Transportador de Membranas/Canal Iónico
Os inibidores de transportadores de membrana e canais iônicos são compostos que bloqueiam a função de proteínas responsáveis pelo transporte de íons, nutrientes e outras moléculas através das membranas celulares. Esses inibidores são cruciais para o estudo da regulação da homeostase celular, transdução de sinais e neurotransmissão. Os inibidores de transportadores de membrana e canais iônicos também são importantes no desenvolvimento de tratamentos para distúrbios como epilepsia, doenças cardiovasculares e síndromes metabólicas. Na CymitQuimica, oferecemos uma ampla seleção de inibidores de alta qualidade de transportadores de membrana e canais iônicos para apoiar sua pesquisa em fisiologia, neurociência e farmacologia.
Subcategorias de "Transportador de Membranas/Canal Iónico"
- ABC(3 produtos)
- ATPase(93 produtos)
- Receptor de adiponectina(5 produtos)
- CFTR(64 produtos)
- Receptor CGRP(51 produtos)
- Canais de Cálcio(493 produtos)
- Canal de cloreto(49 produtos)
- Receptor GABA(336 produtos)
- Transportador de monoamina(23 produtos)
- Transportador de monocarboxilato(17 produtos)
- NKCC(2 produtos)
- NPC1L1(3 produtos)
- Cotransportador Na-K-Cl(8 produtos)
- OAT(27 produtos)
- OCT(7 produtos)
- P-gp(53 produtos)
- Canal de Potássio(276 produtos)
- Bomba de prótons(39 produtos)
- SGLT(30 produtos)
- Canal de Sódio(202 produtos)
- Canal TRP/TRPV(93 produtos)
Exibir 13 mais subcategorias
Foram encontrados 2277 produtos de "Transportador de Membranas/Canal Iónico"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Esomeprazole
CAS:<p>Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis.</p>Fórmula:C17H19N3O3SPureza:97.3%Cor e Forma:SolidPeso molecular:345.42Eperisone hydrochloride
CAS:<p>Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.</p>Fórmula:C17H26ClNOPureza:99.80%Cor e Forma:White Or Similar To White Crystalline Powder With Peculiar Smell And Bitter TastePeso molecular:295.85Epaminurad
CAS:<p>Epaminurad (UR-1102) is an oral URAT1 inhibitor for gout research with a Ki of 0.057 μM, modestly affects OAT1/3.</p>Fórmula:C14H10Br2N2O3Cor e Forma:SolidPeso molecular:414.05ML335
CAS:<p>ML335 is a selective activator of TREK-1 and TREK-2.</p>Fórmula:C15H14Cl2N2O3SPureza:99.73% - 99.79%Cor e Forma:SolidPeso molecular:373.25JNJ-26990990
CAS:<p>"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."</p>Fórmula:C9H10N2O2S2Pureza:97.37%Cor e Forma:SolidPeso molecular:242.32Mitiglinide calcium hydrate
CAS:<p>Mitiglinide calcium hydrate (S-21403 calcium hydrate) is a drug for the treatment of type 2 diabetes.</p>Fórmula:C38H52CaN2O8Pureza:98.97% - 99.96%Cor e Forma:White SolidPeso molecular:704.91Ipidacrine
CAS:<p>Ipidacrine (NIK‐247) (NIK‐247) is an Antidementia Agent</p>Fórmula:C12H16N2Pureza:97.73%Cor e Forma:SolidPeso molecular:188.27AZD-6280
CAS:<p>AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.</p>Fórmula:C20H22N4O3Pureza:98.99%Cor e Forma:SolidPeso molecular:366.41Licarbazepine
CAS:<p>Licarbazepine (10,11-hydroxy-10,11 Dihydrocarbamezer) is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partial</p>Fórmula:C15H14N2O2Pureza:99.11%Cor e Forma:SolidPeso molecular:254.28KCNQ2/3 activator-1
CAS:<p>KCNQ2/3 activator-1 is a Kv7.2/Kv7.3 (KCNQ2/3) potassium channel activator.</p>Fórmula:C23H29FN2OPureza:99.16% - 99.47%Cor e Forma:SolidPeso molecular:368.49Enflurane
CAS:<p>Enflurane (Efrane), a volatile anaesthetic, inhibits Ca2+-activated K+ channels and is used to gauge anesthesia levels in gas chromatography.</p>Fórmula:C3H2ClF5OPureza:99.64%Cor e Forma:Clear Colorless Liquid Ordinary Temperature And Pressure Bp 56 8°C Density 1 50 G Cm-3 At Room Temperature Used As AnPeso molecular:184.49HC-030031
CAS:<p>HC-030031 (TOSLAB 829227) is a potent TRPA1 inhibitor, which antagonizes AITC- and formalin-evoked calcium influx with IC50s of 6.2 and 5.3 μM, respectively.</p>Fórmula:C18H21N5O3Pureza:99.69% - ≥95%Cor e Forma:SolidPeso molecular:355.39UBP710
CAS:<p>UBP710 is an effective and selective NMDA receptor modulator.</p>Fórmula:C18H14O2Pureza:98.05%Cor e Forma:SolidPeso molecular:262.3Tiagabine hydrochloride hydrate
CAS:<p>Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.</p>Fórmula:C20H28ClNO3S2Cor e Forma:SolidPeso molecular:430.02SKF89976A hydrochloride
CAS:<p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>Fórmula:C22H26ClNO2Pureza:98.02%Cor e Forma:SolidPeso molecular:371.9DAAO inhibitor-1
CAS:<p>DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor (IC50: 0.12 μM).</p>Fórmula:C7H5FN2OPureza:97.84%Cor e Forma:SolidPeso molecular:152.13YHO-13177
CAS:<p>YHO-13177 is a potent and specific inhibitor of BCRP; potentiated the cytotoxicity of SN-38 in cancer cells.</p>Fórmula:C20H22N2O3SPureza:98.78%Cor e Forma:SolidPeso molecular:370.47Dihydroergotoxine mesylate
CAS:Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Fórmula:C20H29N3O5SPureza:99.39% - ≥95%Cor e Forma:SolidPeso molecular:423.53Pipequaline hydrochloride
CAS:<p>Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.</p>Fórmula:C22H25ClN2Pureza:99.46%Cor e Forma:SolidPeso molecular:352.9Benzonatate
CAS:<p>Benzonatate is an antagonist of sodium channel protein.</p>Fórmula:C30H53NO11Pureza:99.92%Cor e Forma:Colorless To Faintly Yellow Oil LiquidPeso molecular:603.74Tezacaftor
CAS:<p>Tezacaftor (VX661) is a small molecule that can be used as a corrector of the cystic fibrosis transmembrane conductance regulator (CFTR) gene function.</p>Fórmula:C26H27F3N2O6Pureza:98.84% - >99.99%Cor e Forma:SolidPeso molecular:520.5Aptiganel hydrochloride
CAS:<p>Aptiganel hydrochloride（Cerestat） is the salt form of Aptiganel.Aptiganel is a non-competitive NMDA antagonist with neuroprotective effects used in the treatment of stroke and focal cerebral ischemia.</p>Fórmula:C20H22ClN3Pureza:99.89%Cor e Forma:SolidPeso molecular:339.86Memantine
CAS:<p>Memantine treats moderate to severe Alzheimer's; it's an amantadine derivative blocking NMDA receptors.</p>Fórmula:C12H21NPureza:≥98%Cor e Forma:White PowderPeso molecular:179.3Trans-ACBD
CAS:<p>Trans-ACBD (Trans-1-aminocyclobutane-1,3-dicarboxylic acid) is an effective and specific N-methyl-D-aspartate receptor agonist.</p>Fórmula:C6H9NO4Pureza:99.47%Cor e Forma:SolidPeso molecular:159.14AZ194
CAS:<p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>Fórmula:C34H31F2N3O3Pureza:99.61%Cor e Forma:SolidPeso molecular:567.62AM92016
CAS:<p>AM92016 is a specific blocker of the time dependent delayed rectifier potassium current. AM92016 does not show any β-adrenoceptor blocking activity.</p>Fórmula:C26H30Cl2N2O6SCor e Forma:SolidPeso molecular:569.49SG-209
CAS:<p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>Fórmula:C10H12N2O3Pureza:99.84%Cor e Forma:SolidPeso molecular:208.21Dotinurad
CAS:<p>Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).</p>Fórmula:C14H9Cl2NO4SPureza:97.43% - 98.04%Cor e Forma:SolidPeso molecular:358.2(S)-(-)-5-Fluorowillardiine hydrochloride
CAS:<p>(S)-(-)-5-Fluorowillardiine hydrochloride is a potent and specific agonist of AMPAR.</p>Fórmula:C7H9ClFN3O4Cor e Forma:SolidPeso molecular:253.62GNE-131
CAS:<p>GNE-131 is a potent and specific inhibitor of human sodium channel NaV1.7 (IC50: 3 nM).</p>Fórmula:C23H30N4O3SPureza:98.54% - 99.59%Cor e Forma:SolidPeso molecular:442.57XEN907
CAS:<p>XEN907 is a novel spiro oxindole NaV1.7 blocker. XEN907 also inhibits hNaV1.7 (IC50: 3 nM).</p>Fórmula:C21H21NO4Pureza:99.92%Cor e Forma:SolidPeso molecular:351.4Trofinetide
CAS:<p>Trofinetide (NNZ-2566) is a synthetic analog of the endogenous N-terminus tripeptide. It has been shown to be neuroprotective in animal models of brain injury.</p>Fórmula:C13H21N3O6Pureza:98.70% - 99.50%Cor e Forma:SolidPeso molecular:315.32Esomeprazole magnesium salt
CAS:<p>Esomeprazole magnesium, an oral proton pump inhibitor, curbs gastric acid by blocking H+, K+-ATPase; used in treating GERD.</p>Fórmula:C17H21MgN3O3SCor e Forma:SolidPeso molecular:371.74Propafenone hydrochloride
CAS:<p>Propafenone hydrochloride (Arythmol8) is a classic anti-arrhythmic medication, which treats illnesses associated with rapid heartbeats such as atrial.</p>Fórmula:C21H27NO3·HClPureza:99.67%Cor e Forma:White SolidPeso molecular:377.9Argireline
CAS:<p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>Fórmula:C34H60N14O12SPureza:96.79% - 99.65%Cor e Forma:White PowderPeso molecular:888.99cim0216
CAS:<p>CIM0216 is a synthetic TRPM3 activator whose potency and apparent affinity greatly exceeds that of the canonical TRPM3 agonist.</p>Fórmula:C21H21N3O2Pureza:99.87%Cor e Forma:SolidPeso molecular:347.41Afloqualone
CAS:<p>Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.</p>Fórmula:C16H14FN3OPureza:99.72%Cor e Forma:SolidPeso molecular:283.3PF 05089771
CAS:<p>PF 05089771 is a Selective inhibitor of Nav1.7 (IC50 = 11 nM) that interacts with the voltage-sensor domain of domain IV.</p>Fórmula:C18H12Cl2FN5O3S2Pureza:99.03% - 99.42%Cor e Forma:SolidPeso molecular:500.35Cinacalcet metabolite M4
CAS:<p>Cinacalcet metabolite M4 (Rarechem AL BW 1078) is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.</p>Fórmula:C10H12F3NPureza:97.13%Cor e Forma:SolidPeso molecular:203.2Acecainide hydrochloride
CAS:<p>Acecainide hydrochloride (NAPA) is the major hepatic metabolite of procainamide.Cost-effective and quality-assured.</p>Fórmula:C15H24ClN3O2Pureza:98.023% - 99.81%Cor e Forma:SolidPeso molecular:313.83Tegoprazan
CAS:<p>Tegoprazan is an orally active, highly selective gastric H+/K+-ATPase inhibitor.Cost-effective and quality-assured.</p>Fórmula:C20H19F2N3O3Pureza:98.22%Cor e Forma:SolidPeso molecular:387.38Bisaramil
CAS:<p>Bisaramil is a new class I antiarrhythmic agent.</p>Fórmula:C17H23ClN2O2Cor e Forma:SolidPeso molecular:322.83ML277
CAS:<p>ML277 (CID-53347902) was identified as a potent activator of KCNQ1 channels (EC(50)=260 nM).</p>Fórmula:C23H25N3O4S2Pureza:99.35%Cor e Forma:SolidPeso molecular:471.59Isoflurane
CAS:<p>Isoflurane (Forane) is a stable, non-explosive inhalation anesthetic that has been reported to induce caspase-3 activation.</p>Fórmula:C3H2ClF5OPureza:98%Cor e Forma:Clear Colorless Liquid LiquidPeso molecular:184.49CX614
CAS:<p>CX614 is a positive allosteric modulator of the AMPA receptor concerning AMPA.</p>Fórmula:C13H13NO4Pureza:97.37%Cor e Forma:SolidPeso molecular:247.255,7-Dichlorokynurenic acid
CAS:<p>5,7-Dichlorokynurenic acid (5,7-dichlorokynurenic acid sodium) is an NMDA receptor antagonist.</p>Fórmula:C10H5Cl2NO3Pureza:99.71%Cor e Forma:SolidPeso molecular:258.06TC-I2000
CAS:<p>TC-I2000 is an TRPM8 channel blocker. Inhibits icilin-induced TRPM8 channel activation in rTRPM8-expressing CHO cells with IC50 of 53 nM.</p>Fórmula:C23H18F4N2OPureza:99.778%Cor e Forma:SolidPeso molecular:414.4Ralfinamide
CAS:<p>Ralfinamide (Priralfinamide) is an orally available Na-channel blocker for the treatment of neuropathic pain and other pain conditions.</p>Fórmula:C17H19FN2O2Pureza:99.41%Cor e Forma:SolidPeso molecular:302.34PF-01247324
CAS:<p>PF-01247324 is a selective and orally bioavailable Nav1.8 channel blocker (IC50: 196 nM).</p>Fórmula:C13H10Cl3N3OPureza:99.22%Cor e Forma:SolidPeso molecular:330.6(2S)-6-Prenylnaringenin
CAS:<p>(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.</p>Fórmula:C20H20O5Pureza:99.47%Cor e Forma:SolidPeso molecular:340.37
