Inhibitor Enzymes
Inhibitor enzymes are molecules that decrease or block the activity of enzymes, preventing them from catalyzing their specific reactions. These inhibitors can be reversible or irreversible and are crucial tools in research and drug development for studying enzyme mechanisms, controlling metabolic pathways, and developing therapeutic agents. Inhibitor enzymes are widely used to modulate biological processes and to treat various diseases by targeting specific enzymes. At CymitQuimica, we offer a comprehensive range of high-quality enzyme inhibitors to support your research and pharmaceutical development needs.
Found 123 products of "Inhibitor Enzymes"
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(R)-Pinocembrin
CAS:Controlled Product<p>Applications (2R)-Pinocembrin is the (R)-enantiomer of Pinocembrin, a flavanoid with antioxidant activity found in damiana, honey, and propolis. (2R)-Pinocembrin is a potential inhibitor of PIM1 kinase, an oncogene that has been implicated in the development of leukemias, lymphomas, and prostate cancer.<br>References Zhao, J. et al.: J. Ethnopharmacol., 120, 387 (2008); Holder, S. et al.: Mol. Cancer Ther., 6, 163 (2007); Holder, S. et al.: Bioorg. Med. Chem., 15, 6463 (2007);<br></p>Formula:C15H12O4Color and Shape:WhiteMolecular weight:256.25O,O-Dimethyl Dithiophosphate
CAS:Controlled ProductFormula:C2H7O2PS2Color and Shape:ColourlessMolecular weight:158.18Morusin
CAS:Controlled Product<p>Stability Light Sensitive<br>Applications Morusin is an inhibitor of human cervical cancer stem cell growth, attenuating NF-kB activity, and initiating apoptosis.<br>References Wang, L. et al.: Mol. Cell. Biochem., 379, 7 (2013);<br></p>Formula:C25H24O6Color and Shape:NeatMolecular weight:420.45GDC 0152
CAS:Controlled Product<p>Applications GDC 0152 is a peptidomimetic small molecule antagonist of inhibitor of apoptosis (IAP) proteins with antitumor activity.<br>References Yue, Q., et. al.: Drug Metab. Dispos., 41, 508 (2013)<br></p>Formula:C25H34N6O3SColor and Shape:NeatMolecular weight:498.64Ipidacrine Hydrochloride Hydrate
CAS:Formula:C12H16N2·ClH·H2OColor and Shape:NeatMolecular weight:242.753a,6,7,7a-Tetrahydro-5-(hydroxymethyl)-2-methyl-(3aR,5R,6S,7R,7aR)-5H-pyrano[3,2-d]thiazole-6,7-diol
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications 3a,6,7,7a-Tetrahydro-5-(hydroxymethyl)-2-methyl-(3aR,5R,6S,7R,7aR)-5H-pyrano[3,2-d]thiazole-6,7-diol, can be used in the synthesis of Hexosaminidase inhibitors, which are the new drug candidates for the therapy of osteoarthritis.<br>References Liu, J. et al.: Chem. Bio., 8, 701 (2001);<br></p>Formula:C8H13NO4SColor and Shape:White To Light BeigeMolecular weight:219.26Bisindolylmaleimide VIII Acetic Acid Salt
CAS:Controlled Product<p>Applications It is a potent inhibitor of protein kinase C (PKC) activity. Bisindolylmaleimide VIII (Bis VIII) has been previously shown to enhance Fas-mediated apoptosis through a protein kinase C-independent mechanism.<br>References Emery, J., et al.: J. Biol. Chem., 273, 14363 (1998), Wiley, S., et al.: Immunity, 3, 673 (1995), MacFarlane, M., et al.: Biochem. J., 348, 93 (2000),<br></p>Formula:C26H26N4O4Color and Shape:NeatMolecular weight:458.511-(5-Isoquinolinesulfonyl)-2-methylpiperazine Dihydrochloride
CAS:Controlled Product<p>Applications A selective inhibitor of protein kinase C or cyclic-nucleotide-dependent protein kinases.<br>References Hidaka, H. and Kawamoto, S.: Biochem. and Biophys. Res. Comm., 125, 1, 258 (1984)<br></p>Formula:C14H17N3O2S·2ClHColor and Shape:NeatMolecular weight:364.29O,S-Diethyl Methylphosphonothioate
CAS:Controlled Product<p>Stability Moisture Sensitive<br>Applications An inhibitor of cholinesterase.<br>References Berman, H., et al.: J. Biol. Chem., 264, 3951 (1989), Millard, C., et al.: Biochemistry, 37, 237 (1998), Koellner, G., et al.: J. Mol. Biol., 296, 713 (2000),<br></p>Formula:C5H13O2PSColor and Shape:NeatMolecular weight:168.193-Acetyl-11-keto-β-boswellic Acid
CAS:Controlled ProductFormula:C32H48O5Color and Shape:WhiteMolecular weight:512.721-Propan-1,1,2,2,3,3,3-d7-amine
CAS:Controlled ProductFormula:C3H2D7NColor and Shape:NeatMolecular weight:66.15O-(2,4-Dinitrophenyl)hydroxylamine
CAS:<p>Applications O-(2,4-Dinitrophenyl)hydroxylamine is a rapid active-site-directed inhibitor of D-amino acid oxidase; modification results in specific incorporation of an amine group into an accessible nucleophilic residue with concomitant release of 2,4-dinitrophenol.<br>References D'Silva, C., et al.: Biochemi., 25, 5602 (1986),<br></p>Formula:C6H5N3O5Color and Shape:Brown SolidMolecular weight:199.12N-Acetyl-Lys-Octreotide Trifluoroacetic Acid Salt
CAS:<p>Stability Hygroscopic<br>Applications N-Acetyl-Phe-Octreotide is used as reactant/reagent in inhibition of octreotide acylation inside PLGA microspheres by derivatization of amines of peptide with self-immolative protecting group.<br>References Shirangi, M., et al.: Bioconjugate Chem., 27, 576-585 (2016)<br></p>Formula:C51H68N10O11S2·xC2HF3O2Color and Shape:NeatMolecular weight:1061.284Resolvin E1 Sodium Salt
CAS:Controlled ProductFormula:C20H29NaO5Color and Shape:NeatMolecular weight:372.431(5E)-6-(4-Hydroxy-3-methoxyphenyl)-5-hexene-2,4-dione
CAS:Controlled Product<p>Applications Curcumin (C838500) and gingerdione derivative. A possible human glyoxalase I inhibitor. Flavor modifier.<br>References Yuan, M. et al.; Bioorg. Med. Chem. 19, 1189 (2011); Ley, J. et al.; J. Agr. Food Chem. 56, 6656 (2008)<br></p>Formula:C13H14O4Color and Shape:NeatMolecular weight:234.25(±)-Procinolol Hydrochloride
CAS:Controlled Product<p>Applications (±)-Procinolol is a beta adrenergic receptor antagonist.<br>References Singh, K.: Indian J. Phsiol. Pharmacol., 27, 311 (1983)<br></p>Formula:C15H24ClNO2Color and Shape:NeatMolecular weight:285.81Baohuoside I
CAS:Controlled Product<p>Applications Baohuoside I is an inhibitor of cell growth and also is a down-regulator of durvivin and cyclin D1 expression. Used in the treatment of esophageal cancer. Anti-cancer agent.<br>References Lifang, W. et al.: Oncology Rep., 26, 1149 (2011); Jin, X. et al.: Drug Dev. Ind. Pharm., 39, 1421 (2013);<br></p>Formula:C27H30O10Color and Shape:NeatMolecular weight:514.52Raloxifene 4’-β-D-Glucuronide Lithium Salt
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications Raloxifene 4’-Glucuronide Lithium Salt is a metabolite of Raloxifene (R099995), a nonsteroidal estrogen receptor mixed agonist/antagonist.<br>References Dodge, J., et al.: Bioorg. Med. Chem. Lett., 7, 993 (1997); Jeong, E., et al.: Drug Metab. Dispos., 33, 785 (2005); Trontelj, J., et al.: Pharmacol. Res., 52, 334 (2005); Oswald, S., et al.: Clin. Pharmacol. Ther., 79 206 (2006)<br></p>Formula:C34H34LiNO10SColor and Shape:NeatMolecular weight:655.644-Amino-5-(bromomethyl)-2-methylpyrimidine Dihydrobromide
CAS:Controlled Product<p>Applications A pyrimidine derivative as G protein-coupled receptor kinase (GRK) inhibitor.<br>References Bigham, E., et al.: J. Med. Chem., 35, 1399 (1992), Jansen, M., et al.: Biochem. Pharmacol., 47, 1067 (1994), Hasbi, A., et al.: J. Neurochem., 70, 2129 (1998),<br></p>Formula:C17H17N3O2SColor and Shape:NeatMolecular weight:327.40N-(2-Aminoethyl)-5-chloroisoquinoline-8-sulfonamide Dihydrochloride
CAS:Controlled Product<p>Applications Found to have a potent inhibitory action against casein kinase 1 completely with respect to ATP and a much weaker effect on casein kinase 2 and other protein kinases.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Hidaka, H., et al.: J. of Biol. Chem., 264, 9, 4924 (1989)<br></p>Formula:C11H12ClN3O2S·2ClHColor and Shape:NeatMolecular weight:358.67
![3a,6,7,7a-Tetrahydro-5-(hydroxymethyl)-2-methyl-(3aR,5R,6S,7R,7aR)-5H-pyrano[3,2-d]thiazole-6,7-di…](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTR%2Fthumb-webp%2FT293625.webp&w=3840&q=75)
