Transportador de Membranas/Canal Iónico
Os inibidores de transportadores de membrana e canais iônicos são compostos que bloqueiam a função de proteínas responsáveis pelo transporte de íons, nutrientes e outras moléculas através das membranas celulares. Esses inibidores são cruciais para o estudo da regulação da homeostase celular, transdução de sinais e neurotransmissão. Os inibidores de transportadores de membrana e canais iônicos também são importantes no desenvolvimento de tratamentos para distúrbios como epilepsia, doenças cardiovasculares e síndromes metabólicas. Na CymitQuimica, oferecemos uma ampla seleção de inibidores de alta qualidade de transportadores de membrana e canais iônicos para apoiar sua pesquisa em fisiologia, neurociência e farmacologia.
Subcategorias de "Transportador de Membranas/Canal Iónico"
- ABC(3 produtos)
- ATPase(93 produtos)
- Receptor de adiponectina(5 produtos)
- CFTR(64 produtos)
- Receptor CGRP(52 produtos)
- Canais de Cálcio(496 produtos)
- Canal de cloreto(49 produtos)
- Receptor GABA(337 produtos)
- Transportador de monoamina(23 produtos)
- Transportador de monocarboxilato(17 produtos)
- NKCC(2 produtos)
- NPC1L1(3 produtos)
- Cotransportador Na-K-Cl(8 produtos)
- OAT(27 produtos)
- OCT(7 produtos)
- P-gp(53 produtos)
- Canal de Potássio(277 produtos)
- Bomba de prótons(39 produtos)
- SGLT(30 produtos)
- Canal de Sódio(202 produtos)
- Canal TRP/TRPV(93 produtos)
Exibir 13 mais subcategorias
Foram encontrados 2293 produtos de "Transportador de Membranas/Canal Iónico"
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Quadrol
CAS:<p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>Fórmula:C14H32N2O4Pureza:99.91% - 99.92%Cor e Forma:Viscous Liquid Liquid ViscousPeso molecular:292.41Parimifasor
CAS:<p>Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.</p>Fórmula:C18H11Cl2F4N5OPureza:96.77% - 98.97%Cor e Forma:SolidPeso molecular:460.21TKIM
CAS:<p>TKIM is a TWIK-related potassium channel 1 (TREK-1) inhibitor, binding to the pocket of the intermediate (IM) state of TREK-1.</p>Fórmula:C18H14ClN3O2SPureza:99.47%Cor e Forma:SolidPeso molecular:371.84Budipine
CAS:Budipine is a low affinity, N-methyl-D-aspartate receptor antagonist,is an antiparkinsonian agent.Fórmula:C21H27NPureza:99.64%Cor e Forma:SolidPeso molecular:293.45Guan-fu base A hydrochloride(1394-48-5 free base)
CAS:<p>Guanfu base A HCl, an antiarrhythmic from Aconitum coreanum, inhibits CYP2D6 in humans, monkeys, and dogs.</p>Fórmula:C24H32NO6ClPureza:99.9%Cor e Forma:SolidPeso molecular:465.972'-O-Methylisoliquiritigenin
CAS:<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Fórmula:C16H14O4Pureza:98.75%Cor e Forma:SolidPeso molecular:270.28Cis-ACBD
CAS:<p>Cis-ACBD (cis-1-aminocyclobutane-1,3-dicarboxylic acid) is a potent and selective N-methyl-D-aspartate receptor agonist.</p>Fórmula:C6H9NO4Pureza:99.77%Cor e Forma:SolidPeso molecular:159.14DL-Willardiine
CAS:<p>DL-Willardiine (2-amino-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoic acid) is an unnatural amino acid, a derivative of glutamate.</p>Fórmula:C7H9N3O4Pureza:99.83%Cor e Forma:SolidPeso molecular:199.16Esomeprazole Magnesium
CAS:<p>Esomeprazole Magnesium (NEXIUM) is the S-isomer of omeprazole, can reduce gastric acid secretion with selective and irreversible proton pump inhibitor activity.</p>Fórmula:C34H36MgN6O6S2Pureza:98.76% - 99.73%Cor e Forma:SolidPeso molecular:713.12Eperisone hydrochloride
CAS:<p>Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.</p>Fórmula:C17H26ClNOPureza:99.80%Cor e Forma:White Or Similar To White Crystalline Powder With Peculiar Smell And Bitter TastePeso molecular:295.85AER-271
CAS:<p>AER-271 is an inhibitor of aquaporin-4.</p>Fórmula:C15H9ClF6NO5PPureza:97.45%Cor e Forma:SolidPeso molecular:463.65Ibutilide
CAS:<p>Ibutilide (U70226E) is an antiarrhythmic that prolongs action potential by blocking I Kr in AT-1 cells.</p>Fórmula:C20H36N2O3SCor e Forma:SolidPeso molecular:384.58A2793
CAS:<p>A2793 is a dual inhibitor of TWIK-associated acid-sensitive K+ channel 1 (TASK-1)/TRESK, with an IC50 for mTRESK of 6.8 μM.</p>Fórmula:C13H12ClNO3Pureza:98.54%Cor e Forma:SolidPeso molecular:265.69Pilsicainide
CAS:<p>Pilsicainide (SUN 1165 free acid) is a potent class Ic antiarrhythmic agent. Pilsicainide is a potent sodium channel blocker[1][2].</p>Fórmula:C17H24N2OCor e Forma:SolidPeso molecular:272.39Ilaprazole sodium
CAS:<p>Ilaprazole sodium (IY-81149 sodium) , a substituted benzimidazole prodrug, is a selective and irreversible proton pump inhibitor.</p>Fórmula:C19H17N4NaO2SPureza:99.06%Cor e Forma:SolidPeso molecular:388.42Mitiglinide calcium hydrate
CAS:<p>Mitiglinide calcium hydrate (S-21403 calcium hydrate) is a drug for the treatment of type 2 diabetes.</p>Fórmula:C38H52CaN2O8Pureza:98.97% - 99.96%Cor e Forma:White SolidPeso molecular:704.91Tiagabine
CAS:<p>Tiagabine (NO050328) is an Anti-epileptic Agent.</p>Fórmula:C20H25NO2S2Pureza:99.25%Cor e Forma:White To Off-White Crystalline SolidPeso molecular:375.55Ocinaplon
CAS:<p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>Fórmula:C17H11N5OPureza:99.81%Cor e Forma:SolidPeso molecular:301.37-Chlorokynurenic acid sodium salt
CAS:<p>7-CKA sodium salt: NMDA receptor antagonist, glycine B site (IC50: 0.56 μM), blocks glutamate reuptake (Ki: 0.59 μM).</p>Fórmula:C10H6ClNNaO3Cor e Forma:SolidPeso molecular:246.6(-)-Blebbistatin
CAS:<p>(-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin II inhibitor with IC50 ranging from 0.5 to 5 μM.</p>Fórmula:C18H16N2O2Pureza:99.38% - 99.61%Cor e Forma:SolidPeso molecular:292.33Metaflumizone
CAS:<p>Metaflumizone (BAS-320I) is a sodium channel blocker insecticide.</p>Fórmula:C24H16F6N4O2Pureza:98.73%Cor e Forma:SolidPeso molecular:506.40LY 303511 hydrochloride
CAS:<p>LY 303511 hydrochloride is a potent mTOR inhibitor</p>Fórmula:C19H19ClN2O2Pureza:98.47%Cor e Forma:SolidPeso molecular:342.82NBI-98782
CAS:<p>NBI-98782 ((+)-α-DHTBZ) is an inhibtior of vesicular monoamine transporter (VMAT2) (Ki: 0.97 nM)</p>Fórmula:C19H29NO3Pureza:99.29%Cor e Forma:SolidPeso molecular:319.44SG-209
CAS:<p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>Fórmula:C10H12N2O3Pureza:99.84%Cor e Forma:SolidPeso molecular:208.21Ropivacaine hydrochloride monohydrate
CAS:<p>Ropivacaine hydrochloride monohydrate (LEA-103 HCl) is an anaesthetic agent and blocks impulse conduction through inhibiting sodium ion influx reversibly.</p>Fórmula:C17H29ClN2O2Pureza:99.94% - 99.95%Cor e Forma:White SolidPeso molecular:328.88Arecaidine hydrochloride
CAS:Arecaidine hydrochloride may have carcinogenesis.Fórmula:C7H12ClNO2Pureza:99.69% - ≥95%Cor e Forma:SolidPeso molecular:177.63AZ194
CAS:<p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>Fórmula:C34H31F2N3O3Pureza:99.61%Cor e Forma:SolidPeso molecular:567.62Neboglamine
CAS:<p>Neboglamine, a glycine NMDA-associated agonist, is used potentially for the treatment of schizophrenia.</p>Fórmula:C13H24N2O3Pureza:98%Cor e Forma:SolidPeso molecular:256.34Lansoprazole sulfone
CAS:<p>Lansoprazole sulfone is a metabolite of the gastric pump inhibitor Lansoprazole.</p>Fórmula:C16H14F3N3O3SPureza:99.67%Cor e Forma:SolidPeso molecular:385.36Ralfinamide mesylate
CAS:<p>Ralfinamide mesylate (FCE-26742A (mesylate)) is an orally available Na+ channel blocker.</p>Fórmula:C18H23FN2O5SPureza:99.83%Cor e Forma:SolidPeso molecular:398.45DAAO inhibitor-1
CAS:<p>DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor (IC50: 0.12 μM).</p>Fórmula:C7H5FN2OPureza:97.84%Cor e Forma:SolidPeso molecular:152.13MDR-652
CAS:<p>MDR-652 is a highly specific and efficacious agonist of nonpungent transient receptor potential vanilloid 1 (TRPV1) with Ki value of 11.4 nM and 23.8 nM for</p>Fórmula:C22H23ClFN3O2SPureza:99.96%Cor e Forma:SolidPeso molecular:447.95Kv2-IN-A1
CAS:<p>Kv2-IN-A1 is an inhibitor of Kv2.1 and Kv2.2.</p>Fórmula:C20H17ClN4OSPureza:98.83%Cor e Forma:SolidPeso molecular:396.89Esomeprazole hemistrontium
CAS:<p>Esomeprazole hemistrontium, potent oral proton pump inhibitor, reduces gastric acid by blocking H+, K+-ATPase.</p>Fórmula:C34H36N6O6S2SrCor e Forma:SolidPeso molecular:776.44Adjudin
CAS:<p>Adjudin (AF-2364) is a small molecule compound known to possess antispermatogenic function, attenuates microglia activation by suppression of the NF-κB pathway.</p>Fórmula:C15H12Cl2N4OPureza:96.51% - ≥95%Cor e Forma:SolidPeso molecular:335.19Almitrine mesylate
CAS:<p>Almitrine mesylate targets Ca2+-dependent K+ channels in rat cells, used for chronic lung hypoxemia.</p>Fórmula:C28H37F2N7O6S2Pureza:99.96%Cor e Forma:CoaPeso molecular:669.76Miltirone
CAS:<p>Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.</p>Fórmula:C19H22O2Pureza:99.22% - 99.66%Cor e Forma:SolidPeso molecular:282.38WS-12
CAS:WS-12 is a potent TRPM8 agonist that acts as a cooling agent (EC50 : 193 nM)Fórmula:C18H27NO2Pureza:99.99%Cor e Forma:Whitish To White Solid CrystallinePeso molecular:289.41α-Asarone
CAS:<p>alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.</p>Fórmula:C12H16O3Pureza:99.64% - 99.64%Cor e Forma:Monoclinic Needles From Water Monoclinic Needles From WaterPeso molecular:208.254-Acetamidobutanoic acid
CAS:<p>4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.</p>Fórmula:C6H11NO3Pureza:98.51%Cor e Forma:SolidPeso molecular:145.16Baclofen hydrochloride
CAS:Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.Fórmula:C10H13Cl2NO2Pureza:99.55%Cor e Forma:SolidPeso molecular:250.122Raxatrigine hydrochloride
CAS:Raxatrigine hydrochloride is a state-dependent sodium channel blocker and a Nav1.7 sodium channel inhibitor.Fórmula:C18H20ClFN2O2Pureza:98%Cor e Forma:SolidPeso molecular:350.82Ataluren
CAS:<p>Ataluren (PTC124) is a novel, orally administered drug that targets nonsense mutations.</p>Fórmula:C15H9FN2O3Pureza:99.16% - 99.84%Cor e Forma:SolidPeso molecular:284.24Cyclothiazide
CAS:<p>Cyclothiazide enhances AMPA receptors, prevents desensitization, and boosts glutamic acid response (EC50 = 3.8µM).</p>Fórmula:C14H16ClN3O4S2Pureza:98.23% - 99.49%Cor e Forma:Crystals From Dilute Alcohol SolidPeso molecular:389.88Flecainide hydrochloride
CAS:<p>Flecainide is a medication used to prevent and treat abnormally fast heart rates. This includes ventricular and supraventricular tachycardias.</p>Fórmula:C17H21ClF6N2O3Pureza:97.79%Cor e Forma:SolidPeso molecular:450.81PF-05186462
CAS:<p>PF-05186462 (PF-05150122) is a potent, state-dependent, subtype selective Nav1.7 inhibitor with IC50 of 21 nM, no significant activity against Nav1.5.</p>Fórmula:C19H10ClF4N5O3S2Pureza:99.10% - 99.37%Cor e Forma:SolidPeso molecular:531.89Guanosine 5'-diphosphate disodium salt
CAS:<p>5'-GDP-Na2: a nucleoside diphosphate, iron mobilizer, blocks hepcidin-ferroportin, affects IL-6/stat-3.</p>Fórmula:C10H13N5Na2O11P2Pureza:99.40%Cor e Forma:White PowderPeso molecular:487.16Trofinetide
CAS:Trofinetide (NNZ-2566) is a synthetic analog of the endogenous N-terminus tripeptide. It has been shown to be neuroprotective in animal models of brain injury.Fórmula:C13H21N3O6Pureza:98.70% - 99.50%Cor e Forma:SolidPeso molecular:315.326-Methylflavone
CAS:6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.Fórmula:C16H12O2Pureza:99.69%Cor e Forma:SolidPeso molecular:236.27Nateglinide
CAS:<p>Nateglinide is an oral drug for type 2 diabetes, stimulating insulin release; may cause rare acute liver injury.</p>Fórmula:C19H27NO3Pureza:99.93% - 99.94%Cor e Forma:White Crystalline PowderPeso molecular:317.42
