EGFR
EGFR (epidermal growth factor receptor) inhibitors are compounds that block the signaling of EGFR, a receptor that is often overexpressed in various cancers and plays a critical role in angiogenesis. EGFR inhibitors are used to prevent tumor growth and metastasis by disrupting the pathways that promote blood vessel formation in tumors. These inhibitors are widely used in cancer research and therapy. At CymitQuimica, we offer a diverse selection of high-quality EGFR inhibitors to support your research in oncology and angiogenesis.
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EGFR-IN-82
CAS:2568086-81-5
EGFR-IN-82 (Compound 8a) is a potent, orally active inhibitor of EGFR, exhibiting IC50 values of …
Formula:
C32H41BrN9O2P
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
694.6
Ref: TM-T78788
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
PD 174265
CAS:216163-53-0
PD 174265 is an effective, selective and reversible inhibitor of epidermal growth factor receptor (EGFR) …
Formula:
C17H15BrN4O
Purity:
98.88%
Color and Shape:
Solid
Molecular weight:
371.23
Ref: TM-T28339
| 5mg | 35.00 € | ||
| 10mg | 46.00 € | ||
| 25mg | 63.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 114.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Tarlox-TKI
CAS:2135696-72-7
Tarlox-TKI (Kinase inhibitor-1) is a pan-ErbB inhibitor, the active ingredient of Tarloxotinib, which has antitumor …
Formula:
C19H18BrClN6O
Purity:
97.03%
Color and Shape:
Solid
Molecular weight:
461.74
Ref: TM-T11761
| 1mg | 145.00 € | ||
| 1mL*10mM (DMSO) | 255.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
(E/Z)-CP-724714
CAS:537705-08-1
(E/Z)-CP-724714, comprising racemic mixtures of (E)-CP-724714 and (Z)-CP-724714 isomers, is a potent, selective, and orally …
Formula:
C27H27N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
469.54
Ref: TM-T6046
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
EAI001
CAS:892772-75-7
EAI001 is a potent and selective mutant epidermal growth factor receptor (EGFR) variant inhibitor that …
Formula:
C19H15N3O2S
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
349.41
Ref: TM-T61191
| 5mg | 56.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 283.00 € | ||
| 100mg | 454.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Limertinib
CAS:1934259-00-3
Limertinib (ASK120067) is a EGFR tyrosine kinase inhibitor targeting EGFR T790M, applicable for the study …
Formula:
C29H32ClN7O2
Color and Shape:
Solid
Molecular weight:
546.06
Ref: TM-T35897
| 1mg | 90.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 316.00 € | ||
| 25mg | 637.00 € | ||
| 50mg | 827.00 € | ||
| 100mg | 1,169.00 € | ||
| 200mg | 1,586.00 € | ||
| 1mL*10mM (DMSO) | 250.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Mutated EGFR-IN-2
CAS:2050906-97-1
Mutated EGFR-IN-2 is an inhibitor of mutant-selective EGFR.
Formula:
C29H35FN8O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
562.64
Ref: TM-T12130
| 25mg | 1,586.00 € | ||
| 50mg | 2,072.00 € | ||
| 100mg | 2,660.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
EGFR-IN-5
CAS:2225887-26-1
EGFR-IN-5 inhibits EGFR & mutants; IC50: EGFR 10.4nM, L858R 1.1nM, L858R/T790M 34nM, L858R/T790M/C797S 7.2nM.
Formula:
C31H38FN9O
Purity:
98.17%
Color and Shape:
Solid
Molecular weight:
571.69
Ref: TM-T11160
| 1mg | 105.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 399.00 € | ||
| 25mg | 753.00 € | ||
| 1mL*10mM (DMSO) | 315.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Sunvozertinib
CAS:2370013-12-8
Sunvozertinib (DZD9008) is a potent ErbBs and BTK inhibitor, with inhibitory effects on EGFR, Her2.Cost-effective …
Formula:
C29H35ClFN7O3
Purity:
98.11% - 99.71%
Color and Shape:
Liquid
Molecular weight:
584.08
Ref: TM-T64124
| 1mg | 35.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 131.00 € | ||
| 50mg | 212.00 € | ||
| 100mg | 373.00 € | ||
| 500mg | 1,388.00 € | ||
| 1mL*10mM (DMSO) | 159.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
A-935142
CAS:1031335-85-9
A-935142 enhances hERG (Kv 11.1) channels, slows inactivation, promotes activation, and shortens repolarization.
Formula:
C18H19F3N2O2
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
352.35
Ref: TM-T14077
| 1mg | 200.00 € | ||
| 5mg | 472.00 € | ||
| 10mg | 645.00 € | ||
| 25mg | 905.00 € | ||
| 50mg | 1,121.00 € | ||
| 100mg | 1,425.00 € | ||
| 200mg | 1,863.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Tyrphostin AG 112
CAS:144978-82-5
Tyrphostin AG 112 is an inhibitor of EGFR phosphorylation.
Formula:
C13H8N4O
Purity:
97.01%
Color and Shape:
Solid
Molecular weight:
236.23
Ref: TM-T8534
| 5mg | 47.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 273.00 € | ||
| 500mg | 662.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Epertinib
CAS:908305-13-5
Epertinib is a reversible and selective tyrosine kinase inhibitor of EGFR, HER2, and HER4 (IC50s: …
Formula:
C30H27ClFN5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
560.02
Ref: TM-T11213L
| 25mg | 1,293.00 € | ||
| 50mg | 1,681.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Larotinib
CAS:1438072-11-7
Larotinib is an orally active, potent, and broad-spectrum tyrosine kinase inhibitor (TKI) with an IC50 …
Formula:
C24H26ClFN4O4
Purity:
98.45%
Color and Shape:
Liquid
Molecular weight:
488.94
Ref: TM-T73334
| 1mg | 81.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 259.00 € | ||
| 25mg | 439.00 € | ||
| 50mg | 628.00 € | ||
| 100mg | 882.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
SKLB 1028
CAS:1350544-93-2
SKLB 1028, an oral EGFR/FLT3/Abl inhibitor, excels in AML and CML with Abl mutations.
Formula:
C24H29N9
Purity:
99.71% - 99.85%
Color and Shape:
Solid
Molecular weight:
443.55
Ref: TM-T34656
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 378.00 € | ||
| 50mg | 560.00 € | ||
| 100mg | 800.00 € | ||
| 500mg | 1,644.00 € | ||
| 1mL*10mM (DMSO) | 143.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
CGP77675
CAS:234772-64-6
CGP77675 (ZINC1488120) is a potent and selective inhibitor of Src family kinase with IC50s of …
Formula:
C26H29N5O2
Purity:
98.23%
Color and Shape:
Solid
Molecular weight:
443.54
Ref: TM-T30855
| 1mg | 50.00 € | ||
| 2mg | 70.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 354.00 € | ||
| 50mg | 567.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
DBPR112
CAS:1226549-49-0
DBPR112: oral furanopyrimidine EGFR inhibitor; IC50: 15 nM (EGFRWT), 48 nM (L858R/T790M); blocks ATP site, …
Formula:
C32H31N5O3
Purity:
98.29%
Color and Shape:
Solid
Molecular weight:
533.62
Ref: TM-T10965
| 1mg | 75.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 305.00 € | ||
| 25mg | 495.00 € | ||
| 50mg | 658.00 € | ||
| 100mg | 907.00 € | ||
| 1mL*10mM (DMSO) | 188.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
CHMFL-EGFR-202
CAS:2089381-40-6
CHMFL-EGFR-202 is a potent, irreversible inhibitor of EGFR mutant kinase (IC50s: 5.3 nM and 8.3 …
Formula:
C25H24ClN7O2
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
489.96
Ref: TM-T10802
| 1mg | 115.00 € | ||
| 2mg | 172.00 € | ||
| 5mg | 255.00 € | ||
| 10mg | 375.00 € | ||
| 25mg | 562.00 € | ||
| 50mg | 787.00 € | ||
| 100mg | 1,074.00 € | ||
| 1mL*10mM (DMSO) | 305.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
H-9 dihydrochloride
CAS:116700-36-8
H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.
Formula:
C11H15Cl2N3O2S
Purity:
96.57%
Color and Shape:
Solid
Molecular weight:
324.23
Ref: TM-T22833
| 1mg | 35.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 225.00 € | ||
| 100mg | 331.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
RTC-5
CAS:1423077-49-9
RTC-5 (TRC-382) is a phenothiazine compound that has been specifically enhanced for its potent anti-cancer …
Formula:
C24H22ClF3N2O3S
Purity:
98.14%
Color and Shape:
Solid
Molecular weight:
510.96
Ref: TM-T12777
| 5mg | 52.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 284.00 € | ||
| 100mg | 411.00 € | ||
| 500mg | 867.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Tyrphostin A25
CAS:118409-58-8
Tyrphostin A25 (Tyrphostin AG 82) is a specific EGFR tyrosine kinase inhibitor and GPR35 agonist …
Formula:
C10H6N2O3
Purity:
98.76%
Color and Shape:
Yellow Green Powder /Off-White Solid
Molecular weight:
202.17
Ref: TM-T21622
| 2mg | 39.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 120.00 € | ||
| 50mg | 172.00 € | ||
| 100mg | 255.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
