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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3178 products of "Endocrinology/Hormones"

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  • Endomorphin 2 TFA

    CAS:
    <p>Endomorphin 2 TFA, displays reasonable affinities for kappa3 binding sites, with Ki value between 20 and 30 nM.</p>
    Formula:C34H38F3N5O7
    Color and Shape:Solid
    Molecular weight:685.69
  • Valsartan-d9

    CAS:
    <p>Valsartan D9: deuterium-labeled, angiotensin II receptor antagonist, treats hypertension &amp; heart failure.</p>
    Formula:C24H29N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:444.57
  • Valsartan Ethyl Ester

    CAS:
    <p>Valsartan Ethyl Ester, an impurity in Valsartan, treats hypertension and heart failure by blocking angiotensin II receptors.</p>
    Formula:C26H33N5O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:463.57
  • Azilsartan-d5

    CAS:
    <p>Azilsartan (TAK-536) D5 is the deuterium-labeled Azilsartan. Azilsartan is a specific antagonist of the angiotensin II type 1 receptor.</p>
    Formula:C25H20N4O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:461.48
  • Asimadoline

    CAS:
    <p>Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, Germany.</p>
    Formula:C27H30N2O2
    Color and Shape:Solid
    Molecular weight:414.54
  • VTP-27999 Hydrochloride

    CAS:
    <p>VTP-27999 Hcl is an alkyl amine Renin inhibitor; VTP-27999 is useful for Hypertension and End-Organ Diseases.<br><br>IC50 value:<br><br>Target: Renin</p>
    Formula:C26H42Cl2N4O5
    Color and Shape:Solid
    Molecular weight:561.55
  • ARD-1676

    CAS:
    <p>ARD-1676 is an orally administered androgen receptor (AR) PROTAC degrader that combines an AR ligand with a cereblon ligand.</p>
    Formula:C44H46ClN7O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:788.33
  • GPR41 agonist-1

    CAS:
    <p>GPR41 agonist-1 is a GPR41 agonist, used for studying metabolic diseases such as diabetes and obesity.</p>
    Formula:C24H23N3O4
    Purity:98.40%
    Color and Shape:Solid
    Molecular weight:417.46
  • Protirelin

    CAS:
    <p>Protirelin (Thyroliberin) is a tripeptide that stimulates the release of thyrotropin and prolactin.</p>
    Formula:C16H22N6O4
    Purity:99.76%
    Color and Shape:White Or Almost White Powder
    Molecular weight:362.38
  • GPR40 agonist 6

    CAS:
    <p>GPR40 agonist 6 (Compound 7a) is a potent and selective agonist of free fatty acid receptor 1 ( FFAR1 or GPR40 ) with an EC 50 of 0.058 μM against GPR40 [1].</p>
    Formula:C20H19NO4
    Color and Shape:Solid
    Molecular weight:337.37
  • MS 15203

    CAS:
    <p>MS 15203 is a GPR171 agonist that reduces chronic neuropathic and inflammatory pain in male mice.</p>
    Formula:C12H11NO5
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:249.22
  • Beclomethasone 17-propionate

    CAS:
    <p>Beclomethasone 17-propionate is the active metabolite of BDP. As a GR agonist, 17-BMP inhibits the production of pro-inflammatory cytokines.</p>
    Formula:C25H33ClO6
    Purity:98.06%
    Color and Shape:Solid
    Molecular weight:464.98
  • Hydrocortisone cypionate

    CAS:
    <p>Hydrocortisone cypionate is a corticosteroid ester and synthetic glucocorticoid corticosteroid.</p>
    Formula:C29H42O6
    Color and Shape:Solid
    Molecular weight:486.64
  • AVE 0991 sodium salt

    CAS:
    <p>AVE 0991, a nonpeptide, oral Mas agonist, binds [125I]-Ang-(1-7) with IC50 of 21±35 nM.</p>
    Formula:C29H31N4NaO5S2
    Color and Shape:Solid
    Molecular weight:602.7
  • D4-abiraterone

    CAS:
    <p>D4-abiraterone is the active metabolite of abiraterone.Δ4-Abiraterone is a inhibitor of CYP17A1, 3β-HSD and SRD5A, and an antagonist of the androgen receptor.</p>
    Formula:C24H29NO
    Purity:99.75% - 99.8%
    Color and Shape:Solid
    Molecular weight:347.49
  • Taltirelin

    CAS:
    <p>Taltirelin (TA-0910) is at thyrotropin-releasing hormone receptor (TRH-R) superagonist (IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in</p>
    Formula:C17H23N7O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:405.41
  • (Rac)-PF-998425

    CAS:
    <p>(Rac)-PF-998425: nonsteroidal AR antagonist, potent &amp; selective, IC50: 26 nM (binding), 90 nM (cellular), potential for androgenetic alopecia study.</p>
    Formula:C14H14F3NO
    Color and Shape:Solid
    Molecular weight:269.267
  • Angiotensin II (3-8), human

    CAS:
    <p>Angiotensin II (3-8), human is a less effective agonist at the angiotensin AT1 receptor.</p>
    Color and Shape:Solid
  • Endoxifen Z-isomer hydrochloride

    CAS:
    <p>Endoxifen Z-isomer hydrochloride (Endoxifen HCl) is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.</p>
    Formula:C25H28ClNO2
    Color and Shape:Solid
    Molecular weight:409.95
  • AMG7703

    CAS:
    <p>AMG7703 is a bioactive chemical.</p>
    Formula:C14H15ClN2OS
    Color and Shape:Solid
    Molecular weight:294.8
  • Rezvilutamide

    CAS:
    <p>Rezvilutamide (SHR3680) is an orally available androgen receptor inhibitor that crosses the blood-brain barrier and has antitumor activity.</p>
    Formula:C22H20F3N3O4S
    Purity:99.97%
    Color and Shape:Solid
    Molecular weight:479.47
  • Leelamine hydrochloride

    CAS:
    <p>Leelamine hydrochloride, a pine bark extract, inhibits androgen receptor and CB1, reducing lipid synthesis in prostate cancer.</p>
    Formula:C20H32ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.93
  • Apalutamide-13C-d3


    <p>Apalutamide-13C-d3 is a 13C and 2H labeled Apalutamide. Apalutamide is an androgen receptor (AR) antagonist, used in research on prostate diseases.</p>
    Formula:CC20H12F4N5O2SD3
    Color and Shape:Solid
    Molecular weight:481.45
  • AZD1979

    CAS:
    <p>AZD1979 is a highly potent MCHR1 (Melanin-concentrating hormone receptor 1) antagonist , CNS exposure and insulin sensitivity in steady-state model assessments,</p>
    Formula:C25H26N4O5
    Purity:99.72%
    Color and Shape:Solid
    Molecular weight:462.5
  • Alvimopan dihydrate (LY246736 dihydrate)

    CAS:
    <p>Alvimopan dihydrate is a potent, oral μ-opioid receptor blocker (IC50 1.7 nM, Ki 0.47 nM) used in postoperative ileus research.</p>
    Formula:C25H36N2O6
    Color and Shape:Solid
    Molecular weight:460.56
  • Losartan (D4 Carboxylic Acid)

    CAS:
    <p>Losartan D4 Carboxylic Acid is the deuterium labeled Losartan, which is an angiotensin II receptor antagonist.</p>
    Formula:C22H21ClN6O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.92
  • Pamoic acid disodium

    CAS:
    <p>Pamoic acid disodium is a GPR35 agonist.</p>
    Formula:C23H16NaO6
    Purity:99.73%
    Color and Shape:Yellow Powder
    Molecular weight:411.36
  • 2-Bromoestradiol

    CAS:
    <p>2-Bromoestradiol, an estrogen 2-hydroxylase inhibitor, reduces the irreversible binding of radiolabeled estradiol metabolite(s) to microsomal proteins [1].</p>
    Formula:C18H23BrO2
    Color and Shape:Solid
    Molecular weight:351.28
  • Monomethyl fumarate-d3

    CAS:
    <p>Monomethyl fumarate D3 is a deuterium labeled Monomethyl fumarate.</p>
    Formula:C5H6O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:133.12
  • BMS-986121

    CAS:
    <p>BMS-986121 is a selective positive allosteric modulator (PAM) of the μ opioid receptor with analgesic effects.</p>
    Formula:C15H9Cl2N3O2S
    Purity:99.67%
    Color and Shape:Solid
    Molecular weight:366.22
  • 5β-Dihydroprogesterone

    CAS:
    <p>5β-Dihydroprogesterone (5β-DHP) is a progesterone receptor agonist and metabolite of progesterone .1,2It is formed from progesterone by 5β-reductase.25β-DHP</p>
    Formula:C21H32O2
    Color and Shape:Solid
    Molecular weight:316.485
  • ML334

    CAS:
    <p>ML334 (LH601A) is an NRF2 activator that inhibits cardiac fibroblast activation and proliferation ameliorating myocardial infarction-induced cardiac fibrosis.</p>
    Formula:C26H26N2O5
    Purity:98.06% - 98.06%
    Color and Shape:Solid
    Molecular weight:446.49
  • GDC-0927

    CAS:
    <p>GDC-0927 is a novel,non-steroidal, potent, orally bioavailable, selective estrogen receptor antagonist.</p>
    Formula:C28H28FNO4
    Color and Shape:Solid
    Molecular weight:461.52
  • Prednisolone valerate acetate

    CAS:
    <p>Prednisolone valerate acetate is a prodrug anti-inflammatory and immunosuppressive,converted to the active form of Prednisolone and glucocorticoid receptor.</p>
    Formula:C28H38O7
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:486.6
  • Azilsartan mepixetil

    CAS:
    <p>Azilsartan mepixetil: potent, long-acting angiotensin II blocker, safely lowers blood pressure, protects heart and kidneys.</p>
    Formula:C36H34N6O8
    Color and Shape:Solid
    Molecular weight:678.702
  • Olmesartan-d4

    CAS:
    <p>Olmesartan D4 is the deuterium labeled Olmesartan. Olmesartan is an antagonist of angiotensin II receptor (AT1R) used to treat high blood pressure.</p>
    Formula:C24H26N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:450.53
  • NQO1 substrate

    CAS:
    <p>NQO1 substrate is a highly potent NQO1 substrate with potential antitumor activity for leukemia research.</p>
    Formula:C13H2F2N4O
    Purity:98.02% - 98.02%
    Color and Shape:Solid
    Molecular weight:268.18
  • Vanilpyruvic acid

    CAS:
    <p>Vanillylpyruvic acid is a phenylpyruvic acid derivative applicable in biochemical experiments and drug synthesis research.</p>
    Formula:C10H10O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:210.18
  • GW-1100

    CAS:
    <p>GW-1100 is a selective GPR40 and FFAR1 antagonist for the study of diabetes and metabolic diseases.</p>
    Formula:C27H25FN4O4S
    Purity:97.01%
    Color and Shape:Solid
    Molecular weight:520.58
  • TA 0910 acid-type

    CAS:
    <p>TA 0910 acid-type is a metabolite of TA 0910. TA-0910 is a metabolically stable analog of thyrotropin-releasing hormone.</p>
    Formula:C17H22N6O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:406.39
  • Betamethasone acetate

    CAS:
    <p>Betamethasone acetate, the 21-acetate ester of betamethasone, is a synthetic glucocorticoid corticosteroid and a corticosteroid ester.</p>
    Formula:C24H31FO6
    Color and Shape:Solid
    Molecular weight:434.50
  • PD 123319 ditrifluoroacetate

    CAS:
    <p>PD 123319 ditrifluoroacetate is a selective non-peptide AT2 receptor antagonist with IC50 of 34 nM.</p>
    Formula:C35H34F6N4O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:736.66
  • Diflorasone Diacetate

    CAS:
    <p>Diflorasone Diacetate, a topical glucocorticoid, has immunosuppressive and anti-inflammatory properties.</p>
    Formula:C26H32F2O7
    Color and Shape:Crystals
    Molecular weight:494.53
  • Fenarimol

    CAS:
    <p>Fenarimol, a pyrimidine-type fungicide, exhibits potent inhibitory activity against BR biosynthesis.</p>
    Formula:C17H12Cl2N2O
    Color and Shape:Solid
    Molecular weight:331.2
  • Dienestrol diacetate

    CAS:
    <p>Dienestrol diacetate, a derivative of the synthetic non-steroid phenolic compound, DIENESTROL, exhibits estrogenic activities.</p>
    Formula:C22H22O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:350.41
  • Hydrocortisone buteprate

    CAS:
    <p>Hydrocortisone buteprate is a medium-potent, non-halogenated double-ester of hydrocortisone with a highly favorable benefit-to-risk ratio for inflammatory skin disorders.</p>
    Formula:C28H40O7
    Purity:99.19%
    Color and Shape:Solid
    Molecular weight:488.61
  • Candesartan-d4

    CAS:
    <p>Candesartan D4 is the deuterium labeled Candesartan. Candesartan is an antagonist of angiotensin II receptor.</p>
    Formula:C24H20N6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:444.48
  • Enalaprilat

    CAS:
    <p>Enalaprilat (Enalapril acid) is an ACE inhibitor used in the study of cardiovascular disease.</p>
    Formula:C18H24N2O5
    Purity:97.28%
    Color and Shape:Solid
    Molecular weight:348.39
  • Trans-Diethyl-1,1,1',1'-Stilbestrol-3,3',5,5'-d8

    CAS:
    <p>Trans-Diethyl-1,1,1',1'-Stilbestrol-3,3',5,5'-d8 is a deuterated compound of Trans-Diethyl-Stilbestrol. Trans-Diethyl-Stilbestrol has a CAS number of 56-53-1. Diethylstilbestrol is used in the treatment of menopausal and postmenopausal disorders.</p>
    Formula:C18H12D8O2
    Color and Shape:Solid
    Molecular weight:276.40
  • CGP-42112

    CAS:
    <p>CGP-42112 is an agonist of the Angiotensin-II subtype 2 receptor (AT2 R).</p>
    Formula:C52H69N13O11
    Color and Shape:White Solid
    Molecular weight:1052.18