Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(209 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(49 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(297 products)
- Prostaglandin Receptor(120 products)
- RAAS(87 products)
- Reductase(52 products)
- Somatostatin(49 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
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Found 3183 products of "Endocrinology/Hormones"
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FSH receptor antagonist 1
CAS:<p>FSH receptor antagonist 1 (compound 10) is a potent antagonist of the G(s) protein-coupled human follicle-stimulating hormone (FSH) receptor. It exhibits an IC50 value of 28 nM in cell lines expressing the human FSH receptor. This compound significantly inhibits follicle growth and ovulation in in vitro mouse models.</p>Formula:C33H32N2O2Color and Shape:SolidMolecular weight:488.619L-371,257
CAS:<p>L-371,257 is a competitive antagonist of oxytocin receptor with pA2 of 8.4 and Ki of 19 nM. L-371,257 shows a Ki of 3.7 nM for vasopressin receptor 1a.</p>Formula:C28H33N3O6Purity:99.79%Color and Shape:SolidMolecular weight:507.58GLPG0974
CAS:<p>GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.</p>Formula:C25H25ClN2O4SPurity:99.8%Color and Shape:SolidMolecular weight:484.99ZD 7155 hydrochloride
CAS:<p>ZD 7155 hydrochloride is an angiotensin II receptor type 1 (AT1 receptor) antagonist.</p>Formula:C26H27ClN6OPurity:99.8%Color and Shape:SolidMolecular weight:474.98Cort108297
CAS:<p>Cort108297: selective GR modulator/antagonist, high GR affinity (Ki: 0.45nM), no other steroid receptor affinity.</p>Formula:C26H25F4N3O3SPurity:98.36% - 99.94%Color and Shape:SolidMolecular weight:535.55Nalmefene
CAS:<p>Nalmefene (ORF 11676) is a μ-opioid antagonist and partial κ agonist used in the study of opioid overdose and alcohol dependence.</p>Formula:C21H25NO3Purity:99.86%Color and Shape:SolidMolecular weight:339.43(E/Z)-GSK5182
CAS:<p>GSK5182 is a racemic mix of (E/Z) isomers, a selective ERRγ inverse agonist (IC50: 79 nM), and induces ROS in liver cancer.</p>Formula:C27H31NO3Purity:97.58%Color and Shape:SolidMolecular weight:417.54LSZ-102
CAS:<p>LSZ-102 is an effective and selective degrader of estrogen receptor (IC50 = 0.2 nM) and can be used in studies about ERα positive breast cancer.</p>Formula:C25H17F3O4SPurity:98.56%Color and Shape:SolidMolecular weight:470.46ML314
CAS:<p>ML314 is a brain-permeable nonpeptide β-inhibin-biased neurotensin NTR1 receptor agonist (EC50: 1.9 μM), a biased neurotensin receptor ligand for methamphetamine abuse that inhibits NTR2 and GPR35.</p>Formula:C24H28N4O3Purity:99.52%Color and Shape:SolidMolecular weight:420.504ZK 216348
CAS:<p>ZK 216348 also binds to Progesterone and mineralocorticoid receptors (IC50s: 20.4 nM and 79.9 nM, respectively). ZK 216348 is a nonsteroidal selective glucocorticoid receptor agonist (IC50: 20.3 nM). ZK 216348 has an anti-inflammatory activity similar to</p>Formula:C24H23F3N2O5Purity:98%Color and Shape:SolidMolecular weight:476.45PSN632408
CAS:<p>PSN632408 is an optimized agonist of GPR119 receptors that display similar potency to OEA at both recombinant mouse and human GPR119 receptors (EC50: 5.6 and 7.9 uM, respectively).</p>Formula:C18H24N4O4Purity:98%Color and Shape:SolidMolecular weight:360.41Mapracorat
CAS:<p>Mapracorat (ZK-245186, BOL-303242X) is a selective glucocorticoid receptor agonist,anti-inflammatory agent for atopic dermatitis and allergic conjunctivitis.</p>Formula:C25H26F4N2O2Color and Shape:SolidMolecular weight:462.48(S)-Mapracorat
CAS:<p>(S)-Mapracorat is a selective and less active agonist of the glucocorticoid receptor.</p>Formula:C25H26F4N2O2Color and Shape:SolidMolecular weight:462.48Relacorilant
CAS:<p>Relacorilant is an oral glucocorticoid receptor antagonist with Ki of 7.2 nM, potential for treating Cushing's syndrome.</p>Formula:C27H22F4N6O3SPurity:98.53% - 99%Color and Shape:SolidMolecular weight:586.56Budesonide
CAS:<p>Budesonide (Pulmicort), an anti-inflammatory corticosteroid, has shown the effective glucocorticoid activitie and few mineralocorticoid activities. According to reports, Budesonide has extensively inhibitory effects against multiple cells types and mediators referred to allergic and nonallergic-mediated inflammatory. What's more, the anti-inflammatory action of budesonide has been revealed to contribute to the effectiveness of asthma.</p>Formula:C25H34O6Purity:99.03% - 99.72%Color and Shape:Crystals SolidMolecular weight:430.53Ref: TM-T0094
Discontinued productExemestane
CAS:<p>Exemestane (EXE) is an Aromatase Inhibitor. The mechanism of action of exemestane is as an Aromatase Inhibitor.</p>Formula:C20H24O2Purity:99.35% - 99.35%Color and Shape:White To Light Yellow Crystal PowderMolecular weight:296.421-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione
<p>21-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione is a valuable organic compound for life sciences research [Catalog No.: T67476, CAS No.: 37413-91-5].</p>Formula:C23H26O4Color and Shape:SolidMolecular weight:366.457Phosphoramidon Disodium
CAS:<p>Phosphoramidon Disodium (Phosphoramidon Disodium Salt) Salt is a metalloendopeptidase inhibitor, widely used as a biochemical tool.</p>Formula:C23H34N3Na2O10PPurity:98%Color and Shape:SolidMolecular weight:588.48GPR109 receptor agonist-2
CAS:<p>Compound 5, a selective GPR109a agonist, exhibits a pEC50 value of 5.53 [1].</p>Formula:C7H10N2O2Color and Shape:SolidMolecular weight:154.17PF-998425
CAS:<p>non-steroidal androgen receptor (AR) antagonist</p>Formula:C14H14F3NOPurity:98%Color and Shape:SolidMolecular weight:269.26AZD9496 maleate
CAS:<p>AZD9496 maleate is a highly potent and selective antagonist of the estrogen receptor alpha (ERα), exhibiting an IC50 value of 0.28 nM. This compound, AZD9496 maleate, is an orally bioavailable selective estrogen receptor degrader (SERD).</p>Formula:C29H29F3N2O6Color and Shape:SolidMolecular weight:558.554ERB-196
CAS:<p>Erb-196 is an estrogen receptor-receptor agonist with non-steroidal selectivity.</p>Formula:C17H10FNO2Purity:98%Color and Shape:SolidMolecular weight:279.27L-372662
CAS:<p>L-372662 is bioactive chemical.</p>Formula:C33H38N4O6Color and Shape:SolidMolecular weight:586.68Pamoic acid
CAS:<p>Pamoic acid is the orphan G protein-coupled receptor GPR35 agonist. Pamoic acid activates ERK and beta-arrestin2 and causes antinociceptive activity.</p>Formula:C23H16O6Purity:99.99%Color and Shape:Fine Yellow PowderMolecular weight:388.37SR17018
CAS:<p>SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.</p>Formula:C19H18Cl3N3OPurity:99.89%Color and Shape:SolidMolecular weight:410.72Cebranopadol
CAS:<p>Cebranopadol (GRT6005) is an analgesic NOP and opioid receptor agonist with Kis of 0.9 nM, 0.7 nM, 2.6 nM, 18 nM for human NOP, μ-opioid (MOP), κ-opioid (KOP)</p>Formula:C24H27FN2OPurity:98.32% - 99.78%Color and Shape:SolidMolecular weight:378.48YK11
CAS:<p>YK11 is an androgen receptor partial agonist that activates androgen receptor transcriptional activity in HEK293 cells overexpressing androgen receptors when used at a concentration of 0.1 μM, with osteogenic activity.</p>Formula:C25H34O6Purity:98.91%Color and Shape:SoildMolecular weight:430.53Ceronapril
CAS:<p>Ceronapril (SQ 29852) is an orally active and potent angiotensin-converting enzyme (ACE) inhibitor (IC50 : 36 nM) for the study of dementia and hypertension.</p>Formula:C21H33N2O6PPurity:97.94%Color and Shape:SolidMolecular weight:440.47Ref: TM-T25226
Discontinued productBromadoline maleate
CAS:<p>Bromadoline is an opioid analgesic selective for the μ-opioid receptor.</p>Formula:C19H25BrN2O5Purity:98%Color and Shape:SolidMolecular weight:441.322SR14150
CAS:<p>SR14150 is a partial agonist of high-affinity NOP receptor.</p>Formula:C21H30N2OPurity:98%Color and Shape:SolidMolecular weight:326.48Estrogen receptor modulator 8
CAS:<p>Estrogen Receptor Modulator 8 (compound 4) is an orally active inhibitor targeting Estrogen Receptor/ERR α with potent efficacy (IC50 = 0.437 nM in MCF-7 cells</p>Formula:C25H24F4N2O2Purity:98%Color and Shape:SolidMolecular weight:460.46MOR agonist-1
CAS:<p>MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and is utilized in research concerning pain and associated</p>Formula:C22H26ClFN2O2Purity:98%Color and Shape:SolidMolecular weight:404.91ALS-I-41
CAS:<p>ALS-I-41 is a novel, potent and selective antagonist of oxytocin receptor.</p>Formula:C30H38FN3O6SPurity:98%Color and Shape:SolidMolecular weight:587.7
