Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(229 products)
- Annexin A(16 products)
- Aromatase(23 products)
- Estrogen/progestogen Receptor(66 products)
- GPR(1 products)
- Glucocorticoid Receptor(165 products)
- LHRH(2 products)
- Opioid Receptor(327 products)
- Prostaglandin Receptor(122 products)
- RAAS(89 products)
- Reductase(51 products)
- Somatostatin(57 products)
- Thyroid hormone receptor(THR)(33 products)
- Vasopressin Receptor(48 products)
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Found 3420 products of "Endocrinology/Hormones"
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Olmesartan medoxomil impurity C
CAS:Impurity C of Olmesartan medoxomil is a selective AT1 inhibitor with an IC50 of 66.2 μM.Formula:C29H28N6O5Color and Shape:SolidMolecular weight:540.57Azilsartan Medoxomil Potassium
CAS:Azilsartan Medoxomil Potassium (TAK-491 Potassium) is an orally administered angiotensin II receptor type 1 antagonist with IC50 of 0.62 nM, which used in the treatment of adults with essential hypertension.Formula:C30H23N4O8·KPurity:99.99%Color and Shape:SolidMolecular weight:606.62Hydrocortisone sodium succinate
CAS:Hydrocortisone sodium succinate is a glucocorticoid which is used to alleviate allergic reactions, particularly those of the skin and gums.Formula:C25H34NaO8Color and Shape:SolidMolecular weight:485.529L 363564
CAS:L 363564 is a kidney renin inhibitor.Formula:C54H76N12O10Color and Shape:SolidMolecular weight:1053.276ST-CY14
ST-CY14 is an inhibitor of the Nur77-PPARγ interaction with an EC50 of 3.15 μM. It binds to Nur77 (Kd=32 nM) to prevent its ubiquitination and degradation by PPARγ, reducing fatty acid uptake and mitochondrial respiration, and inhibiting the transcription of CD36 and FABP4. ST-CY14 suppresses proliferation and migration of MCF7 and MDA-MB-231 cancer cells and impedes tumor growth and bone metastasis in mouse models.Formula:C139H237N57O31S2Color and Shape:SolidMolecular weight:3266.86PTP1B/AKR1B1-IN-2
PTP1B/AKR1B1-IN-2 (Compound 7f) is a potent inhibitor targeting both PTP1B and AKR1B1 with IC50 values of 3.2 and 2.1 μM, respectively, and K i values of 4.0Formula:C23H23NO4S2Purity:98%Color and Shape:SolidMolecular weight:441.56AZ 1729
CAS:FFA2 modulator; inhibits cAMP, enhances 35SGTPγS binding (pEC50: 6.9, 7.23); alters Gi/Gq signaling; affects lipolysis, neutrophil migration.Formula:C18H16FN5OSColor and Shape:SolidMolecular weight:369.42Estrogen receptor modulator 6
CAS:ER modulator 6 (3a) is a potent ERβ agonist with a K i of 0.44 nM; 19x more selective for ERβ than ERα.
Formula:C18H16F2O3Color and Shape:SolidMolecular weight:318.32Ro 64-6198
CAS:Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP>opioid affinity.Formula:C26H31N3OPurity:98%Color and Shape:SolidMolecular weight:401.54AKR1B10-IN-1
CAS:AKR1B10-IN-1: potent AKR1B10 inhibitor, IC50 3.5 nM; hinders lung cancer cell growth, spread, and Cisplatin resistance.Formula:C19H16FNO4Color and Shape:SolidMolecular weight:341.338UFP-101
CAS:Strong, selective NOP receptor antagonist with pKi=10.24; >3000x selectivity over δ, μ, κ receptors; blocks nociceptin effects.
Formula:C82H138N32O21Purity:98%Color and Shape:SolidMolecular weight:1908.19T4-ATA (S-isomer)
T4-ATA S-isomer, the active form of the thyroid hormone, represents the S-isomer of T4-ATA.Formula:C19H15I4NO6SPurity:98%Color and Shape:SolidMolecular weight:893.01U-54494A hydrochloride
CAS:U-54494A hydrochloride is a benzamide derivative related to kappa opioid receptor agonists. U-54494A hydrochloride has anticonvulsant activity.Formula:C18H25Cl3N2OColor and Shape:SolidMolecular weight:391.76[Sar1, Ile8]-Angiotensin II TFA
[Sar1,Ile8]-Angiotensin II (TFA) contracts arteries and affects cell growth in vascular muscle.Formula:C48H74F3N13O12Purity:98%Color and Shape:SolidMolecular weight:1082.18Herkinorin
CAS:Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.Formula:C28H30O8Color and Shape:SolidMolecular weight:494.53PROTAC ER Degrader-3
CAS:PROTAC ER Degrader-3 from patent WO2017201449A1 is a PAC synthesis intermediate for ADC/PROTAC antibody conjugates, boosting ERα degradation.Formula:C71H77N7O12Purity:98%Color and Shape:SolidMolecular weight:1220.434Alclometasone
CAS:Alclometasone is a glucocorticoid that reduces inflammation and treats various skin conditions like eczema and psoriasis.Formula:C22H29ClO5Purity:98%Color and Shape:SolidMolecular weight:408.92Dynorphin B (1-13)
CAS:Dynorphin B (1-13) acts as an agonist on opioid κ-receptor.Formula:C74H115N21O17Purity:98%Color and Shape:SolidMolecular weight:1570.84Antihypertensive agent 3
Antihypertensive agent 3 (compound 4a), an angiotensin II receptor 1 antagonist, demonstrates antihypertensive activity in spontaneously hypertensive rats (SHRsFormula:C16H13NO4SColor and Shape:SolidMolecular weight:315.34Neuropeptide AF (human)
CAS:Neuropeptide AF (93-110), Human is an endogenous antiopioid peptide.Formula:C90H132N26O25Purity:98%Color and Shape:SolidMolecular weight:1978.17
