Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
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Subcategories of "Chromatin/Epigenetics"
Products of "Chromatin/Epigenetics"
PF-9366
CAS:72882-78-1
PF-9366 is a human methionine adenosyltransferase 2A (Mat2A) inhibitor (IC50: 420 nM; Kd: 170 nM).
Formula:
C20H19ClN4
Purity:
100% - 98.99%
Color and Shape:
Solid
Molecular weight:
350.84
Ref: TM-T5191
| 1mg | 58.00 € | ||
| 5mg | 122.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 260.00 € | ||
| 50mg | 395.00 € | ||
| 1mL*10mM (DMSO) | 134.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
AG-270
CAS:2201056-66-6
AG-270 is an allosteric and orally active inhibitor of MAT2A.
Formula:
C30H27N5O2
Purity:
98.2% - 98.28%
Color and Shape:
Solid
Molecular weight:
489.57
Ref: TM-T9050
| 1mg | 110.00 € | ||
| 5mg | 256.00 € | ||
| 10mg | 410.00 € | ||
| 25mg | 680.00 € | ||
| 50mg | 938.00 € | ||
| 100mg | 1,301.00 € | ||
| 500mg | 2,593.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
C-82
CAS:1422253-37-9
C-82 is a specific CBP/β-catenin antagonist. It inhibits the binding between β-catenin and CBP and …
Formula:
C33H34N6O4
Purity:
98.86% - 99.66%
Color and Shape:
Solid
Molecular weight:
578.66
Ref: TM-T10641
| 1mg | 430.00 € | ||
| 5mg | 868.00 € | ||
| 10mg | 1,254.00 € | ||
| 25mg | 1,985.00 € | ||
| 1mL*10mM (DMSO) | 1,130.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Itacitinib
CAS:1334298-90-6
Itacitinib (INCB039110) is an orally bioavailable inhibitor of Janus-associated kinase 1 (JAK1) with potential antineoplastic …
Formula:
C26H23F4N9O
Purity:
96.4% - 99.01%
Color and Shape:
Solid
Molecular weight:
553.51
Ref: TM-T3998
| 1mg | 49.00 € | ||
| 2mg | 71.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 325.00 € | ||
| 50mg | 543.00 € | ||
| 100mg | 780.00 € | ||
| 500mg | 1,549.00 € | ||
| 1mL*10mM (DMSO) | 137.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
A-966492
CAS:934162-61-5
A-96649 is a new-type and effective inhibitor. The Ki of A-966492 for PARP1 and PARP2 …
Formula:
C18H17FN4O
Purity:
98.53% - 99.25%
Color and Shape:
Solid
Molecular weight:
324.35
Ref: TM-T6366
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 275.00 € | ||
| 100mg | 394.00 € | ||
| 200mg | 560.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
GSK503
CAS:1346572-63-1
GSK-503, a potent EZH2 inhibitor, has potential antitumor activity.
Formula:
C31H38N6O2
Purity:
98% - 99.74%
Color and Shape:
Solid
Molecular weight:
526.67
Ref: TM-T1775
| 1mg | 37.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 208.00 € | ||
| 50mg | 376.00 € | ||
| 100mg | 560.00 € | ||
| 500mg | 1,216.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
PFI-4
CAS:900305-37-5
PFI-4 is a potent and selective and cell-permeable BRPF1 bromodomain inhibitor.
Formula:
C21H24N4O3
Purity:
99.53% - ≥95%
Color and Shape:
Solid
Molecular weight:
380.44
Ref: TM-T1973
| 5mg | 47.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | 119.00 € | ||
| 50mg | 188.00 € | ||
| 100mg | 311.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
NI-57
CAS:1883548-89-7
NI-57 inhibits BRPF family proteins: BRPF1 (IC50=3.1nM), BRPF2 (IC50=46nM), BRPF3 (IC50=140nM).
Formula:
C19H17N3O4S
Purity:
100% - 99.87%
Color and Shape:
Solid
Molecular weight:
383.42
Ref: TM-TQ0083
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Menin-MLL inhibitor MI-2
CAS:1271738-62-5
Menin-MLL inhibitor MI-2 (MI2) is a potent menin-MLL interaction inhibitor with IC50 of 446 nM.
Formula:
C18H25N5S2
Purity:
97.46%
Color and Shape:
Solid
Molecular weight:
375.55
Ref: TM-T2649
| 2mg | 42.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 243.00 € | ||
| 100mg | 376.00 € | ||
| 200mg | 550.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Molibresib besylate
CAS:1895049-20-3
Molibresib besylate (GSK 525762C) is a BET protein family inhibitor used in the study of …
Formula:
C28H28ClN5O5S
Purity:
99.64% - 99.64%
Color and Shape:
Solid
Molecular weight:
582.07
Ref: TM-T11472L
| 2mg | 146.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Oroxylin A
CAS:480-11-5
Oroxylin A fights tumors, aids RAS therapy, promotes CaCo-2 cell apoptosis, blocks MCF-7 cell invasion …
Formula:
C16H12O5
Purity:
98.72% - 99.55%
Color and Shape:
Solid
Molecular weight:
284.26
Ref: TM-T6S1315
| 20mg | 138.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Tofacitinib
CAS:477600-75-2
Tofacitinib (Tasocitinib) is an orally Janus kinase inhibitor. Tofacitinib is used for the treatment of …
Formula:
C16H20N6O
Purity:
100% - 99.71%
Color and Shape:
Solid
Molecular weight:
312.37
Ref: TM-T6321
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 65.00 € | ||
| 50mg | 85.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 144.00 € | ||
| 500mg | 261.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
GSK126
CAS:1346574-57-9
GSK126 (GSK2816126A) is a excellently specific EZH2 methyltransferase inhibitor ( IC50=9.9 nM).
Formula:
C31H38N6O2
Purity:
98% - 99.67%
Color and Shape:
Solid
Molecular weight:
526.67
Ref: TM-T2079
| 2mg | 44.00 € | ||
| 5mg | 65.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 152.00 € | ||
| 50mg | 227.00 € | ||
| 100mg | 349.00 € | ||
| 200mg | 455.00 € | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Seclidemstat
CAS:1423715-37-0
Seclidemstat (SP-2577) is an effective LSD1 inhibitor, with a mean IC50 of 127 nM.
Formula:
C20H23ClN4O4S
Purity:
98.03% - 98.68%
Color and Shape:
Solid
Molecular weight:
450.94
Ref: TM-T4527
| 5mg | 48.00 € | ||
| 10mg | 72.00 € | ||
| 25mg | 120.00 € | ||
| 50mg | 187.00 € | ||
| 100mg | 354.00 € | ||
| 200mg | 528.00 € | ||
| 500mg | 852.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
GSK778 hydrochloride
CAS:2863657-79-6
GSK778 hydrochloride is a selective BET BD1 bromodomain inhibitor, with IC50s ranging from 41 to …
Formula:
C30H34ClN5O3
Purity:
97.45%
Color and Shape:
Liquid
Molecular weight:
548.08
Ref: TM-T9703L
| 1mg | 115.00 € | ||
| 5mg | 249.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 562.00 € | ||
| 50mg | 787.00 € | ||
| 100mg | 1,054.00 € | ||
| 1mL*10mM (DMSO) | 319.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Veliparib dihydrochloride
CAS:912445-05-7
Veliparib dihydrochloride (ABT-888 dihydrochloride) is a potent inhibitor of PARP1 and PARP2 with Ki of …
Formula:
C13H18Cl2N4O
Purity:
97.09% - 98%
Color and Shape:
Solid
Molecular weight:
317.21
Ref: TM-T2105
| 5mg | 35.00 € | ||
| 10mg | 48.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 116.00 € | ||
| 100mg | 180.00 € | ||
| 200mg | 294.00 € | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Remodelin
CAS:949912-58-7
Remodelin is an effective and specific inhibitor of the acetyl-transferase protein NAT10.
Formula:
C15H14N4S
Purity:
99.39% - 99.78%
Color and Shape:
Solid
Molecular weight:
282.36
Ref: TM-T3499
| 5mg | 55.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 130.00 € | ||
| 50mg | 185.00 € | ||
| 100mg | 274.00 € | ||
| 200mg | 411.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
PT-2385
CAS:1672665-49-4
PT-2385 is a selective HIF-2α inhibitor (Kd<50 nM).
Formula:
C17H12F3NO4S
Purity:
98.69% - 99.55%
Color and Shape:
Solid
Molecular weight:
383.34
Ref: TM-T7848
| 1mg | 66.00 € | ||
| 2mg | 87.00 € | ||
| 5mg | 153.00 € | ||
| 10mg | 258.00 € | ||
| 25mg | 411.00 € | ||
| 50mg | 610.00 € | ||
| 100mg | 868.00 € | ||
| 1mL*10mM (DMSO) | 126.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Venadaparib
CAS:1681017-83-3
Venadaparib, a PARP inhibitor (IC50: 1.4/1.0 nM for PARP1/2), is orally active, selective, not affecting …
Formula:
C23H23FN4O2
Purity:
98.47%
Color and Shape:
Solid
Molecular weight:
406.45
Ref: TM-T9430
| 1mg | 48.00 € | ||
| 2mg | 63.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 283.00 € | ||
| 50mg | 464.00 € | ||
| 100mg | 680.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
RN-1 dihydrochloride
CAS:1781835-13-9
RN-1 dihydrochloride is an effective and selective irreversible inhibitor of lysine-specific demethylase 1 (LSD1, IC50 …
Formula:
C23H31Cl2N3O2
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
452.42
Ref: TM-T21652
| 1mg | 49.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 156.00 € | ||
| 25mg | 255.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 540.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
