Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(208 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(48 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(297 products)
- Prostaglandin Receptor(119 products)
- RAAS(86 products)
- Reductase(52 products)
- Somatostatin(46 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
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Found 3180 products of "Endocrinology/Hormones"
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BI-2081
CAS:<p>BI-2081: GPR40 agonist, EC50=4nM, boosts insulin, lowers blood glucose, potential for type 2 diabetes research.</p>Formula:C32H35FO6Color and Shape:SolidMolecular weight:534.62ES 8891
CAS:<p>ES 8891 is an inhibitor of renin.</p>Formula:C42H60N6O6SPurity:98%Color and Shape:SolidMolecular weight:777.03Fulvestrant (R enantiomer)
CAS:<p>Fulvestrant R enantiomer is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.</p>Formula:C32H47F5O3SPurity:98%Color and Shape:SolidMolecular weight:606.77CITFA
CAS:<p>CITFA, a GPER agonist, enhances neurite outgrowth in rat embryonic (E18) hippocampal neurons [1].</p>Formula:C25H35NO2Color and Shape:SolidMolecular weight:381.55Arzoxifene hydrochloride
CAS:<p>Arzoxifene hydrochloride is a selective estrogen receptor modulator that is a potent estrogen antagonist in mammary and uterine tissue.</p>Formula:C28H30ClNO4SPurity:98%Color and Shape:SolidMolecular weight:512.06LY303336
CAS:<p>LY303336 is an antagonist of AT1 receptor.</p>Formula:C30H37N4O11PSPurity:98%Color and Shape:SolidMolecular weight:692.67H3B-6545
CAS:<p>H3B-6545 is a selective and oral estrogen receptor covalent antagonist (SERCA) used in the research of metastatic ER-positive, HER2-negative breast cancer.</p>Formula:C30H29F4N5O2Color and Shape:SolidMolecular weight:567.58DPI-3290
CAS:<p>DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent</p>Formula:C30H34FN3O2Purity:98%Color and Shape:SolidMolecular weight:487.61RU 59063
CAS:<p>RU 59063 is a prototype of a new class of high-affinity nonsteroidal androgen receptor (AR) ligands.</p>Formula:C17H18F3N3O2SPurity:99.09%Color and Shape:SolidMolecular weight:385.4L-368899 free base
CAS:<p>L-368899: non-peptide, oral oxytocin receptor antagonist (IC50: 8.9 nM), 40x more selective than vasopressin V1a/V2.</p>Formula:C26H42N4O5S2Purity:98%Color and Shape:SolidMolecular weight:554.778,11-Eicosadiynoic acid
CAS:<p>8,11-Eicosadiynoic acid, an unsaturated fatty acid, functions as a steroid 5α-reductase inhibitor and has applications in acne research [1].</p>Formula:C20H32O2Color and Shape:SolidMolecular weight:304.47Conjugated Estrogen sodium
CAS:<p>Conjugated estrogens treat menopause symptoms, vaginal changes, and certain cancers.</p>Formula:C18H19NaO5SPurity:98%Color and Shape:White Needle CrystalMolecular weight:370.39SNC 162
CAS:<p>SNC 162 is a potent and selective delta-opioid receptor (δ-opioid) agonist with analgesic, antidepressant and antiarrhythmic effects.</p>Formula:C27H37N3OPurity:98%Color and Shape:SolidMolecular weight:419.6MCHR1 antagonist 3
CAS:<p>MCHR1 antagonist 3, a potent antagonist of the melanin-concentrating hormone receptor-1 (MCHR1), is employed for the regulation of energy metabolism.</p>Formula:C29H36N4O2Purity:98%Color and Shape:SolidMolecular weight:472.62ER degrader 1
CAS:<p>ER degrader 1 targets estrogen receptor, crucial for cell regulation; shows promise in cancer therapy. (Patent WO2021139756A1, compound 11)</p>Formula:C26H32F4N4O3Color and Shape:SolidMolecular weight:524.55LY2922083
CAS:<p>LY2922083: Potent, selective GPR40 agonist; lowers glucose, boosts insulin and GLP-1.</p>Formula:C31H33NO3SColor and Shape:SolidMolecular weight:499.66Deltakephalin
CAS:<p>Deltakephalin is a synthetic, potent specific opiate delta receptors agonist.</p>Formula:C34H48N6O10Purity:98%Color and Shape:SolidMolecular weight:700.78TP-051
CAS:<p>TP-051 is a FFAR1 agonist.</p>Formula:C29H31FO6SColor and Shape:SolidMolecular weight:526.62MK-8666 Tris
CAS:<p>MK-8666, a partial GPCR agonist, targets GPR40 to enhance insulin secretion, potentially treating type 2 diabetes without adverse effects.</p>Formula:C33H42N2O9SColor and Shape:SolidMolecular weight:642.764LGD-2941
CAS:<p>LGD-2941 is an androgen receptor modulator. LGD-2941 is used for the treatment of hypogonadism, female sexual dysfunction and menopausal syndrome.</p>Formula:C17H16F6N2O2Color and Shape:SolidMolecular weight:394.31AMG 837 sodium salt
CAS:AMG 837 sodium salt: potent GPR40 agonist, EC50=13 nM; enhances insulin secretion; superior pharmacokinetics.Formula:C26H21F3NaO3Purity:98%Color and Shape:SolidMolecular weight:461.436RU28362
CAS:<p>RU28362 is an agonist of glucocorticoid receptor.</p>Formula:C23H28O3Color and Shape:SolidMolecular weight:352.47MK-386
CAS:<p>MK-386 is a potent and selective inhibitor of human type-1 5alpha-reductase.</p>Formula:C28H49NOColor and Shape:SolidMolecular weight:415.69Naloxonazine
CAS:<p>Naloxonazine, a potent, selective opiate mu-1 (μ1) antagonist, also influences leishmania through the modulation of host coding function.</p>Formula:C38H42N4O6Color and Shape:SolidMolecular weight:650.76Nurr1 agonist 4
CAS:<p>Nurr1 agonist 4 (compound 8) serves as a potent Nurr1 agonist, exhibiting an EC50 value of 2.1 μM [1].</p>Formula:C12H10O4Purity:98%Color and Shape:SolidMolecular weight:218.21LY2922470
CAS:<p>LY2922470: Selective GPR40 agonist; EC50=7nM (human), 1nM (mouse), 3nM (rat); lowers glucose, boosts insulin/GLP-1.</p>Formula:C28H29NO4SPurity:95.11% - 97.08%Color and Shape:SolidMolecular weight:475.6μ opioid receptor agonist 3
CAS:<p>Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.</p>Formula:C22H28N2O2Purity:98%Color and Shape:SolidMolecular weight:352.47Glucocorticoid receptor agonist
CAS:<p>Glucocorticoid receptor agonist is an effective glucocorticoid receptor agonist.</p>Formula:C20H20F4N2O2Purity:98%Color and Shape:SolidMolecular weight:396.38BMS-814580
CAS:<p>BMS-814580: potent MCHR1 antagonist, Kb 117 nM, Ki 17 nM (human), 4.9/11.5 nM (monkey/rat), reduces feeding/weight in rodents.</p>Formula:C24H19ClF2N2O4SColor and Shape:SolidMolecular weight:504.93μ opioid receptor agonist 1
CAS:<p>μ opioid receptor agonist 1 (Compound H-1a) is an optically pure oxyheterocyclic substituted pyrroloxypyrazole derivative and an MOR receptor agonist that can</p>Formula:C26H38N4OColor and Shape:SolidMolecular weight:422.61(rel)-BMS-641988
CAS:<p>(rel)-BMS-641988, a relative configuration of the potent nonsteroidal androgen receptor antagonist BMS-641988, holds potential for prostate cancer research.</p>Formula:C20H20F3N3O5SPurity:98%Color and Shape:SolidMolecular weight:471.45AM-1638
CAS:<p>AM-1638 is an orally active GPR40/FFA1 agonist, useful for studying type II diabetes.</p>Formula:C33H35FO4Color and Shape:SolidMolecular weight:514.63TR antagonist 1
CAS:<p>TR antagonist 1 is a highly potent thyroid hormone receptor (TR) antagonist that can be used to study diseases caused by endocrine abnormalities.</p>Formula:C25H23Br2NO4Purity:99.57%Color and Shape:SolidMolecular weight:561.26AMG 837
CAS:<p>Prinaberel (ERB 041) is an ERβ agonist with anticancer activity and anti-inflammatory activity that inhibits the NFκB pro-inflammatory signaling pathway.</p>Formula:C26H21F3O3Purity:98%Color and Shape:SolidMolecular weight:438.44Naloxonazine dihydrochloride
CAS:<p>μ1 receptor antagonist</p>Formula:C38H43ClN4O6Purity:98%Color and Shape:SolidMolecular weight:687.22CYT-1010
CAS:<p>CYT-1010, a mu-opioid receptor agonist; EC50: β-arrestin, 13.1 nM; cAMP, 0.0053 nM. Extracted from patent WO2013173730A2.</p>Formula:C35H40N6O5Purity:98%Color and Shape:SolidMolecular weight:624.73BE-26263
CAS:<p>BE-26263, an antiosteoporotic agent isolated from Scedosporium apiospermum, exhibits an estrogenic effect [1].</p>Formula:C32H38O14Color and Shape:SolidMolecular weight:646.64Dexamethasone palmitate
CAS:<p>DXP, a lipophilic prodrug of Dexamethasone, has 47x less glucocorticoid receptor affinity; it's an agonist & anti-inflammatory.</p>Formula:C38H59FO6Purity:99.28%Color and Shape:SolidMolecular weight:630.87R-84760 hydrochloride
CAS:<p>R-84760, a potent κ-opioid receptor agonist, relieves tonic pain via supraspinal/spinal pathways, activating noradrenergic descent.</p>Formula:C19H25Cl3N2OSColor and Shape:SolidMolecular weight:435.84ADL-08-0011
CAS:<p>ADL-08-0011 is an metabolite of alvimopan.</p>Formula:C23H29NO3Color and Shape:SolidMolecular weight:367.49VPC-14228
CAS:<p>VPC-14228 is a specific AR-DBD inhibitor that acts by inhibiting both Y594A and Q592A mutants.</p>Formula:C13H14N2OSPurity:99.96%Color and Shape:SolidMolecular weight:246.33ICI 204448
CAS:<p>ICI 204448 is a potent and peripherally selective κ-opioid agonist.</p>Formula:C23H26Cl2N2O4Color and Shape:SolidMolecular weight:465.37Glucocorticoid receptor-IN-1
CAS:<p>Glucocorticoid receptor-IN-1 selectively modulates GR with anti-inflammatory effects, represses hMMP1 (IC50: 2.11 nM), and activates MMTV (EC50: 5.59 nM).</p>Formula:C24H19F4N7O2Color and Shape:SolidMolecular weight:513.45TC OT 39
CAS:<p>oxytocin receptor partial agonist</p>Formula:C32H40N8O2SPurity:98%Color and Shape:SolidMolecular weight:600.78IP7e
CAS:<p>IP7e (isoxazolo-pyridinone 7e) is a Nurr1 activator with an EC50 value of 3.9 nM.</p>Formula:C23H22N2O4Purity:99.86%Color and Shape:SolidMolecular weight:390.43Halobetasol
CAS:<p>Halobetasol (Ulobetasol), a corticosteroid, is utilized in the research of severe localized psoriasis [1].</p>Formula:C22H27ClF2O4Purity:98%Color and Shape:SolidMolecular weight:428.9GSK 1440115
CAS:<p>GSK 1440115, an orally active urotensin II receptor antagonist, is used to treat asthma.</p>Formula:C30H29Cl2N3O6Purity:98%Color and Shape:SolidMolecular weight:598.47Spirorenone
CAS:<p>Spirorenone (INN) is a novel aldosterone antagonist with anti-salt corticosteroid activity, used in metabolic disease research.</p>Formula:C24H28O3Purity:98.28% - 99.84%Color and Shape:SolidMolecular weight:364.4810β,17β-dihydroxyestra-1,4-dien-3-one
CAS:<p>10β,17β-dihydroxyestra-1,4-dien-3-one (DHED) has neuroprotective effects, can improve cognitive dysfunction, and can be used to study brain injury.</p>Formula:C18H24O3Color and Shape:SolidMolecular weight:288.38RU 58668
CAS:<p>Pure antiestrogen that downregulates estrogen receptor expression</p>Formula:C34H43F5O5SPurity:98%Color and Shape:SolidMolecular weight:658.76
