EGFR
EGFR (epidermal growth factor receptor) inhibitors are compounds that block the signaling of EGFR, a receptor that is often overexpressed in various cancers and plays a critical role in angiogenesis. EGFR inhibitors are used to prevent tumor growth and metastasis by disrupting the pathways that promote blood vessel formation in tumors. These inhibitors are widely used in cancer research and therapy. At CymitQuimica, we offer a diverse selection of high-quality EGFR inhibitors to support your research in oncology and angiogenesis.
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Limertinib
CAS:1934259-00-3
Limertinib (ASK120067) is a EGFR tyrosine kinase inhibitor targeting EGFR T790M, applicable for the study …
Formula:
C29H32ClN7O2
Purity:
97.44%
Color and Shape:
Solid
Molecular weight:
546.06
Ref: TM-T35897
| 1mg | 90.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 316.00 € | ||
| 25mg | 637.00 € | ||
| 50mg | 827.00 € | ||
| 100mg | 1,169.00 € | ||
| 200mg | 1,586.00 € | ||
| 1mL*10mM (DMSO) | 250.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
A-935142
CAS:1031335-85-9
A-935142 enhances hERG (Kv 11.1) channels, slows inactivation, promotes activation, and shortens repolarization.
Formula:
C18H19F3N2O2
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
352.35
Ref: TM-T14077
| 1mg | 200.00 € | ||
| 5mg | 472.00 € | ||
| 10mg | 645.00 € | ||
| 25mg | 905.00 € | ||
| 50mg | 1,121.00 € | ||
| 100mg | 1,425.00 € | ||
| 200mg | 1,863.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
Sunvozertinib
CAS:2370013-12-8
Sunvozertinib (DZD9008) is a potent ErbBs and BTK inhibitor, with inhibitory effects on EGFR, Her2.Cost-effective …
Formula:
C29H35ClFN7O3
Purity:
98.11% - 99.71%
Color and Shape:
Liquid
Molecular weight:
584.08
Ref: TM-T64124
| 1mg | 35.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 131.00 € | ||
| 50mg | 212.00 € | ||
| 100mg | 373.00 € | ||
| 500mg | 1,388.00 € | ||
| 1mL*10mM (DMSO) | 159.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
EGFR-IN-5
CAS:2225887-26-1
EGFR-IN-5 inhibits EGFR & mutants; IC50: EGFR 10.4nM, L858R 1.1nM, L858R/T790M 34nM, L858R/T790M/C797S 7.2nM.
Formula:
C31H38FN9O
Purity:
98.17%
Color and Shape:
Solid
Molecular weight:
571.69
Ref: TM-T11160
| 1mg | 105.00 € | ||
| 5mg | 250.00 € | ||
| 10mg | 399.00 € | ||
| 25mg | 753.00 € | ||
| 1mL*10mM (DMSO) | 315.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
Mutated EGFR-IN-2
CAS:2050906-97-1
Mutated EGFR-IN-2 is an inhibitor of mutant-selective EGFR.
Formula:
C29H35FN8O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
562.64
Ref: TM-T12130
| 25mg | 1,586.00 € | ||
| 50mg | 2,072.00 € | ||
| 100mg | 2,660.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
SDZ281-977
CAS:150779-71-8
SDZ 281-977 is a derivative of Lavendustin A which is the EGF receptor tyrosine kinase …
Formula:
C18H20O5
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
316.35
Ref: TM-T16866
| 1mg | 99.00 € | ||
| 5mg | 235.00 € | ||
| 10mg | 376.00 € | ||
| 25mg | 753.00 € | ||
| 50mg | 1,169.00 € | ||
| 1mL*10mM (DMSO) | 259.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
RTC-5
CAS:1423077-49-9
RTC-5 (TRC-382) is a phenothiazine compound that has been specifically enhanced for its potent anti-cancer …
Formula:
C24H22ClF3N2O3S
Purity:
98.14%
Color and Shape:
Solid
Molecular weight:
510.96
Ref: TM-T12777
| 5mg | 52.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 284.00 € | ||
| 100mg | 411.00 € | ||
| 500mg | 867.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
H-9 dihydrochloride
CAS:116700-36-8
H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.
Formula:
C11H15Cl2N3O2S
Purity:
96.57%
Color and Shape:
Solid
Molecular weight:
324.23
Ref: TM-T22833
| 1mg | 35.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 225.00 € | ||
| 100mg | 331.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
Nuvenzepine
CAS:96487-37-5
Nuvenzepine is an antagonist of mAChR. It has the potential for gastrospasm treatment.
Formula:
C19H20N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
336.39
Ref: TM-T16362
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
CHMFL-EGFR-202
CAS:2089381-40-6
CHMFL-EGFR-202 is a potent, irreversible inhibitor of EGFR mutant kinase (IC50s: 5.3 nM and 8.3 …
Formula:
C25H24ClN7O2
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
489.96
Ref: TM-T10802
| 1mg | 115.00 € | ||
| 2mg | 172.00 € | ||
| 5mg | 255.00 € | ||
| 10mg | 375.00 € | ||
| 25mg | 562.00 € | ||
| 50mg | 787.00 € | ||
| 100mg | 1,074.00 € | ||
| 1mL*10mM (DMSO) | 305.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
BKI-1369
CAS:1951431-22-3
BKI-1369 is a bumped kinase inhibitor. BKI-1369 increases hERG-inhibitory activity (IC50:1.52 μM).
Formula:
C23H27N7O
Color and Shape:
Solid
Molecular weight:
417.51
Ref: TM-T10556
| 5mg | 450.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
CGP77675
CAS:234772-64-6
CGP77675 (ZINC1488120) is a potent and selective inhibitor of Src family kinase with IC50s of …
Formula:
C26H29N5O2
Purity:
98.23%
Color and Shape:
Solid
Molecular weight:
443.54
Ref: TM-T30855
| 1mg | 50.00 € | ||
| 2mg | 70.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 354.00 € | ||
| 50mg | 567.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
SKLB 1028
CAS:1350544-93-2
SKLB 1028, an oral EGFR/FLT3/Abl inhibitor, excels in AML and CML with Abl mutations.
Formula:
C24H29N9
Purity:
99.71% - 99.85%
Color and Shape:
Solid
Molecular weight:
443.55
Ref: TM-T34656
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 378.00 € | ||
| 50mg | 560.00 € | ||
| 100mg | 800.00 € | ||
| 500mg | 1,644.00 € | ||
| 1mL*10mM (DMSO) | 143.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
Larotinib
CAS:1438072-11-7
Larotinib is an orally active, potent, and broad-spectrum tyrosine kinase inhibitor (TKI) with an IC50 …
Formula:
C24H26ClFN4O4
Purity:
98.45%
Color and Shape:
Liquid
Molecular weight:
488.94
Ref: TM-T73334
| 1mg | 81.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 259.00 € | ||
| 25mg | 439.00 € | ||
| 50mg | 628.00 € | ||
| 100mg | 882.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
EGFR-IN-99
CAS:2068806-31-3
EGFR-IN-99 (JBJ-03-142-02) is an EGFR and HER2 Exon 20 insertion mutation inhibitor for the study …
Formula:
C25H22FN7O3
Purity:
97.75%
Color and Shape:
Liquid
Molecular weight:
487.49
Ref: TM-T35901
| 1mg | 127.00 € | ||
| 5mg | 303.00 € | ||
| 10mg | 449.00 € | ||
| 25mg | 727.00 € | ||
| 50mg | 998.00 € | ||
| 100mg | 1,349.00 € | ||
| 500mg | 2,688.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
LY 456236 hydrochloride
CAS:338736-46-2
LY 456236 hydrochloride (MPMQ hydrochloride) is an mGlu1 receptor antagonist with an ic50 value of …
Formula:
C16H16ClN3O2
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
317.77
Ref: TM-T22954
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 164.00 € | ||
| 50mg | 259.00 € | ||
| 100mg | 374.00 € | ||
| 200mg | 522.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
Cloperastine fendizoate
CAS:85187-37-7
Cloperastine fendizoate (Hustazol) inhibits the hERG K+ currents in a concentration-dependent manner (IC50: 27 nM).
Formula:
C40H38ClNO5
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
648.19
Ref: TM-T13619
| 500mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
EMI1
CAS:35773-42-3
EMI1 targets mutated EGFR in drug-resistant NSCLC research.
Formula:
C20H18N2O3
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
334.37
Ref: TM-T61016
| 5mg | 39.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 117.00 € | ||
| 50mg | 187.00 € | ||
| 100mg | 301.00 € | ||
| 200mg | 425.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
CGP52411
CAS:145915-58-8
CGP52411 is an orally active, and ATP-competitive inhibitor of EGFR (IC50: 0.3 μM).
Formula:
C20H15N3O2
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
329.35
Ref: TM-T10782
| 1mg | 42.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 235.00 € | ||
| 50mg | 358.00 € | ||
| 100mg | 553.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
Selatinib
CAS:1275595-86-2
Selatinib is an orally active and potent dual inhibitor of EGFR and ErbB2 with anticancer …
Formula:
C29H26ClFN4O3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
565.06
Ref: TM-T34602
| 1mg | 99.00 € | ||
| 5mg | 235.00 € | ||
| 10mg | 354.00 € | ||
| 25mg | 645.00 € | ||
| 50mg | 938.00 € |
Estimated delivery in United States, on Thursday 15 May 2025
