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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3178 products of "Endocrinology/Hormones"

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  • Yp537

    CAS:
    <p>Yp537 acts as an estrogen receptor (ER) inhibitor, specifically preventing the dimerization of the human estrogen receptor [1].</p>
    Formula:C64H104N13O22PS
    Color and Shape:Solid
    Molecular weight:1470.62
  • Nurr1 agonist 2

    CAS:
    <p>Nurr1 agonist 2 with EC50 of 0.07 μM, boosts TH &amp; VMAT2 mRNA, binds Nurr1 LBD at Kd 0.14 μM, for parkinsonism study.</p>
    Formula:C18H14O3S
    Purity:98.78%
    Color and Shape:Soild
    Molecular weight:310.37
  • Cgp 38560

    CAS:
    <p>CGP 38560 is a potent renin inhibitor.</p>
    Formula:C40H67N5O9S2
    Color and Shape:Solid
    Molecular weight:826.12
  • Methylprednisolone Acetate


    <p>Methylprednisolone Acetate(Depo-Medrate) has the ability to inhibit oxygen free radicals and can be used to treat acute spinal cord injuries.</p>
    Formula:C24H32O6
    Purity:99.74%
    Color and Shape:Off-White Solid
    Molecular weight:416.51
  • GNE-274

    CAS:
    <p>GNE-274, akin to GDC-0927 but non-degrading, is a partial ER agonist in breast cancer, enhancing chromatin at ER sites, inhibiting ER-LBD.</p>
    Formula:C29H31NO4
    Color and Shape:Solid
    Molecular weight:457.57
  • Axelopran

    CAS:
    <p>Axelopran (TD-1211) treats opioid constipation; it's a potent, selective peripheral opioid blocker.</p>
    Formula:C26H39N3O4
    Color and Shape:Solid
    Molecular weight:457.61
  • Raloxifene 6-glucuronide

    CAS:
    <p>Raloxifene 6-glucuronide is a primary metabolite of Raloxifene. Raloxifene 6-glucuronide is mediated mostly by UGT1A1 and UGT1A8.</p>
    Formula:C34H35NO10S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:649.71
  • GLL 398

    CAS:
    <p>GLL 398 is an orally active and selective degrader of estrogen receptor with an IC50 of 1.14 nM. GLL 398 blocks tumor growth in xenograft breast cancer models.</p>
    Formula:C25H23BO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:398.26
  • OT-R antagonist 2

    CAS:
    <p>OT-R antagonist 2 is a nonpeptide low molecular weight antagonist of OT-R .</p>
    Formula:C28H29N3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:471.55
  • BI 653048

    CAS:
    <p>BI 653048 is a selective and orally active agonist of nonsteroidal glucocorticoid (IC50: 55 nM). BI 653048 is also an HCV NS3 protease inhibitor.</p>
    Formula:C23H25F4N3O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:515.52
  • PROTAC ER Degrader-4

    CAS:
    <p>PROTAC ER Degrader-4 is a PROATC degrader of estrogen receptor (ER)(IC50 of 0.8 nM).</p>
    Formula:C53H67F3N6O8S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1005.2
  • Linuron

    CAS:
    <p>Linuron herbicide disrupts photosynthesis and acts as an androgen receptor antagonist.</p>
    Formula:C9H10Cl2N2O2
    Purity:99.08%
    Color and Shape:White Crystalline Solid Linuron Is A Colorless Crystals Non Corrosive Used As An Herbicide
    Molecular weight:249.09
  • DAMGO (TFA)

    CAS:
    <p>DAMGO is a selective peptide agonist of the µ-opioid receptor .</p>
    Formula:C28H36F3N5O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:627.61
  • 3-epi-25-hydroxy Vitamin D3

    CAS:
    <p>3-epi-25-hydroxy Vitamin D3 lowers serum PTH in male weanling rats at 0.5 and 1 IU/g doses; doesn't affect females.</p>
    Formula:C27H44O2
    Color and Shape:Solid
    Molecular weight:400.64
  • GPR88 agonist 2


    <p>GPR88 agonist 2 (compound 53) serves as a potent, brain-penetrant agonist of GPR88, exhibiting an EC50 of 14 µM in the GPR88 cAMP functional assay [1].</p>
    Color and Shape:Odour Solid
  • Epi-Cryptoacetalide


    <p>Epi-Cryptoacetalide is a useful organic compound for research related to life sciences and the catalog number is T126054.</p>
    Formula:C18H22O3
    Color and Shape:Solid
    Molecular weight:286.371
  • Antitumor agent-195


    <p>Antitumor agent-195 (compound 16c) is a dual-targeting agent that simultaneously targets STAT3 and NQO1. At a concentration of 1 μM, it significantly inhibits the phosphorylation of STAT3 at the Tyr705 site and effectively induces apoptosis in MDA-MB-231 and MDA-MB-468 breast cancer cells. As a substrate of NQO1, Antitumor agent-195 markedly increases ROS production, causing severe DNA damage in a dose-dependent manner. It also demonstrates strong antitumor properties in MDA-MB-231 xenograft models.</p>
    Formula:C22H22N2O4
    Color and Shape:Solid
    Molecular weight:378.42
  • ODM-204

    CAS:
    <p>ODM-204 is novel nonsteroidal dual inhibitor of both androgen receptor and CYP17A1 enzyme(IC50s of 80 nM and 22 nM, respectively).</p>
    Formula:C20H21F3N4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:374.40
  • Ac-RYYRIK-NH2

    CAS:
    <p>NOP site high affinity ligand (Ki=1.5 nM); blocks nociceptin effects in rat brain/heart; agonist in vivo, reduces mouse movement.</p>
    Formula:C44H70N14O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:939.12
  • BigLEN(mouse)

    CAS:
    <p>GPR171 agonist from ProSAAS controls mouse appetite, reduces glutamate in paraventricular neurons via G protein.</p>
    Formula:C78H130N24O22
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1756.03