Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(207 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(49 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(296 products)
- Prostaglandin Receptor(119 products)
- RAAS(86 products)
- Reductase(52 products)
- Somatostatin(46 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
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Found 3178 products of "Endocrinology/Hormones"
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GPR119 agonist 2
CAS:<p>GPR119 agonist 2 (compound 43), an orally active agonist of GPR119, exhibits favorable pharmacokinetic properties in rodents and has demonstrated efficacy in</p>Formula:C23H24FN5O4S2Color and Shape:SolidMolecular weight:517.6Biotin-cholesterol
CAS:<p>Biotin-cholesterol, a biotinylated derivative of cholesterol, serves as a precursor in the manufacturing of biotin-conjugated liposomes and micelles, which are utilized in drug delivery systems [1].</p>Formula:C37H60N2O3SColor and Shape:SolidMolecular weight:612.95GPR88-IN-1
CAS:<p>GPR88-IN-1 is a GPR88 antagonist that may be utilized for the study of central nervous system disorders [1].</p>Formula:C25H28N4O2Color and Shape:SolidMolecular weight:416.52LX-039
CAS:<p>LX-039: Selective oral estrogen receptor degrader with EC50 of 2.99 nM, antitumor activity, C-3 indole chloride, and robust mouse pharmacokinetics.</p>Formula:C27H20Cl2FNO2Color and Shape:SolidMolecular weight:480.36DPP-4/GPR119 modulator 2
CAS:<p>DPP-4/GPR119 modulator 2 is an inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 0.22 μM) and an agonist of GPR119 (EC50: 0.95 μM).</p>Formula:C30H40N8O3Color and Shape:SolidMolecular weight:560.69Nylestriol
CAS:<p>Nylestriol (LY 49825) is an agonist of estrogen receptor.</p>Formula:C25H32O3Purity:98.88%Color and Shape:SolidMolecular weight:380.52TRβ agonist 3
CAS:<p>TRβ agonist 3 (Compound 3) is a potent TRβ agonist that is a new potential TRβ-selective thyromimetics.</p>Formula:C20H25NO3Color and Shape:SolidMolecular weight:327.42RU 58668
CAS:<p>Pure antiestrogen that downregulates estrogen receptor expression</p>Formula:C34H43F5O5SPurity:98%Color and Shape:SolidMolecular weight:658.76VPC-14228
CAS:<p>VPC-14228 is a specific AR-DBD inhibitor that acts by inhibiting both Y594A and Q592A mutants.</p>Formula:C13H14N2OSPurity:99.96%Color and Shape:SolidMolecular weight:246.33Dexamethasone palmitate
CAS:<p>DXP, a lipophilic prodrug of Dexamethasone, has 47x less glucocorticoid receptor affinity; it's an agonist & anti-inflammatory.</p>Formula:C38H59FO6Purity:99.28%Color and Shape:SolidMolecular weight:630.87(rel)-BMS-641988
CAS:<p>(rel)-BMS-641988, a relative configuration of the potent nonsteroidal androgen receptor antagonist BMS-641988, holds potential for prostate cancer research.</p>Formula:C20H20F3N3O5SPurity:98%Color and Shape:SolidMolecular weight:471.45BMS-814580
CAS:<p>BMS-814580: potent MCHR1 antagonist, Kb 117 nM, Ki 17 nM (human), 4.9/11.5 nM (monkey/rat), reduces feeding/weight in rodents.</p>Formula:C24H19ClF2N2O4SColor and Shape:SolidMolecular weight:504.93LY2922470
CAS:<p>LY2922470: Selective GPR40 agonist; EC50=7nM (human), 1nM (mouse), 3nM (rat); lowers glucose, boosts insulin/GLP-1.</p>Formula:C28H29NO4SPurity:95.11% - 97.08%Color and Shape:SolidMolecular weight:475.6Naloxonazine
CAS:<p>Naloxonazine, a potent, selective opiate mu-1 (μ1) antagonist, also influences leishmania through the modulation of host coding function.</p>Formula:C38H42N4O6Color and Shape:SolidMolecular weight:650.76MK-386
CAS:<p>MK-386 is a potent and selective inhibitor of human type-1 5alpha-reductase.</p>Formula:C28H49NOColor and Shape:SolidMolecular weight:415.69RU28362
CAS:<p>RU28362 is an agonist of glucocorticoid receptor.</p>Formula:C23H28O3Color and Shape:SolidMolecular weight:352.47TP-051
CAS:<p>TP-051 is a FFAR1 agonist.</p>Formula:C29H31FO6SColor and Shape:SolidMolecular weight:526.62Deltakephalin
CAS:<p>Deltakephalin is a synthetic, potent specific opiate delta receptors agonist.</p>Formula:C34H48N6O10Purity:98%Color and Shape:SolidMolecular weight:700.78LY2922083
CAS:<p>LY2922083: Potent, selective GPR40 agonist; lowers glucose, boosts insulin and GLP-1.</p>Formula:C31H33NO3SColor and Shape:SolidMolecular weight:499.66SNC 162
CAS:<p>SNC 162 is a potent and selective delta-opioid receptor (δ-opioid) agonist with analgesic, antidepressant and antiarrhythmic effects.</p>Formula:C27H37N3OPurity:98%Color and Shape:SolidMolecular weight:419.6PF 00277343
CAS:<p>PF 00277343, a thyroid receptor agonist, is used for the treatment of androgenetic alopecia.</p>Formula:C24H20FN3O4Purity:98%Color and Shape:SolidMolecular weight:433.43BI-2081
CAS:<p>BI-2081: GPR40 agonist, EC50=4nM, boosts insulin, lowers blood glucose, potential for type 2 diabetes research.</p>Formula:C32H35FO6Color and Shape:SolidMolecular weight:534.62Firuglipel
CAS:<p>Firuglipel is an orally available and selective agonist of GPR119.</p>Formula:C25H26FN3O5Purity:98%Color and Shape:SolidMolecular weight:467.49Azilsartan mopivabil
CAS:<p>Azilsartan mopivabil is the potent antagonist of angiotensin II receptor .</p>Formula:C38H36N4O8Color and Shape:SolidMolecular weight:676.71MK-7246
CAS:<p>MK-7246 is a potent and specific CRTH2 antagonist (Ki: 2.5 nM).</p>Formula:C21H21FN2O4SColor and Shape:SolidMolecular weight:416.47SPH3127
CAS:<p>SPH3127 is a potent oral direct renin inhibitor, effective at 0.4 nM for human renin, used to study hypertension.</p>Formula:C22H32N6O4Color and Shape:SolidMolecular weight:444.53Taragarestrant
CAS:<p>Taragarestrant (D-0502), an oral estrogen receptor degrader, combats ER+ breast cancer in research.</p>Formula:C25H25Cl2FN2O2Color and Shape:SolidMolecular weight:475.38JJH260
CAS:<p>JJH260, a N-hydroxy hydantoin carbamate, inhibits AIG1 and ADTRP with IC50 values of 0.57 μM and 8.5 μM, respectively, and targets ABHD6, LYPLA1/2.</p>Formula:C29H34ClN5O5Color and Shape:SolidMolecular weight:568.06Imlunestrant
CAS:<p>Imlunestrant (LY-3484356) is an orally active, selective estrogen receptor degrader that persistently inhibits ER-dependent gene transcription and cell growth.</p>Formula:C29H24F4N2O3Purity:97.35%Color and Shape:SolidMolecular weight:524.51AMG 837
CAS:<p>Prinaberel (ERB 041) is an ERβ agonist with anticancer activity and anti-inflammatory activity that inhibits the NFκB pro-inflammatory signaling pathway.</p>Formula:C26H21F3O3Purity:98%Color and Shape:SolidMolecular weight:438.44AM-1638
CAS:<p>AM-1638 is an orally active GPR40/FFA1 agonist, useful for studying type II diabetes.</p>Formula:C33H35FO4Color and Shape:SolidMolecular weight:514.63LY303336
CAS:<p>LY303336 is an antagonist of AT1 receptor.</p>Formula:C30H37N4O11PSPurity:98%Color and Shape:SolidMolecular weight:692.67LGD-2941
CAS:<p>LGD-2941 is an androgen receptor modulator. LGD-2941 is used for the treatment of hypogonadism, female sexual dysfunction and menopausal syndrome.</p>Formula:C17H16F6N2O2Color and Shape:SolidMolecular weight:394.31MK-8666 Tris
CAS:<p>MK-8666, a partial GPCR agonist, targets GPR40 to enhance insulin secretion, potentially treating type 2 diabetes without adverse effects.</p>Formula:C33H42N2O9SColor and Shape:SolidMolecular weight:642.7648,11-Eicosadiynoic acid
CAS:<p>8,11-Eicosadiynoic acid, an unsaturated fatty acid, functions as a steroid 5α-reductase inhibitor and has applications in acne research [1].</p>Formula:C20H32O2Color and Shape:SolidMolecular weight:304.47DPI-3290
CAS:<p>DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent</p>Formula:C30H34FN3O2Purity:98%Color and Shape:SolidMolecular weight:487.61Androgen receptor antagonist 5
CAS:<p>AR antagonist 5 blocks AR (IC50: 6.17 μM), hinders LNCaP cell growth, and has anti-tumor effects in mouse models.</p>Formula:C21H15F4N5O3SColor and Shape:SolidMolecular weight:493.43Trap-101 hydrochloride
CAS:<p>nociceptin/orphanin FQ (NOP) receptor antagonist</p>Formula:C24H36ClN3O2Purity:98%Color and Shape:SolidMolecular weight:434.02EPI-7170
CAS:<p>EPI-7170: Ralaniten analogue, blocks androgen receptor, inhibits transcription in AR & variants, fights enzalutamide-resistant prostate cancer.</p>Formula:C22H28Cl3NO6SColor and Shape:SolidMolecular weight:540.88TA-606
CAS:<p>TA-606 is an angiotensin type 1 receptor antagonist with antihypertensive activity.</p>Formula:C33H40ClN7O6Color and Shape:SolidMolecular weight:666.17ER degrader 1
CAS:<p>ER degrader 1 targets estrogen receptor, crucial for cell regulation; shows promise in cancer therapy. (Patent WO2021139756A1, compound 11)</p>Formula:C26H32F4N4O3Color and Shape:SolidMolecular weight:524.55MCHR1 antagonist 3
CAS:<p>MCHR1 antagonist 3, a potent antagonist of the melanin-concentrating hormone receptor-1 (MCHR1), is employed for the regulation of energy metabolism.</p>Formula:C29H36N4O2Purity:98%Color and Shape:SolidMolecular weight:472.62GPR40 Agonist 2
CAS:<p>GPR40 Agonist 2 is a GPR40 agonist. It can be used in the research of diabetes.</p>Formula:C24H30O3Purity:98%Color and Shape:SolidMolecular weight:366.49RTI-13951-33
CAS:<p>RTI-13951-33 is an effective and brain-penetrant GPR88 agonist (EC50: 25 nM, in GPR88 cAMP functional assay).</p>Formula:C28H33N3O3Purity:98%Color and Shape:SolidMolecular weight:459.58Amebucort
CAS:<p>Amebucort is a synthetic glucocorticoid corticosteroid. It may used for the research of inflammatory disorders.</p>Formula:C28H40O7Purity:98%Color and Shape:SolidMolecular weight:488.61ES 8891
CAS:<p>ES 8891 is an inhibitor of renin.</p>Formula:C42H60N6O6SPurity:98%Color and Shape:SolidMolecular weight:777.03Elisartan
CAS:<p>Elisartan is a non-peptide pro-drug of angiotensin II AT1 receptor antagonist HN-12206. It also shows anti-hypertension activities.</p>Formula:C27H29ClN6O5Purity:98%Color and Shape:SolidMolecular weight:553.01GPR120 Agonist 1
CAS:<p>GPR120 Agonist 1 selectively activates human/mouse GPR120 with EC50 of 42/77 nM in HEK293 cells.</p>Formula:C20H12ClF6NO3SPurity:98%Color and Shape:SolidMolecular weight:495.82R-84760 hydrochloride
CAS:<p>R-84760, a potent κ-opioid receptor agonist, relieves tonic pain via supraspinal/spinal pathways, activating noradrenergic descent.</p>Formula:C19H25Cl3N2OSColor and Shape:SolidMolecular weight:435.84Fosdagrocorat
CAS:<p>Fosdagrocorat is an agonist of the dissociated glucocorticoid receptor.</p>Formula:C29H30F3N2O5PColor and Shape:SolidMolecular weight:574.53Estrogen receptor antagonist 5
CAS:<p>Compound 165: Potent estrogen receptor antagonist; useful for metastatic disease research.</p>Formula:C25H31F3N2O3Color and Shape:SolidMolecular weight:464.52GSK 1440115
CAS:<p>GSK 1440115, an orally active urotensin II receptor antagonist, is used to treat asthma.</p>Formula:C30H29Cl2N3O6Purity:98%Color and Shape:SolidMolecular weight:598.47(1S,3R)-GNE-502
CAS:<p>(1S,3R)-GNE-502 degrades ERα in MCF7 cells; potent with EC50 of 13 nM; useful in estrogen-related cancer research.</p>Formula:C25H30FN3O3SColor and Shape:SolidMolecular weight:471.59JNJ-26146900
CAS:<p>JNJ-26146900 is a nonsteroidal androgen receptor (AR) ligand with tissue-selective activity in rats. JNJ-26146900 binds to the rat AR with a K(i) of 400nM.</p>Formula:C15H15F3N2O3SPurity:98%Color and Shape:SolidMolecular weight:360.35THRβ receptor agonist-1
CAS:<p>THRβ receptor agonist-1 is an agonist for the THRβ receptor [1].</p>Formula:C18H12Cl2N6O4Color and Shape:SolidMolecular weight:447.23THR-β modulator-1
CAS:<p>THR-β Modulator-1 (Compound 1a) is a potent modulator of the thyroid hormone receptor β, utilized in the study of thyroid hormone receptor-associated disorders</p>Formula:C17H14Cl2N6O4Color and Shape:SolidMolecular weight:437.24Dagrocorat
CAS:<p>Dagrocorat is a novel and dissociated agonist of glucocorticoid receptor.</p>Formula:C29H29F3N2O2Purity:98%Color and Shape:SolidMolecular weight:494.55GLL398
CAS:<p>GLL398: Oral ERα down-regulator, binds strongly (IC50=1.14nM), degrades ERα in MCF-7 cells (IC50=0.21μM).</p>Formula:C25H23BO4Color and Shape:SolidMolecular weight:398.26GPR120 Agonist 3
CAS:<p>GPR120 Agonist 3 (GPR120-IN-1) is a selective agonist of Gpr120 ( logEC50: -7.62).</p>Formula:C19H23ClF3NO3Purity:99.01%Color and Shape:SolidMolecular weight:405.84Prostaglandin E2-biotin
CAS:<p>Prostaglandin E2-biotin, an analog of prostaglandin, is utilized in the research of Nurr1-related diseases, including cancer and autoimmune diseases [1].</p>Formula:C35H58N4O6SColor and Shape:SolidMolecular weight:662.92Frakefamide
CAS:<p>Frakefamide: potent analgesic, μ-selective agonist, non-CNS penetrating.</p>Formula:C30H34FN5O5Purity:98%Color and Shape:SolidMolecular weight:563.62IP7e
CAS:<p>IP7e (isoxazolo-pyridinone 7e) is a Nurr1 activator with an EC50 value of 3.9 nM.</p>Formula:C23H22N2O4Purity:99.86%Color and Shape:SolidMolecular weight:390.43μ opioid receptor agonist 3
CAS:<p>Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.</p>Formula:C22H28N2O2Purity:98%Color and Shape:SolidMolecular weight:352.47Glucocorticoid receptor-IN-1
CAS:<p>Glucocorticoid receptor-IN-1 selectively modulates GR with anti-inflammatory effects, represses hMMP1 (IC50: 2.11 nM), and activates MMTV (EC50: 5.59 nM).</p>Formula:C24H19F4N7O2Color and Shape:SolidMolecular weight:513.45Icalcaprant
CAS:<p>Icalcaprant is a kappa-opioid receptor antagonist [1].</p>Formula:C23H26N4O3Purity:98%Color and Shape:SolidMolecular weight:406.48Fulvestrant (R enantiomer)
CAS:<p>Fulvestrant R enantiomer is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.</p>Formula:C32H47F5O3SPurity:98%Color and Shape:SolidMolecular weight:606.77Mu opioid receptor antagonist 7
CAS:<p>Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (</p>Formula:C22H27ClN2O2Purity:98%Color and Shape:SolidMolecular weight:386.91Glucocorticoid receptor agonist
CAS:<p>Glucocorticoid receptor agonist is an effective glucocorticoid receptor agonist.</p>Formula:C20H20F4N2O2Purity:98%Color and Shape:SolidMolecular weight:396.38Estrogen receptor antagonist 3
CAS:<p>ER antagonist 3 degrades ER, crucial in cell regulation; ER antagonist 4 may aid cancer research. (Patent WO2021213358A1, compound 7)</p>Formula:C26H29BF6N4O2Color and Shape:SolidMolecular weight:554.34Triiodothyronine Sulfate
CAS:<p>Triiodothyronine sulfate: Hypothyroidism prodrug, metabolizes into active thyroid hormone T3, binds and activates TRβ1.</p>Formula:C15H11I3NNaO7SPurity:98%Color and Shape:SolidMolecular weight:753.02PD 125754
CAS:<p>PD 125754 is a Renin inhibitor, which represents a group of pharmaceutical drugs used primarily to treat essential hypertension.</p>Formula:C42H65N5O7Purity:98%Color and Shape:SolidMolecular weight:751.99Estrogen receptor modulator 7
CAS:<p>Estrogen Receptor Modulator 7 is a potent modulator of estrogen receptors, utilized in cancer research [1].</p>Formula:C30H31BCl2FNO3Purity:98%Color and Shape:SolidMolecular weight:554.29H3B-6545
CAS:<p>H3B-6545 is a selective and oral estrogen receptor covalent antagonist (SERCA) used in the research of metastatic ER-positive, HER2-negative breast cancer.</p>Formula:C30H29F4N5O2Color and Shape:SolidMolecular weight:567.58L-368899 free base
CAS:<p>L-368899: non-peptide, oral oxytocin receptor antagonist (IC50: 8.9 nM), 40x more selective than vasopressin V1a/V2.</p>Formula:C26H42N4O5S2Purity:98%Color and Shape:SolidMolecular weight:554.77Naloxonazine dihydrochloride
CAS:<p>μ1 receptor antagonist</p>Formula:C38H43ClN4O6Purity:98%Color and Shape:SolidMolecular weight:687.22BE-26263
CAS:<p>BE-26263, an antiosteoporotic agent isolated from Scedosporium apiospermum, exhibits an estrogenic effect [1].</p>Formula:C32H38O14Color and Shape:SolidMolecular weight:646.64MCHR1 antagonist 2
CAS:<p>MCHR1 antagonist 2 is an antagonist of melanin-concentratin hormone receptor 1(MCH1-R, IC50 = 65 nM) and also inhibits hERG.</p>Formula:C23H21FN2O5Purity:98.29%Color and Shape:SolidMolecular weight:424.42Fulvestrant (S enantiomer)
CAS:<p>Fulvestrant S enantiomer is the less active S enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.</p>Formula:C32H47F5O3SPurity:98%Color and Shape:SolidMolecular weight:606.77SQ 32970
CAS:<p>SQ 32970 is a potent Endothia aspartic proteinase inhibitor.</p>Formula:C33H51N5O4SColor and Shape:SolidMolecular weight:613.85Nur77 modulator 2
CAS:<p>Nur77 modulator 2: Kd of 0.35 μM, oral anti-inflammatory, affects Nur77/mitochondria localization.</p>Formula:C26H25NO5Color and Shape:SolidMolecular weight:431.48CITFA
CAS:<p>CITFA, a GPER agonist, enhances neurite outgrowth in rat embryonic (E18) hippocampal neurons [1].</p>Formula:C25H35NO2Color and Shape:SolidMolecular weight:381.55Arzoxifene hydrochloride
CAS:<p>Arzoxifene hydrochloride is a selective estrogen receptor modulator that is a potent estrogen antagonist in mammary and uterine tissue.</p>Formula:C28H30ClNO4SPurity:98%Color and Shape:SolidMolecular weight:512.06AMG 837 sodium salt
CAS:<p>AMG 837 sodium salt: potent GPR40 agonist, EC50=13 nM; enhances insulin secretion; superior pharmacokinetics.</p>Formula:C26H21F3NaO3Purity:98%Color and Shape:SolidMolecular weight:461.436TR antagonist 1
CAS:<p>TR antagonist 1 is a highly potent thyroid hormone receptor (TR) antagonist that can be used to study diseases caused by endocrine abnormalities.</p>Formula:C25H23Br2NO4Purity:99.57%Color and Shape:SolidMolecular weight:561.26TC OT 39
CAS:<p>oxytocin receptor partial agonist</p>Formula:C32H40N8O2SPurity:98%Color and Shape:SolidMolecular weight:600.78Spirorenone
CAS:<p>Spirorenone (INN) is a novel aldosterone antagonist with anti-salt corticosteroid activity, used in metabolic disease research.</p>Formula:C24H28O3Purity:98.28% - 99.84%Color and Shape:SolidMolecular weight:364.4810β,17β-dihydroxyestra-1,4-dien-3-one
CAS:<p>10β,17β-dihydroxyestra-1,4-dien-3-one (DHED) has neuroprotective effects, can improve cognitive dysfunction, and can be used to study brain injury.</p>Formula:C18H24O3Color and Shape:SolidMolecular weight:288.38Epelsiban
CAS:<p>Epelsiban is a selective and orally bioavailable oxytocin receptor antagonist (pKi: 9.9 for human oxytocin receptor).</p>Formula:C30H38N4O4Purity:98%Color and Shape:SolidMolecular weight:518.65N-Benzylnaltrindole hydrochloride
CAS:<p>δ2 opioid receptor antagonist</p>Formula:C33H33ClN2O3Purity:98%Color and Shape:SolidMolecular weight:541.08LY3104607
CAS:<p>LY3104607 is an oral GPCR 40 agonist for type 2 diabetes, aimed at reducing glucose.</p>Formula:C27H25N3O3Purity:98%Color and Shape:SolidMolecular weight:439.51CIDD-0149897
CAS:<p>CIDD-0149897 is a potent, selective, and brain-penetrant agonist of ERβ that exhibits antitumor activity in glioblastoma [1].</p>Formula:C15H10FNO3Purity:98%Color and Shape:SolidMolecular weight:271.24H3B-6545 Hydrochloride
CAS:<p>H3B-6545 Hydrochloride is a selective, oral estrogen receptor covalent antagonist (SERCA).</p>Formula:C30H30ClF4N5O2Color and Shape:SolidMolecular weight:604.04HP210
CAS:<p>HP210, a selective glucocorticoid receptor modulator (SGRM), can suppress IL-1β and IL-6 mRNA expression, suggesting its utility in investigating inflammation-</p>Formula:C22H19N3O2S2Purity:98%Color and Shape:SolidMolecular weight:421.54ER degrader 6
CAS:<p>ER degrader 6 (compound 35s) is a potent selective estrogen receptor modulator (SERM) with the capacity to degrade Estrogen Receptor (ER)α.</p>Formula:C33H34FN3O5SSePurity:98%Color and Shape:SolidMolecular weight:682.66Androgen receptor degrader-2
CAS:<p>Androgen Receptor Degrader-2 (Compound 9) is a potent degrader of androgen receptors, with potential application in cancer research [1].</p>Formula:C16H16ClN3O4Purity:98%Color and Shape:SolidMolecular weight:349.77N-Nitrosodicyclohexylamine
CAS:<p>N-Nitrosodicyclohexylamine (NDCHA), an N-nitrosocompound, exhibits anti-androgenic activity by competitively binding to the androgen receptor (AR) in opposition</p>Formula:C12H22N2OPurity:98%Color and Shape:SolidMolecular weight:210.32Androgen receptor degrader-1
CAS:<p>Androgen Receptor Degrader-1 (Compound 18) is a potent agent for androgen receptor degradation, applicable in cancer research [1].</p>Formula:C15H14ClN3O4Purity:98%Color and Shape:SolidMolecular weight:335.74YXG-158
CAS:<p>YXG-158 (Compound 23-h), an orally active androgen receptor (AR) degrader and cytochrome P450 17A1 (CYP17A1) inhibitor, exhibits AR degradation with a DC50 of 1</p>Formula:C30H36FN3OPurity:98%Color and Shape:SolidMolecular weight:473.62Androgen receptor degrader-3
CAS:<p>Androgen Receptor Degrader-3 (ARD-3) is a compound that inhibits androgen receptor signaling and promotes the degradation of the receptor, with potential</p>Formula:C45H51ClN8O5Purity:98%Color and Shape:SolidMolecular weight:819.39N-Demethyl Mifepristone
CAS:<p>N-Demethyl Mifepristone (RU 42633), an active metabolite of Mifepristone, exhibits 61% of the affinity for the glucocorticoid receptor relative to Mifepristone'</p>Formula:C28H33NO2Purity:98%Color and Shape:SolidMolecular weight:415.57
