HIE-124
CAS:<p>HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.</p>Fórmula:C10H12N2O3SPureza:98%Cor e Forma:SolidPeso molecular:240.28Gallopamil HCl, (-)-
CAS:<p>Gallopamil HCl, (-)- is an L-type calcium channel blocker. It is used in the treatment of abnormal heart rhythms.</p>Fórmula:C28H41ClN2O5Pureza:98%Cor e Forma:SolidPeso molecular:521.09Suclofenide
CAS:<p>Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.</p>Fórmula:C16H13ClN2O4SPureza:98%Cor e Forma:SolidPeso molecular:364.8Oe-9000
CAS:<p>Oe-9000 blocks voltage-gated Na(+) currents in neurons at low µM, affecting both TTX-S and TTX-R types.</p>Fórmula:C21H29NO3Pureza:98%Cor e Forma:SolidPeso molecular:343.46A778317
CAS:<p>A778317 is a stereoselective, high-affinity antagonist.</p>Fórmula:C23H25N3OPureza:98%Cor e Forma:SolidPeso molecular:359.46AF-2785
CAS:<p>In epididymal epithelial cells, AF-2785 inhibits cystic fibrosis transmembrane conductance regulator Cl(-) channels.</p>Fórmula:C17H12Cl2N2O2Pureza:98%Cor e Forma:SolidPeso molecular:347.2A 80b
CAS:<p>A-80b: synthetic pyridazinoindole; potent, lasting antihypertensive; lowers diastolic more; no change in heart rate; inhibits Ca2+-induced contraction.</p>Fórmula:C16H17N7Pureza:98%Cor e Forma:SolidPeso molecular:307.35ABP-700
CAS:<p>ABP-700 is a positive allosteric modulator of the GABAA receptor.</p>Fórmula:C17H18N2O4Pureza:98%Cor e Forma:SolidPeso molecular:314.34NS4591
CAS:<p>NS4591 is a modulator of SK-IK channels.</p>Fórmula:C11H12Cl2N2OPureza:98%Cor e Forma:SolidPeso molecular:259.13Methsuximide
CAS:<p>Methsuximide is an anticonvulsant agent which appeared to be effective in petit mal, psychomotor and focal motor attacks [1].</p>Fórmula:C12H13NO2Cor e Forma:Crystals From Dilute Alcohol SolidPeso molecular:203.24Carabersat
CAS:<p>Carabersat(SB 204269) is a novel and effective anticonvulsant and antiepileptic agent.</p>Fórmula:C20H20FNO4Pureza:>99.99%Cor e Forma:SolidPeso molecular:357.38Synthalin dihydrochloride
CAS:<p>Synthalin dihydrochloride is a channel blocker of K+.</p>Fórmula:C12H30Cl2N6Pureza:98%Cor e Forma:SolidPeso molecular:329.313',4'-Dichlorobenzamil HCl
CAS:<p>3',4'-Dichlorobenzamil HCl is an inhibitor of Na+ transport, Na+/Ca2+ exchanger, sarcoplasmic reticulum Ca2+ release channels.</p>Fórmula:C13H12Cl3N7OPureza:98%Cor e Forma:Yellow SolidPeso molecular:388.64BAY-Y-5959
CAS:<p>BAY-Y-5959, a calcium channel agonist, is used potentially for the treatment of arrhythmia, heart failure and myocardial.</p>Fórmula:C26H24N4O2Cor e Forma:SolidPeso molecular:424.49VU0183254
CAS:<p>VU0183254, an insect OR agonist, inhibits odor-driven OR complex activation by targeting the Orco subunit.</p>Fórmula:C22H18N4O2S2Pureza:98%Cor e Forma:SolidPeso molecular:434.53AHR-9294
CAS:<p>AHR-9294 is a novel inhibitor of H, K-ATPase. It also antagonizes gastric HCl secretion in vivo.</p>Fórmula:C22H24N2O3Cor e Forma:SolidPeso molecular:364.44NSC103054
CAS:<p>NSC103054 is an ABCG2 transporter function inhibitor.</p>Fórmula:C18H22Br2O2Pureza:98%Cor e Forma:SolidPeso molecular:430.17AHR-10718
CAS:<p>AHR-10718 has an antiarrhythmic effect.</p>Fórmula:C22H35N3O7SPureza:98%Cor e Forma:SolidPeso molecular:485.6Lubeluzole
CAS:<p>Lubeluzole, a well-known neuroprotective agent, is recently proved useful to potentiate the activity of anti-cancer drugs.</p>Fórmula:C22H25F2N3O2SPureza:98%Cor e Forma:SolidPeso molecular:433.51HENA
CAS:<p>HENA is a novel activator of large conductance, voltage- and Ca2+-gated K+ (BK) channels.</p>Fórmula:C30H48NaO3Pureza:98%Cor e Forma:SolidPeso molecular:479.701Lanceotoxin A
CAS:<p>Lanceotoxin A is a potent Ip blocker.</p>Fórmula:C32H44O12Pureza:98%Cor e Forma:SolidPeso molecular:620.68Dopropidil hydrochloride
CAS:<p>Dopropidil, a calcium channel antagonist, is used potentially for the treatment of arrhymia and angina pectoris.</p>Fórmula:C20H36ClNO2Cor e Forma:SolidPeso molecular:357.96SCH00013
CAS:<p>SCH00013 is a cardiotonic that enhances myofibrillar Ca++ sensitivity, with notable effects at pH 7.2-7.4.</p>Fórmula:C18H20N4O2Pureza:98%Cor e Forma:SolidPeso molecular:324.38GZ4
CAS:<p>GZ4 is a Ca2+ currents inhibitor, acting on cell surface channels.</p>Fórmula:C11H17NO2Pureza:98%Cor e Forma:SolidPeso molecular:195.26AFD-21
CAS:<p>AFD-21 is a class I antiarrhythmic that inhibits sodium channels with moderate kinetics.</p>Fórmula:C28H39NO5Pureza:98%Cor e Forma:SolidPeso molecular:469.61Hexadecylphosphoserine
CAS:<p>Hexadecylphosphoserine is a representative growth inhibitor.</p>Fórmula:C19H40NO6PPureza:98%Cor e Forma:SolidPeso molecular:409.5Metaphit
CAS:<p>Acylator of PCP and σ-receptors</p>Fórmula:C18H24N2SPureza:98%Cor e Forma:SolidPeso molecular:300.46(S)-Baclofen
CAS:<p>(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.</p>Fórmula:C10H12ClNO2Pureza:98%Cor e Forma:SolidPeso molecular:213.66AMG7905
CAS:<p>AMG7905 is a modulator of transient receptor potential vanilloid type 1.</p>Fórmula:C25H24F3N5SPureza:98%Cor e Forma:SolidPeso molecular:483.55Ro18-5362
CAS:<p>Ro18-5362 is the less active prodrug of Ro 18-5364.</p>Fórmula:C22H25N3O2SPureza:98%Cor e Forma:SolidPeso molecular:395.52Ceefourin-2
CAS:<p>Ceefourin-2 is a highly selective multidrug resistance protein 4 inhibitor.</p>Fórmula:C15H9ClF3N3O2Pureza:98%Cor e Forma:SolidPeso molecular:355.7BDF 9148
CAS:<p>BDF 9148, a Na(+)-channel modulator, increases the contractile force of guinea-pig atria and papillary muscles.</p>Fórmula:C28H27N3O3Pureza:98%Cor e Forma:SolidPeso molecular:453.53EO-122
CAS:<p>EO-122, a calcium channel antagonist and sodium channel antagonist, is used potentially for the treatment of arrhythmia.</p>Fórmula:C16H23ClN2OCor e Forma:SolidPeso molecular:294.82DAA-1097
CAS:<p>DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.</p>Fórmula:C24H24ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:409.91Levamlodipine gentisate
CAS:<p>Levamlodipine gentisate, an active amlodipine enantiomer, is a dihydropyridine calcium channel blocker for treating hypertension and angina.</p>Fórmula:C27H31ClN2O9Pureza:98%Cor e Forma:SolidPeso molecular:563JTT-552
CAS:<p>JTT-552, a uric acid transporter 1 (URAT1) inhibitor, is used potentially for the treatment of hyperuricemia.</p>Fórmula:C15H12ClNO3Pureza:98%Cor e Forma:SolidPeso molecular:289.71(S)-3-Carboxy-4-hydroxyphenylglycine
CAS:<p>group I metabotropic glutamate receptor antagonist and group II mGlu agonist</p>Fórmula:C9H9NO5Pureza:98%Cor e Forma:SolidPeso molecular:211.17TAS-4
CAS:<p>TAS-4 is a modulator of metabotropic glutamate receptor 4-positive allosteric.</p>Fórmula:C12H8Cl2N2OPureza:98%Cor e Forma:SolidPeso molecular:267.11Hydroflumethiazide
CAS:<p>Hydroflumethiazide is a thiazide diuretic. It has also shown the activity of anti-hypertensive.</p>Fórmula:C8H8F3N3O4S2Cor e Forma:Crystals SolidPeso molecular:331.29Lombazole
CAS:<p>Lombazole is an antimicrobial agent in the class of imidazole.</p>Fórmula:C22H17ClN2Cor e Forma:SolidPeso molecular:344.84Aladorian
CAS:<p>Aladorian (ARM036), a benzothiazepine, has anti-arrhythmic properties for heart failure and CPVT research.</p>Fórmula:C12H13NO4SPureza:98%Cor e Forma:SolidPeso molecular:267.3Arginylproline
CAS:<p>Arginylproline is a dipeptide composed of arginine and proline. It is an incomplete breakdown product of protein digestion or protein catabolism.</p>Fórmula:C11H21N5O3Cor e Forma:SolidPeso molecular:271.32Ro 8-4304
CAS:<p>Ro 8-4304 Hydrochloride is an antagonist of NMDA receptor with IC50 of 0.4 μM</p>Fórmula:C21H23FN2O3Pureza:98%Cor e Forma:SolidPeso molecular:370.42CS476
CAS:<p>CS476 is a potent drug of hypoglycaemic.</p>Fórmula:C24H29N3O5SPureza:98%Cor e Forma:SolidPeso molecular:471.57Fluzinamide
CAS:<p>Fluzinamide (AHR-8559) has anticonvulsant effects on ignited amygdala seizures.</p>Fórmula:C12H13F3N2O2Pureza:99.38% - >99.99%Cor e Forma:SolidPeso molecular:274.24Laurinterol
CAS:<p>Laurinterol is an antimicrobial from the marine alga Laurencia okamurai.</p>Fórmula:C15H19BrOCor e Forma:SolidPeso molecular:295.21BRL 55834
CAS:<p>BRL 55834, a potassium channel activator, has shown to relax airways and vasculature in vivo.</p>Fórmula:C18H20F5NO3Pureza:98%Cor e Forma:SolidPeso molecular:393.35S-312-d
CAS:<p>S-312d is a calcium channel antagonist. S-312-d can offer marked neuronal protective effects against ischemic injury.</p>Fórmula:C20H22N2O4SPureza:98%Cor e Forma:SolidPeso molecular:386.46Niguldipine Free Base
CAS:<p>Niguldipine Free Base is a calcium channel blocker and a₁-adrenergic receptor antagonist and a clinical modulator of multidrug resistance.</p>Fórmula:C36H39N3O6Pureza:98.97%Cor e Forma:SolidPeso molecular:609.71CGP 28392
CAS:<p>CGP 28392 is used as a partial calcium channel agonist.</p>Fórmula:C18H17F2NO5Pureza:98%Cor e Forma:SolidPeso molecular:365.33RH01617
CAS:<p>RH01617 possesses potent inhibitory activities against Kv1.5.</p>Fórmula:C22H26N2O5SPureza:98%Cor e Forma:SolidPeso molecular:430.52Glypromate
CAS:<p>Glypromate (Gly-Pro-Glu) is a neuroprotective agent, is a weak NMDA receptor agonist</p>Fórmula:C12H19N3O6Pureza:98%Cor e Forma:SolidPeso molecular:301.3SR57227A
CAS:<p>SR 57227A: Selective 5-HT3 receptor inhibitor, affects NMDA responses, has anti-depressant effects and reduces aggression in rats.</p>Fórmula:C10H14ClN3Pureza:98%Cor e Forma:SolidPeso molecular:211.69PNU-107484A
CAS:<p>PNU-107484A is a unique GABA(A) receptor ligand.</p>Fórmula:C18H23ClN6Pureza:98%Cor e Forma:SolidPeso molecular:358.87Dicirenone
CAS:<p>Dicirenone (SC26304) inhibits the Mineralocorticoid receptor (MR), aldosterone regulation of the urinary K+:Na+ ratio, and aldosterone binding to renal</p>Fórmula:C26H36O5Pureza:99.1%Cor e Forma:SolidPeso molecular:428.56Guanosine 5'-diphosphate ditromethamine
CAS:Guanosine 5'-diphosphate ditromethamine (GDP ditromethamine) is a nucleoside diphosphate that activates ATP-sensitive K+ channels. It acts as a potential iron mobilizer, inhibiting the interaction between hepcidin and ferroportin, and modulating the IL-6/STAT-3 pathway. This compound finds application in inflammation research, such as studying anemia of inflammation (AI).Fórmula:C18H37N7O17P2Peso molecular:685.47GSK1702934A
CAS:<p>GSK1702934A is a TRPC3 agonist with pro-arrhythmic and positive inotropic effects and is used in the study of diabetes mellitus.</p>Fórmula:C22H25N3O2SPureza:98.15%Cor e Forma:SolidPeso molecular:395.52N-Oleoyl Valine
CAS:N-Oleoyl valine, an N-acyl amine, antagonizes TRPV3 for thermoregulation; rises post-cold exposure; elevates in mouse lung injury.Fórmula:C23H43NO3Peso molecular:381.59GS 39783
CAS:<p>GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement and</p>Fórmula:C15H23N5O2SPureza:99.92%Cor e Forma:SolidPeso molecular:337.44SM-6586
CAS:<p>SM-6586 is a potent calcium channel antagonist with inhibitory effects on Na+/H+ and Na+/Ca2+ exchange channels, and can be used in the study of cerebrovascular</p>Fórmula:C26H27N5O5Pureza:99.43%Cor e Forma:SolidPeso molecular:489.52(5R)-BW-4030W92
CAS:<p>(5R)-BW-4030W92 is the R-type of BW-4030W92, the active enantiomer.</p>Fórmula:C11H9Cl2FN4Pureza:98.27%Cor e Forma:SolidPeso molecular:287.12AM12
CAS:<p>AM12 inhibits Lanthanide-evoked TRPC5 activity (IC50: 0.28 μM).</p>Fórmula:C15H9BrO5Pureza:98%Cor e Forma:SolidPeso molecular:349.13ML402
CAS:<p>ML402 (ZINC3671497) is an activator of TREK-1 and TREK-2 with EC50s of 13.7 μM and 5.9 μM.</p>Fórmula:C14H14ClNO2SPureza:99.71%Cor e Forma:SolidPeso molecular:295.78Zatebradine hydrochloride
CAS:<p>Zatebradine hydrochloride (UL-FS-49CL) inhibits HCN channels (IC50: ~1.9 µM) blocking human HCN1-4 currents effectively.</p>Fórmula:C26H37ClN2O5Pureza:97%Cor e Forma:SolidPeso molecular:493.04Cyclic ADP-ribose
CAS:<p>cADPR, made from NAD+, boosts calcium in cells via Ryanodine receptors and TRPM2 channels.</p>Fórmula:C15H21N5O13P2Pureza:98%Cor e Forma:Lyophilized PowderPeso molecular:541.3Bifenazate
CAS:<p>Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.</p>Fórmula:C17H20N2O3Pureza:99.62%Cor e Forma:Solid CrystallinePeso molecular:300.35BMS-919373
CAS:<p>BMS-919373 is a potassium channel Kv1.5 (KCNA5) inhibitor for atrial fibrillation and acute coronary syndrome.</p>Fórmula:C25H20N6O2SPureza:98.51% - 99.01%Cor e Forma:SolidPeso molecular:468.53McN5691
CAS:<p>McN5691 is a voltage sensitive calcium channel blocker.</p>Fórmula:C30H35NO3Pureza:98.93% - 99.38%Cor e Forma:SolidPeso molecular:457.6Levosemotiadil
CAS:<p>Levosemotiadil(SA 3212) is a novel calcium antagonist and a very potent inhibitor of low-density lipoprotein oxidation.Levosemotiadil may be used to prevent</p>Fórmula:C29H32N2O6SPureza:98.53% - 99.47%Cor e Forma:SolidPeso molecular:536.64(R)-Baclofen hydrochloride
CAS:<p>Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.</p>Fórmula:C10H13Cl2NO2Pureza:98%Cor e Forma:SolidPeso molecular:250.12Vernakalant
CAS:<p>Vernakalant (RSD-1235) is a mixed ion channel blocker.</p>Fórmula:C20H31NO4Pureza:98%Cor e Forma:SolidPeso molecular:349.46Amsacrine
CAS:<p>Amsacrine (AMSA) (mAMSA) an antineoplastic agent which can intercalate into the DNA of tumor cells.</p>Fórmula:C21H19N3O3SPureza:99.2%Cor e Forma:Yellow Crystalline Powder SolidPeso molecular:393.46SCH 50911
CAS:<p>SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.</p>Fórmula:C8H15NO3Pureza:98%Cor e Forma:SolidPeso molecular:173.21Phenamil
CAS:<p>Phenamil is an inhibitor of epithelial sodium channels, activates the osteomorphin protein pathway to promote bone repair and induces significant fat formation.</p>Fórmula:C12H12ClN7OPureza:99.07%Cor e Forma:SolidPeso molecular:305.72B-TPMF
CAS:<p>B-TPMF is a highly efficient and selective KCa2.1 channel inhibitor with an IC50 of 31 nM, interacting with serine residue at position 293 to inhibit KCa2.1.</p>Fórmula:C19H24N6O2Pureza:99.82%Cor e Forma:SolidPeso molecular:368.43CM-TPMF
CAS:<p>CM-TPMF is a highly efficient and potent activator of the K(Ca)2.1 channel, Ser293 in the transmembrane segment 5, neurological disorders.</p>Fórmula:C16H17ClN6O2Pureza:99.94%Cor e Forma:SolidPeso molecular:360.8TTA-Q6
CAS:<p>TTA-Q6 is a T-type Ca2+ channel antagonist that inhibits the uptake of extracellular calcium ions by tumour cells for the treatment of neurological diseases.</p>Fórmula:C20H15ClF3N3OPureza:99.97%Cor e Forma:SolidPeso molecular:405.818:0 LYSO-PE
CAS:<p>18:0 LYSO-PE is a compound that induces an increase in [Ca2+]i and can be used as a phospholipid (PL) standard for lipid analysis by electrospray mass spectrometry (ESI-MS)/MS.</p>Fórmula:C23H48NO7PPureza:98%Cor e Forma:SolidPeso molecular:481.6ABCG2-IN-1
CAS:<p>ABCG2-IN-1 (compound K2), an analog of Ko143, constitutes an orally active inhibitor targeting ABCG2 with an inhibitory concentration (IC50) of 0.13 μM.</p>Fórmula:C26H36N4O4Pureza:98%Cor e Forma:SolidPeso molecular:468.59E2730
CAS:<p>E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.</p>Fórmula:C9H8F4N2O2SPureza:98.22% - 98.54%Cor e Forma:SolidPeso molecular:284.23TWIK-1/TREK-1-IN-2
CAS:<p>TWIK-1/TREK-1-IN-2 (Compound 2g) serves as an inhibitor of both TWIK-1 and TREK-1, targeting the TREK-1 homodimer and TWIK-1/TREK-1 heterodimer with IC50 values</p>Fórmula:C20H29F3N2O2Pureza:98%Cor e Forma:SolidPeso molecular:386.45ABCG2-IN-2
CAS:<p>ABCG2-IN-2 is a potent inhibitor of ABCG2, exhibiting favorable oral pharmacokinetic profiles in mice, and is applicable for investigating tumor multidrug</p>Fórmula:C25H34N4O4Pureza:98%Cor e Forma:SolidPeso molecular:454.56U-89843A
CAS:<p>U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].</p>Fórmula:C16H24ClN5Pureza:98%Cor e Forma:SolidPeso molecular:321.85TWIK-1/TREK-1-IN-1
CAS:<p>Compound 2a, identified as TWIK-1/TREK-1-IN-1, acts as an inhibitor of the TREK-1, a two-pore domain potassium channel (K2p) that forms TREK-1 homodimers and</p>Fórmula:C21H24F3NO3Pureza:98%Cor e Forma:SolidPeso molecular:395.42D-3263 hydrochloride
CAS:<p>D-3263 hydrochloride (D3263 HCl salt) is enteric-coated, orally bioavailable transient receptor potential melatonin member 8 (TRPM8) agonist.</p>Fórmula:C21H32ClN3O3Pureza:99.93%Cor e Forma:SolidPeso molecular:409.95Vernakalant Hydrochloride
CAS:<p>Vernakalant Hydrochloride (RSD1235 hydrochloride) is a mixed voltage- and frequency-dependent Na+ and atria-preferred K+ channel blocker.</p>Fórmula:C20H32ClNO4Pureza:99.89%Cor e Forma:SolidPeso molecular:385.93YHO-13351 free base
CAS:<p>YHO-13351 free base is the water-soluble prodrug of YHO-13177 which is an inhibitor of BCRP .</p>Fórmula:C26H33N3O4SPureza:99.89%Cor e Forma:SolidPeso molecular:483.62Pinacidil
CAS:<p>Pinacidil (P 1134) is a guanidine that opens potassium channels and directly dilates peripheral blood vessels in small arteries, lowering blood pressure and</p>Fórmula:C13H19N5Pureza:99.9%Cor e Forma:SolidPeso molecular:245.32TRPV4 agonist-1
CAS:<p>TRPV4 agonist-1 is an agonist of TRPV4 (EC50: 60 nM in the hTRPV4 Ca2+ assay).</p>Fórmula:C25H23ClF2N4O2Pureza:98%Cor e Forma:SolidPeso molecular:484.93PF 05089771 tosylate
CAS:<p>PF-05089771 inhibits Nav1.7 channels (IC50: 11-33 nM), selective over Nav1.1-1.6/1.8, Ca+, K+ channels, TRPV1; 1000x affinity for half-inactivated state.</p>Fórmula:C18H12Cl2FN5O3S2·C7H8O3SPureza:98.55%Cor e Forma:SolidPeso molecular:672.56Lesogaberan
CAS:<p>Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).</p>Fórmula:C3H9FNO2PPureza:98%Cor e Forma:SolidPeso molecular:141.08UK 78282 hydrochloride
CAS:<p>UK-78282 hydrochloride, a Kv1.3 blocker.UK-78282 hydrochloride inhibits Kv1.3 voltage-gated potassium channels and suppresses human T cell activation.</p>Fórmula:C29H36ClNO2Pureza:99.68%Cor e Forma:SolidPeso molecular:466.05Puliginurad
CAS:<p>Puliginurad (YL-90148) is a urate transporter protein inhibitor that inhibits the reabsorption of uric acid.Puliginurad is used in the treatment of gout.</p>Fórmula:C19H16N2O2SPureza:99.96% - 99.96%Cor e Forma:SolidPeso molecular:336.41GX-674
CAS:<p>GX-674 is a highly potent and selective voltage-gated sodium channel 1.7 (Nav1.7) antagonist with an IC50 value of 0.1 nM measured at -40 mV for the study of</p>Fórmula:C21H13ClF2N6O3S2Pureza:98.60%Cor e Forma:SolidPeso molecular:534.95TRAM 39
CAS:<p>TRAM 39 (2-Chloro-α,α-diphenylbenzeneacetonitrile) is a selective blocker of intermediate-conductance Ca2+-activated K+channels.</p>Fórmula:C20H14ClNPureza:99.97%Cor e Forma:SolidPeso molecular:303.78Tracazolate hydrochloride
CAS:<p>Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.</p>Fórmula:C16H25ClN4O2Pureza:99.52%Cor e Forma:SolidPeso molecular:340.85TRPM4-IN-2
CAS:<p>NBA, or TRPM4-IN-2, is a potent TRPM4 inhibitor with IC50 of 0.16 μM, used in prostate and colorectal cancer research.</p>Fórmula:C19H14ClNO4Pureza:99.21%Cor e Forma:SolidPeso molecular:355.77RO 4938581
CAS:<p>RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).</p>Fórmula:C13H8BrF2N5Pureza:98%Cor e Forma:SolidPeso molecular:352.14JYL 1421
CAS:<p>JYL 1421 (SC 0030) is an antagonist of TRPV1 receptor (IC50 = 8 nM).</p>Fórmula:C20H26FN3O2S2Pureza:98.83%Cor e Forma:SolidPeso molecular:423.57GDC-0276
CAS:<p>GDC-0276 is an orally active, selective, and potent NaV1.7 inhibitor that can be used for the study of pain-related diseases.</p>Fórmula:C24H31FN2O4SPureza:99.77%Cor e Forma:SolidPeso molecular:462.58RY796
CAS:<p>RY796 is a selective voltage-gated potassium (KV2) channel inhibitor that inhibits KV2.1 and KV2.2, used in research on neurological disorders.</p>Fórmula:C21H27N3O2Pureza:98.59%Cor e Forma:SolidPeso molecular:353.46RN9893
CAS:<p>RN9893 is a selective and potent TRPV4 receptor antagonist with IC50 values of 320, 420 and 660 nM for TRPV4 receptors in mouse, human and rat, respectively.</p>Fórmula:C21H23F3N4O5SPureza:99.89%Cor e Forma:SolidPeso molecular:500.49ATX-II TFA
<p>ATX-II TFA, a specific Na+ channel modulator toxin, is derived from the venom of the sea anemone (Anemonia sulcata).</p>Pureza:98%Cor e Forma:Odour SolidAZD 3043
CAS:<p>AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.</p>Fórmula:C19H29NO5Pureza:98.19% - 99.55%Cor e Forma:SolidPeso molecular:351.44E 0747
CAS:<p>E 0747 is an antiarrhythmic agent of class 1C type. E-0747 suppresses arrhythmia by inhibiting the Na channels of cardiac cells.</p>Fórmula:C21H28ClN3O4Pureza:95.17%Cor e Forma:SolidPeso molecular:421.92TRPV3 antagonist 74a
CAS:<p>TRPV3 antagonist 74a (TRPV3 74a) is a specific TRPV3 antagonist for the study of neurological disorders.</p>Fórmula:C17H17F3N2O2Pureza:≥98.0%Cor e Forma:SolidPeso molecular:338.32AVE1231
CAS:<p>AVE1231 is a TASK-1 channel blocker that inhibits TASK-1 and can be used in the study of atrial fibrillation.</p>Fórmula:C20H27N3O4SPureza:98.03%Cor e Forma:SolidPeso molecular:405.51Phaclofen
CAS:<p>GABAB antagonist</p>Fórmula:C9H13ClNO3PPureza:99.32%Cor e Forma:White SolidPeso molecular:249.63GAL-021 sulfate
CAS:<p>GAL-021 sulfate is a BKCa channel blocker that inhibits the analgesic effects of opioids and is used in the study of respiratory control diseases.</p>Fórmula:C11H24N6O5SPureza:99.92%Cor e Forma:SolidPeso molecular:352.41Istaroxime hydrochloride
CAS:<p>Istaroxime hydrochloride (PST2744 hydrochloride) is a Na+/K+-ATPase inhibitor and SERCA 2 activator, and is a novel positive inotropic compound.</p>Fórmula:C21H33ClN2O3Cor e Forma:SolidPeso molecular:396.95GX-585
CAS:<p>GX-585 is a novel potent inhibitor of NaV1.7 and highly selective against NaV1.5, having limited selectivity against NaV1.1 and NaV1.2.</p>Fórmula:C24H25Cl2FN4O3SPureza:99.02% - 99.03%Cor e Forma:SolidPeso molecular:539.45SRI-37240
CAS:<p>SRI-37240 suppresses CFTR nonsense mutations, aids in fixing premature termination codons, works with G418.</p>Fórmula:C24H23N3O2Pureza:98.73%Cor e Forma:SolidPeso molecular:385.46Aprikalim
CAS:<p>Aprikalim opens KATP channels, protects the heart, and at high doses, dilates blood vessels.</p>Fórmula:C12H16N2OS2Pureza:99.42% - 99.90%Cor e Forma:SolidPeso molecular:268.4Suriclone
CAS:<p>Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.</p>Fórmula:C20H20ClN5O3S2Pureza:99.21% - 99.73%Cor e Forma:SolidPeso molecular:477.99KT-362 fumarate
CAS:<p>KT-362 fumarate, a novel antagonist of Ca, K, and Na channels, induces vasodilation and relaxes rabbit arterial strips.</p>Fórmula:C26H32N2O7SPureza:99.75% - 99.98%Cor e Forma:SolidPeso molecular:516.61AGN-201904
CAS:AGN-201904 is a proton pump inhibitor, an omeprazole prodrug, which delays aging and may be used for the prevention and treatment of peptic ulcers.Fórmula:C25H25N3O8S2Pureza:97.32%Cor e Forma:SolidPeso molecular:559.61DMT1 blocker 1
CAS:<p>DMT1 blocker 1 inhibits DMT1; IC50=0.64μM; may prevent intestinal iron absorption.</p>Fórmula:C16H14N4O2Pureza:99.73%Cor e Forma:SolidPeso molecular:294.31Trombodipine
CAS:<p>Trombodipine (PCA-4230) is a platelet aggregation inhibitor with antithrombotic activity and protection against Listeria monocytogenes.</p>Fórmula:C21H24N2O7SPureza:98.73% - 99.14%Cor e Forma:SolidPeso molecular:448.49Elismetrep
CAS:<p>Elismetrep (MT-8554) is an orally available TRPM8 inhibitor with potential analgesic activity for the study of vasomotor symptoms in postmenopausal women.</p>Fórmula:C27H21F3N2O5SPureza:99.37% - 99.93%Cor e Forma:SolidPeso molecular:542.53R 56865
CAS:<p>R 56865 is a weak potential-operated channel inhibitor that inhibits the late sodium current in human isolated cardiomyocytes.</p>Fórmula:C23H28FN3OSPureza:99.52%Cor e Forma:SolidPeso molecular:413.55Riluzole hydrochloride
CAS:<p>Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).</p>Fórmula:C8H6ClF3N2OSPureza:99.76%Cor e Forma:SolidPeso molecular:270.66SKF96067
CAS:<p>SKF96067 is a reversible gastric H+/K+-ATPase inhibitor that can induce relaxation of human airway smooth muscle in vitro.</p>Fórmula:C21H22N2O2Pureza:99.89%Cor e Forma:SolidPeso molecular:334.41Losigamone
CAS:<p>Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about the treatment of partial seizures.</p>Fórmula:C12H11ClO4Pureza:99.98%Cor e Forma:SolidPeso molecular:254.67TASK-1-IN-1
CAS:<p>TASK-1-IN-1: Potent, selective TASK-1 blocker (IC50: 148 nM), weaker on TASK-3 (IC50: 1750 nM), anticancer properties.</p>Fórmula:C22H20N2O2Pureza:99.57%Cor e Forma:SoildPeso molecular:344.41Nerisopam
CAS:<p>Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.</p>Fórmula:C18H19N3O2Pureza:97.07%Cor e Forma:SolidPeso molecular:309.36Fengabine
CAS:<p>Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.</p>Fórmula:C17H17Cl2NOPureza:99%Cor e Forma:SolidPeso molecular:322.23TAK-653
CAS:<p>TAK-653 is a selective AMPA receptor PAM with minimal agonist activity, showing antidepressant-like effects and safety in rats.</p>Fórmula:C19H23N3O3SPureza:99.89%Cor e Forma:SolidPeso molecular:373.47Neboglamine hydrochloride
CAS:<p>Neboglamine (CR-2249, XY-2401) hydrochloride boosts NMDA receptor, aids schizophrenia research, and is orally active.</p>Fórmula:C13H25ClN2O3Pureza:99.19%Cor e Forma:SolidPeso molecular:292.8DSP-0565
CAS:<p>DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.</p>Fórmula:C14H12FNOPureza:99.51% - 99.56%Cor e Forma:SolidPeso molecular:229.25Alpidem
CAS:<p>Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.</p>Fórmula:C21H23Cl2N3OPureza:99.56% - 99.97%Cor e Forma:White To Off-White SolidPeso molecular:404.33Muscimol HBr
CAS:<p>Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.</p>Fórmula:C4H7BrN2O2Pureza:98.13%Cor e Forma:Off-White PowderPeso molecular:195.01

