Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(229 products)
- Annexin A(16 products)
- Aromatase(23 products)
- Estrogen/progestogen Receptor(66 products)
- GPR(1 products)
- Glucocorticoid Receptor(165 products)
- LHRH(2 products)
- Opioid Receptor(327 products)
- Prostaglandin Receptor(122 products)
- RAAS(89 products)
- Reductase(51 products)
- Somatostatin(57 products)
- Thyroid hormone receptor(THR)(33 products)
- Vasopressin Receptor(48 products)
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Found 3420 products of "Endocrinology/Hormones"
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Inocoterone acetate
CAS:Inocoterone acetate is a nonsteroidal antiandrogen that binds to the androgen receptor and possesses antiandrogenic activity in animal models.Formula:C18H26O3Color and Shape:SolidMolecular weight:290.40AM-5262
CAS:AM-5262 is a potent GPR40 Full Agonist with improved rat PK profile and general selectivity profile.Formula:C33H35FO4Color and Shape:SolidMolecular weight:514.63ER degrader 4
CAS:ER degrader 4, a selective and orally active compound, effectively degrades estrogen receptors and exhibits anti-tumor activity [1].Formula:C26H19FO4SColor and Shape:SolidMolecular weight:446.49Antidiabetic agent 15
Antidiabetic agent 15 (compound 1B15) acts as a dual inhibitor of AT1R and NEP, reducing oxidative stress and restoring mitochondrial membrane potential.Formula:C26H23NO5Color and Shape:SolidMolecular weight:429.15762Nurr1 agonist 12
Nurr1 agonist 12 (Compound 37) acts as an agonist of the nuclear receptor-related protein 1 (Nurr1), enhancing its transcriptional activity with an EC50 of 0.06 μM. It stimulates human response elements NBRE, NurRE, and DR5 with EC50 values of 0.07 μM, 0.027 μM, and 0.014 μM, respectively. Additionally, Nurr1 agonist 12 induces the expression of neurotrophic genes regulated by Nurr1, such as tyrosine hydroxylase (TH), SOD1/2, BDNF, Sestrin 3, and BIRC5 (Survivin). The compound also demonstrates neuroprotective effects against neurotoxicity caused by Paraquat.Formula:C18H12ClN3OColor and Shape:SolidMolecular weight:321.76Myrciacetin
CAS:Myrciacetin from Rhododendron inhibits rat aldose reductase with IC50 of 13 μM.Formula:C17H16O6Color and Shape:SolidMolecular weight:316.309Epi-Cryptoacetalide
Epi-Cryptoacetalide is a useful organic compound for research related to life sciences and the catalog number is T126054.Formula:C18H22O3Color and Shape:SolidMolecular weight:286.371ODM-204
CAS:ODM-204 is novel nonsteroidal dual inhibitor of both androgen receptor and CYP17A1 enzyme(IC50s of 80 nM and 22 nM, respectively).Formula:C20H21F3N4Purity:98%Color and Shape:SolidMolecular weight:374.40MT-7716 hydrochloride
CAS:MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)Formula:C27H29ClN4O2Purity:98%Color and Shape:SolidMolecular weight:477(S,S)-J-113397
CAS:(S,S)-J-113397 is an isomer of J-113397 . J-113397 is an Opioid Receptor antagonist [1] .Formula:C24H37N3O2Color and Shape:SolidMolecular weight:399.57GPR88 agonist 2
GPR88 agonist 2 (compound 53) serves as a potent, brain-penetrant agonist of GPR88, exhibiting an EC50 of 14 µM in the GPR88 cAMP functional assay [1].Color and Shape:Odour SolidGalloylalbiflorin
CAS:Galloylalbiflorin, an AR antagonist with IC50 53.3μM, is sourced from Paeonia lactiflora roots, exhibiting anti-androgenic properties.Formula:C30H32O15Color and Shape:SolidMolecular weight:632.57TD-802
CAS:TD-802, an AR-targeting PROTAC with microsomal stability, shows promise for castration-resistant prostate cancer.Formula:C52H61ClN10O6Color and Shape:SolidMolecular weight:957.56GNE-502
CAS:GNE-502 is an orally active and potent estrogen receptor (ER) degrader, specifically designed for research on breast cancer.Formula:C25H30FN3O3SColor and Shape:SolidMolecular weight:471.59Clocinnamox mesylate
CAS:Clocinnamox mesylate: irreversible μ-opioid blocker; Ki: 0.7 nM (mouse μ), 1.9 nM (δ), 5.7 nM (κ).Formula:C30H33ClN2O7SColor and Shape:SolidMolecular weight:601.11CP 85339
CAS:CP 85339 is an aspartic acid protease inhibitor for X-ray analysis of peptide-renin complexes.Formula:C31H49ClN4O6SColor and Shape:SolidMolecular weight:641.26PSDalpha
PSDalpha, a conjugate of PS, TB, and 17β-estradiol, degrades ERα with peak absorption at 465 nm, effectively inhibiting MCF-7 cell growth.Formula:C44H39N3O2SColor and Shape:SolidMolecular weight:673.86Bufrolin
CAS:Bufrolin is a potent GPR35 agonist, mast cell stabilizer, and anti-inflammatory research agent.Formula:C18H16N2O6Color and Shape:SolidMolecular weight:356.33[Met5]-Enkephalin, amide
CAS:[Met5]-Enkephalin, amide activates δ and ζ opioid receptors; has multiple forms and varying plasma levels.Formula:C27H36N6O6SPurity:98%Color and Shape:SolidMolecular weight:572.68Angiotensin II (1-4), human
CAS:Angiotensin II constricts blood vessels and boosts blood pressure by escalating norepinephrine release.Formula:C24H37N7O8Purity:98%Color and Shape:SolidMolecular weight:551.59Glucocorticoids receptor agonist 2
CAS:Arylpyrazole-based glucocorticoid agonist with potent anti-inflammatory effects; doesn't affect insulin secretion.Formula:C25H25FN2OColor and Shape:SolidMolecular weight:388.48PD 125967
CAS:PD 125967 is a renin inhibitor, which represents a group of pharmaceutical drugs used primarily to treat essential hypertension.Formula:C51H67N5O4Color and Shape:SolidMolecular weight:814.111-Methyl-2-[(6Z,9Z)-6,9-pentadecadienyl]-4(1H)-quinolone
CAS:Methyl-2-quinolone from Evodia rutaecarpa blocks angiotensin II receptor with 48.2 μM IC50.Formula:C25H35NOColor and Shape:SolidMolecular weight:365.55PD 132002
CAS:PD 132002 is a renin inhibitor.Formula:C31H50N4O9SColor and Shape:SolidMolecular weight:654.82Boc-ypgflt(O-tbu)
CAS:Boc-ypgflt(O-tbu) is a delta-receptor-selective opioid antagonist.Formula:C44H64N6O11Color and Shape:SolidMolecular weight:853.01Faznolutamide
CAS:Faznolutamide is an antiandrogen agent [1] [2] .Formula:C19H17FN4O2SColor and Shape:SolidMolecular weight:384.43PROTAC ERα Y537S degrader-1
CAS:PROTAC ERα Y537S degrader-1 comprises a ubiquitin E3 ligase binding group, a linker and a protein binding group.Formula:C46H49N5O6Color and Shape:SolidMolecular weight:767.91(Rac)-SNC80
CAS:(Rac)-SNC80, a racemic δ-opioid agonist (K i 1.78 nM), shows potential for treating various headache disorders.Formula:C28H39N3O2Color and Shape:SolidMolecular weight:449.63[Ala17]-MCH
CAS:Potent MCH receptor agonist with EC50 of 17 nM (MCH1) & 54 nM (MCH2); prefers MCH1 (Ki 0.16 nM) over MCH2 (Ki 34 nM).Formula:C97H155N29O26S4Purity:98%Color and Shape:SolidMolecular weight:2271.71Raloxifene 4-Monomethyl Ether
CAS:Raloxifene 4-Monomethyl Ether (Compound 37), an estrogen receptor α inhibitor, has an IC50 of 1 μM against MCF-7 cells.Formula:C29H29NO4SColor and Shape:SolidMolecular weight:487.61Saralasin
CAS:Competitive non-selective angiotensin II antagonist.Formula:C42H65N13O10Purity:98%Color and Shape:PowderMolecular weight:912Triamcinolone Benetonide
CAS:Triamcinolone benetonide is a synthetic glucocorticoid corticosteroid exhibiting potent anti-inflammatory properties.Formula:C35H42FNO8Purity:98%Color and Shape:SolidMolecular weight:623.71Ac-RYYRWK-NH2
CAS:Selective NOP receptor partial agonist peptide; Ki=0.71 nM; >4000 nM for μ, δ, κ receptors; boosts food intake in vivo.Formula:C49H69N15O9Purity:98%Color and Shape:SolidMolecular weight:1012.17AZ'6421
CAS:"AZ'6421: A PROTAC degrading estrogen receptor alpha; potent in anti-tumor activity, useful for cancer research."Formula:C52H65F3N6O7SColor and Shape:SolidMolecular weight:975.17Naldemedine
CAS:Naldemedine (S 297995), developed by Shionogi, is a drug for opioid side effects like constipation. It's well tolerated with minor GI issues.Formula:C32H34N4O6Color and Shape:SolidMolecular weight:570.64BigLEN(rat)
CAS:Potent GPR171 agonist (EC50 = 1.6 nM). ProSAAS-derived peptide. Regulates body weight in mice and promotes the outgrowth of neurites in Neuro2A cells.Formula:C76H128N24O23Purity:98%Color and Shape:SolidMolecular weight:1746ER degrader 5
CAS:ER degrader 5: potent ER degrader, anti-cancer, for breast cancer research.Formula:C26H18F2O4SColor and Shape:SolidMolecular weight:464.48C-Type Natriuretic Peptide (1-53), human
CAS:CNP, from natriuretic family, first in pigs, now in other species, processes into CNP-22/CNP-53, similar to ANP/BNP, with varying potencies.Formula:C251H417N81O71S3Purity:98%Color and Shape:SolidMolecular weight:5801.77RLA-5331
RLA-5331: iron activator with anti-androgen properties; inhibits mCRPC cell proliferation.Formula:C40H43F3N6O7SColor and Shape:SolidMolecular weight:808.87PD 123177
CAS:PD 123177 is an inhibitor of Nonpeptide angiotensin AII-2.Formula:C29H28N4O3Purity:98%Color and Shape:SolidMolecular weight:480.56AKR1Cs-IN-1
AKR1Cs-IN-1 (Compound 29) is an effective and broad-spectrum inhibitor of the Aldo-Keto Reductase 1C family (AKR1C1-1C4). It achieves subtype inhibition by simultaneously binding to the SP2 and SP3 pockets, thereby blocking metabolic pathways related to drug resistance. In enzyme assays, AKR1Cs-IN-1 exhibits significant inhibitory activity with IC50 values of 0.09, 0.28, 0.05, and 0.51 µM for AKR1C1, AKR1C2, AKR1C3, and AKR1C4, respectively. The compound shows excellent resensitizing effects in doxorubicin (DOX)-resistant breast cancer cell line MCF-7/ADR, effectively enhancing the cytotoxicity of DOX. AKR1Cs-IN-1 holds promise for research on breast cancer resistance.Color and Shape:Odour Solid[Orn8]-Urotensin II
CAS:[Orn8]-Urotensin II is a Urotensin receptor ligand and a partial agonist at Urotensin receptors.Formula:C63H83N13O18S2Color and Shape:SolidMolecular weight:1374.5517-Epiestriol
CAS:17-Epiestriol, metabolite of estrone, forms via 16α-hydroxy intermediate and binds ERα and ERβ with affinity less than 17β-estradiol.Formula:C18H24O3Purity:99.72%Color and Shape:SolidMolecular weight:288.38Emd 55068
CAS:Emd 55068 is a synthetic antagonist of renin.Formula:C41H65N9O6Color and Shape:SolidMolecular weight:780.01(S)-CVN424
CAS:(S)-CVN424 modulates GPR6, key for neurological/psychiatric research, including Parkinson's.Formula:C24H29F2N5O3Color and Shape:SolidMolecular weight:473.525Nocistatin
CAS:Nocistatin, a neuropeptide, blocks Nociceptin effects and inhibits 5-HT release, acting on an opioid-related receptor.Formula:C32H56N10O12Color and Shape:SolidMolecular weight:772.85Helianorphin-19
Helianorphin-19: Potent KOR agonist (Ki=25 nM; EC50=45 nM), 200x selective over μ/δ receptors, effective in mouse pain model, non-sedative.Color and Shape:LiquidTRV056
CAS:TRV056 is a Gq-biased AT1R agonist effective in Gq-mediated signaling and a basis for similar drug development.Formula:C52H74N14O13Color and Shape:SolidMolecular weight:1103.249β-Lipotropin (60-65)
CAS:β-Lipotropin (60-65) (β-LPH (60-65)), an opioid agonist, is a significant [1] opioid peptide.Formula:C33H47N9O8SColor and Shape:SolidMolecular weight:729.85DP32
CAS:DP32 is a dual-function compound incorporating an opioid receptor (MOP) agonist and a neuropeptide FF receptor (NPFFR) antagonist. It is applicable in analgesia-related research.Formula:C57H77N13O7Color and Shape:SolidMolecular weight:1056.30[DAla2, DArg6] Dynorphin A, (1-13) (porcine)
CAS:'[DAla2, DArg6] Dynorphin A (1-13) porcine is a potent opioid peptide resistant to enzymatic degradation.'Formula:C76H128N24O15Color and Shape:SolidMolecular weight:1617.98β-Endorphin (rat)
CAS:β-Endorphin (β-EP) is an endogenous opioid neuropeptide with diverse biological activities.Formula:C157H254N42O44SColor and Shape:SolidMolecular weight:3466.07Dynorphin B (1-13) (TFA)
Dynorphin B (1-13) TFA acts as an agonist on opioid κ-receptor .Formula:C76H116N21F3O19Color and Shape:SolidMolecular weight:1684.86Kylo-0603
CAS:KYLO-0603 is an orally active and selective THR-β agonist with an EC50 of 31.07 nM. It effectively reduces serum cholesterol and low-density lipoprotein cholesterol levels. By activating THR-β receptors, KYLO-0603 enhances the expression of THR-regulated genes like iodothyronine deiodinase 1 (Dio1), malic enzyme 1 (Me1), and thyroid hormone-responsive (Thrsp) gene, while it inhibits the expression of inflammatory and fibrosis-related genes, including low-density lipoprotein receptor (LDL-R) gene. This compound is applicable for the study of metabolic associated steatohepatitis (MASH) and liver fibrosis.Formula:C81H134N8O28Color and Shape:SolidMolecular weight:1667.97(N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8)
CAS:E-2078, known chemically as (N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8), is a stable analog of Dynorphin A (1–8) and functions as a kappa opioidFormula:C50H81N15O9Color and Shape:SolidMolecular weight:1036.27PRL 3195
CAS:PRL 3195: Somatostatin antagonist, Ki: 6 nM (sst5), 17 nM (sst2), 66 nM (sst3), 1 μM (sst1/4).Formula:C58H69ClN12O9S2Color and Shape:SolidMolecular weight:1177.83ALR2-IN-6
ALR2-IN-6 (compound 9) is a potent competitive inhibitor of ALR2, with a Ki value of 0.064 μM. It is applicable in research related to neuropathy, retinopathy, and nephropathy.Formula:C21H19BrFN3OColor and Shape:SolidMolecular weight:427.06955Prepro-TRH-(160-169)
CAS:Prepro-TRH-(160-169), a pro-TRH peptide, enhances TRH-stimulated TSH secretion.Formula:C54H75N11O18SColor and Shape:SolidMolecular weight:1198.3THR-β agonist 2 diacetate
THR-β agonist 2 diacetate (Compound 3) is a potent THR-β agonist with potential applications in researching metabolic disorders such as obesity, hyperlipidemia, hypercholesterolemia, and diabetes, as well as other conditions like steatosis and non-alcoholic steatohepatitis (NASH), atherosclerosis, and other related diseases and conditions.Color and Shape:Odour SolidAc-RYYRWK-NH2 TFA
CAS:Ac-RYYRWK-NH2: potent, specific NOP receptor partial agonist with 0.071 nM affinity; no affinity for μ/κ/δ-opioid receptors.Formula:C51H70F3N15O11Color and Shape:SolidMolecular weight:1126.21PROTAC ERα Degrader-7
CAS:PROTAC ERα Degrader-7 (Compound i-320) is a powerful PROTAC degrader targeting the estrogen receptor alpha (ERα), exhibiting a DC50 of 0.000006 µM. This compound consists of a cereblon-binding segment, LBM, connected to ERBM, an ERα-binding ligand that includes a benzofused partially saturated 6-membered carbocyclic or heterocyclic ring [1].Formula:C46H49F2N5O4Color and Shape:SolidMolecular weight:773.91Melanin Concentrating Hormone, salmon TFA
MCH (salmon) TFA is a 19-amino-acid neuropeptide affecting appetite, energy, sleep, and heart health via GPCR SLC-1/GPR24 and MCHR2.Formula:C91H140F3N27O26S4Color and Shape:SolidMolecular weight:2213.5Aclerastide
CAS:Aclerastide, an angiotensin receptor agonist, decreases fibrosis in wounds; effect increases with use duration, blocked by AT antagonist.Formula:C42H64N12O11Color and Shape:SolidMolecular weight:913.03PROTAC ERα Degrader-8
CAS:PROTAC ERα Degrader-8 (compound ii-56), a highly potent degrader of Erα, achieves a DC50 of just 0.000006 μM in MCF7 cells [1].Formula:C47H51N5O4Color and Shape:SolidMolecular weight:749.94[Nphe1]Nociceptin(1-13)NH2 TFA
[Nphe1]Nociceptin(1-13)NH2 is a selective nociceptin receptor antagonist with potential analgesic properties, pKi=8.4, pA2=6.0.Formula:C63H101F3N22O17Color and Shape:SolidMolecular weight:1495.61Floramanoside C
CAS:Floramanoside C exhibits 2,2-diphenyl-1-picrylhydrazyl scavenging and aldose reductase inhibitory activities [1].Formula:C21H18O15Color and Shape:SolidMolecular weight:510.36[Ala17]-MCH TFA
'[Ala17]-MCH TFA is an MCH analogue, a selective MCHR1 ligand (Ki=0.16 nM) with high affinity (Kd=0.37 nM), and low MCHR2 affinity (Ki=34 nM).Formula:C99H156F3N29O28S4Color and Shape:SolidMolecular weight:2385.73MCH(human, mouse, rat) TFA
MCH TFA, a peptide, selectively binds MCH1R and MCH2R with IC50 of 0.3nM, 1.5nM; EC50s are 3.9nM (MCH1R) and 0.1nM (MCH2R) in CHO cells.Formula:C107H161F3N30O28S4Color and Shape:SolidMolecular weight:2500.86Abaloparatide
CAS:Abaloparatide (BA 058) is a selective PTHR1 analog that promotes bone growth and may be researched for osteoporosis.Formula:C174H300N56O49Color and Shape:SolidMolecular weight:3960.59hFSH-β-(33-53) (TFA)
hFSH-β-(33-53) TFA, a thiol-containing peptide representing the second follicle-stimulating hormone receptor (FSHR) binding domain, acts as an FSHR antagonist.Formula:C115H183N31O32SxC2HF3O2Color and Shape:SolidMolecular weight:2657.96Yp537
CAS:Yp537 acts as an estrogen receptor (ER) inhibitor, specifically preventing the dimerization of the human estrogen receptor [1].Formula:C64H104N13O22PSColor and Shape:SolidMolecular weight:1470.62(d(CH2)51,Tyr(Me)2,Thr4,Orn8,des-Gly-NH29)-Vasotocin
CAS:'(d(CH2)51,Tyr(Me)2,Thr4,Orn8,des-Gly-NH29)-Vasotocin blocks oxytocin receptors, stopping oxytocin effects on CA1 neuron currents.'Formula:C45H69N9O12S2Color and Shape:SolidMolecular weight:992.21Eprosartan
CAS:Eprosartan is a selective AT1 receptor blocker with IC50s of 9.2 nM (rat) and 3.9 nM (human), used for hypertension.Formula:C23H24N2O4SPurity:99.99%Color and Shape:SolidMolecular weight:424.51TrxR1 prodrug-1
TrxR1 prodrug-1 (compound 5u) is a potent inhibitor of TrxR1, demonstrating significant antitumor activity in nude mice and NSCLC organoids.Formula:C22H30N2O6S2Color and Shape:SolidMolecular weight:482.6139,10-Dihydrophenanthrene
CAS:9,10-Dihydrophenanthrene has inhibitory activity against the androgen receptor and can be used in related research in the field of life sciences.Formula:C14H12Purity:98.76%Color and Shape:SolidMolecular weight:180.25DDHF20
DDHF20 is an inhibitor of Staphylococcus aureus, specifically targeting and inhibiting its thioredoxin reductase (TrxR) by acting as a competitive inhibitor at the NADPH binding site. DDHF20 shows potential for research in combating infections related to Staphylococcus aureus.Formula:C34H28O4Color and Shape:SolidMolecular weight:500.58Rimexolone
CAS:Rimexolone is a glucocorticoid steroid used to treat inflammation in the eye.Formula:C24H34O3Color and Shape:SolidMolecular weight:370.52Tetrahydro Aldosterone
CAS:Tetrahydro Aldosterone is a steroidal compound that inhibits the adrenal angiotensin II receptor, with an IC50 of 10 μM.Formula:C21H32O5Color and Shape:SolidMolecular weight:364.48PRL 2915
CAS:PRL 2915 is a potent antagonist of the human somatostatin subtype 2 receptor (hsst 2), exhibiting a binding affinity (K_i) of 12 nM [1].Formula:C59H71ClN12O8S2Color and Shape:SolidMolecular weight:1175.85PRO20
PRO20 is a specific and competitive antagonist of the (pro)renin receptor (PRR). It inhibits the calcium influx induced by Proproin with an IC50 value of 81 nmol/L. By blocking the binding of Prorenin to PRR, PRO20 inhibits the activation of the renin-angiotensin system (RAS), reducing the production of angiotensin II (Ang II) and exerting antihypertensive effects. PRO20 holds promise for research in antihypertensive agents.
Color and Shape:Odour SolidDPC-AJ1951 TFA
DPC-AJ1951 TFA is a 14 amino acid peptide, potent PTH/PPR agonist, tested in bone resorption assays.Formula:C78H128F3N23O21Color and Shape:SolidMolecular weight:1781.02(Glu2)-TRH
CAS:(Glu2)-TRH: Stable TRH analog; reduces TRH's cholinergic action; no thyroliberinase metabolism; neuroprotective with antidepressant, anticonvulsant effects.Formula:C15H22N4O6Color and Shape:SolidMolecular weight:354.36Osteostatin
CAS:Osteostatin, derived from parathyroid hormone-related protein (PTHrP) 107-111, has demonstrated properties conducive to bone repair in animal models presentingFormula:C27H41N9O8Color and Shape:SolidMolecular weight:619.677α-(Thiomethyl)spironolactone
CAS:7α-(Thiomethyl)spironolactone is a steroid receptor antagonist and major spironolactone metabolite, steroid metabolism, nuclear receptor, and coronavirus.Formula:C23H32O3SPurity:>99.99%Color and Shape:SolidMolecular weight:388.56NPFF1-R antagonist 1
NPFF1-R antagonist 1 (compound 8b) is a piperidine analog and an effective neuropeptide FF (NPFF) receptor antagonist. It exhibits 15-fold selectivity for the NPFF1-R subtype, with Ki values of 211 nM and 3270 nM for NPFF1-R and NPFF2-R, respectively.Formula:C37H44N4OMolecular weight:560.35151VinclozolinM2-2204
VinclozolinM2-2204 is an androgen receptor AUTOTAC degrader with a DC50 of 200 nM in LNCaP prostate cancer cells. It induces the formation of AR+LC3+ autophagic membranes and is applicable for cancer research.Formula:C43H51Cl2N3O9Molecular weight:823.30024DP50
DP50 is a bifunctional compound containing both an opioid receptor agonist (MOP) and a neuropeptide FF receptor (NPFFR) antagonist. It can be utilized in studies related to analgesia.Formula:C58H72N8O7Molecular weight:992.5524PIPE-3297
PIPE-3297 (compound 25) is a selective kappa opioid receptor (KOR) agonist that activates the G protein signaling pathway with an EC50 of 1.1 nM and exhibits low β-arrestin-2 recruitment activity (10%). Additionally, PIPE-3297 promotes myelination and has anti-inflammatory properties.Formula:C23H30N2OMolecular weight:350.23581Nurr1 agonist 9
Nurr1 agonist 9 (Compound 36) acts as an agonist for Nurr1, with an EC50 of 0.090 µM and a Kd of 0.17 µM. It activates Nurr1 homodimers (NurRE, EC50 = 0.094 µM) and Nurr1-RXR heterodimers (DR5, EC50 = 0.165 µM). This compound induces the expression of Nurr1-regulated tyrosine hydroxylase (TH) in Parkinson's disease organoid models and can penetrate the human brain endothelial cell barrier.
Formula:C21H19ClN4O2Molecular weight:394.11965Awl 60
CAS:Awl 60 is a substance P (6-11) non-competitive antagonist.Formula:C57H65N9O8SPurity:98%Color and Shape:SolidMolecular weight:1036.25SB 205607 dihydrobromide
CAS:non-peptide δ1 opioid receptor agonistFormula:C23H24N2OPurity:98%Color and Shape:SolidMolecular weight:344.45Ethamoxytriphetol
CAS:Ethamoxytriphetol is a non-steroidal estrogen antagonist.Formula:C27H33NO3Color and Shape:SolidMolecular weight:419.56Bradykinin potentiator-5
CAS:Bradykinin potentiator-5 is a peptide inflammatory mediator, causes blood vessels to dilate (enlarge), and therefore causes blood pressure to fall.Formula:C30H41N7O7Purity:98%Color and Shape:SolidMolecular weight:611.69Enalapril
CAS:Enalapril is a dicarbocyl-containing peptide and angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.Formula:C20H28N2O5Purity:99.47% - 99.51%Color and Shape:SolidMolecular weight:376.455-O-β-D-Glucopyranosylmyricanol
5-O-beta-D-Glucopyranosylmyricanol is a useful organic compound for research related to life sciences and the catalog number is T123967.Formula:C27H36O10Color and Shape:SolidMolecular weight:520.575RU-39411
CAS:RU-39411 is a steroidal anti-estrogen.Formula:C28H37NO3Purity:98%Color and Shape:SolidMolecular weight:435.60Acetiromate
CAS:Acetiromate is a drug of antilipidemic. It is used to treat hyperlipidemia.Formula:C15H9I3O5Purity:98%Color and Shape:SolidMolecular weight:649.94LY301875
CAS:LY301875 is an antagonist of nonpeptide angiotensin receptor.Formula:C31H36N4O10SColor and Shape:SolidMolecular weight:656.70AT2R antagonist 2
Compound I-16 (AT2R antagonist 2) is an orally active AT2R antagonist.Formula:C20H23F3N8SColor and Shape:SolidMolecular weight:464.51TRIP13-IN-1
TRIP13-IN-1 (compound 20) is a potent ligand and inhibitor of TRIP13, demonstrating anticancer effects both in vivo and in vitro.Formula:C24H25NO9SColor and Shape:SolidMolecular weight:503.52
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