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Endocrinology/Hormones

Endocrinology/Hormones

Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.

Subcategories of "Endocrinology/Hormones"

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Found 3183 products of "Endocrinology/Hormones"

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  • Zuclomiphene citrate

    CAS:
    <p>Zuclomiphene citrate, a cis isomer of Clomiphene, has stronger antiestrogenic effects and better inhibits LH secretion.</p>
    Formula:C32H36ClNO8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:598.08
  • Ono-3805 sodium

    CAS:
    <p>Ono-3805 is an inhibitor of nonsteroidal 5 alpha-reductase.</p>
    Formula:C31H37NNaO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:526.629
  • SC 51316

    CAS:
    <p>SC 51316 is a nonpeptidic angiotensin II (AII) receptor antagonist.</p>
    Formula:C24H29N7O
    Color and Shape:Solid
    Molecular weight:431.53
  • Estrogen receptor β antagonist 2

    CAS:
    <p>Estrogen receptor β antagonist 2 is a selective, potent estrogen receptor β (ERβ) antagonist that acts on Erα (IC50: 109.10 μM) and Erβ (IC50: 0.63 μM).</p>
    Formula:C23H26N2O6
    Color and Shape:Solid
    Molecular weight:426.46
  • LGD-2226

    CAS:
    <p>LGD-2226: selective oral androgen receptor modulator, EC50: 0.2nM, Ki: 1.5nM. Treats muscle loss, osteoporosis, sexual issues.</p>
    Formula:C14H9F9N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:392.22
  • LY191704

    CAS:
    <p>LY 191704 is a 5α-reductase type 1 inhibitor.</p>
    Formula:C14H16ClNO
    Color and Shape:Solid
    Molecular weight:249.74
  • L-159282

    CAS:
    <p>L-159282 is an orally active and nonpeptide angiotensin II receptor antagonist. It also has anti-hypertensive activity.</p>
    Formula:C30H28N4O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:524.63
  • DK1

    CAS:
    <p>DK1: potent ERRα modulator, lowers blood glucose, promising for diabetes research.</p>
    Formula:C16H13ClN2O2
    Color and Shape:Solid
    Molecular weight:300.74
  • Carbazole derivative 1

    CAS:
    <p>Carbazole derivative 1 is used to reduce androgen or oestrogen levels in mammals.</p>
    Formula:C18H13FN2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:276.31
  • (R)-DPN

    CAS:
    <p>estrogen receptor (ER) β agonist</p>
    Formula:C15H13NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:239.27
  • AT2R antagonist 1

    CAS:
    <p>AT2R antagonist 1: potent, selective ligand, Ki 29 nM, inhibits CYP enzymes, stable in liver microsomes.</p>
    Formula:C23H30N4O4S2
    Color and Shape:Solid
    Molecular weight:490.64
  • JTC-801 free base

    CAS:
    <p>JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).</p>
    Formula:C26H25N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:411.5
  • Viminol

    CAS:
    <p>Viminol is an opioid analgesic. Viminol is based on the α-pyrryl-2-aminoethanol structure, unlike any other class of opioids.</p>
    Formula:C21H31ClN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:362.94
  • Lubabegron fumarate

    CAS:
    <p>Lubabegron (LY591281, LY488756 fumarate) is a beta-agonist approved in 2018 to lower ammonia in cattle waste, aiding environment and health.</p>
    Formula:C29H29N3O3SC4H4O4
    Color and Shape:Solid
    Molecular weight:557.66
  • GSK706

    CAS:
    <p>GSK706 is a novel effective agonist of the GPR119.</p>
    Formula:C23H29N5O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:471.57
  • GPR35 agonist 3

    CAS:
    <p>GPR35 agonist 3 is a synthetic GPR35 agonist used in the study of cancer, type 2 diabetes and cardiovascular disease.</p>
    Formula:C12H9NO5S
    Purity:98.80%
    Color and Shape:Solid
    Molecular weight:279.27
  • NNC45-0781

    CAS:
    <p>NNC45-0781 is a tissue-selective partial-agonist of estrogen.</p>
    Formula:C27H29NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:415.52
  • AZD2906

    CAS:
    <p>AZD2906: selective GR agonist with human/rat IC50s - 2.2/0.3 nM (PBMC), 41.6/7.5 nM (blood); induces rat bone marrow micronuclei.</p>
    Formula:C26H25FN4O3
    Color and Shape:Solid
    Molecular weight:460.5
  • PF-3882845

    CAS:
    <p>PF-3882845, a high affinity MR antagonist (IC50=2.7 nM) for hypertension, also targets progesterone receptor (IC50: 310 nM).</p>
    Formula:C24H22ClN3O2
    Purity:99.63%
    Color and Shape:Solid
    Molecular weight:419.9
  • FK-739 free acid

    CAS:
    <p>FK-739, an angiotensin II receptor blocker, inhibits rat aorta binding (IC50=8.6 nM) but not bovine cerebellum.</p>
    Formula:C24H23N7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:409.49
  • CAY10595

    CAS:
    <p>CAY10595 is an antagonist of the CRTh2 (DP2) receptor with a Ki of 10 nM.</p>
    Formula:C20H13Cl2FN2O5
    Purity:99.95% - 99.97%
    Color and Shape:Solid
    Molecular weight:451.23
  • Chlorothiazide Sodium

    CAS:
    <p>diuretic and antihypertensive</p>
    Formula:C7H6ClN3NaO4S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:318.71
  • Aldose reductase-IN-2

    CAS:
    <p>Aldose reductase-IN-2 (5f) inhibits AR with antioxidant effects; potential anti-diabetic drug.</p>
    Formula:C25H28N4O5
    Color and Shape:Solid
    Molecular weight:464.51
  • CR-665 Acetate

    CAS:
    <p>CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.</p>
    Formula:C38H53N9O6
    Color and Shape:Solid
    Molecular weight:731.899
  • AZ12216052

    CAS:
    <p>AZ12216052 is a GRP8 antagonist with anxiolytic and anti-inflammatory activity and can be used to study obesity and metabolic disorders.</p>
    Formula:C19H22BrNOS
    Purity:99.29%
    Color and Shape:Solid
    Molecular weight:392.35
  • (R)-Viloxazine Hydrochloride

    CAS:
    <p>(R)-Viloxazine Hydrochloride, the R-isomer of Viloxazine.</p>
    Formula:C13H20ClNO3
    Purity:99.88% - 99.94%
    Color and Shape:Solid
    Molecular weight:273.76
  • CRTh2 antagonist 1

    CAS:
    <p>CRTh2 antagonist 1 is a CRTh2 antagonist (IC50: 89 nM).</p>
    Formula:C23H25N3O5S
    Purity:97.24%
    Color and Shape:Solid
    Molecular weight:455.53
  • L 364918

    CAS:
    <p>L 364918 is an oxytocin antagonist.</p>
    Formula:C40H54N8O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:742.91
  • HG122

    CAS:
    <p>HG122 promotes AR degradation via proteasome, inhibiting castration-resistant prostate cancer.</p>
    Formula:C15H13N5O5
    Color and Shape:Solid
    Molecular weight:343.29
  • (1R,2R)-2-PCCA hydrochloride

    CAS:
    <p>(1R,2R)-2-PCCA HCl: Potent, selective GPR88 agonist, crosses BBB, EC50 1140 nM in mouse striatum. Useful for CNS research.</p>
    Formula:C30H39Cl2N3O
    Purity:98.75% - 99.67%
    Color and Shape:Solid
    Molecular weight:528.56
  • CPSA

    CAS:
    <p>CPSA is an effective and selective AKR1C1 inhibitor.</p>
    Formula:C13H9ClO3
    Color and Shape:Solid
    Molecular weight:248.66
  • Bopindolol fumarate

    CAS:
    <p>Bopindolol fumarate: non-selective β1/β2-adrenoceptor blocker, partial agonist, low β3 affinity, treats hypertension.</p>
    Formula:C27H32N2O7
    Color and Shape:Solid
    Molecular weight:496.56
  • LY2444296

    CAS:
    <p>LY2444296 (FP3FBZ) is an orally active and selective antagonist of kappa opioid receptor(Ki = 1 nM).</p>
    Formula:C24H22F2N2O2
    Purity:99.18%
    Color and Shape:Solid
    Molecular weight:408.44
  • TUG-469

    CAS:
    <p>TUG-469 is an agonist of free fatty acid 1(FFA) receptor.</p>
    Formula:C23H23NO2
    Purity:99.73%
    Color and Shape:Solid
    Molecular weight:345.43
  • Fispemifene

    CAS:
    <p>Fispemifene (HM-101) is an estrogen receptor modulator (SERM) used to treat genitourinary syndromes and vaginal atrophy.</p>
    Formula:C26H27ClO3
    Purity:98.74% - 99.67%
    Color and Shape:Solid
    Molecular weight:422.94
  • Renin inhibitor-1

    CAS:
    <p>Renin inhibitor-1 (compound 26) is a potent, orally active renin inhibitor capable of acting on rh-renin (IC50: 0.9 nM) and hPRA (IC50: 1.8 nM). renal disease.</p>
    Formula:C22H30N4O4
    Color and Shape:Solid
    Molecular weight:414.5
  • Desketoraloxifene

    CAS:
    <p>Desketoraloxifene is a selective estrogen receptor modulator, inhibiting mammalian PLD (PLD1 and PLD2).</p>
    Formula:C27H27NO3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:445.57
  • Org-34517

    CAS:
    <p>Org-34517, a glucocorticoid receptor (GR) antagonist, is used potentially for the treatment of depression.</p>
    Formula:C28H30O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:430.54
  • GW7604

    CAS:
    <p>GW7604 is an antiestrogen and it also is the metabolite of GW5638. GW5638 is an antagonist of high-affinity estrogen receptor (ER).</p>
    Formula:C25H22O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:370.44
  • ICI 154,129

    CAS:
    <p>Selective δ opioid antagonist</p>
    Formula:C34H46N4O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:638.82
  • Prednisolone Tebutate

    CAS:
    <p>Prednisolone Tebutate is a synthetic glucocorticoid, and is an antiinflammatory and immunosuppressant.</p>
    Formula:C27H38O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:458.59
  • SR8993

    CAS:
    <p>SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.</p>
    Formula:C25H37FN4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:412.59
  • LY2048978

    CAS:
    <p>LY2048978: orally-active kappa antagonist, shows promise for mood and addiction in animal studies.</p>
    Formula:C19H24N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:312.41
  • AZD7268

    CAS:
    <p>AZD7268 is a potent, selective, reversible, and orally bioavailable agonist of δ-opioid receptor with CNS penetration.</p>
    Formula:C29H30N4O2S
    Color and Shape:Solid
    Molecular weight:498.64
  • Tolonidine

    CAS:
    <p>Tolonidine is orally active and has been shown to possess hypotensive. Tolonidine is a derivative of imidazoline.</p>
    Formula:C10H12ClN3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:209.68
  • AT-076

    CAS:
    <p>AT-076: κ-opioid (Ki=1.14 nM) &amp; nociceptin (Ki=1.75 nM) noncompetitive antagonist; μ-opioid (Ki=1.67 nM) &amp; δ-opioid (Ki=19.6 nM) competitive antagonist.</p>
    Formula:C26H35N3O3
    Color and Shape:Solid
    Molecular weight:437.57
  • RU 45144

    CAS:
    <p>RU 45144 is an estradiol derivative with antiestrogenic activity.</p>
    Formula:C28H37NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:435.6
  • Zuclomiphene

    CAS:
    <p>Zuclomiphene is a nonsteroidal selective estrogen receptor modulator (SERM) with triphenylethylene group.</p>
    Formula:C26H28ClNO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:405.96
  • AC-7954

    CAS:
    <p>AC-7954 is a potent and efficacious agonist of urotensin II receptor.</p>
    Formula:C19H20ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.82
  • Fidarestat

    CAS:
    <p>Fidarestat (SNK 860),Aldose reductase inhibitor (IC50=26 nM). Targets AKR1B10 (33 μM) and V301L AKR1B10 (1.8 μM). Potential diabetes treatment.</p>
    Formula:C12H10FN3O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:279.22