Endocrinology/Hormones
Endocrinology/hormone inhibitors are compounds that block the action of hormones or interfere with hormone signaling pathways. These inhibitors are essential for studying the regulation of endocrine systems and for developing treatments for hormone-related diseases, such as diabetes, thyroid disorders, and hormone-dependent cancers. By modulating hormone activity, these inhibitors can help elucidate the complex interactions within the endocrine system. At CymitQuimica, we offer a wide range of high-quality endocrinology/hormone inhibitors to support your research in endocrinology, pharmacology, and medical sciences.
Subcategories of "Endocrinology/Hormones"
- Androgen Receptor(207 products)
- Annexin A(11 products)
- Aromatase(20 products)
- Estrogen/progestogen Receptor(49 products)
- GPR(1 products)
- Glucocorticoid Receptor(153 products)
- LHRH(1 products)
- Opioid Receptor(296 products)
- Prostaglandin Receptor(119 products)
- RAAS(86 products)
- Reductase(52 products)
- Somatostatin(46 products)
- Thyroid hormone receptor(THR)(26 products)
- Vasopressin Receptor(44 products)
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Found 3178 products of "Endocrinology/Hormones"
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Estrogen receptor antagonist 5
CAS:<p>Compound 165: Potent estrogen receptor antagonist; useful for metastatic disease research.</p>Formula:C25H31F3N2O3Color and Shape:SolidMolecular weight:464.52GSK 1440115
CAS:<p>GSK 1440115, an orally active urotensin II receptor antagonist, is used to treat asthma.</p>Formula:C30H29Cl2N3O6Purity:98%Color and Shape:SolidMolecular weight:598.47(1S,3R)-GNE-502
CAS:<p>(1S,3R)-GNE-502 degrades ERα in MCF7 cells; potent with EC50 of 13 nM; useful in estrogen-related cancer research.</p>Formula:C25H30FN3O3SColor and Shape:SolidMolecular weight:471.59JNJ-26146900
CAS:<p>JNJ-26146900 is a nonsteroidal androgen receptor (AR) ligand with tissue-selective activity in rats. JNJ-26146900 binds to the rat AR with a K(i) of 400nM.</p>Formula:C15H15F3N2O3SPurity:98%Color and Shape:SolidMolecular weight:360.35THRβ receptor agonist-1
CAS:<p>THRβ receptor agonist-1 is an agonist for the THRβ receptor [1].</p>Formula:C18H12Cl2N6O4Color and Shape:SolidMolecular weight:447.23THR-β modulator-1
CAS:<p>THR-β Modulator-1 (Compound 1a) is a potent modulator of the thyroid hormone receptor β, utilized in the study of thyroid hormone receptor-associated disorders</p>Formula:C17H14Cl2N6O4Color and Shape:SolidMolecular weight:437.24Dagrocorat
CAS:<p>Dagrocorat is a novel and dissociated agonist of glucocorticoid receptor.</p>Formula:C29H29F3N2O2Purity:98%Color and Shape:SolidMolecular weight:494.55GLL398
CAS:<p>GLL398: Oral ERα down-regulator, binds strongly (IC50=1.14nM), degrades ERα in MCF-7 cells (IC50=0.21μM).</p>Formula:C25H23BO4Color and Shape:SolidMolecular weight:398.26GPR120 Agonist 3
CAS:<p>GPR120 Agonist 3 (GPR120-IN-1) is a selective agonist of Gpr120 ( logEC50: -7.62).</p>Formula:C19H23ClF3NO3Purity:99.01%Color and Shape:SolidMolecular weight:405.84Prostaglandin E2-biotin
CAS:<p>Prostaglandin E2-biotin, an analog of prostaglandin, is utilized in the research of Nurr1-related diseases, including cancer and autoimmune diseases [1].</p>Formula:C35H58N4O6SColor and Shape:SolidMolecular weight:662.92Frakefamide
CAS:<p>Frakefamide: potent analgesic, μ-selective agonist, non-CNS penetrating.</p>Formula:C30H34FN5O5Purity:98%Color and Shape:SolidMolecular weight:563.62IP7e
CAS:<p>IP7e (isoxazolo-pyridinone 7e) is a Nurr1 activator with an EC50 value of 3.9 nM.</p>Formula:C23H22N2O4Purity:99.86%Color and Shape:SolidMolecular weight:390.43μ opioid receptor agonist 3
CAS:<p>Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.</p>Formula:C22H28N2O2Purity:98%Color and Shape:SolidMolecular weight:352.47Glucocorticoid receptor-IN-1
CAS:<p>Glucocorticoid receptor-IN-1 selectively modulates GR with anti-inflammatory effects, represses hMMP1 (IC50: 2.11 nM), and activates MMTV (EC50: 5.59 nM).</p>Formula:C24H19F4N7O2Color and Shape:SolidMolecular weight:513.45Icalcaprant
CAS:<p>Icalcaprant is a kappa-opioid receptor antagonist [1].</p>Formula:C23H26N4O3Purity:98%Color and Shape:SolidMolecular weight:406.48Fulvestrant (R enantiomer)
CAS:<p>Fulvestrant R enantiomer is the less active R enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.</p>Formula:C32H47F5O3SPurity:98%Color and Shape:SolidMolecular weight:606.77Mu opioid receptor antagonist 7
CAS:<p>Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (</p>Formula:C22H27ClN2O2Purity:98%Color and Shape:SolidMolecular weight:386.91Glucocorticoid receptor agonist
CAS:<p>Glucocorticoid receptor agonist is an effective glucocorticoid receptor agonist.</p>Formula:C20H20F4N2O2Purity:98%Color and Shape:SolidMolecular weight:396.38Estrogen receptor antagonist 3
CAS:<p>ER antagonist 3 degrades ER, crucial in cell regulation; ER antagonist 4 may aid cancer research. (Patent WO2021213358A1, compound 7)</p>Formula:C26H29BF6N4O2Color and Shape:SolidMolecular weight:554.34Triiodothyronine Sulfate
CAS:<p>Triiodothyronine sulfate: Hypothyroidism prodrug, metabolizes into active thyroid hormone T3, binds and activates TRβ1.</p>Formula:C15H11I3NNaO7SPurity:98%Color and Shape:SolidMolecular weight:753.02PD 125754
CAS:<p>PD 125754 is a Renin inhibitor, which represents a group of pharmaceutical drugs used primarily to treat essential hypertension.</p>Formula:C42H65N5O7Purity:98%Color and Shape:SolidMolecular weight:751.99Estrogen receptor modulator 7
CAS:<p>Estrogen Receptor Modulator 7 is a potent modulator of estrogen receptors, utilized in cancer research [1].</p>Formula:C30H31BCl2FNO3Purity:98%Color and Shape:SolidMolecular weight:554.29H3B-6545
CAS:<p>H3B-6545 is a selective and oral estrogen receptor covalent antagonist (SERCA) used in the research of metastatic ER-positive, HER2-negative breast cancer.</p>Formula:C30H29F4N5O2Color and Shape:SolidMolecular weight:567.58L-368899 free base
CAS:<p>L-368899: non-peptide, oral oxytocin receptor antagonist (IC50: 8.9 nM), 40x more selective than vasopressin V1a/V2.</p>Formula:C26H42N4O5S2Purity:98%Color and Shape:SolidMolecular weight:554.77Naloxonazine dihydrochloride
CAS:<p>μ1 receptor antagonist</p>Formula:C38H43ClN4O6Purity:98%Color and Shape:SolidMolecular weight:687.22BE-26263
CAS:<p>BE-26263, an antiosteoporotic agent isolated from Scedosporium apiospermum, exhibits an estrogenic effect [1].</p>Formula:C32H38O14Color and Shape:SolidMolecular weight:646.64MCHR1 antagonist 2
CAS:<p>MCHR1 antagonist 2 is an antagonist of melanin-concentratin hormone receptor 1(MCH1-R, IC50 = 65 nM) and also inhibits hERG.</p>Formula:C23H21FN2O5Purity:98.29%Color and Shape:SolidMolecular weight:424.42Fulvestrant (S enantiomer)
CAS:<p>Fulvestrant S enantiomer is the less active S enantiomer of Fulvestrant. Fulvestrant is a potent estrogen receptor antagonist with an IC50 of 9.4 nM.</p>Formula:C32H47F5O3SPurity:98%Color and Shape:SolidMolecular weight:606.77SQ 32970
CAS:<p>SQ 32970 is a potent Endothia aspartic proteinase inhibitor.</p>Formula:C33H51N5O4SColor and Shape:SolidMolecular weight:613.85Nur77 modulator 2
CAS:<p>Nur77 modulator 2: Kd of 0.35 μM, oral anti-inflammatory, affects Nur77/mitochondria localization.</p>Formula:C26H25NO5Color and Shape:SolidMolecular weight:431.48CITFA
CAS:<p>CITFA, a GPER agonist, enhances neurite outgrowth in rat embryonic (E18) hippocampal neurons [1].</p>Formula:C25H35NO2Color and Shape:SolidMolecular weight:381.55Arzoxifene hydrochloride
CAS:<p>Arzoxifene hydrochloride is a selective estrogen receptor modulator that is a potent estrogen antagonist in mammary and uterine tissue.</p>Formula:C28H30ClNO4SPurity:98%Color and Shape:SolidMolecular weight:512.06AMG 837 sodium salt
CAS:<p>AMG 837 sodium salt: potent GPR40 agonist, EC50=13 nM; enhances insulin secretion; superior pharmacokinetics.</p>Formula:C26H21F3NaO3Purity:98%Color and Shape:SolidMolecular weight:461.436TR antagonist 1
CAS:<p>TR antagonist 1 is a highly potent thyroid hormone receptor (TR) antagonist that can be used to study diseases caused by endocrine abnormalities.</p>Formula:C25H23Br2NO4Purity:99.57%Color and Shape:SolidMolecular weight:561.26TC OT 39
CAS:<p>oxytocin receptor partial agonist</p>Formula:C32H40N8O2SPurity:98%Color and Shape:SolidMolecular weight:600.78Spirorenone
CAS:<p>Spirorenone (INN) is a novel aldosterone antagonist with anti-salt corticosteroid activity, used in metabolic disease research.</p>Formula:C24H28O3Purity:98.28% - 99.84%Color and Shape:SolidMolecular weight:364.4810β,17β-dihydroxyestra-1,4-dien-3-one
CAS:<p>10β,17β-dihydroxyestra-1,4-dien-3-one (DHED) has neuroprotective effects, can improve cognitive dysfunction, and can be used to study brain injury.</p>Formula:C18H24O3Color and Shape:SolidMolecular weight:288.38Epelsiban
CAS:<p>Epelsiban is a selective and orally bioavailable oxytocin receptor antagonist (pKi: 9.9 for human oxytocin receptor).</p>Formula:C30H38N4O4Purity:98%Color and Shape:SolidMolecular weight:518.65N-Benzylnaltrindole hydrochloride
CAS:<p>δ2 opioid receptor antagonist</p>Formula:C33H33ClN2O3Purity:98%Color and Shape:SolidMolecular weight:541.08LY3104607
CAS:<p>LY3104607 is an oral GPCR 40 agonist for type 2 diabetes, aimed at reducing glucose.</p>Formula:C27H25N3O3Purity:98%Color and Shape:SolidMolecular weight:439.51CIDD-0149897
CAS:<p>CIDD-0149897 is a potent, selective, and brain-penetrant agonist of ERβ that exhibits antitumor activity in glioblastoma [1].</p>Formula:C15H10FNO3Purity:98%Color and Shape:SolidMolecular weight:271.24H3B-6545 Hydrochloride
CAS:<p>H3B-6545 Hydrochloride is a selective, oral estrogen receptor covalent antagonist (SERCA).</p>Formula:C30H30ClF4N5O2Color and Shape:SolidMolecular weight:604.04HP210
CAS:<p>HP210, a selective glucocorticoid receptor modulator (SGRM), can suppress IL-1β and IL-6 mRNA expression, suggesting its utility in investigating inflammation-</p>Formula:C22H19N3O2S2Purity:98%Color and Shape:SolidMolecular weight:421.54ER degrader 6
CAS:<p>ER degrader 6 (compound 35s) is a potent selective estrogen receptor modulator (SERM) with the capacity to degrade Estrogen Receptor (ER)α.</p>Formula:C33H34FN3O5SSePurity:98%Color and Shape:SolidMolecular weight:682.66Androgen receptor degrader-2
CAS:<p>Androgen Receptor Degrader-2 (Compound 9) is a potent degrader of androgen receptors, with potential application in cancer research [1].</p>Formula:C16H16ClN3O4Purity:98%Color and Shape:SolidMolecular weight:349.77N-Nitrosodicyclohexylamine
CAS:<p>N-Nitrosodicyclohexylamine (NDCHA), an N-nitrosocompound, exhibits anti-androgenic activity by competitively binding to the androgen receptor (AR) in opposition</p>Formula:C12H22N2OPurity:98%Color and Shape:SolidMolecular weight:210.32Androgen receptor degrader-1
CAS:<p>Androgen Receptor Degrader-1 (Compound 18) is a potent agent for androgen receptor degradation, applicable in cancer research [1].</p>Formula:C15H14ClN3O4Purity:98%Color and Shape:SolidMolecular weight:335.74YXG-158
CAS:<p>YXG-158 (Compound 23-h), an orally active androgen receptor (AR) degrader and cytochrome P450 17A1 (CYP17A1) inhibitor, exhibits AR degradation with a DC50 of 1</p>Formula:C30H36FN3OPurity:98%Color and Shape:SolidMolecular weight:473.62Androgen receptor degrader-3
CAS:<p>Androgen Receptor Degrader-3 (ARD-3) is a compound that inhibits androgen receptor signaling and promotes the degradation of the receptor, with potential</p>Formula:C45H51ClN8O5Purity:98%Color and Shape:SolidMolecular weight:819.39N-Demethyl Mifepristone
CAS:<p>N-Demethyl Mifepristone (RU 42633), an active metabolite of Mifepristone, exhibits 61% of the affinity for the glucocorticoid receptor relative to Mifepristone'</p>Formula:C28H33NO2Purity:98%Color and Shape:SolidMolecular weight:415.57
