Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(208 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(48 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(297 products)
- Prostaglandin Receptor(119 products)
- RAAS(86 products)
- Reductase(52 products)
- Somatostatin(46 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
Show 6 more subcategories
Found 3180 products of "Endocrinology/Hormones"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Norleual
CAS:<p>Angiotensin IV analog, potent HGF/c-MET inhibitor (IC50=3 pM), halts MDCK cell growth and invasion, AT4 antagonist, impairs LTP, antiangiogenic.</p>Formula:C41H58N8O7Purity:98%Color and Shape:SolidMolecular weight:774.95Herkinorin
CAS:<p>Herkinorin: μ-opioid agonist with 100x μ-affinity, 50x less κ-affinity than Salvinorin A, from Salvia divinorum. Semi-synthetic from Salvinorin B.</p>Formula:C28H30O8Color and Shape:SolidMolecular weight:494.53PROTAC ER Degrader-3
CAS:<p>PROTAC ER Degrader-3 from patent WO2017201449A1 is a PAC synthesis intermediate for ADC/PROTAC antibody conjugates, boosting ERα degradation.</p>Formula:C71H77N7O12Purity:98%Color and Shape:SolidMolecular weight:1220.434Methylpiperidino pyrazole
CAS:<p>Methylpiperidino pyrazole is an ERα inhibitor and can prevent the BPS-induced Rb phosphorylation and cell cycle progression.</p>Formula:C29H31N3O3Purity:98.84%Color and Shape:SolidMolecular weight:469.57[Orn5]-URP
CAS:<p>Urotensin-II receptor antagonist, no agonist effect, pEC50 7.24, blocks U-II in rat aorta assay.</p>Formula:C48H62N10O10S2Purity:98%Color and Shape:SolidMolecular weight:1003.2PL-017
CAS:<p>μ opioid receptor agonist; IC50: 5.5 nM (μ), >10,000 nM (δ). Induces reversible analgesia, catalepsy, hyperthermia in rats.</p>Formula:C29H37N5O5Purity:98%Color and Shape:SolidMolecular weight:535.64[Met5]-Enkephalin, amide
CAS:<p>[Met5]-Enkephalin, amide activates δ and ζ opioid receptors; has multiple forms and varying plasma levels.</p>Formula:C27H36N6O6SPurity:98%Color and Shape:SolidMolecular weight:572.68(Rac)-SNC80
CAS:<p>(Rac)-SNC80, a racemic δ-opioid agonist (K i 1.78 nM), shows potential for treating various headache disorders.</p>Formula:C28H39N3O2Color and Shape:SolidMolecular weight:449.63Melanin Concentrating Hormone, salmon TFA
<p>MCH (salmon) TFA is a 19-amino-acid neuropeptide affecting appetite, energy, sleep, and heart health via GPCR SLC-1/GPR24 and MCHR2.</p>Formula:C91H140F3N27O26S4Color and Shape:SolidMolecular weight:2213.5(Rac)-Finerenone
CAS:<p>Rac-Finerenone, or (Rac)-BAY 94-8862, is an oral nonsteroidal MR antagonist with high selectivity and an IC50 of 18 nM.</p>Formula:C21H22N4O3Color and Shape:SolidMolecular weight:378.432Montirelin
CAS:<p>Montirelin is an analog of thyrotropin-releasing hormone.</p>Formula:C17H24N6O4SColor and Shape:SolidMolecular weight:408.483-Cl-Pyridine-amide-acrylaldehyde-piperazine
<p>3-Cl-Pyridine-amide-acrylaldehyde-piperazine serves as a synthetic intermediate for LO-4-25. LO-4-25 is a ligand for the androgen receptor (AR) DNA binding domain and is linked to a truncated fumaramide handle via a connector. In 22Rv1 cells, LO-4-25 demonstrates potent degradation of both AR and AR-V7.</p>Color and Shape:Odour SolidAkuammicine
CAS:<p>Akuammicine, as an indole alkaloid from Catharanthus roseus, can be used in cancer cell eradication.</p>Formula:C20H22N2O2Color and Shape:SolidMolecular weight:322.408Glucocorticoids receptor agonist 1
CAS:<p>GRA-1, an arylpyrazole, is a potent glucocorticoid receptor agonist with robust anti-inflammatory effects and preserves insulin secretion.</p>Formula:C20H23FN2OColor and Shape:SolidMolecular weight:326.41CP 85339
CAS:<p>CP 85339 is an aspartic acid protease inhibitor for X-ray analysis of peptide-renin complexes.</p>Formula:C31H49ClN4O6SColor and Shape:SolidMolecular weight:641.26Nociceptin(1-7)
CAS:<p>Bioactive metabolite of nociceptin, antagonist of nociceptin-induced hyperalgesia</p>Formula:C31H41N7O9Purity:98%Color and Shape:SolidMolecular weight:655.709Brain Natriuretic Peptide (1-32), rat
CAS:<p>Rat Brain Natriuretic Peptide (1-32) is a 32-amino-acid peptide from heart, released when ventricles stretch excessively.</p>Formula:C146H239N47O44S3Purity:98%Color and Shape:SolidMolecular weight:3452.944',2-Dihydroxy-4,6-dimethoxydihydrochalcone
CAS:<p>4',2-Dihydroxy-4,6-dimethoxydihydrochalcone, an estrogen-like compound, binds to bovine estrogen receptors, IC50 15 μM.</p>Formula:C17H18O5Color and Shape:SolidMolecular weight:302.32Lyciumin A
CAS:<p>Lyciumin A, a cyclic octapeptide, inhibits proteases and could aid in hypertension studies.</p>Formula:C42H51N9O12Color and Shape:SolidMolecular weight:873.921[(pF)Phe4]Nociceptin(1-13)NH2
CAS:<p>Potent, selective OP4 agonist; pKi=10.68, pEC50=9.80. >8000x selectivity vs other opioid receptors; long-lasting in vivo effects.</p>Formula:C61H99FN22O15Purity:98%Color and Shape:SolidMolecular weight:1399.6PSDalpha
<p>PSDalpha, a conjugate of PS, TB, and 17β-estradiol, degrades ERα with peak absorption at 465 nm, effectively inhibiting MCF-7 cell growth.</p>Formula:C44H39N3O2SColor and Shape:SolidMolecular weight:673.86PROTAC ERRα Degrader-2
CAS:<p>PROTAC ERRα Degrader-2 is a compound consisting of an MDM2 ligand binding group, a linker, and an estrogen-related receptor alpha (ERRα) binding group.</p>Formula:C57H55Cl2F6N7O8Purity:98%Color and Shape:SolidMolecular weight:1150.99Aliskiren D6 Hydrochloride
CAS:<p>Aliskiren (CGP 60536) D6 Hydrochloride is a deuterium-labeled Aliskiren. Aliskiren hemifumarate is a direct and orally active renin inhibitor (IC50: 1.5 nM).</p>Formula:C30H54ClN3O6Purity:98%Color and Shape:SolidMolecular weight:594.26Rofleponide
CAS:<p>Rofleponide is a synthetic glucocorticosteroid with a high affinity for the rat thymus glucocorticoid receptor.</p>Formula:C25H34F2O6Purity:99.32%Color and Shape:SolidMolecular weight:468.53Dermorphin Analog
<p>Dermorphin Analog, a heptapeptide from amphibian skin, binds μ-opioid receptors selectively and strongly.</p>Formula:C44H59N11O10Purity:98%Color and Shape:SolidMolecular weight:901.43Imidaprilate
CAS:<p>Imidaprilate, an active TA-6366 metabolite, is a potent ACE inhibitor with an IC50 of 2.6 nM, researched for hypertension.</p>Formula:C18H23N3O6Purity:98%Color and Shape:SolidMolecular weight:377.39Potassium Channel Targeted Library
<p>A unique collection of xnum potassium channel blockers and agonists for high throughput and high content screening;</p>Color and Shape:Odour SolidAngiotensin II (5-8), human
CAS:<p>Angiotensin II (5-8) is an endogenous C-terminal fragment of the peptide vasoconstrictor angiotensin II</p>Formula:C26H36N6O5Purity:98%Color and Shape:SolidMolecular weight:512.6Dipropyl phthalate
CAS:<p>Dipropyl phthalate is a weak androgen receptor inhibitor, and can be used in biochemical experiments and drug synthesis.</p>Formula:C14H18O4Purity:98.62%Color and Shape:SolidMolecular weight:250.29UFP-803
CAS:<p>UT receptor ligand acts mainly as silent antagonist with slight agonist effects; blocks U-II in rat aorta, pIC50 = 7.46, & inhibits plasma leakage in mice.</p>Formula:C50H64N10O12S2Purity:98%Color and Shape:SolidMolecular weight:1061.24[Ala17]-MCH
CAS:<p>Potent MCH receptor agonist with EC50 of 17 nM (MCH1) & 54 nM (MCH2); prefers MCH1 (Ki 0.16 nM) over MCH2 (Ki 34 nM).</p>Formula:C97H155N29O26S4Purity:98%Color and Shape:SolidMolecular weight:2271.71Aclerastide
CAS:<p>Aclerastide, an angiotensin receptor agonist, decreases fibrosis in wounds; effect increases with use duration, blocked by AT antagonist.</p>Formula:C42H64N12O11Color and Shape:SolidMolecular weight:913.03Yp537
CAS:<p>Yp537 acts as an estrogen receptor (ER) inhibitor, specifically preventing the dimerization of the human estrogen receptor [1].</p>Formula:C64H104N13O22PSColor and Shape:SolidMolecular weight:1470.62Methylprednisolone Acetate
<p>Methylprednisolone Acetate(Depo-Medrate) has the ability to inhibit oxygen free radicals and can be used to treat acute spinal cord injuries.</p>Formula:C24H32O6Purity:99.74%Color and Shape:Off-White SolidMolecular weight:416.51Nurr1 agonist 2
CAS:<p>Nurr1 agonist 2 with EC50 of 0.07 μM, boosts TH & VMAT2 mRNA, binds Nurr1 LBD at Kd 0.14 μM, for parkinsonism study.</p>Formula:C18H14O3SPurity:98.78%Color and Shape:SoildMolecular weight:310.37Axelopran
CAS:<p>Axelopran (TD-1211) treats opioid constipation; it's a potent, selective peripheral opioid blocker.</p>Formula:C26H39N3O4Color and Shape:SolidMolecular weight:457.61Cgp 38560
CAS:<p>CGP 38560 is a potent renin inhibitor.</p>Formula:C40H67N5O9S2Color and Shape:SolidMolecular weight:826.12Raloxifene 6-glucuronide
CAS:<p>Raloxifene 6-glucuronide is a primary metabolite of Raloxifene. Raloxifene 6-glucuronide is mediated mostly by UGT1A1 and UGT1A8.</p>Formula:C34H35NO10SPurity:98%Color and Shape:SolidMolecular weight:649.71GPR88 agonist 2
<p>GPR88 agonist 2 (compound 53) serves as a potent, brain-penetrant agonist of GPR88, exhibiting an EC50 of 14 µM in the GPR88 cAMP functional assay [1].</p>Color and Shape:Odour SolidGLL 398
CAS:<p>GLL 398 is an orally active and selective degrader of estrogen receptor with an IC50 of 1.14 nM. GLL 398 blocks tumor growth in xenograft breast cancer models.</p>Formula:C25H23BO4Purity:98%Color and Shape:SolidMolecular weight:398.26BI 653048
CAS:<p>BI 653048 is a selective and orally active agonist of nonsteroidal glucocorticoid (IC50: 55 nM). BI 653048 is also an HCV NS3 protease inhibitor.</p>Formula:C23H25F4N3O4SPurity:98%Color and Shape:SolidMolecular weight:515.523-epi-25-hydroxy Vitamin D3
CAS:<p>3-epi-25-hydroxy Vitamin D3 lowers serum PTH in male weanling rats at 0.5 and 1 IU/g doses; doesn't affect females.</p>Formula:C27H44O2Color and Shape:SolidMolecular weight:400.64DAMGO (TFA)
CAS:<p>DAMGO is a selective peptide agonist of the µ-opioid receptor .</p>Formula:C28H36F3N5O8Purity:98%Color and Shape:SolidMolecular weight:627.61Linuron
CAS:<p>Linuron herbicide disrupts photosynthesis and acts as an androgen receptor antagonist.</p>Formula:C9H10Cl2N2O2Purity:99.08%Color and Shape:White Crystalline Solid Linuron Is A Colorless Crystals Non Corrosive Used As An HerbicideMolecular weight:249.09OT-R antagonist 2
CAS:<p>OT-R antagonist 2 is a nonpeptide low molecular weight antagonist of OT-R .</p>Formula:C28H29N3O4Purity:98%Color and Shape:SolidMolecular weight:471.55GNE-274
CAS:<p>GNE-274, akin to GDC-0927 but non-degrading, is a partial ER agonist in breast cancer, enhancing chromatin at ER sites, inhibiting ER-LBD.</p>Formula:C29H31NO4Color and Shape:SolidMolecular weight:457.57Galloylalbiflorin
CAS:<p>Galloylalbiflorin, an AR antagonist with IC50 53.3μM, is sourced from Paeonia lactiflora roots, exhibiting anti-androgenic properties.</p>Formula:C30H32O15Color and Shape:SolidMolecular weight:632.57PTP1B/AKR1B1-IN-1
<p>PTP1B/AKR1B1-IN-1 is a dual inhibitor targeting protein tyrosine phosphatase 1B (PTP1B) and aldose reductase (AKR1B1), exhibiting inhibitory potency with IC50s</p>Formula:C22H21NO4S2Purity:98%Color and Shape:SolidMolecular weight:427.54BigLEN(mouse)
CAS:<p>GPR171 agonist from ProSAAS controls mouse appetite, reduces glutamate in paraventricular neurons via G protein.</p>Formula:C78H130N24O22Purity:98%Color and Shape:SolidMolecular weight:1756.03ODM-204
CAS:<p>ODM-204 is novel nonsteroidal dual inhibitor of both androgen receptor and CYP17A1 enzyme(IC50s of 80 nM and 22 nM, respectively).</p>Formula:C20H21F3N4Purity:98%Color and Shape:SolidMolecular weight:374.40
![[Orn5]-URP](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1928.webp&w=3840&q=75)
![[Met5]-Enkephalin, amide](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1255.webp&w=3840&q=75)
![[(pF)Phe4]Nociceptin(1-13)NH2](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1885.webp&w=3840&q=75)
![[Ala17]-MCH](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1997.webp&w=3840&q=75)
