BTK
BTK (Bruton's tyrosine kinase) inhibitors are compounds that specifically target and inhibit BTK, a crucial enzyme involved in B-cell receptor signaling and the regulation of angiogenesis. BTK plays a significant role in the proliferation and survival of cancer cells, particularly in hematological malignancies. By inhibiting BTK, these compounds can disrupt angiogenesis and tumor growth, making them valuable in cancer therapy. At CymitQuimica, we offer a range of high-quality BTK inhibitors to support your research in oncology, immunology, and angiogenesis.
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IBT6A
CAS:1022150-12-4
IBT6A is an impurity of Ibrutinib. Ibrutinib is a Btk inhibitor (IC50: 0.5 nM). IBT6A …
Formula:
C22H22N6O
Purity:
99.8% - 99.88%
Color and Shape:
Solid
Molecular weight:
386.45
Ref: TM-T10625
| 100mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Orelabrutinib
CAS:1655504-04-3
Orelabrutinib (ICP-022) is an orally active and irreversible inhibitor of Bruton's tyrosine kinase (BTK).
Formula:
C26H25N3O3
Purity:
97.77% - 99.44%
Color and Shape:
Solid
Molecular weight:
427.49
Ref: TM-T12317
| 1mg | 89.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 309.00 € | ||
| 25mg | 511.00 € | ||
| 50mg | 707.00 € | ||
| 100mg | 925.00 € | ||
| 500mg | 1,859.00 € | ||
| 1mL*10mM (DMSO) | 216.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Tirabrutinib hydrochloride
CAS:1439901-97-9
Tirabrutinib hydrochloride is a potent, highly selective, irreversible oral BTK inhibitor.Cost-effective and quality-assured.
Formula:
C25H23ClN6O3
Purity:
99.04% - 99.27%
Color and Shape:
Solid
Molecular weight:
490.94
Ref: TM-T12311
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 193.00 € | ||
| 100mg | 343.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Rilzabrutinib
CAS:1575596-29-0
Rilzabrutinib (PRN1008) is a reversible covalent, selective and oral active inhibitor of Bruton’s Tyrosine Kinase …
Formula:
C36H40FN9O3
Purity:
97.87% - 99.76%
Color and Shape:
Solid
Molecular weight:
665.76
Ref: TM-T12542
| 1mg | 95.00 € | ||
| 5mg | 227.00 € | ||
| 10mg | 363.00 € | ||
| 25mg | 631.00 € | ||
| 50mg | 909.00 € | ||
| 100mg | 1,273.00 € | ||
| 500mg | 2,545.00 € | ||
| 1mL*10mM (DMSO) | 332.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Btk inhibitor 2
CAS:1558036-85-3
Btk inhibitor 2 (BGB-3111 analog) is a BTK inhibitor.
Formula:
C24H25N5O3
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
431.49
Ref: TM-T10629
| 1mg | 37.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 222.00 € | ||
| 50mg | 370.00 € | ||
| 100mg | 450.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
MT-802
CAS:2231744-29-7
MT-802 is an effective BTK degrader based on PROTAC technology (DC50: 1 nM). MT-802 has …
Formula:
C41H41N9O8
Purity:
95.93% - 97.00%
Color and Shape:
Solid
Molecular weight:
787.82
Ref: TM-T16157
| 1mg | 93.00 € | ||
| 5mg | 181.00 € | ||
| 10mg | 273.00 € | ||
| 25mg | 519.00 € | ||
| 50mg | 703.00 € | ||
| 100mg | 903.00 € | ||
| 200mg | 1,272.00 € | ||
| 1mL*10mM (DMSO) | 236.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
ARQ 531
CAS:2095393-15-8
ARQ-531: potent oral BTK inhibitor, anti-cancer potential, IC50 of 0.85/0.39 nM for WT/C481S-BTK.
Formula:
C25H23ClN4O4
Purity:
98.69% - 99.59%
Color and Shape:
Solid
Molecular weight:
478.93
Ref: TM-T14323
| 2mg | 49.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 209.00 € | ||
| 50mg | 333.00 € | ||
| 100mg | 532.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
evobrutinib
CAS:1415823-73-2
Evobrutinib(M2951) , also known as M-2951 and MSC-2364447C, is a highly selective inhibitor of the …
Formula:
C25H27N5O2
Purity:
98.04% - 99.42%
Color and Shape:
Solid
Molecular weight:
429.51
Ref: TM-T4387
| 1mg | 41.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 223.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 461.00 € | ||
| 500mg | 995.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
DBt-10
DBt-10 is a potent Bruton's tyrosine kinase (BTK) degrader [1].
Formula:
C68H86ClFN16O6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1277.97
Ref: TM-T79890
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
PROTAC BTK Degrader-6
CAS:2767204-39-5
PROTAC BTK Degrader-6 (Compound 15), with a DC50 of 3.18 nM, exhibits anti-inflammatory properties by …
Formula:
C45H47N11O6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
837.92
Ref: TM-T78782
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
Atuzabrutinib
CAS:1581714-49-9
Atuzabrutinib (SAR 444727) is a selective BTK inhibitor and can be used to study arthritis …
Formula:
C30H30FN7O2
Purity:
97.27%
Color and Shape:
Liquid
Molecular weight:
539.6
Ref: TM-T39056
| 1mg | 176.00 € | ||
| 5mg | 446.00 € | ||
| 10mg | 738.00 € | ||
| 25mg | 1,461.00 € | ||
| 50mg | 2,465.00 € | ||
| 100mg | 3,842.00 € | ||
| 1mL*10mM (DMSO) | 529.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
AS-1763
CAS:2227211-00-7
AS-1763 is an orally available and selective BTK inhibitor with an IC50 of 0.85 nM.
Formula:
C33H31FN6O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
578.64
Ref: TM-T39707
| 1mg | 218.00 € | ||
| 5mg | 542.00 € | ||
| 10mg | 811.00 € | ||
| 25mg | 1,387.00 € | ||
| 50mg | 2,075.00 € | ||
| 100mg | 3,117.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Acalabrutinib enantiomer
CAS:1952316-43-6
R-Acalabrutinib, a BTK inhibitor,enantiomer, is researched for cancer, autoimmune diseases, and inflammation.
Formula:
C26H23N7O2
Purity:
96.68%
Color and Shape:
Solid
Molecular weight:
465.51
Ref: TM-T67881
| 1mg | 113.00 € | ||
| 5mg | 251.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 551.00 € | ||
| 50mg | 776.00 € | ||
| 100mg | 1,043.00 € | ||
| 500mg | 2,103.00 € | ||
| 1mL*10mM (DMSO) | 279.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
BTK inhibitor 17
CAS:1858206-76-4
BTK inhibitor 17 is a potent irreversible BTK inhibitor (IC50 = 2.1 nM). BTK inhibitor …
Formula:
C25H24N6O3
Purity:
99.29% - 99.57%
Color and Shape:
Solid
Molecular weight:
456.5
Ref: TM-T9706
| 1mg | 91.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 255.00 € | ||
| 25mg | 409.00 € | ||
| 50mg | 542.00 € | ||
| 100mg | 758.00 € | ||
| 200mg | 998.00 € | ||
| 1mL*10mM (DMSO) | 169.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
PROTAC BTK Degrader-5
PROTAC BTK Degraders-5 (Compound 3e) is a selective Bruton's tyrosine kinase (BTK) degrader with a …
Formula:
C52H57ClFN9O6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
958.52
Ref: TM-T79292
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
PCI-33380
CAS:1022899-36-0
PCI-33380 is an irreversible inhibitor of Bruton's Tyrosine Kinase.
Formula:
C46H52BF2N11O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
855.8
Ref: TM-T16441
| 25mg | 940.00 € | ||
| 50mg | 1,482.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
N-piperidine Ibrutinib hydrochloride
CAS:2231747-18-3
N-piperidine Ibrutinib hydrochloride is a BTK inhibitor that inhibits WT BTK and C481S BTK , …
Formula:
C22H23ClN6O
Purity:
98.83%
Color and Shape:
Solid
Molecular weight:
422.91
Ref: TM-T12152
| 1mg | 52.00 € | ||
| 5mg | 110.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 329.00 € | ||
| 50mg | 489.00 € | ||
| 100mg | 707.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GDC-0834
CAS:1133432-49-1
GDC-0834 inhibits BTK with an in vitro IC50 of 5.9 and 6.4 nM in biochemical …
Formula:
C33H36N6O3S
Color and Shape:
Solid
Molecular weight:
596.74
Ref: TM-T11379
| 2mg | 186.00 € | ||
| 5mg | 374.00 € | ||
| 1mL*10mM (DMSO) | 516.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Tirabrutinib
CAS:1351636-18-4
Tirabrutinib, an oral Btk inhibitor (IC50=6.8 nM), crosses the BBB and halts B cell signaling …
Formula:
C25H22N6O3
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
454.48
Ref: TM-TQ0236
| 10mg | 50.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 114.00 € | ||
| 100mg | 206.00 € | ||
| 200mg | 307.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
N-piperidine Ibrutinib
CAS:330785-90-5
N-piperidine Ibrutinib is a potent BTK inhibitor with IC50s of 51.0 for WT BTK and …
Formula:
C22H22N6O
Purity:
96.65%
Color and Shape:
Solid
Molecular weight:
386.45
Ref: TM-T9408
| 1mg | 94.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 271.00 € | ||
| 25mg | 433.00 € | ||
| 50mg | 615.00 € | ||
| 100mg | 817.00 € | ||
| 200mg | 1,080.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
